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DERWENT

DRUG FILE
Thesaurus Part 3 Appendices
2004 Thomson. All rights reserved

Edition 11 ISBN: 1 903836 66 1

2004 Thomson

Published by Thomson Scientific 14 Great Queen Street, London WC2B 5DF, United Kingdom Visit the Thomson Scientific web site at http://www.thomson.com/scientific Edition 10 published August 1998 Edition 11 published March 2004 ISBN: ISBN: ISBN: ISBN: ISBN: ISBN: 0 901157 11 2 0 901157 16 3 0 901157 21 X 1 903836 64 5 1 903836 65 3 1 903826 66 1 (Edition 10 part 1) (Edition 10 part 2) (Edition 10 part 3) (Edition 11 part 1) (Edition 11 part 2) (Edition 11 part 3)

All rights reserved. No part of this publication may be reproduced, stored in a retrieval system or transmitted in any form or by any means electronic, mechanical, recording, photocopying or otherwise without express written permission from the copyright owner.

Derwent Drug File Thesaurus

CONTENTS

INTRODUCTION ................................... 1 A .......................................................... 5 B ........................................................ 83 C ...................................................... 135 D ...................................................... 223 E ...................................................... 279 F ...................................................... 315 G ..................................................... 347 |H ..................................................... 377 I ....................................................... 415 J ....................................................... 449 K ...................................................... 455 L ...................................................... 469 M ..................................................... 511 N ...................................................... 571 O ..................................................... 611

P ...................................................... 633 Q ..................................................... 709 R ...................................................... 713 S ...................................................... 755 T ...................................................... 833 U ...................................................... 885 V ...................................................... 899 W ..................................................... 915 X ...................................................... 927 Y ...................................................... 931 Z ...................................................... 937 NUMBERS ........................................ 945 APPENDIX A ..................................... 951 APPENDIX B ..................................... 975 APPENDIX C ................................... 1029 APPENDIX D ................................... 1043

Derwent Drug File 951 Thesaurus

APPENDIX A
The following list provides definitions of terms whose meaning is not self-evident nor to be found in standard reference books. Many terms also have Related Terms, More Specific Terms and/ or suggested strategy (Codeless Scanning) for searching the older files. Only the appropriate elements are included for each term, so an entry may have only a definition, or only a Codeless Scanning strategy, etc. The entries under * More Specific comprise more precise keywords for that concept, but do not include specific examples. The entry for ANALGESICS, for instance, does not list all the drugs covered by this term. Where corresponding drug activity and classification terms exist, (e.g. ANALGESIC and ANALGESICS), only the plural, classification terms are included in this Appendix. Because one pharmacological Index Term was routinely assigned to most drugs in Codeless Scanning, whether or not that activity was actually studied, it is not always possible to distinguish between drug activity and classification in Codeless Scanning. The suggested search strategies may therefore find all references to the particular class of drugs whether or not the appropriate activity is being investigated. Searches for classes of drugs in the older files can be conducted via the Derwent Drug Registry rather than by the sometimes very cumbersome strategy indicated here.

ACT.
Active.

ADJUVANTS
Substances injected with antigens during immunization (usually mixed with them but sometimes given prior to or following the antigen) which non-specifically enhance or modify the immune response to that antigen. * Related VACCINES ANTIBODY-RESPONSE IMMUNE-RESPONSE IMMUNITY

ADOLESCENT
An individual during the period of secondary sexual development - roughly 11 to 19 years of age. * Related * More Specific CASES HUMAN INFANT NEONATE PEDIATRICS

AEROSOL
A system with very fine liquid or solid particles dispersed in a gas. * Related SPRAY

A.V.
Atrioventricular.

AGE-DEPENDENCE
Term used for papers concerned with effects of age on e.g. response to drugs.

ABORTIFACIENT
Activity of drug that causes abortion i.e. induces premature delivery of the conceptus as an embryo or non-viable fetus. * Related OBSTETRICS

ALONE
Term used for papers where the effects of single drugs are compared with those of combinations of drugs. * Related COMB. COMB.PREP.

ABS.
Absolute.

AMINOACID-METAB.
Metabolism of aminoacids in man and animals excluding involvement in protein, monoamine and neurotransmitter metabolism. * Related AMINOACID-METAB.DISORDER N-METAB. PROTEIN-METAB.

ACARICIDES
Drugs that destroy mites, ticks and spiders.

ACE-INHIBITORS
Angiotensin converting enzyme inhibitors. Drugs which inhibit the enzyme that catalyzes the cleavage of angiotensin I to form angiotensin II. * Related ANGIOTENSIN-ANTAGONISTS RENIN-INHIBITORS

AMINOACID-METAB.DISORDER
Disease produced by an inborn error in the metabolism of an aminoacid, e.g. PHENYLKETONURIA. * Related AMINOACID-METAB. CONGENITAL-DISEASE

952 APPENDIX A

ANABOLICS
Drugs which promote food utilization and the building up of the body tissues. * Related ANDROGENS

ANTIAGGREGANTS
Drugs which prevent aggregation of platelets.

ANTIALCOHOLICS
Drugs for the treatment of alcoholism.

ANALEPTICS
Drugs that stimulate the respiratory and vasomotor centers in the medulla of the brain.

ANTIANAPHYLACTICS
Drugs which control allergic reactions such as anaphylaxis other than by blocking the action of histamine. Includes drugs which control histamine release. Does not cover desensitizing drugs. * Related ANTIHISTAMINES-H1

ANALGESICS Drugs which relieve pain.


* Related * More Specific * C/S LOCAL-ANESTHETICS OPIOIDS NARCOTICS /IT,FT ANALGESIC OR AMINOPYRINE OR ANTIPYRINE OR ASPIRIN OR CODEINE OR METHADONE OR MORPHINE OR OPIUM OR PETHIDINE OR PHENACETIN OR SALICYLIC-ACID

ANTIARRHYTHMICS
Drugs which act to correct variations from normal heart rhythm. * Related * More Specific * C/S CARDIANTS CHRONOTROPIC INOTROPIC /IT,FT ANTIARRHYTHMIA OR LIDOCAINE OR PHENYTOIN OR PRACTOLOL OR PROPRANOLOL OR SPARTEINE

ANDROGEN-METAB.
Metabolism of endogenous androgens in man and animals. * Related * C/S ANDROGENS /IT,FT ALL HORMONE-METAB.: AND (ANDROGEN OR TESTOSTERONE)

ANTIASTHMATICS
Drugs which relieve asthmatic spasm. * More Specific * C/S ANTIANAPHYLACTICS BRONCHODILATORS /IT,FT ANTIASTHMATIC OR ADRENALINE OR ISOPRENALINE OR THEOPHYLLINE s.a. CORTICOSTEROID OR HYDROCORTISONE OR PREDNISONE

ANIMAL-MODEL
Term used for papers describing new animal models of disease. Not to be used routinely for studies of diseases in laboratory animals. * Related * C/S LAB.ANIMAL SCREENING-METHOD LAB.ANIMAL/IT AND MODEL/FT

ANTIBIOTICS
Antimicrobial agents produced by microorganisms and their synthetic or semisynthetic analogs. * Related * More Specific ANTISEPTICS PHYTONCIDES TUBERCULOSTATICS ANTILEPROTICS VI/PN (from 1967 only) If all references from 1964 are required: /IT,FT ANTIBIOTIC OR BACITRACIN OR CHLORAMPHENICOL OR CYCLOSERINE OR ERYTHROMYCIN OR GRISEOFULVIN OR KANAMYCIN OR NEOMYCIN OR NYSTATIN OR OLEANDOMYCIN OR PENICILLIN OR POLYMYXIN OR STREPTOMYCIN OR TETRACYCLINE OR VIOMYCIN OR VI/PN

ANORECTICS
Drugs that reduce the desire to eat by an action exerted in the central nervous system.

* C/S

ANTAGONIST
Compound which blocks the pharmacological activity of another drug. Not used for: routine blocking activity of pharmacological tools; where the term ANTIDOTE is applicable; physiological antagonism of endogenous compounds.

ANTHELMINTICS
Drugs which paralyse or kill parasitic worms.

Derwent Drug File 953 Thesaurus

ANTICONVULSANTS
Drugs which prevent epileptic and related types of convulsions. * C/S /IT,FT ANTICONVULSANT OR DIAZEPAM OR PHENYTOIN OR PHENOBARBITAL

ANTIPYRETICS
Substances relieving or reducing fever. * C/S /IT,FT ANTIPYRETIC OR AMINOPYRINE OR ANTIPYRINE OR ASPIRIN OR PHENACETIN OR SALICYLIC-ACID

ANTIDEPRESSANTS
Drugs which elevate the mood of depressed patients. * Related PSYCHOSTIMULANTS PSYCHOTONICS

ANTIRHEUMATICS
Drugs which relieve or prevent rheumatism. * Related ANALGESICS ANTIINFLAMMATORIES CORTICOSTEROIDS /IT,FT ANTIRHEUMATIC OR ASPIRIN OR CHLOROQUINE OR INDOMETACIN OR PHENYLBUTAZONE OR SALICYLIC-ACID s.a. CORTICOSTEROID

ANTIDOTES
An agent administered to prevent or counteract the action of a poison or of drug intoxication. * C/S

ANTIGOUTS
Drugs used to treat gout which is a consequence of abnormally high biosynthesis of uric acid and its deposition in the joints. * Related URICOSURICS

ANTISEPTICS
Substances, other than antibiotics, which inhibit the growth and development of bacteria without necessarily destroying them. * More Specific * C/S TUBERCULOSTATICS ANTILEPROTICS /IT,FT ANTISEPTIC OR ISONIAZID OR NITROFURAL OR PAS OR ALL SULFA-DRUG: OR (SULFONAMIDE AND M/TG)

ANTIINFLAMMATORIES
Non-steroidal antiinflammatory agents. * Related * More Specific * C/S CORTICOSTEROIDS PROSTAGLANDIN-ANTAGONISTS ANTIRHEUMATICS /IT,FT ANTIPHLOGISTIC OR ANTIRHEUMATIC OR ASPIRIN OR INDOMETACIN OR PHENYLBUTAZONE OR SALICYLIC-ACID

APPL.
Application. * Related DRUG-APPL.

ANTILEPROTICS
Drugs inhibiting the growth and development of Mycobact. leprae. * Related ANTIBIOTICS ANTISEPTICS

ART.
Artificial.

ASYM. ANTIMANICS Drugs which reduce mania and euphoria. ANTITUSSIVES


Drugs used to suppress coughing. * Related MUCOLYTICS EXPECTORANTS Asymmetrical.

AUSTR.
Australia.

AUXILIARY-INGREDIENT
Term applied to compounds used in pharmaceutical formulations as carrier-materials, fillers and so-called inert additives. * Related * More Specific PHARMACEUTICS PHARM.PREP. FILLER PROPELLANT SOLVENT FLOCCULANT STABILIZER

954 APPENDIX A

B.I.D.
Dosage schedule in which a drug is administered twice a day. * Related DOSAGE

BIOSYNTH.
Biosynthesis.

BLIND-TEST BACT.
Bacterium. Term used for bacterial species excluding actinomycetes, streptomycetes and Rickettsiales. * More Specific * C/S GRAM-NEG. GRAM-POS. /IT,FT ALL BACT: OR CLOSTR. OR ESCHERICHIA OR MYCOBACT. OR SALM. OR STAPH. OR STREPT. A study of the effects of a drug in which the recipient is unaware whether the test drug or a comparison agent (e.g. placebo) is being given. * Related * More Specific CLIN.TRIAL PLACEBO DOUBLE BLIND-TEST

BLOOD-BRAIN-BARRIER
The biological separation between the blood and the brain that restricts or prevents the transfer of a drug from one to the other.

BEHAVIOR
Term used for studies on human behavior. * Related ANIMAL-BEHAVIOR

BLOOD-CLOTTING-FACTOR
* C/S (/FT FIBRINOGEN OR PLASMINOGEN OR COBYRIC-ACID) OR (/IT,FT PROTHROMBIN OR THROMBOPLASTIN) OR (BLOODCLOTTING/IT AND ALL FACTOR-:)

BIOAVAILABILITY
The proportion of active drug in a formulation that is absorbed and therefore available to exert its pharmacological effect. * Related * More Specific BIOPHARM. BIOEQUIVALENCE

BOLUS
A concentrated mass of a pharmaceutical preparation given i.v.. *Related DRUG-APPL.

BIOEQUIVALENCE
Equivalence of bioavailability and hence of biological activity of two products with the same active principle but different formulations. * Related BIOAVAILABILITY BIOPHARM.

BOTANY
Term used for all plants. * More Specific BARK FLOWER FRUIT HEARTWOOD LEAF ROOT SEED SEEDLING VEGETABLE WOOD /IT,FT ALL BOTANY: OR ACONITUM OR CINCHONA OR DIGITALIS OR IPECAC OR LOBELIA OR RAUWOLFIA OR STROPHANTHUS OR TOBACCO OR VERATRUM OR VINCA (N.B. The terms for specific genera will also retrieve alkaloids isolated from these plants).

BIOL. Biological. BIOMETRICS


Term used for studies describing mathematical analysis of biological data and mathematical models of e.g. pharmacokinetics. * Related MATHEMATICS STATISTICS * C/S

BRONCHODILATORS
Drugs which dilate the respiratory airways by acting directly on the lungs; not used when bronchodilatation is achieved by inhibiting the effects of an allergic mediator. * Related ANTIASTHMATICS

BIOPHARM.
Biopharmaceutics. Term used for studies of the effects of formulation on drug activity or metabolism, e.g. comparison of different tablets, evaluation of bioavailability, comparison of the different salts or esters of a compound. * More Specific BIOAVAILABILITY DRUG-DELIVERY

Derwent Drug File 955 Thesaurus

BUN
Blood urea nitrogen.

CASES
Term used for diseased patients. However, the term is not used in studies using patients (e.g. surgical patients) whose condition is not relevant to the subject of the investigation. * Related CASE-HISTORY HUMAN

CALCIUM-ANTAGONISTS
Drugs that inhibit the entry of Ca++ into cardiac and smooth muscle cells through specific voltage dependent or receptor operated calcium ion channels. * Related CALMODULIN-ANTAGONISTS

CELL.
Cellular.

CALMODULIN-ANTAGONISTS
Drugs which bind to calmodulin and thereby interfere with its ability to bind Ca++. * Related CALCIUM-ANTAGONISTS

CEREBROPROTECTIVE
Activity of a drug which protects brain cells from ischemic damage following cerebrovascular accidents, thrombosis etc. * Related NEUROPROTECTIVE

CARCINOGEN
Activity of a compound which induces tumor formation. * Related COCARCINOGEN MUTAGEN

CHEM.
Chemical.

CHOLAGOGUES CARDIOGLYCOSIDES
Term used for plant glycosides with cardiovascular activity. The singular activity term should be used in addition to CARDIANT where this activity is studied. * C/S /IT,FT CARDIOGLYCOSIDE OR STROPHANTHUS OR DIGITALIS Drugs that stimulate evacuation of the gallbladder or increase bile formation. * Related LITHOLYTICS

CHRON.
Chronic.

CARDIOPATHY
Any disease of the heart. * More Specific * C/S ARRHYTHMIA CORONARY-DISEASE /IT,FT CARDIOPATHY OR ANGINA-PECTORIS OR ARRHYTHMIA OR ENDOCARDITIS OR MYOCARD.INFARCT.

CLATHRATE
Used when a drug forms an inclusion complex with a host molecule, typically a cyclodextrin derivative. * Related COMPLEX

CLIN.
Clinical.

CARDIOPROTECTIVE
Activity of a drug which protects myocardial cells from ischemic damage.

CLIN.TRIAL
A carefully and ethically designed experiment to answer a precisely framed question having therapeutic relevance. * Related * More Specific PLACEBO BLIND-TEST PHASE-I PHASE-II PHASE-III PHASE-IV

CASE-HISTORY
Term used for papers describing in some detail the chronological course of illness(es) in individual patients, generally containing information on pathological features, diagnostic procedures and therapy. The singular term is used regardless of the number of cases presented. * Related CASES

COATING
Refers to the actual substance used to coat a dosage form.

956 APPENDIX A

COCARCINOGEN
Activity of a compound which does not induce tumor formation on its own, but which enhances the carcinogenic activity of another compound or which, when combined with another inert compound induces tumor formation. * Related CARCINOGEN MUTAGEN

CONTRACEPTIVES
Hormones or other drugs preventing conception. The term is not used for mechanical methods of contraception. * Related CONTRACEPTION INTRAUTERINE-DEVICE

CORONARY-DISEASE COLL.
Collective. Disease of the blood vessels of the heart. * Related * More Specific CARDIOPATHY ANGINA-PECTORIS MYOCARD.INFARCT.

COMB.
Combination. Term used for drugs used in conjunction with other drugs, e.g. combination chemotherapy. * Related ALONE COMB.PREP.

CORTICOSTEROID-METAB.
Metabolism of endogenous glucocorticoids in man and animals. * Related * C/S CORTICOSTEROIDS MINERALOCORTICOID-METAB. /IT,FT ALL HORMONE-METAB.: AND (CORTICOSTEROID OR CORTICOSTERONE OR CORTISONE OR HYDROCORTISONE)

COMB.PREP.
Combination preparation, i.e. a pharmaceutical formulation containing two or more active ingredients. * Related COMB.

COMP .
Component or composition.

CORTICOSTEROIDS
Natural or synthetic glucocorticoids. N.B. CORTICOSTEROID is used for antiinflammatory activity of steroids. * Related * C/S MINERALOCORTICOIDS CORTICOSTEROID-METAB. /IT,FT CORTICOSTEROID OR BETAMETHASONE OR CORTICOSTERONE OR CORTISONE OR DEXAMETHASONE OR METHYLPREDNISOLONE OR PREDNISOLONE OR PREDNISONE OR TRIAMCINOLONE

COMPATIBILITY
Ability of two or more drugs to be mixed without adverse effects on the physical, chemical or pharmacological properties of the components. * Related INCOMPATIBILITY

COMPLEX
Used for a drug forming a coordination compound with other (inorganic or organic) substances. * More Specific CLATHRATE CYTOSTATICS

Agents which suppress the growth and multiplication of cells, especially cancer cells. * C/S /IT,FT CYTOSTATIC OR ACTINOMYCIN OR ASPARAGINASE OR BLEOMYCIN OR COLCHICUM OR CYCLOHEXIMIDE OR CYCLOPHOSPHAMIDE OR CYTARABINE OR FLUOROURACIL OR MERCAPTOPURINE OR METHOTREXATE OR PUROMYCIN OR RIFAMYCIN OR TETRACYCLINE OR VINCA

COND.
Condensed.

CONFIG.
Configuration.

CONGENITAL-DISEASE
Diseases present at birth. * Related TERATOGENESIS

CYTOTOX.
Cytotoxicity.

Derwent Drug File 957 Thesaurus

DER.
Derivative.

DIGEST.
Digestive.

DEPOT
Term used for drug preparations with timed, or slow-release properties. * Related PHARM.PREP. IMPLANT DRUG-DELIVERY

DIGITALIS
Term used for Digitalis species, i.e. not for alkaloids. * C/S DIGITALIS/IT,FT (N.B. Will give references to cardioglycosides as well as the plants).

DISCUSSION DERMATOLOGICAL
Topical application of drugs for the treatment of skin disorders. * Related ANTIPRURITIC ANTIPSORIATIC Term used for short, review-type papers with few or no references. * Related REVIEW EDITORIAL

DISINTEGRATION DERMATOLOGY
Any disease of the skin. * C/S /IT,FT DERMATOLOGY OR ACNE OR ECZEMA OR PSORIASIS OR SCABIES Physical break down of tablets, dragees, etc. in-vivo or in-vitro. * Related DISSOLUTION PHARMACEUTICS

DISPERSION
Formulation in which particles of the drug are dispersed in the form of suspensions or colloidal solutions.

DESENSITIZERS
Allergens used to induce tolerance in the therapy of allergic disorders.

DISSOLUTION
Process of a solid dosage form going into solution. Separate from (and subsequent to) physical disintegration. * Related DISINTEGRATION PHARMACEUTICS

DET.
Detection.

DIAGNOSIS
Term used for papers describing diagnostic methods or where diagnosis is particularly stressed. Not used for routine diagnosis. * Related DIAGNOSTICS

DISTR.
Distribution.

DIURETICS
Drugs which increase the excretion of urine. * C/S /IT,FT DIURETIC OR ETACRYNIC-ACID OR FUROSEMIDE OR MANNITOL OR SORBITOL OR SPIRONOLACTONE OR THEOPHYLLINE

DIAGNOSTICS
Compounds or products used as aids in diagnosis. * Related DIAGNOSIS RADIOPAQUES

DIET
The customary, day to day, allowance of food and drink. The term is used particularly in relation to modifications for special purposes, e.g. therapy. * More Specific FASTING THERAPEUTIC-FASTING

DOSAGE
Term used only for papers where dosages are evaluated, or are unusual, or are in any other respect important. * Related LONG-TERM-THERAPY SHORT-TERM-THERAPY

958 APPENDIX A

DOUBLE BLIND-TEST
A study of the effects of a drug in which both the investigator and the recipient are unaware whether the test drug or a comparison agent (e.g. placebo) is being given. * Related BLIND-TEST CLIN.TRIAL PLACEBO

EMBOLIZATION
Introduction of a substance into a vessel to occlude it, especially for therapeutic purposes.

EMIT
Enzyme-Multiplied Immunoassay Technique. * Related ENZYME-IMMUNODET. IMMUNODET.

DRUG-APPL.
Drug application. Term used only when the route of administration of a drug is itself significant, e.g. where different routes are compared.

ENCEPHALOPATHY
Diseases of the brain, excluding cerebrovascular and psychiatric disorders. * Related * C/S CEREBROVASCULAR-DISEASE MENTAL-DISORDER /IT,FT ENCEPHALOPATHY OR MENINGITIS OR NEUROLOGY OR OLIGOPHRENIA OR PARKINSONISM OR COMA OR EPILEPSY OR CHOREA

DRUG-COMPARISON
Term used for papers where the actions of two or more drugs are compared. * Related BLIND-TEST CLIN.TRIAL

DRUG-DELIVERY
Term used for studies of drug delivery systems, e.g. osmotic pumps, controlled release systems, prodrugs. * Related * More Specific BIOPHARM. PHARM.PREP. DEPOT PRODRUG

ENDOCRINE-DISEASE
Any disease of the endocrine glands. * Related OVARY-DISEASE TESTIS-DISEASE THYMUS-DISEASE ADRENOPATHY HYPOTHALAMUS-DISEASE PITUITARY-DISEASE PANCREOPATHY PARATHYROID-DISEASE THYROID-DISEASE /IT,FT ADRENOPATHY OR DIABETES OR DIAB.INSIP. OR GOITER OR HYPOTHYROIDISM OR THYROTOXICOSIS

EDITORIAL
Used for all editorial review-type papers. * Related DISCUSSION REVIEW * More Specific

EL.
Electrical. * C/S

ELECTROCHEM.
Electrochemistry.

ENERGY-METAB.
Term used for the catabolic process by which energy is produced when no more specific term can be applied. * Related * More Specific BASAL-METAB. GLYCOLYSIS OX.PHOSPHORYLATION RESPIRAT.CHAIN

ELECTROPHYSIOL.
Term used for studies of conduction in nerve and muscle (including heart).

ELECTROSHOCK
Electroconvulsive therapy.

