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Contents…………

Titles Page No.

1. Introduction 01
2. Definition 01

3. Correlation between Preformulation and formulation 02

4. Steps in Preformulation Process Pharmaceutical Research 03


4.1. Stability
4.2. Solid State Compatibility
4.3. Physico-chemical Properties
4.4. Physico-mechanical Properties
4.5. In Vitro Availability Properties
4.6. Other Studies

5. Preformulation drug characterization program 05

5.1 UV Spectroscopy

5.2 Solubility Determination

5.3 Melting Point

5.4 Particle Size, Shape and Surface Area

5.5 Power Flow Properties

5.6 Chemical stability profile

5.7 Compatibility studies

5.8 Solution phase stability

5.9 Absorption behavior

6. Conclusion 19
References 20

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