ENTEROSOLUBILITY ELIMINATION
Excretion, e.g. in urine or feces. Solubility of pharmaceutical preparations, e.g. tablets, in enteric juice. * Related DISINTEGRATION

Derwent Drug File 959 Thesaurus

ENZYME-MODEL
Chemicals and chemical reactions used as models for the demonstration of enzyme reaction mechanisms.

FIRST-PASS-EFFECT
The proportion of an orally administered drug that is removed by the liver before entering the general circulation. *Related MICROSOME-DRUG-METAB.

ENZYMES
Term used only to classify enzymes which are drugs, e.g. ASPARAGINASE. The term is not used for endogenous enzyme activity. N.B. To find all enzymes use ALL EC-:/FT

FLOCCULANT
Pharmacologically inert auxiliary ingredient that promotes flocculation. * Related AUXILIARY-INGREDIENT FLOCCULATION PHARM.PREP. PHARMACEUTICS

ESS.
Essential.

ESTROGEN-METAB.
Metabolism of endogenous estrogens in man and animals. * Related * C/S ESTROGENS /IT,FT ALL HORMONE-METAB.: AND (ESTROGEN OR ESTRADIOL)

FLOCCULATION
A colloid phenomenon in which the disperse phase separates in discrete, usually visible, particles rather than in continuous mass. * Related FLOCCULANT FORMULATION PHARM.PREP. PHARMACEUTICS

EXPECTORANTS
Drugs which promote the ejection of mucus or exudate from the lungs, bronchi and trachea by decreasing mucus viscosity or by increasing the secretion of mucus in a dry, unproductive cough. * Related MUCOLYTICS ANTITUSSIVES

FORMULATION
Term used for papers describing the process of formulation of pharmaceutical preparations. * Related PHARM.PREP. PHARMACEUTICS AUXILIARY-INGREDIENT

FUNGICIDES EXTRACELL.
Extracellular. Substances, including antibiotics, which inhibit fungal growth or destroy fungi. * C/S /IT,FT FUNGICIDE OR AMPHOTERICIN OR CYCLOHEXIMIDE OR GRISEOFULVIN OR NYSTATIN

EXUD.
Exudative.

FUNGUS FERMENTATION
Term used for papers describing culture conditions, etc. for production of compounds (especially antibiotics) by microorganisms with possible relevance to industrial processes. * Related CULTURE-MEDIUM Term used for fungi other than those with macroscopic fruiting bodies. Includes actinomycetes and streptomycetes. * Related * More Specific * C/S LICHEN MUSHROOM YEAST /IT,FT FUNGUS OR YEAST OR CANDIDA

FILLER
Inert packing substance used in drug formulations. *Related AUXILIARY-INGREDIENT PHARMACEUTICS PHARM.PREP. FORMULATION

G.U.TRACT
Term used for parts of the genito-urinary tract not covered by the more specific terms below. * More Specific KIDNEY OVARY PENIS PROSTATE TESTIS UTERUS VAGINA

960 APPENDIX A

GANGLIONOPLEGICS
Drugs that block the transmission of impulses through the sympathetic or parasympathetic ganglia.

GONADOTROPIN-METAB.
Metabolism of endogenous gonadotropins in man and animals. * Related GONADOTROPINS GONADOTROPIN-METAB. PITUITARY-HORMONE-METAB. /IT,FT ALL HORMONE-METAB.: AND GONADOTROPIN

GANGLION-STIMULANTS
Drugs that stimulate the transmission of impulses through the autonomic ganglia. * C/S

GASTROENTEROPATHY
Any disease of the gastrointestinal tract. * C/S /IT,FT GASTROENTEROPATHY OR AMEBIASIS OR CHOLERA OR CONSTIPATION OR DIARRHEA OR DYSENTERY OR ILEUS OR SPRUE OR TYPHOID OR ULCER

GROWTH
Term used for growth of whole organisms or organs, but not for proliferation of tissue-cultures or microorganisms.

GYNECOLOGY
Term used for diseases of the female pelvic and adjacent organs not covered by more specific terms. * Related * More Specific OBSTETRICS OVARY-DISEASE UTERUS-DISEASE VAGINA-DISEASE

GASTROINTEST.HORMONES
Gastrointestinal hormones such as gastrin, secretin, gastric inhibitory polypeptide, etc. * Related * C/S GASTROINTEST.HORMONE-METAB. Input terms for individual hormones.

GASTROINTEST.HORMONE-METAB.
Metabolism of gastrointestinal hormones in man and animals. * Related * C/S GASTROINTEST.HORMONES /IT,FT ALL HORMONE-METAB.: plus terms for individual hormones.

H-K-ATPASE-INHIBITORS
Drugs which inhibit H+,K+-ATPase.

HAL.
Halogenated.

GEN.
General.

HELMINTH
* C/S /IT,FT ALL HELMINTH: OR ALL CESTOD: OR ALL NEMATOD: OR ALL TREMATOD: N.B. Will retrieve references to in-vitro studies and infestations.

GEN.PHARMACOL.
General pharmacology. A series of tests which aim to determine the effects of an established (named) drug on the different organ systems of the body. Not used for drug screening papers.

HEM.
Hemorrhagic

GLAND
Term used for exocrine glands, e.g. salivary glands. * Related MAMMA PANCREAS

HEM.DIATHESIS
Hemorrhagic diathesis. Predisposition to hemorrhagic disease.

Derwent Drug File 961 Thesaurus

HEMIC-DISEASE
Not a search term in the UDB. To search for this concept, OR the keywords listed under More Specific. * Related * More Specific LYMPH-DISEASE LYMPHOPROLIFERATIVE-DISEASE ANEMIA HEM.DIATHESIS LEUKOCYTE-DISORDER MARROW-DISEASE THROMBOSIS /IT,FT ANEMIA OR AGRANULOCYTOSIS OR PERNICIOSA OR HEM.DIATHESIS OR THROMBOSIS

HORMONES
Exogenous hormones. Not a search term in the UDB. To search the concept, OR the keywords listed under More Specific. * More Specific ANABOLICS ANDROGENS CORTICOSTEROIDS ESTROGENS GASTROINTEST.HORMONES GONADOTROPINS KININS MINERALOCORTICOIDS PANCREAS-HORMONES PITUITARY-HORMONES PROGESTOGENS PROSTAGLANDINS RELEASING-FACTORS RELEASING-FACTOR-INHIBITORS THYMUS-HORMONES THYROID-HORMONES

* C/S

HEPARINOIDS
Substances with heparin-like activity; sulfonated polysaccharides with anticoagulant and lipolytic activities.

HORMONE-METAB.
Metabolism of endogenous hormones not covered by more specific terms. * More Specific ANDROGEN-METAB. CORTICOSTEROID-METAB. ESTROGEN-METAB. GASTROINTEST.HORMONE-METAB. GONADOTROPIN-METAB. KININ-METAB. MINERALOCORTICOID-METAB. PANCREAS-HORMONE-METAB. PITUITARY-HORMONE-METAB. PROGESTOGEN-METAB. PROSTAGLANDIN-METAB. RELEASING-FACTOR-METAB. THYMUS-HORMONE-METAB. THYROID-HORMONE-METAB. ALL HORMONE-METAB.: (N.B. Covers exogenous and endogenous hormones.)

HEPATOPATHY
Any disease of the liver. * C/S /IT,FT HEPATOPATHY OR ALCOHOLISM OR ICTERUS OR VIRUS-HEPATITIS

HEPATOTROPICS
Drugs used in liver protection therapy.

HETE
12-Hydroxy-5,8,10,14-eicosatetraenoic acid. * C/S 12-HYDROXY-5,8,10,14-EICOSATETRAENOIC-ACID/FT C/S

HISTOPATHOL.
Histopathology.

HPLC
High performance/pressure liquid chromatography. * Related * C/S CHROMATOGRAPHY HPL-CHROMATOGRAPHY OR (ALL HIGH-P: AND LIQUID-CHROMATOGRAPHY)

HMG-COA-REDUCTASE-INHIBITORS
Drugs which inhibit hydroxymethylglutaryl-CoA reductase. * Related ANTIARTERIOSCLEROTIC

HUMAN
Term used for normal, healthy humans. * Related * More Specific CASES INFANT PEDIATRICS ADOLESCENT GERIATRICS ADULT NEONATE

962 APPENDIX A

HYPERACT.
Hyperactive.

IMAGING-AGENTS
Diagnostic agents used to visualize specific tissues by means of scintillography, NMR (magnetic resonance imaging agents), positron emission tomography (PET), ultrasonics etc. Excludes radiopaques (X-rays contrast media). * Related RADIOPAQUES DIAGNOSIS

HYPERALIMENTATION
Term used for i.v. feeding, e.g. total parenteral nutrition.

HYPOTENSIVES
Drugs which reduce blood pressure. * C/S /IT,FT HYPOTENSIVE OR CLONIDINE OR GUANETHIDINE OR METHYLDOPA OR PARGYLINE OR PHENOXYBENZAMINE OR PRACTOLOL OR PROPRANOLOL OR RESERPINE

IMMUNOMODULATOR
Drugs which control or modulate the function of cells of the immune system. Not used when a more specific term is appropriate. * More Specific IMMUNOSUPPRESSIVES IMMUNOSTIMULANTS

HYPOVITAMINOSIS
A condition due to a deficiency of one or more vitamins. * C/S /IT,FT HYPOVITAMINOSIS OR BERIBERI OR PELLAGRA OR RACHITIS OR SCURVY

IMMUNOSTIMULANTS
Drugs which enhance the intensity of the immune response. * Related IMMUNOMODULATOR

IMMUNOSUPPRESSIVES I.A.
Intraarterial. * Related DRUG-APPL. Drugs which suppress the immune response. Does not include antihistamines or antianaphylactics. * Related IMMUNOMODULATOR

I.C.
Intracardial. * Related DRUG-APPL.

IMPLANT
Solid drug formulation for inserting into the body tissues. Used to provide a regular and long-term release of active component. * Related DEPOT DRUG-DELIVERY

I.M.
Intramuscular. * Related DRUG-APPL.

INCOMPATIBILITY
Inability of two or more drugs to be mixed without adverse effects on the physical, chemical or pharmacological properties of the components. * Related DRUG-APPL. COMPATIBILITY

I.P.
Intraperitoneal. * Related

IND.
Industrial.

I.V.
Intravenous. * Related DRUG-APPL.

INFANT
Term used for children up to the age of 2 years. * Related * More Specific CASES HUMAN PEDIATRICS NEONATE

Derwent Drug File 963 Thesaurus

INFECTION,BACT. Any bacterial infection.


* C/S /IT,FT INFECTION,BACT. OR ANTHRAX OR BRUCELLOSIS OR CHOLERA OR DIPHTHERIA OR DYSENTERY OR LEPROSY OR LEPTOSPIROSIS OR MASTITIS OR MENINGITIS OR MYCOPLASMOSIS OR PASTEURELLOSIS OR PERTUSSIS OR PSEUDOMONIASIS OR PYELONEPHRITIS OR SCARLATINA OR SEPSIS OR TETANUS OR TUBERCULOSIS OR TYPHOID

INFUSION
Gradual introduction (usually i.v.) of a solution of a drug for therapeutic or pharmacological purposes. * Related DRUG-APPL.

INJECTABLE
Galenical preparation of a drug in injectable form, including infusions. * Related FORMULATION PHARM.PREP. PHARMACEUTICS

INFECTION,FUNGUS
Any fungal infection. * C/S /IT,FT INFECTION,FUNGUS OR CANDIDIASIS

INJECTION
Introduction of a drug etc. into the body by force e.g. via a needle. * Related * More Specific DRUG-APPL. I.A. I.C. I.M. I.P. I.V.

INFECTION,PROTOZOON
Any protozoal infection. * C/S /IT,FT INFECTION,PROTOZOON OR AMEBIASIS OR BABESIASIS OR COCCIDIOSIS OR HISTOMONIASIS OR LEISHMANIASIS OR MALARIA OR THEILERIASIS OR TOXOPLASMOSIS OR TRICHOMONIASIS OR TRYPANOSOMIASIS

INSECT
* C/S /IT,FT ARTHROPOD OR ALL FLY: OR MITE OR TICK

INSECT-HORMONES
* C/S /IT,FT HORMONE AND (INSECT OR JUVENILE)

INFECTION,RICKETTSIALES
Any rickettsial infection. * C/S /IT,FT INFECTION,RICKETTSIALES OR ANAPLASMOSIS OR TRACHOMA

INTERN.
International.

INTEST. INFECTION,VIRUS
All viral infections. * C/S /IT,FT INFECTION,VIRUS OR HERPES OR MENINGITIS OR POLIOMYELITIS OR VIRUS-HEPATITIS OR INFLUENZA OR COMMON-COLD Intestinal.

INTOXICATION
Poisoning * Related * More Specific ALCOHOLISM HYPERVITAMINOSIS THYROTOXICOSIS ADDICTION ERGOTISM

INFESTATION,ECTOPARASITE
Parasitic attack or subsistence on the skin and its appendages by insects, mites or ticks. * C/S ALL INFESTATION: OR SCABIES/IT,FT

INVERSE-AGONIST
Activity of a drug which binds to the same receptor as an agonist but produces the opposite pharmacological effect. Usually applies to benzodiazepine drugs. * Related BENZODIAZEPINE-AGONIST

INFLAMMATION
Term used only for non-specific inflammatory conditions which cannot be classified by a more specific disease term.

964 APPENDIX A

KERATOLYTICS
Drugs that promote keratolysis i.e. softening or peeling of the horny layer of the epidermis. * Related DERMATOLOGICAL

LIPOXYGENASE-INHIBITORS
Drugs which inhibit lipoxygenase.

LITHOLYTICS
Drugs which dissolve stones or calculi. * Related CHOLAGOGUES

KININ-METAB.
Metabolism of kinins in man and animals. * Related * C/S KININS /IT,FT ALL HORMONE-METAB.: AND (KININ OR BRADYKININ)

LOCAL-ANESTHETICS
Anesthetics whose action is limited to an area around the site of application. * Related ANESTHESIA-CAUDAL ANESTHESIA-EPIDURAL ANESTHESIA-HYPOTENSIVE ANESTHESIA-INTRATHECAL ANESTHESIA-NERVE-BLOCK ANESTHESIA-PERIDURAL ANESTHESIA-SADDLE-BLOCK ANESTHESIA-SPINAL /IT,FT LOCAL-ANESTHETIC OR COCAINE OR LIDOCAINE OR PROCAINE

LAB.
Laboratory.

LAB.ANIMAL
Laboratory animals. Term used for all animals used for experimental purposes. * Related ANIMAL-MODEL

* C/S

LD10
Concentration of a compound that kills 10% of the animals tested.

LYMPHOPROLIFERATIVE-DISEASE
Term applied to a group of diseases characterized by proliferation of lymphoid tissue such as lymphocytic leukemia and malignant lymphoma.

LD100
Concentration of a compound that kills 100% of the animals tested.

MAIN-TOPIC
Term applied to a concept which is the main subject of a review paper. (N.B. the term is not used in conjunction with DISCUSSION). * Related REVIEW

LD50
Concentration of a compound that kills 50% of the animals tested.

MAMMAL LD90
Concentration of a compound that kills 90% of the animals tested. Term used for mammals only when they appear in a context other than use as experimental animals, e.g. isolation of compounds.

LEUKOTRIENE-ANTAGONISTS
Drugs which antagonise the effects of leukotrienes.

MATHEMATICS
Term used for papers concerned with mathematics, other than analysis of biological data or mathematical models of pharmacokinetics. * Related BIOMETRICS STATISTICS

LIPOSOME
Microscopic vesicle formed from a lipid membrane. Used to carry active compounds for purposes of drug delivery. * Related DRUG-DELIVERY

MED.
Medical or medicine.

Derwent Drug File 965 Thesaurus

MEDITER.
Mediterranean.

MORPHINE-ANTAGONISTS
Compounds which antagonise the activity of morphine, and of plant and synthetic morphine-like compounds. N.B. The term is not used for antagonists of endogenous opioid peptides. * Related * C/S OPIOID-ANTAGONIST /IT,FT MORPHINE AND ANTAGONIST

MENTAL-DISORDER
Any psychiatric disorder. * More Specific ANXIETY-DISORDER PERSONALITYDISORDER EATING-DISORDER FACTITIOUSDISORDER MOOD-DISORDER PSYCHOTICDISORDER /IT,FT ANXIETY OR DEPRESSION OR NEUROSIS OR SCHIZOPHRENIA OR PSYCHIATRY

MUCOLYTICS
Drugs which reduce the viscosity of mucus. * Related EXPECTORANTS ANTITUSSIVES

* C/S

MUSC. METABOLISM
* C/S /IT,FT AMINOACID-METAB. OR CARBOHYDRATE-METAB. OR CITRIC-ACID-CYCLE OR ALL DRUG-METAB.: OR ELECTROLYTE-METAB. OR GLYCOLYSIS OR ALL HORMONE-METAB.: OR LIPID-METAB. OR N-METAB. OR NUCLEIC-ACID-METAB. OR PROTEIN-METAB. OR VITAMIN-METAB. Muscular.

MUSCLE
Skeletal muscle. * Related SMOOTH-MUSCLE

MUSCULOSKELETAL-DISEASE
* C/S /IT,FT MYOPATHY OR OSTEOPATHY OR RHEUMATISM

MICROSOME-DRUG-METAB.
Term used for studies of microsomal drug metabolizing systems. * C/S /IT,FT ALL DRUG-METAB.: AND MICROSOME

MUTAGEN
Compound which induces gene mutation. * Related CARCINOGEN COCARCINOGEN

MILIT.
Military.

MUTATION
A change in the structure of DNA or in the number of genes or chromosomes in a cell that results in the expressions of genetic abnormalities. * More Specific SISTER-CHROMATID EXCHANGE CHROMOSOME ABERRATION

MODE-OF-ACT.
Term used for studies of the mechanism of action of drugs.

MODEL
Term used for e.g. mathematical models. * Related ANIMAL-MODEL ENZYME-MODEL

MYDRIATICS
Drugs which produce dilatation of the pupil. * Related OPHTHALMOLOGICAL

MOL.
Molecular.

MYOCARD.
Myocardial.

966 APPENDIX A

NA-K-ATPASE-INHIBITORS
Drugs which inhibit Na+,K+-ATPase.

NEUROLOGICAL-DISEASES
* C/S /IT,FT ENCEPHALOPATHY OR MENINGITIS OR NEURITIS OR NEUROLOGY OR OLIGOPHRENIA OR PARALYSIS OR PARKINSONISM (For psychiatric diseases see MENTAL-DISORDER).

NARCOTICS
Drugs which produce narcosis (reversible depression of the central nervous system). * Related OPIOIDS ANALGESICS

NEUROMUSC.
Neuromuscular.

NEG.
Negative.

NEUROMUSC.BLOCKERS
Drugs with a curare-like action i.e. which relax skeletal muscles by acting peripherally on the motor end-plates. * Related RELAXANTS

NEONATE
Term used for newborn children (up to the age of about 4 weeks) and laboratory animals. * Related HUMAN CASES INFANT PEDIATRICS LAB.ANIMAL

NEUROMUSC.DISEASE
Disorders of neuromuscular function such as myasthenia gravis.

NEOPLASM
Malignant and benign human tumors other than leukemias and lymphomas. * Related ANIMAL-NEOPLASM LYMPHOPROLIFERATIVE-DISEASE

NEUROPROTECTIVE
Activity of a drug which protects peripheral nerves from damage. * Related CEREBROPROTECTIVE

NEPHROTROPIC
Activity of a drug that improves kidney function by a specific or nonspecific mechanism of action.

NEW
Term applied to compounds appearing in the file for the first time which are screened for pharmacological activity.

NEUROLEPTANALGESIA
A state of quiescence, altered awareness and analgesia produced by the administration of a combination of a narcotic analgesic and a neuroleptic drug. * Related NEUROLEPTICS NARCOTICS

NEW-ACT.
Term applied on the first mention of a novel activity for an established drug.

NO.
Number.

NEUROLEPTANESTHESIA
A state of neuroleptanalgesia and unconsciousness produced by the administration of a narcotic analgesic and a neuroleptic drug with the inhalation of nitrous oxide and oxygen. * Related NEUROLEPTICS NARCOTICS GEN.ANESTHETICS

NOMENCLATURE
Term used when compounds (other than trial-preparations) are given trivial names.

NOOTROPICS NEUROLEPTICS
Drugs used to control the signs and symptoms of psychotic disorders. * Related PSYCHOSEDATIVES TRANQUILIZERS Drugs which enhance learning and improve memory.

Derwent Drug File 967 Thesaurus

OBSTETRICS
Term used for management of pregnancy, labor and the puerperium, and for diseases complicating pregnancy. * Related PREGNANCY

PANCREAS-HORMONES
* C/S /IT,FT INSULIN OR GLUCAGON OR PANCREATIC-POLYPEPTIDE

PANCREAS-HORMONE-METAB. ODONTOLOGY
Term used for diseases of the teeth. Metabolism of endogenous pancreas hormones in man and animals. * Related PANCREAS-HORMONES /IT,FT ALL HORMONE-METAB.: AND (INSULIN OR GLUCAGON OR PANCREATIC-POLYPEPTIDE)

OPHTHALMOLOGICAL
Use of drugs for the treatment of eye diseases.

* C/S

OPIOID-ANTAGONIST
Compounds which antagonise the activity of naturally occurring opioid peptides and their synthetic analogs. N.B. The term is not used for antagonists of plant opiates. * Related MORPHINE-ANTAGONISTS

PARASYMPATHOMIMETICS
Drugs simulating the effects of parasympathetic stimulation. * C/S /IT,FT PARASYMPATHOMIMETIC OR ACETYLCHOLINE OR CHOLINE OR DFP OR MUSCARINE OR NEOSTIGMINE OR NICOTINE OR PHYSOSTIGMINE OR PILOCARPINE

OPIOIDS
Naturally occurring peptides, e.g. enkephalins, or synthetic analogs, with opiate-like activity. * Related ANALGESICS NARCOTICS

PARTIAL-AGONIST
A term to denote an agonist that fails to produce a maximal response of a tissue when all the receptors are occupied.

OPT.
Optical.

PATHOL.
Pathological.

ORG.
Organic.

PEDIATRICS
Term used for children between 0 and 19 years of age. * Related * More Specific CASES HUMAN INFANT NEONATE

ORL
Otorhinolaryngology.

OX.
Oxidative.

PENETRATION-ENHANCERS
Excipients in a drug formulation which have no pharmacological activity but which promote the percutaneous absorption of a drug. * Related DRUG-APPL. AUXILIARY-INGREDIENT FORMULATION PHARM.PREP. PHARMACEUTICS

P.O.
Per os, by mouth. * Related

PAF-ANTAGONISTS
Drugs which antagonise the effects of platelet activating factor (PAF).

PERCUTANEOUS
Term applied to drug absorption via the skin e.g. following transdermal administration. * Related TRANSDERMAL

968 APPENDIX A

PERIPHERAL-NERVE-DISEASE
Diseases of the peripheral nervous system. * C/S /IT,FT NEURITIS OR NEUROLOGY OR PARALYSIS

PHYTONCIDES
Antimicrobial substances isolated from higher plants and from macroscopic thallophytes. * Related ANTIBIOTICS FUNGICIDES

PHARM.PREP.
Pharmaceutical preparation. Term used for papers describing particular formulations, e.g. tablets, capsules. * Related FORMULATION

PITUITARY-HORMONE-METAB.
Metabolism of endogenous pituitary hormones, other than gonadotropins, in man and animals. * Related PITUITARY-HORMONES /IT,FT HORMONE-METAB. AND (ACTH OR INTERMEDIN OR PROLACTIN OR SOMATOTROPIN OR LIPOTROPIN OR OXYTOCIN OR THYROTROPIN OR VASOPRESSIN)

PHARMACEUTICS
Term used for papers dealing with the preparation and examination of pharmaceutical forms of drugs. * Related FORMULATION PHARM.PREP. AUXILIARY-INGREDIENT

* C/S

PITUITARY-HORMONES PHARMACOKINETICS
Term used for papers describing time-related aspects of drug metabolism, e.g. HALF-LIFE. For more general studies of drug metabolism use DM. Pituitary hormones other than gonadotropins. * C/S /IT,FT SOMATOTROPIN OR ACTH OR INTERMEDIN OR LIPOTROPIN OR PROLACTIN OR OXYTOCIN OR THYROTROPIN OR VASOPRESSIN

PHASE-I
Clinical trials of a drug to determine human pharmacology and safety studies. * Related CLIN.TRIAL BLIND-TEST PLACEBO

PLACEBO
Comparison medication that has no inherant pharmacological activity, but which might exert a psychological one. * Related BLIND-TEST CLIN.TRIAL

PHASE-II
Early clinical trials with small patient numbers. Monitoring very stringent. * Related CLIN.TRIAL BLIND-TEST PLACEBO

PNEUMOPATHY
Diseases of the lungs. * C/S /IT,FT PNEUMOPATHY OR ASTHMA OR BRONCHITIS OR INFECTION,RESPIRAT. OR PERTUSSIS OR TUBERCULOSIS

PHASE-III
Clinical trials using greater numbers of patients to attain statistical significance. Monitoring correspondingly less stringent. * Related CLIN.TRIAL BLIND-TEST PLACEBO

POS.
Positive.

POT.
Potential (adjective).

PHASE-IV
Clinical trials monitoring the incidence of side-effects etc. which are carried out after the drug is registered and being actively marketed. * Related CLIN.TRIAL BLIND-TEST PLACEBO

POTASSIUM-AGONIST
Activity of a drug that facilitates the passage of K+ through membrane potassium channels. Also called potassium channel activators.

Derwent Drug File 969 Thesaurus

POTENTIAL
Potential (noun).

PROTEIN-KINASE-C-INHIBITORS
Drugs which inhibit protein-kinase C.

PREGNANCY
Normal pregnancy, i.e. that period from conception to delivery, in humans and animals. * Related OBSTETRICS

PROTOZOACIDES
Drugs destroying protozoa. * Related * More Specific * C/S ANTIBIOTICS AMEBICIDES COCCIDIOSTATICS /IT,FT PROTOZOACIDE OR AMEBICIDE OR BABESIACIDE OR CHLOROQUINE OR COCCIDIOSTATIC OR DIMETRIDAZOLE OR DIMINAZENE OR FURAZOLIDONE OR METHYLDINITROBENZAMIDE OR TIABENDAZOLE

PRESERVATIVE
Action of a compound to prevent chemical degradation of a drug by microbial contaminants, oxidation, etc. * Related * C/S PRESERVATION PRESERVATION/IT,FT

PROTOZOON PRIM.
Primary. * C/S /IT,FT PROTOZOON OR AMEBIASIS OR BABESIASIS OR COCCIDIOSIS OR HISTOMONIASIS OR LEISHMANIASIS OR MALARIA OR THEILERIASIS OR TOXOPLASMOSIS OR TRICHOMONIASIS OR TRYPANOSOMIASIS (N.B. With the exception of PROTOZOON, these terms will give both in-vitro and in-vivo studies).

PRODRUG
A drug precursor which, on administration, undergoes metabolic conversion to an active agent. * Related DRUG-DELIVERY

PSYCHOSEDATIVES PROGESTOGEN-METAB.
Metabolism of endogenous progestogens in man and animals. * Related * C/S PROGESTOGENS /IT,FT ALL HORMONE-METAB.: AND (PROGESTOGEN OR PROGESTERONE) Drugs which calm and relieve anxiety while producing minimal motor and sensory impairment. * More Specific * C/S NEUROLEPTICS TRANQUILIZERS /IT,FT PSYCHOSEDATIVE OR CHLORDIAZEPOXIDE OR CHLORPROMAZINE OR CHLORPROTHIXENE OR DIAZEPAM OR HALOPERIDOL OR MEPROBAMATE OR PHENOTHIAZINE

PROP .
Property.

PSYCHOSTIMULANTS PROPELLANT
Pharmacologically inert vehicle for aerosol packs, consisting of packed gas. * Related AUXILIARY-INGREDIENT PHARM.PREP. FORMULATION PHARMACEUTICS Drugs which produce transient increases in psychomotor activity. * More Specific * C/S ANTIDEPRESSANTS PSYCHOTONICS /IT,FT PSYCHOSTIMULANT OR AMITRIPTYLINE OR AMPHETAMINE OR CAFFEINE IMIPRAMINE OR PARGYLINE

PROSTAGLANDIN-METAB.
Metabolism of endogenous prostaglandins in man and animals. * Related * C/S PROSTAGLANDINS /IT,FT ALL HORMONE-METAB.: AND ALL PROSTAGLANDIN:

PSYCHOTOMIMETICS
Drugs which produce psychosis-like symptoms, e.g. hallucination. * C/S /IT,FT PSYCHOTOMIMETIC OR CANNABINOID OR LSD OR MESCALINE

970 APPENDIX A

PURINE-ANTAGONISTS
Drugs which have antagonist activity at the adenosine receptor.

RENIN-INHIBITORS
Drugs which inhibit renin, the enzyme which catalyzes the conversion of angiotensinogen to angiotensin. * Related ACE-INHIBITORS ANGIOTENSIN-ANTAGONISTS

PURINERGICS
Drugs which have agonist activity at the adenosine receptor.

Q.I.D.
Dosage schedule in which the drug is administered four times a day. * Related DOSAGE

RES
Reticuloendothelial system.

RESISTANCE
Natural and acquired resistance of microorganisms and pests to chemotherapeutic agents and pests. Term also used for resistance of e.g. tumor cell lines to cytostatic drugs.

QUAT.
Quaternary.

RESPIRATION-DISORDER RADIOSENSITIZERS
Drugs that increase the sensitivity of cells to electromagnetic radiation. * Related RADIOTHERAPY IRRADIATION Disturbances in control, especially autonomic control, of respiration.

RESPIRATORY-TRACT-DISEASE
* C/S /IT,FT ASTHMA OR BRONCHITIS OR INFECTION,RESPIRAT. OR PERTUSSIS OR PNEUMOPATHY OR TUBERCULOSIS

RADIOTHERAPY
The use of electromagnetic waves, such as those of light or ionizing rays, for therapeutic purposes. * Related RADIOSENSITIZERS IRRADIATION

REUPTAKE-INHIBITOR
Activity of a drug that inhibits the uptake of serotonin into platelets and the neuronal uptake of serotonin and noradrenaline.

REACTION-MECHANISM
Term used for studies of the mechanism of chemical reactions.

REVIEW
Term used for papers which review topics in some detail and which provide significant numbers of literature references. * Related EDITORIAL MAIN-TOPIC DISCUSSION

RED.
Reduced.

REDOX
Reduction/oxidation potential or system. * Related RESPIRAT.CHAIN

S.C.
Subcutaneous. * Related DRUG-APPL.

RELAXANTS
Drugs which relax skeletal muscle by a central action. * Related NEUROMUSC.BLOCKERS

SAFETY
Term used for accident prevention and associated problems e.g. in hospitals, pharmaceutical manufacturing, etc.

SCREENING
Examination of a group for the existence of a disease, etc.

Derwent Drug File 971 Thesaurus

SCREENING-METHOD
Term used for papers describing methods applicable to testing of drugs for particular activities.

SPASMOLYTICS
Smooth muscle relaxants; anticholinergics. * C/S /IT,FT SPASMOLYTIC OR ATROPINE OR PAPAVERINE OR SCOPOLAMINE

SEC.
Secondary.

SPERMATOCIDES
Drugs that kill spermatozoa or hasten their degeneration by impeding their passage through the cervical canal.

SEDATIVES
Substances inducing sleep. * C/S /IT,FT SEDATIVE OR BARBITURATE OR CHLORAL OR DIAZEPAM OR PHENOBARBITAL OR SCOPOLAMINE OR THIOBARBITURATE

SPRAY
Liquid droplets propelled by a gas. * Related AEROSOL

SEROLOGY
Term used for immunological techniques, e.g. radioimmunoassay.

STABILITY
Studies of the change in chemical or pharmacological activity of drugs in pharmaceutical preparations. * Related PHARMACEUTICS FORMULATION PHARM.PREP.

SEROTHERAPY
Therapy using antisera, globulins, etc.

STABILIZER
Pharmacologically inert substances used to maintain the integrity of pharmaceutical formulations. * Related AUXILIARY-INGREDIENT FORMULATION PHARM.PREP. PHARMACEUTICS

SEX
Applied when there is a difference in response, e.g. to drug action, between males and females.

SEX-HORMONE, FEMALE
* C/S /IT,FT ESTRADIOL OR ESTROGEN OR GONADOTROPIN OR PROGESTERONE OR PROGESTOGEN

STEADY-STATE
Situation when levels of a drug in body fluids and tissues has reached equilibrium, such that absorption and elimination of the drug are balanced.

SEX-HORMONE, MALE
* C/S /IT,FT ANDROGEN OR TESTOSTERONE

STERILIZATION
Term used for physical methods for killing microorganisms.

SIDE-EFFECT
An adverse reaction to a drug during clinical use. * C/S /IT,FT ALL SIDE-EFFECT: OR AGRANULOCYTOSIS OR EMBRYOPATHY OR (RING76 only) XXXV/PN

STRESS
Term used for any external stress, either natural or experimental, applied to man and animals.

STRUCT.ACT. SOLVENT
The medium, usually a liquid, which dissolves a solute to form a solution. * Related AUXILIARY-INGREDIENT FORMULATION PHARM.PREP. PHARMACEUTICS Term used for studies of relationships between chemical structure and chemical, or, especially, pharmacological activity.

SUBCELL.STRUCT.
Subcellular structure.

972 APPENDIX A

SUBCHRON.
Subchronic.

TACHYPHYLAXIS
A rapid diminution in response to each of a succession of repeated doses of a drug.

SUBCLIN.
Subclinical.

TARGETING
Term used for methods of directing delivery or release of a drug at a specific organ or tissue. * Related DRUG-DELIVERY

SUBST.
Substituted.

SYM.
Symmetrical.

TERATOGEN
Compound which induces malformation of the embryo.

SYMPATHOLYTICS
Adrenergic blocking drugs. Term used only for drugs which cannot be classified as alpha or beta blockers. * More Specific * C/S SYMPATHOLYTICS-ALPHA SYMPATHOLYTICS-BETA /IT,FT SYMPATHOLYTIC OR GUANETHIDINE OR PHENOXYBENZAMINE OR PHENTOLAMINE OR PRACTOLOL OR PROPRANOLOL

TERATOGENESIS
Malformation of the embryo. * Related * C/S CONGENITAL-DISEASE EMBRYOPATHY/IT,FT OR TERATOGENESIS/FT

TERT.
Tertiary.

THROMBOXANE-ANTAGONISTS
Drugs which antagonise the effects of thromboxanes and thromboxane mimetics.

SYMPATHOMIMETICS
Adrenergic agonists. Used only for drugs which cannot be classified as alpha or beta agonists. * More Specific * C/S SYMPATHOMIMETICS-ALPHA SYMPATHOMIMETICS-BETA /IT,FT SYMPATHOMIMETIC OR ADRENALINE OR AMPHETAMINE OR EPHEDRINE OR ISOPRENALINE OR NORADRENALINE OR TYRAMINE

THYMUS-HORMONE-METAB.
Metabolism of endogenous thymus hormones in man and animals. * Related * C/S THYMUS-HORMONES /IT,FT ALL HORMONE-METAB.: AND THYMUS AND HORMONE

SYNERGISTS
Drugs which enhance the pharmacological activity of other drugs e.g. beta-lactamase-inhibitors. * Related BETA-LACTAMASE-INHIBITORS

THYROID-HORMONES
* C/S /IT,FT THYROID-HORMONE OR DIIODOTYROSINE OR THYRONINE OR THYROXINE OR TRIIODOTHYRONINE

SYNTH.
Synthesis.

THYROID-HORMONE-METAB.
Metabolism of endogenous thyroid hormones in man and animals. * Related THYROID-HORMONES /IT,FT ALL HORMONE-METAB.: AND (THYROID-HORMONE OR DIIODOTYROSINE OR THYRONINE OR THYROXINE OR TRIIODOTHYRONINE)

T.I.D.
Dosage schedule in which the drug is administered three times a day. * Related DOSAGE

* C/S

Derwent Drug File 973 Thesaurus

THYROLIBERIN
* C/S /FT THYROLIBERIN OR LOPREMONE OR PROTIRELIN OR ((/FT ALL TSH: OR ALL THYROTROPIN:) AND ALL RELEASING:)

TRIAL-PREP.
A compound prepared for pharmacological testing which is identified by a code (usually alpha-numeric).

TROP . TISSUE-CULTURE
Term used for all in-vitro cultures of tissues or organs, including neoplastic cells. Tropical.

TUBERCULOSTATICS
Drugs inhibiting the growth and development of Mycobacterium tuberculosis and related species, but not Mycobact. leprae. * Related * C/S ANTIBIOTICS ANTISEPTICS /IT,FT TUBERCULOSTATIC OR CYCLOSERINE OR ISONIAZID OR PAS OR STREPTOMYCIN OR VIOMYCIN

TOCOLYTICS
Drugs that suppress premature labor by inhibiting contractions of the uterus. * Related LABOR OBSTETRICS

TOLERANCE
The state whereby drugs, usually in a clinical situation, have to be given in progressively larger doses to produce the desired effect.

UNCOUPLER
Activity of a drug that acts in the mitochondria to uncouple the production of ATP in the electron transport chain. * Related OX.PHOSPHORYLATION RESPIRAT.CHAIN

TOPICAL
Term used for application of drug to a particular site, where such application cannot be described by a more specific term. * More Specific DERMATOLOGICAL OPHTHALMOLOGICAL

URICOSURICS
Drugs that produce an increase in the urinary excretion of uric acid. * Related ANTIGOUTS

TOX.
Toxic/toxicity. Term used for studies of toxic effects in animals, e.g. LD50, mutagenesis, teratogenesis.

URINARY-TRACT-DISEASE
Term used for diseases of the urinary tract not covered by the more specific terms below. * More Specific * C/S BLADDER-DISEASE NEPHROPATHY /IT,FT G.U.DISEASE OR G.U.-INFECTION

TRACE-ELEMENT
Term used for chemical elements, which, in very small amounts, are essential in nutrition.

TRANQUILIZERS
Drugs which have anti-anxiety actions for use in anxiety neuroses. * Related NEUROLEPTICS PSYCHOSEDATIVES

UTEROTONICS
Drugs which increase the tone of the uterine muscle. * Related OBSTETRICS UTERUS

TRANSDERMAL
Administration of a drug via the surface of the skin. * Related PERCUTANEOUS

VACCINES
A suspension of killed or attenuated microorganisms, or other antigenic material, used for the induction of immunity. * Related ADJUVANTS ANTIBODY-RESPONSE IMMUNE-RESPONSE IMMUNITY

974 APPENDIX A

VASCULAR-DISEASE
Term used for diseases of blood vessels, other than brain and coronary vessels. * Related * C/S CEREBROVASCULAR-DISEASE CORONARY-DISEASE /IT,FT ARTERIOPATHY OR VENOPATHY

VET.
Vetinary.

VIS.
Visible.

YEAST
Term used only for commercially useful yeasts such as Saccharomyces cerevisiae. * Related FUNGUS

ZOOLOGY
Term used for animals, other than birds, fish, or mammals, only when compounds are isolated from them, or when they appear in a context other than use as experimental animals.

Derwent Drug File 975 Thesaurus

APPENDIX B
CHEMICAL SUBSTRUCTURE TERMS
1. INTRODUCTION

2.

APPLICATION TO OLDER FILES

A further entry provides the strategy needed to find such substructures in the older Derwent Drug and Veterinary Drug files. In many cases a Codeless Scanning (C/S) strategy is given. Some substructures are given no strategy at all because no suitable word exists in Codeless Scanning. It must also be stressed that the strategies provided cannot be guaranteed to afford comprehensive retrieval. They have been designed for users who are unfamiliar with the principles of the indexing systems used and therefore represent a simplified approach. The following points must be borne in mind when using Codeless Scanning concepts for substructure retrieval: (a) Generally only one substructure term was used for a drug or other standard compound, however many might have been applicable; the term used is indicated in the Codeless Scanning Thesaurus, Instruction Bulletin No. 3. Substructure terms were given for other compounds (e.g. synthesized chemicals) only if they actually appeared in a Codeless Scanning heading, and some may have been omitted because of limitations of space; heterocyclic terms can be searched fairly confidently since they were almost always included when appropriate, but this is not true of other terms. Where a More Specific term exists (usually for a well-known drug), the recommended strategy will not retrieve this term, e.g. MORPHINAN would give no references to MORPHINE or CODEINE; this difficulty can be overcome online by using the Derwent Drug Registry (DDR) to establish which compounds possess the substructure, and then cross-filing the drug names into the older files.

The following list provides definitions and searching hints for chemical substructure terms. All such terms are included, with the exception of most of the elements (e.g. SODIUM), where the definitions are self-evident.Most entries also have Related Terms. These are mainly wider terms which would have been used if the more precise defined term had not existed (e.g. ALCOHOL is a Related Term for AMINOALCOHOL); however, it must be stressed that ALCOHOL is not a higher term for (i.e. it is not assigned together with) AMINOALCOHOL. The major purpose of these Related Terms is to give an indication of how a strategy might be widened if an insufficient number of answers were found because the question was too specific. More Specific Terms have also been given for many entries. These indicate other substructure terms which are encompassed by the one which is defined, e.g. AMINOCYCLITOL for CYCLITOL; the latter is not included as a higher term when AMINOCYCLITOL is used as a keyword. Therefore, More Specific Terms should be included as alternatives in a search strategy for complete retrieval of all answers, e.g. a search for all cyclitols should be entered as: CYCLITOL--FT OR AMINOCYCLITOL--FT CYCLITOL-FT OR AMINOCYCLITOL-FT CYCLITOL *FT OR AMINOCYCLITOL *FT (DIALOG) (DataStar) (STN)

(b)

(c)

to ensure comprehensive retrieval unless, of course, such a substructure is definitely not required. Some of these More Specific Terms are given within parentheses, e.g. (IMIDE,CYCLIC) and (THIOLACTAM) for LACTAM; these represent possible alternatives in a strategy, but careful consideration should be given as to whether or not to use them - in this particular case, it might well be decided that thio lactams were acceptable but that cyclic imides were not. Thus More Specific terms which are not enclosed within parentheses are more or less mandatory alternatives for a strategy, whilst those within parentheses are merely possible alternatives. In one case, viz. COND.RING, there are so many More Specific Terms that these have not been quoted. More Specific Terms are again not given for MACROCYCLE, but in this case they are unnecessary since MACROCYCLE is automatically assigned as a higher term for all such keywords.

976 APPENDIX B

AA-LINKED Direct linkage between any two alicyclic rings via a single or double bond, including unsaturated analogs. * Related * More Specific * C/S ACETAL Used for compounds of the form R-CH(OR)-OR, where R = C, R or R = H or C. Either OR or OR may be part of ring systems, but the term is not used when both are in the same ring, e.g. in 1,3-dioxole. * Related * More Specific * C/S ACETYLENE Used for any carbon-to-carbon triple bond, where the carbon atoms may or may not be substituted. Usually acyclic, but may be within a ring. * Related * More Specific ACRIDINE Including all hydrogenated derivatives. * Related * More Specific * C/S ACYLHALIDE Used for compounds of the form R-C(=X)-Hal, where R = C, Hal = Br, Cl, F, I etc. X = O or (with CS-ACID) S. The appropriate substructure term for the halogen is also given. * Related * More Specific ADAMANTANE Including dehydrogenated derivatives. * Related * More Specific * C/S AH-LINKED-CC Direct linkage of carbon-to-carbon between any alicyclic ring and any heterocyclic ring, via a single or double bond. * Related * More Specific * C/S BRIDGE-STRUCT. CYCLOHEXANE ADAMANTANE/IT,FT BROMINE CHLORINE FLUORINE IODINE COND.RING PIPERIDINE PYRIDINE QUINOLINE ACRIDINE/IT,FT (UNSAT.FATTY-ACID) ALCOHOL ETHER POLYALCOHOL (GLYCOSIDE) (ORTHO-C-ESTER) THIOACETAL ACETAL/IT,FT -

AH-LINKED-CX Direct linkage of a carbon-to-heteroatom between any alicyclic ring and any heterocyclic ring, via a double or single bond. * Related * More Specific * C/S ALCOHOL Used for compounds of the form R-OH, where R = C, except aryl. * Related * More Specific (ACETAL) AMINOALCOHOL (AMINOCYCLITOL) ENOL (GLYCERIDE) HYDROXYACID (KETAL) (PHENOL) POLYALCOHOL RETINOID ALCOHOL/IT,FT -

* C/S ALDEHYDE

Used for compounds of the form R-CHO, where R = C, but not aryl. * Related * More Specific ARYLALDEHYDE POLYALDEHYDE THIOALDEHYDE (URONIC-ACID)

ALDIMINE Used for compounds of the form R-CH=NR, where R,R = H or C. * Related * More Specific ALKALOID Organic nitrogen-containing bases, mainly of plant origin. * Related * More Specific * C/S /IT ALKALOID OR ACONITUM OR CINCHONA OR CLAVICEPS OR COLCHICUM OR CURARE OR IPECAC OR LOBELIA OR OPIUM OR PSILOCYBE OR RAUWOLFIA OR VERATRUM OR VINCA OR ATROPINE OR CAFFEINE OR COCAINE OR CODEINE OR EMETINE OR EPHEDRINE OR MESCALINE OR MORPHINE OR MUSCARINE OR NICOTINE OR PAPAVERINE OR PHYSOSTIGMINE OR PILOCARPINE OR QUININE OR SCOPOLAMINE OR SPARTEINE OR STRYCHNINE OR THEOPHYLLINE OR YOHIMBINE OR LSD OR LYSERGIC-ACID (OXIME)

Derwent Drug File 977 Thesaurus

ALKANE Any unsubstituted straight or branched-chain acyclic saturated hydrocarbon. * Related * More Specific * C/S ALKYLBROMIDE Used for compounds of the form R-Br, where R = any C (including alicyclic rings) other than aryl. * Related * More Specific ALKYLCHLORIDE Used for compounds of the form R-Cl, where R = any C (including alicyclic rings) other than aryl. * Related * More Specific ALKYLFLUORIDE Used for compounds of the form R-F, where R = any C (including alicyclic rings) other than aryl. * Related * More Specific ALKYLIODIDE Used for compounds of the form R-I, where R = any C (including alicyclic rings) other than aryl. * Related * More Specific IODINE (N-MUSTARD) (SEMI-N-MUSTARD) FLUORINE (N-MUSTARD) (SEMI-N-MUSTARD) CHLORINE N-MUSTARD SEMI-N-MUSTARD BROMINE (N-MUSTARD) (SEMI-N-MUSTARD) ALKANE/IT

AMIDINE Used for compounds with two nitrogen atoms attached to a single carbon atom, of the form (i) R-C(=NR)-NRR or (ii) R-C(-NRR)-NRR, where R = H or C; each R may be anything and may be the same or different from other R. * Related * More Specific AMINE KETIMINE POLYAMINE AMIDINE,CYCLIC AMIDRAZONE CARBODIIMIDE FORMAZAN

AMIDINE,CYCLIC As for AMIDINE but the central carbon andone (but not two) of the nitrogens must be part of the same ring. * Related * More Specific AMIDRAZONE Used for compounds of the type R-C(NRR)-NR-NRR, where R = anything and may be the same or different. Includes analogs with C=N bonds. * Related * More Specific * C/S AMINE Used for compounds of the form R-NR-R, where R = C, R or R = H or C, but excluding those where any R is aryl. * Related * More Specific (AMIDINE) (AMIDINE,CYCLIC) AMINOACID AMINOALCOHOL AMINOCYCLITOL AMINOSUGAR ARALKYLAMINE ARYLAMINE (GUANIDINE) (GUANIDINE,CYCLIC) (HYDRAZINE) HYDROXYLAMINE N-MUSTARD POLYAMINEQUAT.AMINE SEMI-N-MUSTARD AMIDINE HYDRAZINE POLYAMINE FORMAZAN AMIDINE AMINE PTERIDINE PURINE

ALUMINUM-COMPLEX Used for compounds where an organic component is coordinated with aluminum. * Related * More Specific ALUMINUM COMPLEX AMINOACID

ALUMINUM-SALT Used for an aluminum salt of an organic acid. * Related * More Specific ALUMINUM -

Used for all carboxylic acids or their derivatives (esters, amides, etc.) with an amino group (substituted or not) attached to a carbon atom which forms part of the parent acid. * Related * More Specific * C/S AMINE C-ACID (BETAINE) PEPTIDE PROTEIN -

978 APPENDIX B

AMINOALCOHOL All compounds possessing a nitrogen atom and a hydroxyl group (which may be esterified but not otherwise substituted) provided that the groups are linked via carbon atoms in chains and/or rings. * Related * More Specific * C/S AMINOCYCLITOL Cyclohexanes substituted on each C by hydroxyl or amino groups (at least one of each). Includes derivatives such as ethers and esters. * Related ALCOHOL AMINEAMINOALCOHOL CYCLITOL CYCLOHEXANE POLYALCOHOL POLYAMINE ALCOHOL AMINE AMINOCYCLITOL (AMINOSUGAR) -

ANHYDRIDE,CYCLIC As for anhydride, but the group must form part of a ring. * Related * More Specific ANTHRACENE Including hydrogenated derivatives. * Related * More Specific BENZENE COND.RING NAPHTHALENE ANTHRACYCLINES (ARENE) TETRACYCLINES ANHYDRIDE LACTONE -

ANTHRACYCLINES Tetracycline analogs with a quinone B-ring possessing antibiotic and/or cytostatic activity. * Related * More Specific ANTHRACENE ARENE COND.RING NAPHTHALENE QUINONE TETRACYCLINES -

* More Specific AMINOSUGAR

Any sugar with one or more OH-groups replaced by amino groups (substituted or not). Includes derivatives such as ethers, esters, etc. * Related * More Specific * C/S AMMONIA Used for free ammonia and unsubstituted ammonium salts. See also QUAT.AMINE. * Related * More Specific * C/S ANDROSTANE Any steroid with both angular Me-groups and no C-atom at C17-beta. * Related * More Specific * C/S ANHYDRIDE Used for compounds of the form R-CO-O-OC-R, where R and R = C. * Related * More Specific C-ACID C-ESTER ANHYDRIDE,CYCLIC STEROID ANDROSTANE/IT,FT AMMONIA/IT,FT AMINE AMINOALCOHOL FURAN GLYCOSIDE POLYAMINE PYRAN SUGAR (NUCLEOSIDE) (NUCLEOTIDE) (POLYSACCHARIDE) AMINOSUGAR/IT,FT

ANTIMONY-COMPLEX Used for compounds where an organic component is coordinated with antimony. * Related * More Specific ANTIMONY COMPLEX -

ANTIMONY-SALT Used for an antimony salt of an organic acid. * Related * More Specific ARALKYLAMINE Used for a benzene ring which has one substituent of the form -R-NRR or -R-CR=NR, and where R = alkyl or alkenyl (substituted or not), R,R = anything, including cyclic NRR derivatives such as piperidine. * Related * More Specific * C/S ARENE Condensed aromatic ring systems with 4 or more rings. Includes hydrogenated derivatives, but excludes steroids and triterpenes. * Related ANTHRACENE BENZENE COND.RING NAPHTHALENE PHENANTHRENE ANTHRACYCLINES TETRACYCLINES AMINE ARALKYLAMINE/IT,FT ANTIMONY -

* More Specific

Derwent Drug File 979 Thesaurus

ARYL-C-ACID Used for compounds of the type aryl-COOH. Also used for derivatives other than the amides or esters. * Related * More Specific ARYL-C-AMIDE Used for compounds of the type aryl-CONRR, where RR = anything. * Related * More Specific ARYL-C-ESTER Used for compounds of the type aryl-COOR, where R = C. * Related * More Specific ARYLALDEHYDE Used for compounds of the type aryl-CHO. * Related * More Specific ARYLAMINE Used for compounds of the type aryl-NRR, where R = anything, and RR= anything including cyclic NRRderivatives. * Related * More Specific ARYLBROMIDE Used for compounds of the type aryl-Br. * Related * More Specific ARYLCHLORIDE Used for compounds of the type aryl-Cl. * Related * More Specific ARYLFLUORIDE Used for compounds of the type aryl-F. * Related * More Specific ARYLIODIDE Used for compounds of the type aryl-I. * Related * More Specific IODINE THYRO-C-ACID FLUORINE CHLORINE BROMINE AMINE ALDEHYDE C-ESTER DEPSIDE C-AMIDE C-ACID SALICYLIC-ACID THYRO-C-ACID

ARYLKETONE Used for compounds of the type aryl-CO-R, where R = C. * Related * More Specific ARYLSULFIDE Used for compounds of the type aryl-SR, where R = C. * Related * More Specific PHENOL-ETHER SULFIDE KETONE BUTYROPHENONE CHALCONE

AZACYCLODODECANE Any 12-membered ring with 1 N atom and 11 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

AZACYCLOHENEICOSANE Any 21-membered ring with 1 N atom and 20 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

AZACYCLONONACOSANE Any 29-membered ring with 1 N atom and 28 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

AZACYCLONONADECANE Any 19-membered ring with 1 N atom and 18 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

AZACYCLOPENTADECANE Any 15-membered ring with 1 N atom and 14 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

980 APPENDIX B

AZACYLOTETRADECANE Any 14-membered ring with 1 N atom and 13 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

AZAPHENOTHIAZINE Used when an N atom replaces a C atom in a phenothiazine ring (excluding the C atoms at the junctions of the rings). Includes hydrogenated derivatives. * Related * More Specific * C/S AZAPHOSPHOLE Any 5-membered ring with 1 N atom, 1 P atom and 3 C atoms. * Related * More Specific COND.RING PIPERIDINE PYRIDINE THIAZINE AZAPHENOTHIAZINE/IT,FT

AZACYCLOTRICOSANE Any 23-membered ring with 1 N atom and 22 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

AZACYCLOTRIDECANE Any l3-membered ring with 1 N atom and 12 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

AZAPHOSPHORINE Any 6-membered ring with 1 N atom, 1 P atom and 4 C atoms. * Related * More Specific -

AZATETRAOXACYCLOPENTADECANE Any 15-membered ring with 1 N atom, 4 O atoms and 10 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S AZECINE Any 10-membered ring with 1 N-atom and 9 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S AZEPINE Any 7-membered ring with 1 N atom and 6 C atoms. * Related * More Specific * C/S AZETIDINE Any 4-membered ring with 1 N atom and 3 C atoms. * Related * More Specific * C/S CEPHALOSPORINS PENICILLINS AZETIDINE/IT,FT DIBENZAZEPINE AZEPINE/IT,FT MACROCYCLE AZECINE/FT MACROCYCLE -

AZACYCLOUNDECANE Any 11-membered ring with 1 N atom and 10 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

AZACYCLOUNTRIACONTANE Any 3l-membered ring with 1 N-atom and 30 C-atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

AZAPENTAOXACYCLOHEXADECANE Any 16-membered ring with 1 N atom, 5 O atoms and 10 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

Derwent Drug File 981 Thesaurus

AZIDE Used for compounds of the form R-N=N+=N, where R = anything. See also TRIAZENE. * Related * More Specific AZIRIDINE Any 3-membered ring with 1 N atom and 2 C atoms. * Related * More Specific * C/S AZO Used for compounds of the form R-N=N-R, where R or R = C. * Related * More Specific AZOCINE Any 8-membered ring containing 1 N atom and 7 C atoms. * Related * More Specific * C/S AZONINE Any 9-membered ring with 1 N atom and 8 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S AZULENE Including hydrogenated derivatives. * Related * More Specific * C/S BA-LINKED Direct linkage between a benzene ring and any alicyclic (saturated or dehydrogenated) ring via a single bond. * Related * More Specific * C/S COND.RING CYCLOHEPTANE CYCLOPENTANE AZULENE/IT,FT MACROCYCLE AZONINE/IT,FT AZOCINE/IT,FT HYDRAZINE DIAZONIUM (FORMAZAN) TRIAZENE AZIRIDINE/IT,FT -

BARBITURATES Used for barbituric acid or any derivative thereof. * Related * More Specific * C/S IMIDE,CYCLIC PYRIMIDINE UREA,CYCLIC THIOBARBITURATES BARBITURATE/IT,FT

BARIUM-COMPLEX Used for compounds where an organic component is coordinated with barium. * Related * More Specific BARIUM-SALT Used for a barium salt of an organic acid. * Related * More Specific BB-LINKED Direct linkage between two benzene rings via a single bond, as in biphenyl and all derivatives thereof. * Related * More Specific * C/S BENZENE Used for benzene itself and simple derivatives (e.g. toluene) for which there is no other substructure term. * Related * More Specific ANTHRACENE ARENE BIPHENYL DIPHENYLMETHANE NAPHTHALENE PHENANTHRENE STILBENE BIPHENYL BIPHENYL/IT,FT BARIUM BARIUM COMPLEX -

BENZIMIDAZOLE Including hydrogenated derivatives. * Related * More Specific COND.RING IMIDAZOLE -

BENZODIAZEPINE Used when a benzene ring is condensed to a seven-membered ring containing any two N atoms, the other atoms in the ring being C atoms. Includes hydrogenated derivatives. * Related * More Specific * C/S COND.RING DIAZEPINE BENZODIAZEPINE/IT,FT

982 APPENDIX B

BENZOFURAN Including hydrogenated derivatives. See also ISOBENZOFURAN. * Related * More Specific * C/S BENZOPYRAN Including hydrogenated derivatives. See also ISOBENZOPYRAN. * Related * More Specific * C/S COND.RING PYRAN CANNABINOIDS COUMARIN FLAVONOID XANTHENE BENZOPYRAN/IT,FT COND.RING FURAN BENZOFURAN/IT,FT

BH-LINKED-CX Direct linkage of carbon-to-hetero atom between a benzene ring and any heterocyclic ring via a single bond. * Related * More Specific * C/S BILE-ACID Any steroid with a carboxylic or sulfonic acid in the C-17 side chain. Also used for derivatives such as esters and amides. * Related * More Specific * C/S BIPHENYL Used when two benzene rings are connected via a single bond. Includes all derivatives and hydrogenated analogs. BB-LINKED or BA-LINKED always appear in addition. * Related * More Specific BENZENE (CANNABINOIDS) C-ACID CHOLESTANE STEROID SULFONIC-ACID 17-BETA-ALKYLSTEROID BILE-ACID/IT,FT -

BENZOQUINOLIZINE Any quinolizine condensed with a benzene ring, including hydrogenated derivatives. * Related COND.RING ISOQUINOLINE PIPERIDINE PYRIDINE QUINOLINE QUINOLIZINE BENZOQUINOLIZINE/IT,FT

* More Specific * C/S

BERYLLIUM-COMPLEX Used for compounds where an organic component is coordinated with beryllium. * Related * More Specific BETAINE Used for compounds of the form R-N RR-R-COO , where each R = C and may be the same or different. Also used for analogs of the quaternary amine (e.g. oxonium) or carboxylate (e.g. sulfonate); in such cases the additional term for the analog (e.g. ONIUM, SULFONIC-ACID) is also used. Not used for zwitterionic forms. * Related * More Specific * C/S BH-LINKED-CC Direct linkage of carbon-to-carbon between a benzene ring and any heterocyclic ring via a single bond. * Related * More Specific * C/S FLAVONOID AMINOACID C-ACID QUAT.AMINE BETAINE/IT,FT
+

BISMUTH-COMPLEX Used for compounds where an organic component is coordinated with bismuth. * Related * More Specific BISMUTH-SALT Used for a bismuth salt of an organic acid. * Related * More Specific BISMUTH BISMUTH COMPLEX -

BERYLLIUM COMPLEX -

BORON-COMPLEX Used for compounds where an organic component is coordinated with boron. * Related * More Specific BRIDGE-STRUCT. Any two-ring system with three or more atoms common to both rings. * Related * More Specific ADAMANTANE PORPHYRIN QUINUCLIDINE TROPANE BORON COMPLEX -

Derwent Drug File 983 Thesaurus

BROMINE Used for the element itself and also for bromine attached to a heterocyclic ring or to any atom other than carbon. * Related * More Specific ALKYLBROMIDE ARYLBROMIDE

CALCIUM-COMPLEX Used for compounds where an organic component is coordinated with calcium. * Related * More Specific CALCIUM-SALT Used for a calcium salt of an organic acid. * Related * More Specific CANNABINOIDS Active components of marihuana such as tetrahydrocannabinol, and close analogs (including a broken pyran ring) thereof. * Related * More Specific * C/S CARBAMATE Used for compounds of the form R-NR-COOR, where R,R,R = anything. * Related * More Specific CARBAMATE,CYCLIC DITHIOCARBAMATE THIOCARBAMATE THIOCARBAMATE,CYCLIC BA-LINKED BENZOPYRAN BIPHENYL COND.RING ISOBENZOPYRAN CANNABINOID/IT,FT (from 1974 only) CALCIUM CALCIUM COMPLEX -

BUTYROPHENONE Used when a benzene ring has the substituent -COCH2CH2CH3. Includes any substituted derivative. * Related * More Specific * C/S C-ACID Used for compounds of the form R-COOH, where R = substituted alkyl, unless a more specific term is applicable. * Related * More Specific AMINOACID ANHYDRIDE ARYL-C-ACID BETAINE BILE-ACID CS-ACID FATTY-ACID HAL.FATTY-ACID HYDROXY ACID KETO ACID POLY-C-ACID THYRO-C-ACID ARYLKETONE KETONE BUTYROPHENONE/IT,FT

C-AMIDE Used for compounds of the form R-CONRR, where R = any C except aryl. Also used for acyclic imides of the type R-CO-NR-CO-R. * Related * More Specific ARYL-C-AMIDE DEPSIPEPTIDE (HYDROXAMIC-ACID) (LACTAM) PEPTIDE (THIOHYDROXAMIC-ACID) (THIOLACTAM)

CARBAMATE,CYCLIC As for CARBAMATE, but the central carbon must be part of a ring. * Related * More Specific CARBAZOLE Including hydrogenated derivatives. * Related * More Specific COND.RING INDOLE PYRROLE PYRROLIDINE CARBAZOLE/IT,FT CARBAMATE -

C-ESTER Used for compounds of the form R-COOR, where R = any C except aryl, R = anything. * Related * More Specific (ANHYDRIDE) ARYL-C-ESTER CS-ESTER DEPSIDE DEPSIPEPTIDE GLYCERIDE (LACTONE) PHOSPHOLIPID (THIOLACTONE)

CADMIUM-COMPLEX Used for compounds where an organic component is coordinated with cadmium. * Related * More Specific CADMIUM-SALT Used for a cadmium salt of an organic acid. * Related * More Specific CADMIUM CADMIUM COMPLEX -

* C/S CARBODIIMIDE

Used for compounds of the type R-N=C=N-R,where R,R = anything. * Related * More Specific AMIDINE -

984 APPENDIX B

CARBOLINE Includes hydrogenated derivatives. * Related * More Specific * C/S CARBONATE Used for carbonic acid and all derivatives there of. * Related * More Specific CAROTENOID Used for beta-carotene and close analogs thereof. * Related * More Specific * C/S CYCLOHEXANE POLYOLEFIN TERPENE RETINOID CAROTENOID/IT,FT COND.RING INDOLE PIPERIDINE PYRIDINE PYRIDINE PYRROLE PYRROLIDINE CARBOLINE/IT,FT

CHOLESTANE Steroids with two angular methyl groups and a C17-beta side-chain of the type -CHMe-(CH2)3-CH(CH3)2 * Related * More Specific STEROID 17-BETA-ALKYLSTEROID (BILE-ACID)

CHROMIUM-COMPLEX Used for compounds where an organic component is coordinated with chromium. * Related * More Specific CHROMIUM COMPLEX -

CHROMIUM-SALT Used for a chromium salt of an organic acid. * Related * More Specific CINNOLINE Including hydrogenated derivatives. * Related * More Specific * C/S COND.RING PYRIDAZINE CINNOLINE/IT,FT CHROMIUM -

CEPHALOSPORINS Used for antibiotics with a thiazine beta-lactam ring. * Related * More Specific * C/S CERIUM-SALT Used for a cerium salt of an organic acid. * Related * More Specific CERIUM AMINOACID AZETIDINE COND.RING LACTAM THIAZINE CEPHALOSPORINS/IT,FT

COBALT-COMPLEX Used for compounds where an organic component is coordinated with cobalt. * Related * More Specific COBALT-SALT Used for a cobalt salt of an organic acid. * Related * More Specific COMPLEX Used for all inorganic and organic coordination compounds; in the former case a further term, e.g. ALUMINUM-COMPLEX, is used in addition. * Related * More Specific COND.RING Any two-ring system with two atoms common to both rings. * Related * More Specific * C/S COBALT COBALT COMPLEX -

CESIUM-COMPLEX Used for compounds where an organic component is coordinated with cesium. * Related * More Specific CHALCONE Used for compounds of the form Ar-CO-CH=CH-Ar, where Ar, Ar = any aryl. * Related * More Specific * C/S CHLORINE Used for the element itself and for chlorine attached to a heterocyclic ring or to any atom other than carbon. * Related * More Specific ALKYLCHLORIDE ARYLCHLORIDE ARYLKETONE KETONE CHALCONE/IT,FT OLEFIN CESIUM COMPLEX -

Derwent Drug File 985 Thesaurus

COPPER-COMPLEX Used for compounds where an organic component is coordinated with copper. * Related * More Specific COPPER-SALT Used for a copper salt of an organic acid. * Related * More Specific CORRINOID Including hydrogenated derivatives. Applied to many vitamin B12 compounds. * Related BRIDGE-STRUCT. MACROCYCLE OLEFIN POLYOLEFIN PYRROLE TETRAAZACYCLOPENTADECANE CORRINOID/IT,FT COPPER COPPER COMPLEX -

CYCLOBUTANE Any 4-membered carbocyclic ring, saturated or not. * Related * More Specific CYCLODECANE Any 10-membered carbocyclic ring, saturated or not. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE CYCLODECANE/FT -

CYCLODODECANE Any 12-membered carbocyclic ring, saturated or not. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

* More Specific * C/S COUMARIN

CYCLOHEPTADECANE Any 17-membered carbocyclic ring, saturated or not. MACROCYCLE always appears in addition. * Related * More Specific * C/S CYCLOHEPTANE Any 7-membered carbocyclic ring, saturated or not. * Related * More Specific AZULENE DIBENZOCYCLOHEPTADIENE TROPANE MACROCYCLE -

Including hydrogenated derivatives. * Related * More Specific CS-ACID Used for compounds of the form R-CS-OH, R-CS-SH, or R-CO-SH, where R = C. Also used for thio-analogs of oxygen-containing terms where the specific term does not exist, e.g. CS-ACID, C-AMIDE for R-CS-NH2. * Related * More Specific CS-ESTER Any ester of a CS-acid. * Related * More Specific CYANATE Used for compounds containing an R-O-function attached to a carbon atom which is triply-bonded to an N atom, where R = anything. See also ISOCYANATE. * Related * More Specific CYCLITOL Includes derivatives such as ethers and esters. * Related * More Specific CYCLOHEXANE POLYALCOHOL AMINOCYCLITOL ETHER NITRILE THIOCYANATE C-ESTER C-ACID (THIOHYDROXAMIC-ACID) BENZOPYRAN COND.RING LACTONE PYRAN -

CYCLOHEXADECANE Any 16-membered carbocyclic ring, saturated or not. MACROCYCLE always appears in addition. * Related * More Specific * C/S CYCLOHEXANE Any 6-membered carbocyclic ring, saturated or not, except those with three double bonds. * Related * More Specific ADAMANTANE AMINOCYCLITOL CAROTENOID CYCLITOL RETINOID MACROCYCLE -

986 APPENDIX B

CYCLONONANE Any 9-membered carbocyclic ring, saturated or not. MACROCYCLE always appears in addition. * Related * More Specific CYCLOOCTANE Any 8-membered carbocyclic ring, saturated or not. * Related * More Specific MACROCYCLE -

CYCLOTETRADECANE Any 14-membered carbocyclic ring, saturated or not. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

CYCLOTRIDECANE Any 13-membered carbocyclic ring, saturated or not. MACROCYCLE always appears in addition. * Related MACROCYCLE * More Specific * C/S

CYCLOPENTADECANE Any 15-membered carbocyclic ring, saturated or not. MACROCYCLE always appears in addition. * Related * More Specific * C/S CYCLOPENTANE Any 5-membered carbocyclic ring, saturated or not. * Related * More Specific CYCLOPROPANE Any 3-membered carbocyclic ring, saturated or not. * Related * More Specific CYCLOSTEROID A steroid containing an additional 3- or more membered ring within the nucleus.The additional ring must be formed by a direct bond between two of the steroid nucleus C-atoms, additional bridge atoms prohibiting the use of this term. * Related * More Specific * C/S STEROID CYCLOSTEROID/IT,FT AZULENE FLUORENE INDENE MACROCYCLE -

CYCLOUNDECANE Any 11-membered carbocyclic ring, saturated or not. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

DECAOXAZACYCLOTRITRIACONTANE Any 33-membered ring with 10 O atoms, 1 N atom and 22 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S DEPSIDE An ester of an aromatic hydroxy acid with a hydroxy acid. * Related * More Specific * C/S DEPSIPEPTIDE Mixed esters and amides of amino acids and hydroxy acids. PEPTIDE,CYCLIC is used in addition for cyclic depsipeptides. * Related * More Specific * C/S C-AMIDE C-ESTER PEPTIDE DEPSIPEPTIDE/IT,FT ARYL-C-ESTER C-ESTER HYDROXYACID DEPSIDE/IT,FT MACROCYCLE -

CYCLOTETRACOSANE Any 24-membered carbocyclic ring, saturated or not. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

DIAZACYCLODOCOSANE Any 22-membered ring with 2 N atoms and 20 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

Derwent Drug File 987 Thesaurus

DIAZACYCLODODECANE Any 12-membered ring with 2 N atoms and 10 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

DIAZADIPHOSPHOCINE Any 8-membered ring with 2 N atoms, 2 P atoms and 4 C atoms. MACROCYCLE always appears in addition. * Related * More Specific -

DIAZAPHOSPHEPINE Any 7-membered ring with 2 N atoms, 1 P atom and 4 C atoms. * Related * More Specific -

DIAZACYCLONONADECANE Any 19-membered ring with 2 N atoms and 17 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

DIAZAPHOSPHOCINE Any 8-membered ring with 2 N atoms, 1 P atom and 5 C atoms. * Related * More Specific * C/S DIAZAPHOSPHOCINE

DIAZACYCLOOCTADECANE Any 18-membered ring with 2 N atoms and 16 O atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

DIAZAPHOSPHOLE Any 5-membered ring with 2 N atoms, 1 P atom and 2 C atoms. * Related * More Specific * C/S DIAZAPHOSPHOLE

DIAZACYCLOPENTADECANE Any 15-membered ring with 2 N atoms and 13 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

DIAZAPHOSPHORANE Any 6-membered ring with 2 N atoms, 1 P atom and 3 C atoms. * Related * More Specific * C/S DIAZEPINE Any 7-membered ring with 2 N atoms and 5 C atoms. * Related * More Specific * C/S DIAZETIDINE Any 4-membered ring with 2 N atoms and 2 C atoms. * Related * More Specific DIAZIRIDINE Any 3-membered ring with 2 N atoms and 1 C atom. * Related * More Specific * C/S DIAZIRIDINE/FT BENZODIAZEPINE DIAZEPINE/IT,FT DIAZAPHOSPHORANE/FT

DIAZACYCLOTETRADECANE Any 14-membered ring with 2 N atoms and 12 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

DIAZACYCLOTRIDECANE Any 13-membered ring with 2 N atoms and 11 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

DIAZACYCLOUNDECANE Any 11-membered ring with 2 N atoms and 9 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

988 APPENDIX B

DIAZOCINE Any 8-membered ring with 2 N atoms and 6 C atoms. * Related * More Specific * C/S DIAZONINE Any 9-membered ring with 2 N atoms and 7 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S DIAZONIUM Used for compounds where an N atom is triply bonded to N-R, where R = C. * Related * More Specific DIBENZAZEPINE Including hydrogenated derivatives. * Related * More Specific * C/S AZEPINE COND.RING DIBENZAZEPINE/IT,FT AZO HYDRAZINE MACROCYCLE DIAZONINE/FT DIAZOCINE/FT

DIOXACYCLODODECANE Any 12-membered ring with 2 O atoms and 10 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

DIOXACYCLODOTRIACONTANE Any 32-membered ring with 2 O atoms and 30 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

DIOXACYCLOEICOSANE Any 20-membered ring with 2 O atoms and 18 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

DIOXACYCLOHENEICOSANE Any 21-membered ring with 2 O atoms and 19 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

DIBENZOCYCLOHEPTADIENE Including hydrogenated derivatives. * Related * More Specific * C/S DIOXABORIN Any 6-membered ring with 2 O atoms, 1 B atom and 3 C atoms. * Related * More Specific BORON COND.RING CYCLOHEPTANE DIBENZOCYCLOHEPTADIENE /IT,FT

DIOXACYCLOHEPTACOSANE Any 27-membered ring with 2 O atoms and 25 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

DIOXACYCLOHEPTADECANE Any 17-membered ring with 2 O atoms and 15 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

DIOXACYCLODOCOSANE Any 22-membered ring with 2 O atoms and 20 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

DIOXACYCLOHEXADECANE Any 16-membered ring with 2 O atoms and 14 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

Derwent Drug File 989 Thesaurus

DIOXACYCLOHEXATRIACONTANE Any 36-membered ring with 2 O atoms and 34 C atoms. * Related * More Specific * C/S MACROCYCLE -

DIOXACYCLOTETRACOSANE Any 24-membered ring with 2 O atoms and 22 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

DIOXACYCLONONADECANE Any 19-membered ring with 2 O atoms and 17 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE DIOXACYCLOTETRADECANE Any 14-membered ring with 2 O atoms and 12 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S DIOXACYCLOOCTACOSANE Any 28-membered ring with 2 O atoms and 26 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE DIOXACYCLOTETRATRIACONTANE Any 34-membered ring with 2 O atoms and 32 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S DIOXACYCLOOCTADECANE Any 18-membered ring with 2 O atoms and 16 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE DIOXACYCLOTRIACONTANE Any 30-membered ring with 2 O atoms and 28 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S,R/S DIOXACYCLOPENTACOSANE Any 25-membered ring with 2 O atoms and 23 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE DIOXACYCLOTRIDECANE Any 13-membered ring with 2 O atoms and 11 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S DIOXACYCLOPENTADECANE Any 15-membered ring with 2 O atoms and 13 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE DIOXACYCLOUNDECANE Any 11-membered ring with 2 O atoms and 9 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S DIOXACYCLOTETRACONTANE Any 40-membered ring with 2 O atoms and 38 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE DIOXADIAZACYCLODOTRIACONTANE Any 32-membered ring with 2 O atoms, 2 N atoms and 28 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE MACROCYCLE MACROCYCLE MACROCYCLE MACROCYCLE MACROCYCLE -

990 APPENDIX B

DIOXADIAZACYCLOOCTACOSANE Any 28-membered ring with 2 O atoms, 2 N atoms and 24 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

DIOXADITHIEPIN Any 7-membered ring with 2 O atoms, 2 S atoms and 3 C atoms. * Related * More Specific * C/S DIOXADITHIEPIN

DIOXADIAZACYCLOPENTACOSANE Any 25-membered ring with 2 O atoms, 2 N atoms and 21 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S,R/S MACROCYCLE -

DIOXADITHIOCIN Any 8-membered ring with 2 O atoms, 2 S atoms and 4 C atoms. * Related * More Specific -

DIOXADITHIONIN Any 9-membered ring with 2 O atoms, 2 S atoms and 5 C atoms. MACROCYCLE always appears in addition. * Related * More Specific MACROCYCLE -

DIOXADIAZACYCLOPENTADECANE Any 15-membered ring with 2 O atoms, 2 N atoms and 11 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S,R/S MACROCYCLE -

DIOXAHEXAAZACYCLOTETRACOSANE Any 24-membered ring with 2 O atoms, 6 N atoms and 16 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S DIOXANE Any 6-membered ring with 2 O atoms and 4 C atoms. * Related * More Specific * C/S DIOXANE/IT,FT MACROCYCLE -

DIOXADIAZACYCLOTETRACOSANE Any 24-membered ring with 2 O atoms, 2 N atoms and 20 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE _

DIOXADIAZACYCLOTRIACONTANE Any 30-membered ring with 2 O atoms 2 N atoms and 26 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

DIOXAPHOSPHABORIN Any 6-membered ring with 2 O atoms, 1 P atom, 1 B atom and 2 C atoms. * Related * More Specific BORON -

DIOXADIAZOCINE Any 8-membered ring with 2 O atoms, 2 N atoms and 4 C atoms. * Related * More Specific * C/S DIOXADIAZOCINE

DIOXAPHOSPHEPIN Any 7-membered ring with 2 O atoms, 1 P atom and 4 C atoms. * Related * More Specific

DIOXADITHIATETRAAZACYCLOOCTACOSANE Any 28-membered ring with 2 O atoms, 2 S atoms, 4 N atoms and 20 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

DIOXAPHOSPHOLANE Any 5-membered ring with 2 O atoms, 1 P atom and 2 C atoms. * Related * More Specific -

Derwent Drug File 991 Thesaurus

DIOXAPHOSPHORINANE Any 6-membered ring with 2 O atoms, 1 P atom and 3 C atoms. * Related * More Specific * C/S DIOXARSOLE Any 5-membered ring with 2 O atoms, 1 As atom and 2 C atoms. * Related * More Specific * C/S DIOXASTANNIN Any 6-membered ring with 2 O atoms, 1 Sn atom and 3 C atoms. * Related * More Specific TIN ORGANOMETALLIC ARSENIC DIOXARSOLE DIOXAPHOSPHORINANE/FT

DIOXATHIOLANE Any 5-membered ring with 2 O atoms, 1 S atom and 2 C atoms. * Related * More Specific -

DIOXATRITHIAHEXAAZACYCLOTETRACONTANE Any 40-membered ring with 2 O atoms, 3 S atoms, 6 N atoms and 29 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S -

DIOXAZACYCLOHENEICOSANE Any 21-membered ring with 2 O atoms, 1 N atom and 18 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

DIOXASTANNOLE Any 5-membered ring with 2 O atoms, 1 Sn atom and 2 C atoms. * Related * More Specific TIN ORGANOMETALLIC -

DIOXAZACYCLOHEPTACOSANE Any 27-membered ring with 2 O atoms, 1 N atom and 24 C atoms. MACROCYCLE always appears in addition * Related * More Specific * C/S MACROCYCLE -

DIOXATHIADIAZACYCLOUNDECANE Any 11-membered ring with 2 O atoms, 1 S atom, 2 N atoms and 6 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S DIOXATHIANE Any 6-membered ring with 2 O atoms, 1 S atom and 3 C atoms. * Related * More Specific * C/S DIOXATHIEPIN Any 7-membered ring with 2 O atoms, 1 S atom and 4 C atoms. * Related * More Specific DIOXATHIANE/FT MACROCYCLE -

DIOXAZACYCLOHEXACOSANE Any 26-membered ring with 2 O atoms, 1 N atom and 23 C atoms. MACROCYCLE always appears in addition * Related * More Specific * C/S MACROCYCLE -

DIOXAZACYCLOHEXADECANE Any 16-membered ring with 2 O atoms, 1 N atom and 13 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

DIOXAZACYCLONONACOSANE Any 29-membered ring with 2 O atoms, 1 N atom and 26 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

992 APPENDIX B

DIOXAZACYCLOPENTACOSANE Any 25-membered ring with 2 O atoms, 1 N atom and 22 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

DIOXAZINE Any 6-membered ring with 2 O atoms, 1 N atom and 3 C atoms. * Related * More Specific DIOXAZOCINE Any 8-membered ring with 2 O atoms, 1 N atom and 5 C atoms. * Related * More Specific * C/S DIOXECIN Any 10-membered ring with 2 O atoms and 8 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S DIOXEPIN Any 7-membered ring with 2 O atoms and 5 C atoms. * Related * More Specific DIOXETANE Any 4-membered ring with 2 O atoms and 2 C atoms. * Related * More Specific * C/S DIOXOCIN Any 8-membered ring with 2 O atoms and 6 C atoms. * Related * More Specific * C/S DIOXOLE Any 5-membered ring with 2 O atoms and 3 C atoms. * Related * More Specific DIOXONIN Any 9-membered ring with 2 O atoms and 7 C atoms. MACROCYCLE always appears in addition. * Related * More Specific MACROCYCLE DIOXOCIN/FT DIOXETANE MACROCYCLE DIOXAZOCINE/FT -

DIOXAZACYCLOPENTADECANE Any 15-membered ring with 2 O atoms, 1 N atoms and 12 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

DIOXAZAPHOSPHOCIN Any 8-membered ring with 2 O atoms, 1 N atom, 1 P atom and 4 C atoms. * Related * More Specific -

DIOXAZASILACYCLOOCTADECANE Any 18-membered ring with 2 O atoms, 1 N atom, 1 Si atom and 14 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE SILICON -

DIOXAZASILACYCLOOCTANE Any 8-membered ring with 2 O atoms, 1 N atom, 1 Si atom and 4 C atoms. * Related * More Specific * C/S -

DIOXAZASTANNECINE Any 10-membered ring with 2 O atoms, 1 N atom, 1 Sn atom and 6 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S DIOXAZEPINE Any 7-membered ring with 2 O atoms, 1 N atom and 4 C atoms. * Related * More Specific * C/S DIOXAZEPINE MACROCYCLE TIN ORGANOMETALLIC -

Derwent Drug File 993 Thesaurus

DIPHENYLMETHANE Used for compounds of the form Ph2-CRR or Ph2-C=R, where R or R = anything. Includes hydrogenated derivatives. * Related * More Specific * C/S DISULFIDE Used for compounds of the form R-S-S-R,where R or R = C. * Related * More Specific SULFIDE SULFUR THIURAM BENZENE DIPHENYLMETHANE/IT,FT

DITHIATETRASTANNEPIN Any 7-membered ring with 2 S atoms, 4 Sn atoms and 1 C atom. * Related * More Specific DITHIAZEPINE Any 7-membered ring with 2 S atoms, 1 N atom and 4 C atoms. * Related * More Specific * C/S DITHIAZEPINE/FT TIN ORGANOMETALLIC -

DITHIADIAZECINE Any 10-membered ring with 2 S atoms, 2 N atoms and 6 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE DITHIADIAZECINE DITHIAZINE Any 6-membered ring with 2 S atoms, 1 N atom and 3 C atoms. * Related * More Specific DITHIAZOCINE Any 8-membered ring with 2 S atoms, 1 N atom and 5 C atoms. * Related * More Specific DITHIAZOLE Any 5-membered ring with 2 S atoms, 1 N atom and 2 C atoms. * Related * More Specific DITHIETANE Any 4-membered ring with 2 S atoms and 2 C atoms. * Related * More Specific -

DITHIADIAZEPINE Any 7-membered ring with 2 S atoms, 2 N atoms and 3 C atoms. * Related * More Specific DITHIANE Any 6-membered ring with 2 S atoms and 4 C atoms. * Related * More Specific DITHIARSOLE Any 5-membered ring with 2 S atoms, 1 As atom and 2 C atoms. * Related * More Specific DITHIASTIBOLE Any 5-membered ring with 2 S atoms, 1 Sb atom and 2 C atoms. * Related * More Specific ANTIMONY ARSENIC -

DITHIOCARBAMATE Used for compounds of the type R-NR-C(=S)-S-R, where R,R,R = anything. If the central C is part of a ring, THIOCARBAMATE,CYCLIC is also used. * Related * More Specific DITHIOLE Any 5-membered ring with 2 S atoms and 3 C atoms. * Related * More Specific CARBAMATE THIOCARBAMATE THIURAM

DITHIATETRAAZACYCLOHEPTADECANE Any 17-membered ring with 2 S atoms, 4 N atoms and 11 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

994 APPENDIX B

DYSPROSIUM-COMPLEX Used for compounds where an organic component is coordinated with dysprosium. * Related * More Specific DYSPROSIUM COMPLEX -

FATTY-ACID Any straight- or branched-chain, unsubstituted, saturated monocarboxylic acid with a total of 3 or more C atoms. Includes derivatives such as esters and amides, and includes analogs with cycloalkyl substituents in the chain. * Related * More Specific * C/S C-ACID GLYCERIDE HAL.FATTY-ACID PHOSPHOLIPID UNSAT.FATTY-ACID FATTY-ACID/IT,FT N.B. GLYCERIDE/IT,FT could also be considered for additional hits. FLAVONOID Used for compounds with a benzopyran ring substituted at C-2 or C-3 by an aryl group. * Related * More Specific * C/S FLUORENE Including hydrogenated derivatives. * Related * More Specific FLUORINE Used for the element itself and for fluorine attached to a heterocyclic ring or to any atom other than carbon. * Related * More Specific FORMAZAN These are compounds of the type R-N=N-CR-N=N-R, where R,R,R = anything. Includes analogs with single N-N or C-N bonds. * Related * More Specific * C/S FURAN Any 5-membered ring with 1 O atom and 4 C atoms. * Related * More Specific (AMINOSUGAR) BENZOFURAN (GLYCOSIDE) ISOBENZOFURAN NITROFURAN (SUGAR) (THIOSUGAR) FURAN/IT,FT AMIDINE AMIDRAZONE AZO POLYAMINE FORMAZAN/FT ALKYLFLUORIDE ARYLFLUORIDE COND.RING CYCLOPENTANE INDENE BH-LINKED-CC BENZOPYRAN /IT,FT FLAVONOID OR BIOFLAVONOID PYRAN

DYSPROSIUM-SALT Used for a dysprosium salt of an organic acid. * Related * More Specific ENOL Used for compounds of the form R-CR=CR-OH, where R, R = anything, R =C. Also used if the C atoms form part of a ring (other than benzene rings). * Related * More Specific ERBIUM-SALT Used for an erbium salt of an organic acid. * Related * More Specific ESTRANE Any steroid with no C atom at C-10. * Related * More Specific * C/S ETHER These have the structure R-O-R, where R,R = C except for aryl groups when PHENOL-ETHER is used. * Related * More Specific (ACETAL) (CYANATE) (KETAL) (PHENOL-ETHER) STEROID ESTRANE/IT,FT ERBIUM ALCOHOL OLEFIN DYSPROSIUM -

EUROPIUM-COMPLEX Used for compounds where an organic component is coordinated with europium. * Related * More Specific EUROPIUM-SALT Used for a europium salt of an organic acid. * Related * More Specific EUROPIUM EUROPIUM COMPLEX -

* C/S

Derwent Drug File 995 Thesaurus

GADOLINIUM-COMPLEX Used for compounds where an organic component is coordinated with gadolinium. * Related * More Specific GADOLINIUM COMPLEX -

GOLD-COMPLEX Used for compounds where an organic component is coordinated with gold. * Related * More Specific GOLD-SALT Used for a gold salt of an organic acid. * Related * More Specific GUANIDINE Used to include structures of the form RRN-C(=NR)-NRR, where R = anything and may or may not be the same. * Related * More Specific AMINE POLYAMINE GUANIDINE,CYCLIC GOLD GOLD COMPLEX -

GADOLINIUM-SALT Used for a gadolinium salt of an organic acid. * Related * More Specific GADOLINIUM -

GALLIUM-COMPLEX Used for compounds where an organic component is coordinated with gallium. * Related * More Specific GALLIUM-SALT Used for a gallium salt of an organic acid. * Related * More Specific GERMANIN Any 6-membered ring with 1 Ge atom and 5 C atoms. * Related * More Specific GLYCERIDE Mono-, di- or tri-esters of glycerol with saturated and/or unsaturated fatty acids. * Related * More Specific * C/S GLYCOPROTEIN Any protein with a carbohydrate group attached. * Related * More Specific * C/S GLYCOSIDE An acetal or ketal formed between a sugaror polysaccharide and a non-sugar moiety. * Related * More Specific ACETAL FURAN KETAL PYRAN SUGAR POLYSACCHARIDE PROTEIN GLYCOPROTEIN/IT,FT ALCOHOL C-ESTER FATTY-ACID POLYALCOHOL UNSAT.FATTY-ACID PHOSPHOLIPID GLYCERIDE/IT,FT GERMANIUM ORGANOMETALLIC GALLIUM GALLIUM COMPLEX -

GUANIDINE,CYCLIC As for GUANIDINE, but the central carbon must form part of a ring. * Related * More Specific AMINE GUANIDINE POLYAMINE -

HAFNIUM-COMPLEX Used for compounds where an organic component is coordinated with hafnium. * Related * More Specific HAL.FATTY-ACID Any fatty acid (but including acetic acidin this case) substituted in the chain by halogen; includes derivatives such as esters and amides. Another term is used to indicate the halogen, e.g. ALKYLBROMIDE * Related ALKYLBROMIDE ALKYLCHLORIDE ALKYLFLUORIDE ALKYLIODIDE C-ACID FATTY-ACID HAL.FATTY-ACID/IT,FT HAFNIUM COMPLEX -

* More Specific * C/S

HEPTAOXACYCLOTETRATRIACONTANE Any 34-membered ring with 7 O atoms and 27 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

996 APPENDIX B

HEPTAOXACYCLOTETRACOSANE Any 24-membered ring with 7 O atoms and 17 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S HETEROSTEROID Any steroid with one or more ring C atom replaced by a heteroatom. Terms for the resulting heterocyclic and alicyclic rings are also used. * Related * More Specific * C/S STEROID HETEROSTEROID/IT,FT MACROCYCLE -

HEXAOXACYCLOEICOSANE Any 20-membered ring with 6 O atoms and 14 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

HEXAOXACYCLOHENEICOSANE Any 21-membered ring with 6 O atoms, and 15 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

HEXAOXACYCLOOCTADECANE HEXAAZACYCLODOTRIACONTANE Any 32-membered ring with 6 N atoms and 26 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE HEXAOXACYCLOTETRIACONTANE HEXAAZACYCLOOCTADECANE Any 18-membered ring with 6 N atoms and 12 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE HEXAOXACYCLOTRICOSANE HEXAAZACYCLOOCTATRIACONTANE Any 38-membered ring with 6 N atoms and 32 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE HEXAOXAZACYCLOHENEICOSANE HEXAAZACYCLOTETRACOSANE Any 24-membered ring with 6 N atoms and 18 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE Any 21-membered ring with 6 O atoms, 1 N atom and 14 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE Any 23-membered ring with 6 O atoms and 17 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE Any 34-membered ring with 6 O atoms and 28 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE Any 18-membered ring with 6 O atoms and 12 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

HEXAOXACYCLODOCOSANE Any 22-membered ring with 6 O atoms and 16 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

Derwent Drug File 997 Thesaurus

HEXATHIACYCLOOCTADECANE Any 18-membered ring with 6 S atoms and 12 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S HH-LINKED-CC Direct linkage of carbon-to-carbon between any two heterocyclic rings, via a single or double bond. * Related * More Specific * C/S HH-LINKED-CX Direct linkage of carbon-to-heteroatom between any two heterocyclic rings, via a single or double bond. * Related * More Specific * C/S HH-LINKED-XX Direct linkage of heteroatom-to-heteroatom between any two heterocyclic rings, via a single or double bond. * Related * More Specific * C/S NUCLEOSIDE NUCLEOTIDE MACROCYCLE -

HYDRAZINE Used for compounds of the form R-NR-NR-R, where R = C and may or may not be the same. * Related * More Specific AMINE AMIDRAZONE (AZO) (DIAZONIUM) (SEMICARBAZIDE) (SEMICARBAZIDE,CYCLIC) (THIOSEMICARBAZIDE) (THIOSEMICARBAZIDE,CYCLIC) TRIAZENE HYDRAZINE/IT,FT

* C/S HYDRIDE

Used for any metal hydride such as LiAlH4 or NaH. * Related * More Specific * C/S HYDRIDE/IT,FT

HYDROXAMIC-ACID Used for compounds of the type R-C(=N-OR)-OR or R-C(=O)-NOR where R,R,R = anything and may be the same or different. Includes analogs with monovalent N or O bonds to the central C. * Related * More Specific * C/S HYDROXYACID Any compound possessing an alcoholic function attached via carbon atoms in chains and/or rings to a carboxylic acid function. Includes simple derivatives. * Related * More Specific * C/S ALCOHOL C-ACID DEPSIDE ONIC-ACID URONIC-ACID HYDROXYACID/IT,FT (from 1972) C-AMIDE HYDROXYLAMINE IMIDATE THIOHYDROXAMIC-ACID HYDROXAMIC-ACID/IT,FT

HOLMIUM-COMPLEX Used for compounds where an organic component is coordinated with holmium. * Related * More Specific HOMOSTEROID Any ring-enlarged steroid. Terms for the resultant alicyclic rings are also used. * Related * More Specific HYDANTOIN Used for compounds which posess animidazole ring with keto groups at positions 2 and 4, and with groups R and R at position 5, where R and R = anything. * Related * More Specific * C/S IMIDAZOLE IMIDE,CYCLIC UREA,CYCLIC THIOHYDANTOIN HYDANTOIN/IT,FT STEROID HOLMIUM COMPLEX -

HYDROXYLAMINE Used for compounds of the form R-NR-OR, where R, R = C but not acyl. R = anything. * Related * More Specific * C/S IMIDATE These have the form R-C(=NR)-OR, where R,R,R = C. * Related * More Specific HYDROXAMIC-ACID AMINE HYDROXAMIC-ACID OXIME HYDROXYLAMINE/IT,FT

998 APPENDIX B

IMIDAZOLE Including hydrogenated derivatives. * Related * More Specific * C/S IMIDE,CYCLIC Used for situations where the sequence O=C-N(R)-C=O |______| appears, where R = anything. * Related * More Specific LACTAM BARBITURATES HYDANTOIN PHTHALIMIDE BENZIMIDAZOLE HYDANTOIN THIOHYDANTOIN IMIDAZOLE/IT,FT PURINE

IODINE Used for the element itself and for iodine attached to a heterocyclic ring or to any atom other than carbon. * Related * More Specific ALKYLIODIDE ARYLIODIDE

IODINE-COMPLEX Used for compounds where an organic component is coordinated with iodine * Related * More Specific IODINE COMPLEX -

IRIDIUM-COMPLEX Used for compounds where an organic component is coordinated with iridium. * Related * More Specific IRON-COMPLEX Used for compounds where an organic component is coordinated with iron. * Related * More Specific IRON-SALT Used for an iron salt of an organic acid. * Related * More Specific IRON IRON COMPLEX IRIDIUM COMPLEX -

INDAZOLE Including hydrogenated derivatives. * Related * More Specific INDENE Including hydrogenated derivatives. * Related * More Specific COND.RING CYCLOPENTANE FLUORENE COND.RING PYRAZOLE -

INDIUM-COMPLEX Used for compounds where an organic component is coordinated with indium. * Related * More Specific INDIUM-SALT Used for an indium salt of an organic acid. * Related * More Specific INDOLE Including hydrogenated derivatives. * Related * More Specific * C/S INDOLIZINE Including hydrogenated derivatives. * Related * More Specific * C/S COND.RING PIPERIDINE PYRIDINE PYRROLE PYRROLIDINE INDOLIZINE/IT,FT COND.RING PYRROLE CARBAZOLE CARBOLINE INDOLE/IT,FT PYRROLIDINE INDIUM INDIUM COMPLEX -

ISOBENZOFURAN Including hydrogenated derivatives. * Related * More Specific BENZOFURAN COND.RING FURAN -

ISOBENZOPYRAN Including hydrogenated derivatives. * Related * More Specific ISOCYANATE Used for compounds of the type R-N=C=O where R = anything. * Related * More Specific ISOINDOLE Including hydrogenated derivatives. * Related * More Specific * C/S COND.RING PYRROLE PHTHALIMIDE ISOINDOLE/IT,FT PYRROLIDINE MUSTARD-OIL BENZOPYRAN COND.RING PYRAN CANNABINOIDS

Derwent Drug File 999 Thesaurus

ISOQUINOLINE Including hydrogenated derivatives. * Related * More Specific * C/S ISOSTEROID A steroid with unusual configuration at the ring junctions, i.e. with one or more of the following (X = H or a substituent): 8-alpha-X, 9-beta-X, 10-alpha-X, 13-alpha-X, 14-beta-X. The appropriate steroid term for the system is also used. * Related * More Specific * C/S ISOTHIAZOLE Including hydrogenated derivatives. * Related * More Specific ISOXAZOLE Including hydrogenated derivatives. * Related * More Specific * C/S KETAL Used for structures of the form RR-C(OR)-OR, where R = C (may be the same or different) , and R,R = anything. Either OR or OR or both may be part of a ring system. * Related * More Specific * C/S KETENE Used for compounds of the form R-C=C=O, where R = anything. * Related * More Specific KETIMINE This includes compounds of the type RRC=N-R, where R, R = C, and R = anything. * Related * More Specific (AMIDINE) OXIME KETONE OLEFIN ALCOHOL ETHER POLYALCOHOL (GLYCOSIDE) (ORTHO-C-ESTER) THIOKETAL KETAL/IT,FT ISOXAZOLE/IT,FT STEROID ISOSTEROID/IT,FT COND.RING PIPERIDINE PYRIDINE (BENZOQUINOLIZINE) PHENANTHRIDINE ISOQUINOLINE/IT,FT MORPHINAN

KETOACID Any compound possessing a ketone function attached via carbon atoms in chains and/or rings to a carboxylic acid function. Includes simple derivatives. * Related * More Specific * C/S KETONE Ketones have the general formula R-C(=O)-R, where R, R = any C except aryl. * Related * More Specific ARYLKETONE BUTYROPHENONE CHALCONE KETENE KETOACID KETONE,CYCLIC POLYKETONE THIOKETONE C-ACID KETONE (URONIC-ACID) KETOACID/IT,FT [from 1972]

KETONE,CYCLIC As for KETONE, but the group forms part of a ring. * Related * More Specific LACTAM A cyclic amide which has the structure R-NR-CR=O, and |_____| where R, R, R = anything. * Related * More Specific C-AMIDE (IMIDE,CYCLIC) PEPTIDE,CYCLIC THIOBARBITURATES (THIOHYDANTOIN) THIOLACTAM LACTAM/IT,FT KETONE QUINONE

* C/S LACTONE

A cyclic ester of the form R-O-CR=O, where R, R = C. |___| * Related * More Specific * C/S C-ESTER ANHYDRIDE,CYCLIC COUMARIN THIOLACTONE LACTONE/IT,FT

LANTHANUM-COMPLEX Used for compounds where an organic component is coordinated with lanthanum. * Related * More Specific LANTHANUM COMPLEX -

LANTHANUM-SALT Used for a lanthanum salt of an organic acid. * Related * More Specific LANTHANUM -

1000 APPENDIX B

LEAD-COMPLEX Used for compounds where an organic component is coordinated with lead. * Related * More Specific LEAD-SALT Used for a lead salt of an organic acid. * Related * More Specific LIPOPROTEIN Any compound containing a protein and a lipid moiety. * Related * More Specific * C/S PROTEIN LIPOPROTEIN/IT,FT LEAD LEAD COMPLEX -

MAGNESIUM-SALT Used for a magnesium salt of an organic acid. * Related * More Specific MAGNESIUM -

MANGANESE-COMPLEX Used for compounds where an organic component is coordinated with manganese. * Related * More Specific MANGANESE COMPLEX -

MANGANESE-SALT Used for a manganese salt of an organic acid. * Related * More Specific MERCAPTAN Used for compounds R-SH, where R = any C except aryl. * Related * More Specific (THIOACETAL) (THIOKETAL) (THIOPHENOL) (THIOSUGAR) MANGANESE -

LITHIUM-COMPLEX Used for compounds where an organic component is coordinated with lithium. * Related * More Specific LITHIUM-SALT Used for a lithium salt of an organic acid. * Related * More Specific LUTETIUM-SALT Used for a lutetium salt of an organic acid. * Related * More Specific MACROCYCLE Any ring with 9 or more members. Used in association with a specific term for the ring itself. * Related * More Specific * C/S MACROCYCLE/IT,FT LUTETIUM LITHIUM LITHIUM COMPLEX -

MERCURY-COMPLEX Used for compounds where an organic component is coordinated with mercury. * Related * More Specific MERCURY-SALT Used for a mercury salt of an organic acid. * Related * More Specific MERCURY MERCURY COMPLEX -

MOLYBDENUM-COMPLEX Used for compounds where an organic component is coordinated with molybdenum. * Related * More Specific MORPHINAN Including hydrogenated derivatives. * Related BRIDGE-STRUCT. ISOQUINOLINE NAPHTHALENE PHENANTHRENE PIPERIDINE PYRIDINE MORPHINAN/IT,FT MOLYBDENUM COMPLEX -

MAGNESIUM-COMPLEX Used for compounds where an organic component is coordinated with magnesium. * Related * More Specific MAGNESIUM COMPLEX -

* More Specific * C/S

Derwent Drug File 1001 Thesaurus

MORPHOLINE Used for morpholine itself and derivatives thereof. Dehydrogenated analogs are indexed with OXAZINE. * Related * More Specific * C/S MUSTARD-OIL Any isothiocyanate of the form R-N=C=S, where R = anything. * Related * More Specific N-ACID Nitrogen oxyacids. * Related * More Specific * C/S N-ESTER Esters of nitric or nitrous acid which have the form R-O-NO2 or R-O-N=O, where R= anything. * Related * More Specific * C/S N-MUSTARD Used for compounds which have the structure alkylhalide-NR-alkylhalide where R = anything. * Related ALKYLBROMIDE ALKYLCHLORIDE ALKYLFLUORIDE ALKYLIODIDE AMINE SEMI-N-MUSTARD N-MUSTARD/IT,FT N-ESTER/IT,FT N-ACID/IT,FT ISOCYANATE OXAZINE (PHENOXAZINE) MORPHOLINE/IT,FT

NAPHTHALENE Including hydrogenated derivatives. * Related * More Specific BENZENE COND.RING ANTHRACENE ARENE MORPHINAN PHENANTHRENE

NAPHTHYRIDINE Any pyridopyridine (1,5-, 1,6-, 1,7-,1,8-, 2,6- or 2,7-diazanaphthalene) or hydrogenated derivative. * Related * More Specific * C/S COND.RING PIPERIDINE PYRIDINE NAPHTHYRIDINE/IT,FT [from 1974]

NEODYMIUM-COMPLEX Used for compounds where an organic component is coordinated with neodymium. * Related * More Specific NEODYMIUM COMPLEX -

NEODYMIUM-SALT Used for a neodymium salt of an organic acid. * Related * More Specific NEODYMIUM SALT -

NICKEL-COMPLEX Used for compounds where an organic component is coordinated with nickel. * Related * More Specific NICKEL-SALT Used for a nickel salt of an organic acid. * Related * More Specific NITRILE Used for organic cyanides. * Related * More Specific NITRO (CYANATE) (THIOCYANATE) NICKEL NICKEL COMPLEX -

* More Specific * C/S N-OXIDE

These compounds have the formula R-(R)N(R)-O, where R,R,R = C. * Related * More Specific N-OXIDE,CYCLIC As for N-oxide, but the nitrogen atom is part of a ring. * Related * More Specific N-OXIDE N-OXIDE,CYCLIC

These compounds are of the type R-NO2, where R = any C except aryl or furyl. * Related * More Specific NITROARENE NITROFURAN

1002 APPENDIX B

NITROARENE Used for compounds of the type aryl-NO2. * Related * More Specific NITROFURAN Any furan substituted by a nitro group. * Related * More Specific * C/S FURAN NITRO NITROFURAN/IT,FT [from 1969] NITRO/IT,FT AND FURAN/IT,FT [1964-1968] NITRO -

NORSTEROID Any ring-contracted steroid. Terms forthe resultant alicyclic rings are also used. * Related * More Specific NUCLEOSIDE Any heterocyclic system attached via an N atom to a sugar moiety. Appropriate term(s) for the heterocyclic system are also used. * Related * More Specific * C/S NUCLEOTIDE A nucleoside with a phosphate group attached to the sugar moiety. Appropriate term(s) for the heterocyclic system are also used. * Related * More Specific * C/S HH-LINKED-CX AMINOSUGAR NUCLEOSIDE P-ESTER NUCLEOTIDE/IT,FT HH-LINKED-CX AMINOSUGAR (NUCLEOTIDE) NUCLEOSIDE/IT,FT STEROID -

NITROSO Used for the compounds of the form R-N=O, where R = anything. * Related * More Specific -

NONAOXACYCLOHEPTACOSANE Any 27-membered ring with 9 O atoms and 18 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

OCTAAZACYCLODOTRIACONTANE Any 32-membered ring with 8 N atoms and 24 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

NONAOXACYCLOTRIACONTANE Any 30-membered ring with 9 O atoms and 21 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

OCTAAZACYCLOHEXACOSANE Any 26-membered ring with 8 N atoms and 18 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

NONAOXAZACYCLOHEPTACOSANE Any 27-membered ring with 9 O atoms and 18 C atoms. MACROCYCLE always appears in addition. * Related * C/S MACROCYCLE -

* More Specific

OCTAAZACYCLOHEXADECANE Any 16-membered ring with 8 N atoms and 8 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

NONAOXAZACYCLOTRIACONTANE Any 30-membered ring with 9 O atoms, 1 N atom and 20 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

OCTAAZACYCLOTETRACOSANE Any 24-membered ring with 8 N atoms and 16 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

Derwent Drug File 1003 Thesaurus

OCTAOXACYCLODOTRIACONTANE Any 32-membered ring with 8 O atoms and 24 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

OLEFIN Any C=C double bond in a carbon chain, any cycloalkane or any macro cyclic heterocyclic ring. Used when there is only one double bond in the whole compound indexed. * Related * More Specific CHALCONE ENOL KETENE POLYOLEFIN (PORPHYRIN) STILBENE (UNSAT.FATTY-ACID) OLEFIN/IT,FT

OCTAOXACYCLOHEPTACOSANE Any 27-membered ring with 8 O atoms and 19 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE * C/S ONIC-ACID

The oxidation product of an aldose in which the -CHO group is converted to -COOH or of a ketose in which the CH2OH closest to the keto group is converted to -COOH. * Related * More Specific * C/S ONIUM Any organic compound containing a charged heteroatom except for those where a more specific term (see below) exists. * Related * More Specific PHOSPHONIUM QUAT.AMINE SULFONIUM HYDROXYACID POLYALCOHOL SUGAR (URONIC-ACID) ONIC-ACID/IT,FT

OCTAOXACYCLOHEXACOSANE Any 26-membered ring with 8 O atoms and 18 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

OCTAOXACYCLOOCTACOSANE Any 28-membered ring with 8 O atoms and 20 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

ORGANOMETALLIC Any compound with a carbon-metal linkage. * Related * More Specific ORTHO-C-ESTER This is used for compounds containing three O atoms attached to a single C atom, of the form R-C(OR)(OR)-OR, where R = H or C, and R = C. (The R groups may be the same or different). * Related * More Specific * C/S ACETAL KETAL ORTHO-C-ESTER/IT,FT METAL GERMANIN etc.

OCTAOXACYCLOTETRACOSANE Any 24-membered ring with 8 O atoms and 16 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

OCTAOXACYCLOTETRATRIACONTANE Any 34-membered ring with 8 O atoms and 26 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

OSMIUM-COMPLEX Used for compounds where an organic component is coordinated with osmium. * Related * More Specific OSMIUM COMPLEX -

OCTAOXACYCLOHEPTACOSANE Any 27-membered ring with 8 O atoms, 1 N atom and 18 O atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE OXACYCLODOCOSANE Any 22-membered ring with 1 O atom and 21 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

1004 APPENDIX B

OXACYCLODODECANE Any 12-membered ring with 1 O atom and 11 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

OXACYCLOHEXATRIACONTANE Any 36-membered ring with 1 O atom and 35 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

OXACYCLODOTETRACONTANE Any 42-membered ring with 1 O atom and 41 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

OXACYCLOOCTACOSANE Any 28-membered ring with 1 O atom and 27 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

OXACYCLODOTRIACONTANE Any 32-membered ring with 1 O atom and 31 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

OXACYCLOOCTADECANE Any 18-membered ring with 1 O atom and 17 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

OXACYCLOEICOSANE Any 20-membered ring with 1 O atom and 19 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

OXACYCLOOCTATRIACONTANE Any 38-membered ring with 1 O atom and 37 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

OXACYCLOHEPTADECANE Any 17-membered ring with 1 O atom and 16 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

OXACYCLOPENTACOSANE Any 25-membered ring with 1 O atom and 24 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

OXACYCLOHEXACOSANE Any 26-membered ring with 1 O atom and 25 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

OXACYCLOPENTADECANE Any 15-membered ring with 1 O atom and 14 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

OXACYCLOHEXADECANE Any 16-membered ring with 1 O atom and 15 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

OXACYCLOPENTATRIACONTANE Any 35-membered ring with 1 O atom and 34 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

Derwent Drug File 1005 Thesaurus

OXACYCLOTETRACOSANE Any 24-membered ring with 1 O atom and 23 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

OXADIAZACYCLODODECANE Any 12-membered ring with 1 O atom, 2 N atoms and 9 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

OXACYCLOTETRADECANE Any 14-membered ring with 1 O atom and 13 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

OXADIAZACYCLOHEPTADECANE Any 17-membered ring with 1 O atom, 2 N atoms and 14 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

OXACYCLOTETRATETRACONTANE Any 44-membered ring with 1 O atom and 43 C atoms. MACROCYCLE always appear in addition. * Related * More Specific * C/S MACROCYCLE -

OXADIAZACYCLOHEXADECANE Any 16-membered ring with 1 O atom, 2 N atoms and 13 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

OXACYCLOTETRATRIACONTANE Any 34-membered ring with 1 O atom and 33 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

OXADIAZACYCLONONADECANE Any 19-membered ring with 1 O atom, 2 N atoms and 16 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

OXACYCLOTRIACONTANE Any 30-membered ring with 1 O atom and 29 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

OXADIAZACYCLOOCTADECANE Any 18-membered ring with 1 O atom, 2 N atoms and 15 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

OXACYCLOTRIDECANE Any 13-membered ring with 1 O atom and 12 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

OXADIAZACYCLOPENTADECANE Any 15-membered ring with 1 O atom, 2 N atoms and 12 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

OXACYCLOUNDECANE Any 11-membered ring with 1 O atom and 10 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

OXADIAZACYCLOTETRACOSANE Any 24-membered ring with 1 O atom, 2 N atoms and 21 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

1006 APPENDIX B

OXADIAZACYCLOTETRADECANE Any 14-membered ring with 1 O atom, 2 N atoms and 11 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

OXADIAZOCINE Any 8-membered ring with 1 O atom, 2 N atoms and 5 C atoms. * Related * More Specific * C/S OXADIAZOLE Any 5-membered ring with 1 O atom, 2 N atoms and 2 C atoms. * Related * More Specific * C/S OXADIAZONINE Any 9-membered ring with 1 O atom, 2 N atoms and 6 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE OXADIAZONINE OXADIAZOLE/IT,FT OXADIAZOCINE/FT

OXADIAZACYCLOTRICOSANE Any 23-membered ring with 1 O atom, 2 N atoms and 20 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

OXADIAZACYCLOTRIDECANE Any 13-membered ring with 1 O atom, 2 N atoms and 10 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

OXADIAZAPHOSPHORINE Any 6-membered ring with 1 O atom, 2 N atoms, 1 P atom and 2 C atoms. * Related * More Specific * C/S OXADIAZECINE Any 10-membered ring with 1 O atom, 2 N atoms and 7 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S OXADIAZEPINE Any 7-membered ring with 1 O atom, 2 N atoms and 4 C atoms. * Related * More Specific * C/S OXADIAZINE Any 6-membered ring with 1 O atom, 2 N atoms and 3 C atoms. * Related * More Specific * C/S OXADIAZINE/IT,FT OXADIAZEPINE/FT MACROCYCLE OXADIAZECINE OZADIAZAPHOSPHORINE

OXAMERCURETANE Any 4-membered ring with 1 O atom, 1 Hg atom and 2 C atoms. * Related MERCURY

ORGANOMETALLIC * More Specific * C/S OXAMERCURETANE

OXAPENTAAZACYCLOHEXACOSANE Any 26-membered ring with 1 O atom, 5 N atoms and 20 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

OXAPENTAAZACYCLOOCTACOSANE Any 28-membered ring with 1 O atom, 5 N atoms and 22 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

Derwent Drug File 1007 Thesaurus

OXAPENTAAZACYCLOOCTADECANE Any 18-membered ring with 1 O atom, 5 N atoms and 12 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

OXATHIAZEPINE Any 7-membered ring with 1 O atom, 1 N atom and 5 C atoms. * Related * More Specific OXATHIAZINE Any 6-membered ring with 1 O atom, 1 S atom, 1 N atom and 3 C atoms. * Related * More Specific -

OXAPHOSPHOLE Any 5-membered ring with 1 O atom, 1 P atom and 3 C atoms. * Related * More Specific * C/S OXAPHOSPHOLE/FT

OXATHIAZONINE Any 9-membered ring with 1 O atom, 1 S atom, 1 N atom and 6 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S OXATHIECIN Any 10-membered ring with 1 O atom, 1 S atom and 8 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S OXATHIEPIN Any 7-membered ring with 1 O atom, 1 S atom and 5 C atoms. * Related * More Specific * C/S OXATHIEPIN/FT MACROCYCLE OXATHIECIN MACROCYCLE OXATHIAZONINE/FT

OXAPHOSPHORIN Any 6-membered ring with 1 O atom, 1 P atom and 4 C atoms. * Related * More Specific OXASELENOLE Any 5-membered ring with 1 O atom, 1 Se atom and 3 C atoms. * Related * More Specific * C/S OXATHIANE Any 6-membered ring with 1 O atom, 1 S atom and 4 C atoms. * Related * More Specific SELENIUM OXASELENOLE -

OXATHIAZABORONINE Any 9-membered ring with 1 O atom, 1 S atom, 1 N atom, 1 B atom and 5 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S OXATHIAZECINE Any 10-membered ring with 1 O atom, 1 S atom, 1 N atom and 7 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE OXATHIAZECINE OXATRIAZACYCLONONADECANE Any 19-membered ring with 1 O atom, 3 N atoms and 15 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE MACROCYCLE BORON OXATRIAZACYCLOHEPTACOSANE Any 27-membered ring with 1 O atom, 3 N atoms and 23 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE OXATHIOLE Any 5-membered ring with 1 O atom, 1 S atom and 3 C atoms. * Related * More Specific -

1008 APPENDIX B

OXATRIAZACYCLOTRICOSANE Any 23-membered ring with 1 O atom, 3 N atoms and 19 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S OXATRIAZOLE Any 5-membered ring with 1 O atom, 3 N atoms and 1 C atom. * Related * More Specific * C/S OXATRIAZOLE/FT MACROCYCLE -

OXAZACYCLOPENTACOSANE Any 25-membered ring with 1 O atom, 1 N atom and 23 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

OXAZACYCLOPENTADECANE Any 15-membered ring with 1 O atom, 1 N atom and 13 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

OXATRITHIADIAZACYCLONONADECANE Any 19-membered ring with 1 O atom, 3 S atoms, 2 N atoms and 13 C atoms.MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE OXAZACYCLOTETRACOSANE Any 24-membered ring with 1 O atom, 1 N atom and 22 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S OXAZACYCLOEICOSANE Any 20-membered ring with 1 O atom, 1 N atom and 18 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE OXAZACYCLOTETRADECANE Any 14-membered ring with 1 O atom, 1 N atom and 12 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S OXAZACYCLOHEXADECANE Any 16-membered ring with 1 O atom, 1 N atom and 14 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE OXAZACYCLOTRICOSANE Any 23-membered ring with 1 O atom, 1 N atom and 21 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S OXAZACYCLONONADECANE Any 19-membered ring with 1 O atom, 1 N atom and 17 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE OXAZADISILACYCLOHEXANE Any 6-membered ring with 1 O atom, 1 N atom, 2 Si atoms and 2 C atoms. * Related * More Specific SILICON MACROCYCLE MACROCYCLE MACROCYCLE -

OXAZACYCLOOCTACOSANE Any 28-membered ring with 1 O atom, 1 N atom and 26 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

OXAZAPHOSPHEPINE Any 7-membered ring with 1 O atom, 1 N atom, 1 P atom and 4 C atoms. * Related * More Specific -

Derwent Drug File 1009 Thesaurus

OXAZAPHOSPHORINE Any 6-membered ring with 1 O atom, 1 N atom, 1 P atom and 3 C atoms. * Related * More Specific OXAZECINE Any 10-membered ring with 1 O atom, 1 N atom and 8 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S OXAZEPINE Any 7-membered ring with 1 O atom, 1 N atom and 5 C atoms. * Related * More Specific * C/S OXAZINE Any 6-membered ring with 1 O atom, 1 N atom and 4 C atoms, except morpholine. * Related * More Specific * C/S OXAZIRIDINE Any 3-membered ring with 1 O atom, 1 N atom and 1 C atom. * Related * More Specific * C/S OXAZOCINE Any 8-membered ring with 1 O atom, 1 N atom and 6 C atoms. * Related * More Specific * C/S OXAZOLE Including hydrogenated derivatives. * Related * More Specific * C/S OXAZOLE/IT,FT OXAZOCINE/IT,FT [from 1971] MORPHOLINE PHENOXAZINE OXAZINE/IT,FT OXAZEPINE/IT,FT [from 1972] MACROCYCLE OXAZECINE -

OXAZONINE Any 9-membered ring with 1 O atom, 1 N atom and 7 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S OXECIN Any 10-membered ring with 1 O atom and 9 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S OXEPIN Any 7-membered ring with 1 O atom and 6 C atoms. * Related * More Specific * C/S OXETANE Any 4-membered ring with 1 O atom and 3 C atoms. * Related * More Specific OXIME Used for compounds of the form RRC=N-OR, where R,R,R = H or C. * Related * More Specific OXIRANE Any 3-membered ring with 1 O atom and 2 C atoms (i.e. epoxides). * Related * More Specific * C/S OXOCIN Any 8 membered ring with 1 O atom and 7 C atoms. * Related * More Specific P-ACID Inorganic oxides and oxyacids of phosphorus * Related * More Specific * C/S PHOSPHONIC-ACID PS-ACID P-ACID/IT,FT EPOXIDE/IT,FT ALDIMINE HYDROXYLAMINE KETIMINE OXEPIN/IT,FT MACROCYCLE MACROCYCLE OXAZONINE

1010 APPENDIX B

P-AMIDE This group of compounds has the structure RRRP=NR, where R = anything and may be the same or different. Includes analogs with a single P-N bond. * Related * More Specific P-ESTER An ester of any acid of phosphorus. * Related * More Specific * C/S NUCLEOTIDE (PHOSPHOLIPID) P-ESTER/IT,FT (TRIAZATRIPHOSPHORINE)

PENTAOXACYCLODOCOSANE Any 22-membered ring with 5 O atoms and 17 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

PENTAOXACYCLOOCTADECANE Any 18-membered ring with 5 O atoms and 13 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

PALLADIUM-COMPLEX Used for compounds where an organic component is coordinated with palladium. * Related * More Specific PALLADIUM COMPLEX -

PENTAOXACYCLOPENTADECANE Any 15-membered ring with 5 O atoms and 10 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

PALLADIUM-SALT Used for a palladium salt of an organic acid. * Related * More Specific PENICILLINS Antibiotics with a thiazole beta-lactam ring, and any derivative thereof. * Related * More Specific * C/S AMINOACID AZETIDINE COND.RING LACTAM THIAZOLE PENICILLIN/IT,FT PALLADIUM -

PENTAOXADIAZACYCLOHENEICOSANE Any 21-membered ring with 5 O atoms, 2 N atoms and 14 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

PENTAOXAZACYCLOOCTADECANE Any 18-membered ring with 5 O atoms, 1 N atom and 12 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S PEPTIDE A compound formed by the linking of two or more amino acids by CO-NH groups up to a molecular weight of about 12,000. * Related * More Specific * C/S PEPTIDE,CYCLIC As for peptide or depsipeptide, but part of all of the peptide chain forming a ring. * Related * More Specific LACTAM PEPTIDE POLYMER AMINOACID C-AMIDE PROTEIN PEPTIDE/IT,FT POLYMER MACROCYCLE -

PENTAAZACYCLOHEXADECANE Any 16-membered ring with 5 N atoms and 11 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

PENTAAZACYCLOPENTADECANE Any 15-membered ring with 5 N atoms and 10 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

DEPSIPEPTIDE PEPTIDE,CYCLIC PROTEIN

Derwent Drug File 1011 Thesaurus

PEROXIDE Used for compounds of the form R-O-O-R, where R, R = anything. Includes peracids R-CO-OOH. * Related * More Specific * C/S PEROXIDE/IT,FT

PHENOXAZINE Including hydrogenated derivatives. * Related * More Specific * C/S PHOSPHINE COND.RING MORPHOLINE OXAZINE PHENOXAZINE/IT,FT

PHENANTHRENE Including hydrogenated derivatives. * Related * More Specific BENZENE COND.RING (ARENE) MORPHINAN MORPHINAN

Used for compounds of the form R-PR-R, where R,R,R = H or C. * Related * More Specific PHOSPHOLE Any 5-membered ring with 1 P atom and 4 C atoms. * Related * More Specific PHOSPHOLIPID Esters of fatty acids formed with alcohol components containing a phosphate group. * Related * More Specific * C/S C-ESTER FATTY-ACID GLYCERIDE P-ESTER PHOSPHOLIPID/IT,FT PHOSPHONIUM

PHENANTHRIDINE Including hydrogenated derivatives. * Related * More Specific * C/S PHENAZINE Including hydrogenated derivatives. * Related * More Specific * C/S PHENOL Used in cases where a phenol ring is substituted with a group R, such that R = anything except an oxygen function. * Related * More Specific * C/S PHENOL-ETHER Used for compounds of the type aryl-OR, where R= C. * Related * More Specific * C/S PHENOTHIAZINE Including hydrogenated derivatives. * Related * More Specific * C/S COND.RING THIAZINE PHENOTHIAZINE/IT,FT ETHER ARYLSULFIDE THYRO-C-ACID PHENOL-ETHER/IT,FT ALCOHOL POLYPHENOL SALICYLIC-ACID THIOPHENOL PHENOL/IT,FT COND.RING PIPERAZINE PYRAZINE QUINOXALINE PHENAZINE/IT,FT COND.RING ISOQUINOLINE PIPERIDINE PYRIDINE QUINOLINE PHENANTHRIDINE/IT,FT [from 1969]

PHOSPHONIC-ACID These compounds have the form RRP(=O)-OR where Ror R= H or C,and R = H or OR. * Related * More Specific PHOSPHONIUM Used for compounds of the form R3-P-R, where R = C, and may be the same or different. * Related * More Specific PHTHALAZINE Including hydrogenated derivatives. * Related * More Specific * C/S PHTHALIMIDE Used for phthalimide itself, substituted derivatives and hydrogenated analogs. * Related * More Specific COND.RING IMIDE,CYCLIC PYRROLE ISOINDOLE COND.RING PYRIDAZINE PHTHALAZINE/IT,FT ONIUM PHOSPHINE P-ACID -

1012 APPENDIX B

PIPERAZINE Used for piperazine itself and derivatives thereof. * Related * More Specific * C/S PIPERIDINE Used for piperidine itself and derivatives thereof, excluding dehydrogenated analogs. * Related * More Specific PYRIDINE (ACRIDINE) (AZAPHENOTHIAZINE) (BENZOQUINOLIZINE) (CARBOLINE) (INDOLIZINE) (ISOQUINOLINE) MORPHINAN (NAPHTHYRIDINE) (PHENANTHRIDINE) (QUINOLINE) (QUINOLIZINE) QUINUCLIDINE TROPANE PIPERIDINE/IT,FT (PHENAZINE) (PTERIDINE) (QUINOXALINE) PIPERAZINE/IT,FT

POLYALCOHOL Any compound with two or more non-phenolic hydroxyl groups, unless a more specific term exists. * Related * More Specific ALCOHOL (ACETAL) AMINOCYCLITOL CYCLITOL (GLYCERIDE) (KETAL) ONIC-ACID SUGAR (THIOSUGAR) URONIC-ACID POLYALCOHOL/IT,FT

* C/S POLYALDEHYDE

Any compound containing two or more aldehyde groups. * Related * More Specific POLYAMINE Any compound containing two or more amino groups, or simple derivatives thereof. * Related * More Specific AMINE (AMIDINE) (AMIDRAZONE) (AMINOCYCLITOL) (AMINOSUGAR) (FORMAZAN) (GUANIDINE) (GUANIDINE,CYCLIC) ALDEHYDE -

* C/S

PLANT-SUBSTANCE Any compound of plant origin for which the structure is unknown and for which no more specific term (e.g. ALKALOID, FLAVONOID) exits. * Related * More Specific * C/S PLANT-SUBSTANCE/IT,FT

POLYKETONE Any compound containing two or more ketone groups. * Related * More Specific * C/S POLYMER Used for all polymeric compounds for which no specific term exists. * Related * More Specific POLYOLEFIN Any compound containing two or more olefinic bonds as defined under OLEFIN. * Related * More Specific * C/S OLEFIN CAROTENOID (PORPHYRIN) RETINOID (UNSAT.FATTY-ACID) POLYOLEFIN/IT,FT (PEPTIDE) (PEPTIDE,CYCLIC) (PROTEIN) KETONE QUINONE POLYKETONE/IT,FT

PLATINUM-COMPLEX Used for compounds where an organic component is coordinated with platinum. * Related * More Specific PLATINUM-SALT Used for a platinum salt of an organic acid. * Related * More Specific PLATINUM PLATINUM COMPLEX -

PLUTONIUM-SALT Used for a plutonium salt of an organic acid. * Related * More Specific POLY-C-ACID Any compound containing two or more carboxyl groups; includes simple derivatives such as esters or amides. * Related * More Specific * C/S C-ACID POLY-C-ACID/IT,FT PLUTONIUM -

POLYPHENOL Any compound with two or more -OH or -OR groups attached to benzene rings. * Related * More Specific * C/S PHENOL THYRO-C-ACID POLYPHENOL/IT,FT

Derwent Drug File 1013 Thesaurus

POLYSACCHARIDE Used for compounds comprising 7 or more connected monosaccharide units. * Related * More Specific * C/S PORPHYRIN Including hydrogenated derivatives. * Related BRIDGE-STRUCT. MACROCYCLE OLEFIN POLYOLEFIN PYRROLE TETRAAZACYCLOHEXADECANE PORPHYRIN/IT,FT AMINOSUGAR SUGAR THIOSUGAR GLYCOPROTEIN POLYSACCHARIDE/IT,FT

PS-ACID Used for any phosphorus acid analog for which one or more oxygen atom is replaced by sulfur. The appropriate term(s) for the parent acid is also applied. * Related * More Specific * C/S PTERIDINE Including hydrogenated derivatives. * Related * More Specific * C/S PURINE Including hydrogenated derivatives. * Related * More Specific * C/S PYRAN Any 6-membered ring with 1 O atom and 5 C atoms. * Related * More Specific (AMINOSUGAR) BENZOPYRAN COUMARIN FLAVONOID (GLYCOSIDE) ISOBENZOPYRAN (SUGAR) (THIOSUGAR) XANTHENE PYRAN/IT,FT AMIDINE,CYCLIC COND.RING IMIDAZOLE PYRIMIDINE PURINE/IT,FT AMIDINE,CYCLIC COND.RING PIPERAZINE PYRAZINE PYRIMIDINE PTERIDINE/IT,FT P-ACID PS-ACID/IT,FT

* More Specific * C/S

POTASSIUM-COMPLEX Used for compounds where an organic component is coordinated with potassium. * Related * More Specific POTASSIUM COMPLEX -

POTASSIUM-SALT Used for a potassium salt of an organic acid. * Related * More Specific POTASSIUM -

PRASEODYMIUM-COMPLEX Used for compounds where an organic component is coordinated with praseodymium. * Related * More Specific PRASEODYMIUM COMPLEX -

* C/S PYRAZINE

PRASEODYMIUM-SALT Used for a praseodymium salt of an organic acid. * Related * More Specific PREGNANE Any steroid with both angular Me-groups and a two carbon chain at C17. * Related * More Specific PROTEIN As for peptide, but for compounds of molecular weight greater than about 12,000. * Related * More Specific * C/S AMINOACID PEPTIDE POLYMER GLYCOPROTEIN LIPOPROTEIN PROTEIN/IT,FT (PEPTIDE) STEROID 17-BETA-ALKYLSTEROID PRASEODYMIUM -

Including di- and tetra-hydro analogs. * Related * More Specific * C/S PYRAZOLE Including hydrogenated derivatives. * Related * More Specific * C/S PYRIDAZINE Including hydrogenated derivatives. * Related * More Specific * C/S CINNOLINE PHTHALAZINE PYRIDAZINE/IT,FT INDAZOLE PYRAZOLE/IT,FT PHENAZINE PIPERAZINE PTERIDINE QUINOXALINE PYRAZINE/IT,FT

1014 APPENDIX B

PYRIDINE Including di- and tetra-hydro derivatives. * Related * More Specific ACRIDINE AZAPHENOTHIAZINE BENZOQUINOLIZINE CARBOLINE ISOQUINOLINE (MORPHINAN) NAPHTHYRIDINE PHENANTHRIDINE PIPERIDINE QUINOLINE QUINOLIZINE QUINUCLIDINE (TROPANE) PYRIDINE/IT,FT

QUINAZOLINE Including hydrogenated derivatives. * Related * More Specific * C/S QUINOLINE Including hydrogenated derivatives. * Related * More Specific COND.RING PIPERIDINE PYRIDINE ACRIDINE (BENZOQUINOLIZINE) PHENANTHRIDINE QUINOLINE/IT,FT COND.RING PYRIMIDINE QUINAZOLINE/IT,FT

* C/S PYRIMIDINE

Including hydrogenated derivatives. * Related * More Specific * C/S PYRROLE Including any dihydro derivative. * Related * More Specific CARBAZOLE CARBOLINE CORRINOID INDOLE INDOLIZINE ISOINDOLE PHTHALIMIDE PORPHYRIN PYRROLIDINE PYRROLIZINE (TROPANE) PYRROLE/IT,FT BARBITURATES PTERIDINE PURINE QUINAZOLINE THIOBARBITURATES PYRIMIDINE/IT,FT

* C/S QUINOLIZINE

Including hydrogenated derivatives. * Related * More Specific * C/S QUINONE Used for benzoquinone, the 1,2 -dioxo analog, and any derivative; includes analogs with =X in place of =O. * Related * More Specific * C/S QUINOXALINE Including hydrogenated derivatives. * Related * More Specific * C/S QUINUCLIDINE Including dehydrogenated derivatives. * Related * More Specific * C/S RETINOID Used for retinol and close analogs with similar biological activity. * Related * More Specific ALCOHOL CAROTENOID CYCLOHEXANE POLYOLEFIN BRIDGE-STRUCT. PIPERIDINE PYRIDINE QUINUCLIDINE/IT,FT [from 1972] COND.RING PIPERAZINE PYRAZINE PHENAZINE QUINOXALINE/IT,FT KETONE,CYCLIC POLYKETONE ANTHRACYCLINES QUINONE/IT,FT COND.RING PIPERIDINE PYRIDINE BENZOQUINOLIZINE QUINOLIZINE/IT,FT

* C/S PYRROLIDINE

Used for pyrrolidine itself and derivatives thereof. * Related * More Specific PYRROLE (CARBAZOLE) (CARBOLINE) (INDOLE) (INDOLIZINE) (ISOINDOLE) (PYRROLIZINE) TROPANE

PYRROLIZINE Including hydrogenated derivatives. * Related * More Specific * C/S QUAT.AMINE Any organic ammonium salt of the form +RRNRR, where R = C, which may be the same or different. * Related * More Specific AMINE ONIUM (BETAINE) COND.RING PYRROLE PYRROLIDINE PYRROLIZINE/IT,FT [from 1972]

Derwent Drug File 1015 Thesaurus

RHENIUM-COMPLEX Used for compounds where an organic component is coordinated with rhenium. * Related * More Specific RHENIUM COMPLEX -

SAMARIUM-SALT Used for a samarium salt of an organic acid. * Related * More Specific SAMARIUM -

SCANDIUM-COMPLEX RHODIUM-COMPLEX Used for compounds where an organic component is coordinated with rhodium. * Related * More Specific RHODIUM-SALT Used for a rhodium salt of an organic acid. * Related * More Specific RHODIUM RHODIUM COMPLEX SECOSTEROID Any steroid in which one ring of the nucleus has been broken. Appropriate terms are added for the residual alicyclic system. * Related * More Specific * C/S SELENADIAZOLE Any 5-membered ring with 1 Se atom, 2 N atoms and 2 C atoms. * Related * More Specific SELENAZINE Any 6-membered ring with 1 Se atom, 1 N atom and 4 C atoms. * Related * More Specific * C/S SELENAZOCINE Any 8-membered ring with 1 Se atom, 1 N atom and 6 C atoms. * Related S-ESTER Used for any ester of a sulfur acid. * Related * More Specific * C/S SALICYLIC-ACID Used for salicylic acid itself and for derivatives of the acid and/or phenolic functions. Not used when the benzene ring is further substituted. * Related * More Specific * C/S ARYL-C-ACID PHENOL SALICYLIC-ACID/IT,FT SULTONE S-ESTER/IT,FT * More Specific * C/S SELENAZOLE Any 5-membered ring with 1 Se atom, 1 N atom and 3 C atoms. * Related * More Specific * C/S SELENEPIN Any 7-membered ring with 1 Se atom and 6 C atoms. * Related * More Specific SELENIUM SELENIUM SELENAZOLE/FT SELENIUM SELENAZOCINE SELENIUM SELENAZINE SELENIUM SECOSTEROID/IT,FT Used for compounds where an organic component is coordinated with scandium. * Related * More Specific SCANDIUM COMPLEX -

RUBIDIUM-COMPLEX Used for compounds where an organic component is coordinated with rubidium. * Related * More Specific RUBIDIUM COMPLEX -

RUTHENIUM-COMPLEX Used for compounds where an organic component is coordinated with rhodium. * Related * More Specific S-ACID Inorganic oxides and oxyacids of sulfur. * Related * More Specific * C/S SULFONIC-ACID S-ACID/IT,FT RUTHENIUM COMPLEX -

1016 APPENDIX B

SELENIN Any 6-membered ring with 1 Se atom and 5 C atoms. * Related * More Specific * C/S SELENIUM SELENIN

SILVER-SALT Used for a silver salt of an organic acid. * Related * More Specific SILVER -

SODIUM-COMPLEX Used for compounds where an organic component is coordinated with sodium. * Related * More Specific SODIUM-SALT Used for a sodium salt of an organic acid. * Related * More Specific SPIRO Two rings connected by one shared atom. * Related * More Specific STEROID Used for any compound with a gonane system not covered by a More Specific steroidal term. * Related * More Specific ANDROSTANE BILE-ACID CHOLESTANE CYCLOSTEROID ESTRANE HETEROSTEROID HOMOSTEROID ISOSTEROID NORSTEROID PREGNANE SECOSTEROID (TRITERPENE) 17-BETA-ALKYLSTEROID STEROID/IT,FT SODIUM SODIUM COMPLEX -

SEMI-N-MUSTARD These compounds have the formula R-NR-CH2-CH2-X, where R,R = H or C, and X = halogen. * Related * More Specific * C/S SEMICARBAZIDE Used for compounds of the form R-NR-C(=O)-NR-NRR, where the R groups maybe the same or different, and where R = anything. Includes analogous structures with a single C-O bond. * Related * More Specific HYDRAZINE UREA SEMICARBAZIDE,CYCLIC THIOSEMICARBAZIDE THIOSEMICARBAZIDE,CYCLIC ALKYLBROMIDE ALKYLCHLORIDE ALKYLFLUORIDE ALKYLIODIDE AMINE (N-MUSTARD) -

SEMICARBAZIDE,CYCLIC As for SEMICARBAZIDE, but the central C atom must form part of a ring. * Related * More Specific * C/S HYDRAZINE SEMICARBAZIDE UREA,CYCLIC SEMICARBAZIDE/IT,FT AND XIX/PN [from 1966]

* C/S STILBENE

SILACYCLOHEXANE Any 6-membered ring with 1 Si atom and 5 C atoms. * Related * More Specific * C/S SILICON SILACYCLOHEXANE

This has the structure Ar-CR=CR-Ar, where the R groups may be the same or different, and where R = anything. * Related * More Specific * C/S BENZENE OLEFIN STILBENE/IT,FT

SILACYCLOPENTANE Any 5-membered ring with 1 Si atom and 4 C atoms. * Related * More Specific * C/S SILVER-COMPLEX Used for compounds where an organic component is coordinated with silver. * Related * More Specific SILVER COMPLEX SILICON SILACYCLOPENTANE

STRONTIUM-COMPLEX Used for compounds where an organic component is coordinated with strontium. * Related * More Specific STRONTIUM COMPLEX -

Derwent Drug File 1017 Thesaurus

SUGAR Used for mono- to hexa-saccharides. * Related * More Specific FURAN POLYALCOHOL PYRAN AMINOSUGAR GLYCOSIDE ONIC-ACID POLYSACCHARIDE URONIC-ACID SUGAR/IT,FT

SULFONIC-ACID Used for compounds of the form R-SO2-OR or R-SO-OR, where R= C, R= H or C. Includes thio-analogs with S in place of O. * Related * More Specific SULFONIUM Compounds in this group have the structure +R-SR-R, where the R groups may be the same or different, and where R, R,R = C. * Related * More Specific ONIUM SULFIDE S-ACID (BILE-ACID)

* C/S SULFENAMIDE

Used for compounds of the form R-S-NRR, where R = C, R = anything. (The R groups may be the same or different). * Related * More Specific * C/S SULFIDE Used for compounds of the form R-S-R, where R, R = any C except aryl. * Related * More Specific ARYLSULFIDE DISULFIDE (SULFONE) SULFONIUM (SULFOXIDE) (THIOACETAL) (THIOCYANATE) (THIOKETAL) SULFUR (THIOHYDROXAMIC-ACID) SULPHENAMIDE/FT

SULFONYL-HALIDE Used for compounds of the form R-SO2-X or R-SO-X, where R = C, X = halogen. * Related * More Specific SULFOXIDE Used for compounds of the form R-SO-R, where R, R = C. * Related * More Specific SULFIDE (SULFONE) SULFOXIDE,CYCLIC BROMINE CHLORIDE FLUORINE IODINE -

SULFINAMIDE Used for compounds of the form R-SO-NRR, where R = C and R, R = anything. * Related * More Specific SULFONAMIDE Used for compounds of the form R-SO2-NRR, where R = C and R, R = anything. * Related * More Specific SULFONE Used for compounds of the form R-SO2-R, where R, R = C. * Related * More Specific SULFONE,CYCLIC As for sulfone, but the S atom must form part of a ring. * Related * More Specific SULFONE SULFIDE SULFOXIDE SULFONE,CYCLIC SULFINAMIDE SULTAM (SULFOXIMIDE) (SULFONAMIDE)

SULFOXIDE,CYCLIC As for SULFOXIDE, but the S atom must form part of a ring. * Related * More Specific SULFOXIMIDE Used for structures of the type RRS(=O)=N-R, where R, R = C, and R = anything. * Related * More Specific SULTAM Used for a cyclic sulfonamide of the form R-SO-NR-R or |____| R-SO2-NR-R, where R, R= C, and R= anything. |_____| * Related * More Specific SULTONE Used for any cyclic S-ester R-SO-O-R or R-SO2-O-R, where R, |______| |_______| R= C. * Related * More Specific S-ESTER SULFONAMIDE SULFONAMIDE SULFOXIDE -

1018 APPENDIX B

TECHNETIUM-COMPLEX Used for compounds where an organic component is coordinated with technetium. * Related * More Specific TELLURAPYRAN Any 6-membered ring with 1 Te atom, and 5 C atoms. * Related * More Specific * C/S TELLURAZINE Any 6-membered ring with 1 Te atom, 1 N atom and 4 C atoms. * Related * More Specific * C/S TELLURIUM TELLURAZINE/FT TELLURIUM TELLURAPYRAN/FT TECHNETIUM COMPLEX -

TETRAAZACYCLODODECANE Any 12-membered ring with 4 N atoms and 8 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

TETRAAZACYCLOEICOSANE Any 20-membered ring with 4 N atoms and 16 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

TETRAAZACYCLOHEXADECANE Any 16-membered ring with 4 N atoms and 12 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE PORPHYRIN -

TELLURIUM-COMPLEX Used for compounds where an organic component is coordinated with tellurium. * Related * More Specific TELLURIUM COMPLEX -

TETRAAZACYCLOPENTADECANE Any 15-membered ring with 4 N atoms and 11 C atoms. MACROCYCLE always appears in addition. * Related MACROCYCLE CORRINOID * More Specific * C/S

TERBIUM-COMPLEX Used for compounds where an organic component is coordinated with terbium. * Related * More Specific * C/S TERBIUM-SALT Used for a terbium salt of an organic acid. * Related * More Specific TERPENE Any natural product or analog thereof which is built up from isoprene units. * Related * More Specific * C/S CAROTENOID TRITERPENE TERPENE/IT,FT TERBIUM TERBIUM COMPLEX

TETRAAZACYCLOTETRADECANE Any 14-membered ring with 4 N atoms and 10 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

TETRAAZACYCLOTRIDECANE Any 13-membered ring with 4 N atoms and 9 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

TETRAAZATETRAPHOSPHOCINE Any 8-membered ring with 4 N atoms and 4 P atoms. * Related * More Specific * C/S TETRAAZATETRAPHOSPHOCINE

Derwent Drug File 1019 Thesaurus

TETRACYCLINES Used for tetracycline itself and for close analogs and derivatives. * Related * More Specific * C/S ANTHRACENE ARENE COND.RING NAPHTHALENE (ANTHRACYCLINES) TETRACYCLINE/IT,FT N.B. This will also retrieve anthracyclines.

TETRAOXACYCLOHEXATRIACONTANE Any 36-membered ring with 4 O atoms and 32 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

TETRAOXACYCLONONADECANE TETRAOXACYCLODOCOSANE Any 22-membered ring with 4 O atoms and 18 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE TETRAOXACYCLOOCTACOSANE TETRAOXACYCLODODECANE Any 12-membered ring with 4 O atoms and 8 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE TETRAOXACYCLOOCTADECANE TETRAOXACYCLOEICOSANE Any 20-membered ring with 4 O atoms and 16 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE TETRAOXACYCLOTETRADECANE TETRAOXACYCLOHENEICOSANE Any 21-membered ring with 4 O atoms and 17 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE TETRAOXACYCLOTETRATRIACONTANE TETRAOXACYCLOHENTRIACONTANE Any 31-membered ring with 4 O atoms and 27 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE TETRAOXADIAZACYCLOOCTADECANE TETRAOXACYCLOHEXADECANE Any 16-membered ring with 4 O atoms and 12 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE Any 18-membered ring with 4 O atoms, 2 N atoms and 12 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE Any 34-membered ring with 4 O atoms and 30 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE Any 14-membered ring with 4 O atoms and 10 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE Any 18-membered ring with 4 O atoms and 14 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE Any 28-membered ring with 4 O atoms and 24 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE Any 19-membered ring with 4 O atoms and 15 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

1020 APPENDIX B

TETRAOXADIAZECINE Any 10-membered ring with 4 O atoms, 2 N atoms and 4 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S TETRAOXANE Any 6-membered ring with 4 O atoms and 2 C atoms. * Related * More Specific MACROCYCLE MACROCYCLE TETRAOXADIAZECINE

TETRATHIAZOCINE Any 8-membered ring with 4 S atoms, 1 N atom and 3 C atoms. * Related * More Specific * C/S TETRAZECINE Any 10-membered ring with 4 N atoms and 6 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S TETRAZINE Any 6-membered ring with 4 N atoms and 2 C atoms. * Related * More Specific * C/S TETRAZOCINE Any 8-membered ring with 4 N atoms and 4 C atoms. * Related * More Specific TETRAZOLE Any 5-membered ring with 4 N atoms and 1 C atom. * Related * More Specific * C/S TETRAZOLE/IT,FT TETRAZINE/IT,FT MACROCYCLE TETRAZECINE TETRATHIAZOCINE

TETRAOXASILACYCLOUNDECANE Any 11-membered ring with 4 O atoms, 1 Si atom and 6 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE SILICON -

TETRAOXATETRASILACYCLOOCTANE Any 8-membered ring with 4 O atoms and 4 Si atoms. * Related * More Specific * C/S SILICON -

TETRATHIACYCLODODECANE Any 12-membered ring with 4 S atoms and 8 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

THIACYCLOHENEICOSANE TETRATHIAHEPTAAZACYCLOTRIACONTANE Any 30-membered ring with 4 S atoms, 7 N atoms and 19 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE THALLIUM-SALT TETRATHIATETRAAZACYCLODOCOSANE Any 22-membered ring with 4 S atoms, 4 N atoms and 14 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE Used for a thallium salt of an organic acid. * Related * More Specific THALLIUM Any 21-membered ring with 1 S atom and 20 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

THIADIAZACYCLONONADECANE Any 19-membered ring with 1 S atom, 2 N atoms and 16 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

Derwent Drug File 1021 Thesaurus

THIADIAZEPINE Any 7-membered ring with 1 S atom, 2 N atoms and 4 C atoms. * Related * More Specific THIADIAZINE Any 6-membered ring with 1 S atom, 2 N atoms and 3 C atoms. * Related * More Specific * C/S THIADIAZOCINE Any 8-membered ring with 1 S atom, 2 N atoms and 5 C atoms. * Related * More Specific * C/S THIADIAZOLE Any 5-membered ring with 1 S atom, 2 N atoms and 2 C atoms. * Related * More Specific * C/S THIAPYRAN Any 6-membered ring with 1 S atom and 5 C atoms. * Related * More Specific * C/S THIASELENOLE Any 5-membered ring with 1 S atom, 1 Se atom and 3 C atoms. * Related * More Specific * C/S SELENIUM THIASELENOLE THIAXANTHENE (THIOSUGAR) THIAPYRAN/IT,FT THIADIAZOLE/IT,FT THIADIAZINE/IT,FT -

THIATRIAZACYCLODODECANE Any 12-membered ring with 1 S atom, 3 N atoms and 8 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

THIATRIAZACYCLOEICOSANE Any 20-membered ring with 1 S atom, 3 N atoms and 16 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

THIATRIAZACYCLOTRIDECANE Any 13-membered ring with 1 S atom, 3 N atoms and 9 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

THIATRIAZADIPHOSPHORANE Any 6-membered ring with 1 S atom, 3 N atoms and 2 P atoms. * Related * More Specific * C/S THIATRIAZINE Any 6-membered ring with 1 S atom, 3 N atoms and 2 C atoms. * Related * More Specific * C/S THIAXANTHENE Including hydrogenated derivatives. * Related * More Specific * C/S COND.RING THIAPYRAN THIAXANTHENE/IT,FT THIATRIAZADIPHOSPHORANE/FT

THIATETRAAZACYCLOHEXADECANE Any 16-membered ring with 1 S atom, 4 N atoms and 11 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

THIAZAGERMOLANE Any 5-membered ring with 1 S atom, 1 N atom, 1 Ge atom and 2 C atoms. * Related * More Specific * C/S GERMANIUM THIAZAGERMOLANE/FT

1022 APPENDIX B

THIAZASILACYCLOPENTANE Any 5-membered ring with 1 S atom, 1 N atom, 1 Si atom and 2 C atoms. * Related * More Specific * C/S THIAZEPINE Any 7-membered ring with 1 S atom, 1 N atom and 5 C atoms. * Related * More Specific * C/S THIAZINE Any 6-membered ring with 1 S atom, 1 N atom and 4 C atoms. * Related * More Specific * C/S THIAZOCINE Any 8-membered ring with 1 S atom, 1 N atom and 6 C atoms. * Related * More Specific * C/S THIAZOLE Including hydrogenated derivatives; see also ISOTHIAZOLE. * Related * More Specific * C/S PENICILLINS THIAZOLE/IT,FT N.B. This will also retrieve isothiazoles. THIAZOCINE/FT AZAPHENOTHIAZINE CEPHALOSPORINS PHENOTHIAZINE THIAZINE/IT,FT THIAZEPINE/IT,FT SILICON THIAZASILACYCLOPENTANE/FT

THIOACETAL As for ACETAL, but with one or both O atoms replaced by S. * Related * More Specific * C/S THIOALDEHYDE Used for compounds of the form R-CH=S, where R = C. * Related * More Specific ALDEHYDE ACETAL MERCAPTAN SULFIDE -

THIOBARBITURATES Used for thiobarbituric acid and any derivative thereof. * Related * More Specific * C/S BARBITURATES LACTAM PYRIMIDINE THIOUREA,CYCLIC THIOBARBITURATE/IT,FT

THIOCARBAMATE Used for compounds of the form (i)R-NR-C(=S)OR or (ii) R-NR-C(=O)SR, where R,R,R = anything. Includes analogs with a single C-S or C-O bond. * Related * More Specific CARBAMATE DITHIOCARBAMATE THIOCARBAMATE,CYCLIC

THIOCARBAMATE,CYCLIC As for THIOCARBAMATE or DITHIOCARBAMATE, but the central atom must be part of aring. * Related * More Specific THIOCIN Any 8-membered ring with 1 S atom and 7 C atoms. * Related * More Specific * C/S THIOCYANATE Used for groups of the form R-S-nitrile, where R = anything. * Related * More Specific CYANATE NITRILE SULFIDE THIOCIN CARBAMATE DITHIOCARBAMATE THIOCARBAMATE -

THIEPIN Any 7-membered ring with 1 S atom and 6 C atoms. * Related * More Specific * C/S THIIRANE Any 3-membered ring with 1 S atom and 2 C atoms. * Related * More Specific THIEPIN/IT,FT

Derwent Drug File 1023 Thesaurus

THIOHYDANTOIN As for HYDANTOIN, but with an S atom in place of either or both of the O atoms. * Related HYDANTOIN IMIDAZOLE LACTAM THIOLACTAM THIOUREA,CYCLIC UREA,CYCLIC -

THIOPHENE Any 5-membered ring with 1 S atom and 4 C atoms. * Related * More Specific * C/S THIOPHENOL Used for compounds of the type aryl-SH. * Related * More Specific * C/S MERCAPTAN PHENOL THIOPHENOL/IT,FT (THIOSUGAR) THIOPHENE/IT,FT

* More Specific

THIOHYDROXAMIC-ACID Used for compounds of the form R-C(=N-OR)-SR or R-C(=S)-NR-OR, where R,R,R = anything. Includes analogs where the O and S atoms are interchanged and/or where the N,O or S bond to the central C is monovalent. * Related * More Specific THIOIMIDATE As for IMIDATE, but with an S atom replacing the O atom. * Related * More Specific THIOKETAL As for KETAL, but with one or both O atoms replaced by S. * Related * More Specific * C/S THIOKETONE Used for compounds of the form R-CS-R, where R, R = C. * Related * More Specific THIOLACTAM A cyclic thio-amide of the form |___________| where R, R= C, R-NR-C(=S)-R R = anything. * Related * More Specific THIOLACTONE A cyclic thio-ester of the form |_________| or R-S-C(=O)-R R-X-C(=S)-R |_________| where X = O or S, and R, R = C. * Related * More Specific C-ESTER LACTONE C-AMIDE LACTAM (THIOHYDANTOIN) KETONE KETAL MERCAPTAN SULFIDE THIOKETAL/FT IMIDATE THIOHYDROXAMIC-ACID C-AMIDE CS-ACID HYDROXAMIC-ACID SULFENAMIDE THIOIMIDATE -

THIOSEMICARBAZIDE As for SEMICARBAZIDE, but with the O atom being replaced by S. Includes analogous structures with a single C-S bond. * Related * More Specific HYDRAZINE SEMICARBAZIDE THIOUREA THIOSEMICARBAZIDE,CYCLIC

THIOSEMICARBAZIDE,CYCLIC As for THIOSEMICARBAZIDE, but the central C atom must form part of a ring. * Related HYDRAZINE SEMICARBAZIDE SEMICARBAZIDE,CYCLIC THIOSEMICARBAZIDE THIOUREA,CYCLIC THIOSEMICARBAZIDE/IT,FT AND XIX/PN

* More Specific * C/S THIOSUGAR

Any mono- to hexa-saccharide moiety with one or more O atoms replaced by S atoms. GLYCOSIDE is used in addition where appropriate. * Related * More Specific * C/S THIOUREA Applied to structures of the form R-NR-C(=S)-NR-R, where the R = anything and may be the same or different. * Related * More Specific * C/S UREA THIOSEMICARBAZIDE THIOUREA,CYCLIC THIOUREA/IT,FT FURAN MERCAPTAN POLYALCOHOL PYRAN THIAPYRAN THIOPHENE (POLYSACCHARIDE) THIOSUGAR/FT

THIOUREA,CYCLIC As for THIOUREA, but the central C atom must form part of a ring. * Related * More Specific * C/S THIOUREA UREA,CYCLIC THIOBARBITURATES (THIOHYDANTOIN) THIOSEMICARBAZIDE,CYCLIC THIOUREA/IT,FT AND XIX/PN

1024 APPENDIX B

THIURAM Used for compounds of the form R-NR-C(=S)-S-S-C(=S)-NR-R, where the R = anything, and may be the same or different. * Related * More Specific DISULFIDE DITHIOCARBAMATE -

TRIAZATRIPHOSPHORINE Any 6-membered ring with 3 N atoms and 3 P atoms. * Related * More Specific TRIAZENE P-AMIDE -

THORIUM-COMPLEX Used for compounds where an organic component is coordinated with thorium. * Related * More Specific THORIUM COMPLEX -

Used for compounds of the form R-NR-N=N-R, where R,R,R = anything. * Related * More Specific TRIAZEPINE AZO HYDRAZINE -

THULIUM-COMPLEX Used for compounds where an organic component is coordinated with thulium. * Related * More Specific THULIUM-SALT Used for a thulium salt of an organic acid. * Related * More Specific THYRO-C-ACID Analogs of p-HO-Ph-O-Ph-COOH-p orp-HO-Ph-O-Ph-X-COOH-p, where X = CH2 or C2H4. This structure almost invariably has iodine substituent(s) on one or both benzene rings. * Related * More Specific * C/S TIN-COMPLEX Used for compounds where an organic component is coordinated with tin. * Related * More Specific TIN COMPLEX ARYL-C-ACID ARYLIODIDE C-ACID PHENOL-ETHER POLYPHENOL THYRO-C-ACID/IT,FT THULIUM THULIUM COMPLEX -

Any 7-membered ring with 3 N atoms and 4 C atoms. * Related * More Specific TRIAZINE Any 6-membered ring with 3 N atoms and 3 C atoms. * Related * More Specific * C/S TRIAZOCINE Any 8-membered ring with 3 N atoms and 5 C atoms. * Related * More Specific TRIAZOLE Any 5-membered ring with 3 N atoms and 2 C atoms. * Related * More Specific * C/S TRIAZONINE Any 9-membered ring with 3 N atoms and 6 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE TRIAZONINE TRIAZOLE/IT,FT TRIAZINE/IT,FT -

TITANIUM-COMPLEX Used for compounds where an organic component is coordinated with titanium. * Related * More Specific TITANIUM-SALT Used for a titanium salt of an organic acid. * Related * More Specific TITANIUM TITANIUM COMPLEX -

TRIOXACYCLODODECANE Any 12-membered ring with 3 O atoms and 9 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

Derwent Drug File 1025 Thesaurus

TRIOXACYCLOEICOSANE Any 20-membered ring with 3 O atoms and 17 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

TRIOXACYCLOPENTADECANE Any 15-membered ring with 3 O atoms and 12 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

TRIOXACYCLOHENEICOSANE Any 21-membered ring with 3 O atoms and 18 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S TRIOXACYCLOHENTRIACONTANE Any 31-membered ring with 3 O atoms and 28 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE MACROCYCLE -

TRIOXACYCLOTETRACOSANE Any 24-membered ring with 3 O atoms and 21 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

TRIOXACYCLOTETRADECANE Any 14-membered ring with 3 O atoms and 11 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

TRIOXACYCLOHEXADECANE Any 16-membered ring with 3 O atoms and 13 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

TRIOXACYCLOTRIACONTANE Any 30-membered ring with 3 O atoms and 27 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

TRIOXACYCLONONADECANE Any 19-membered ring with 3 O atoms and 16 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

TRIOXACYCLOTRICOSANE Any 23-membered ring with 3 O atoms and 20 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

TRIOXACYCLOOCTADECANE Any 18-membered ring with 3 O atoms and 15 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

TRIOXADIAZACYCLOPENTADECANE Any 15-membered ring with 3 O atoms, 2 N atoms and 10 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

TRIOXACYCLOPENTACOSANE Any 25-membered ring with 3 O atoms and 22 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

TRIOXADISILACYCLOOCTANE Any 8-membered ring with 3 O atoms, 2 Si atoms and 3 C atoms. * Related * More Specific SILICON -

1026 APPENDIX B

TRIOXANE Any 6-membered ring with 3 O atoms and 3 C atoms. * Related * More Specific -

TUNGSTEN-COMPLEX Used for compounds where an organic component is coordinated with tungsten. * Related * More Specific TUNGSTEN COMPLEX -

TRIOXAZACYCLOTRIDECANE Any 13-membered ring with 3 O atoms, 1 N atom and 9 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S TRIOXEPIN Any 7-membered ring with 3 O atoms and 4 C atoms. * Related * More Specific TRIOXONIN Any 9-membered ring with 3 O atoms and 6 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S TRITERPENE A natural C-30 terpene with a steroid or D-homosteroid nucleus. The appropriate keyword for the steroid nucleus is used in addition. * Related * More Specific * C/S TRITHIAZEPINE Any 7-membered ring with 3 S atoms, 1 N atom and 3 C atoms. * Related * More Specific * C/S TROPANE Including dehydrogenated and other derivatives. * Related BRIDGE-STRUCT. CYCLOHEPTANE PIPERIDINE PYRIDINE PYRROLE PYRROLIDINE TROPANE/IT,FT TRITHIAZEPINE HOMOSTEROID STEROID TRITERPENE/IT,FT [from 1972] TERPENE UNSAT.FATTY-ACID As for FATTY-ACID except that one or more double and/or triple bonds are to be found in the chain. The type of multiple bond is also specified. * Related * More Specific * C/S ACETYLENE FATTY-ACID OLEFIN POLYOLEFIN (GLYCERIDE) UNSAT.FATTY-ACID/IT,FT MACROCYCLE TRIOXONIN UNDECAOXACYCLOTRITRIACONTANE Any 33-membered ring with 11 O atoms and 22 C atoms. MACROCYLE always appears in addition. * Related * More Specific * C/S MACROCYCLE MACROCYCLE TUNGSTEN-SALT Used for a tungsten salt of an organic acid. * Related * More Specific TUNGSTEN -

UNDECAAZACYCLOPENTATRIACONTANE Any 35-membered ring with 11 N atoms and 24 C atoms. MACROCYCLE always appears in addition. * Related * More Specific * C/S MACROCYCLE -

URANIUM-COMPLEX Used for compounds where an organic component is coordinated with uranium. * Related * More Specific URANIUM-SALT Used for a uranium salt of an organic acid. * Related * More Specific URANIUM URANIUM COMPLEX -

* More Specific * C/S

Derwent Drug File 1027 Thesaurus

UREA Used for compounds of the form RRN-C(=O)-NRR, where R = anything but N, and may be the same or different. * Related * More Specific * C/S UREA,CYCLIC As for UREA, but the central C atom must form part of a ring. * Related * More Specific UREA BARBITURATES HYDANTOIN SEMICARBAZIDE,CYCLIC (THIOHYDANTOIN) UREA/IT,FT + XIX/PN SEMICARBAZIDE THIOUREA UREA,CYCLIC UREA/IT,FT

YTTERBIUM-COMPLEX Used for compounds where an organic component is coordinated with ytterbium. * Related * More Specific YTTERBIUM COMPLEX -

YTTERBIUM-SALT Used for a ytterbium salt of an organic acid. * Related * More Specific YTTERBIUM -

YTTRIUM-COMPLEX Used for compounds where an organic component is coordinated with yttrium. * Related * More Specific YTTRIUM-SALT Used for a yttrium salt of an organic acid. * Related * More Specific ZINC-COMPLEX Used for compounds where an organic component is coordinated with zinc. * Related * More Specific ZINC-SALT Used for a zinc salt of an organic acid. * Related * More Specific ZINC ZINC COMPLEX YTTRIUM YTTRIUM COMPLEX -

* C/S URONIC-ACID

The oxidation product of an aldose in which the CH2-OH is converted to COOH or of a ketose in which the CH2-OH furthest from the keto group is similarly oxidized. * Related * More Specific * C/S ALDEHYDE HYDROXYACID KETOACID ONIC-ACID POLYALCOHOL SUGAR URONIC-ACID/IT,FT

VANADIUM-COMPLEX Used for compounds where an organic component is coordinated with vanadium. * Related * More Specific XANTHENE Including hydrogenated derivatives. * Related * More Specific * C/S BENZOPYRAN COND.RING PYRAN XANTHENE/IT,FT VANADIUM COMPLEX -

ZIRCONIUM-COMPLEX Used for compounds where an organic component is coordinated with zirconium. * Related * More Specific ZIRCONIUM COMPLEX -

XANTHOGENATE Applied to compounds of the form R-O-C(=S)-SR, where R, R = anything. * Related * More Specific * C/S YLIDE All compounds with a charge separation, other than those covered by more specific terms. * Related * More Specific * C/S YLIDE/IT,FT XANTHOGENATE/IT,FT

17-BETA-ALKYLSTEROID Any steroid with both angular methyl groups and with a carbon chain attached at the C17-beta position, excluding bile acids, cholestanes and pregnanes. * Related * More Specific * C/S STEROID BILE-ACID CHOLESTANE PREGNANE 17-BETA-ALKYLSTEROID/FT

1028 APPENDIX B

Derwent Drug File 1029 Thesaurus

APPENDIX C
CLASSIFIED HIGHER TERMS
INTRODUCTION This Appendix provides lists of UDB higher terms grouped into a series of classifications. It should indicate to searchers the higher terms available in the various fields of interest. All higher terms used in UDB indexing are included. However, there seemed little point in including both the singular and plural forms of higher terms used to represent biological activities, so only the plural form has been included in these cases. Obviously the singular form will be appropriate in the same classification. Many higher terms, particularly those used for chemical substructures, fall into more than one category. In such cases, the higher terms have been included in all appropriate groups. The classifications are arranged into four main groups, and a number of sub-groups, as follows: 1. BIOLOGICAL ACTIVITIES 1.1 1.2 1.3 1.4 1.5 1.6 1.7 1.8 1.9 1.10 1.11 1.12 1.13 1.14 1.15 1.16 1.17 Pesticides and plant hormones Anesthetics and drugs relieving fever, inflammation and pain Antimicrobials and chemotherapeutics Hormones and antagonists Enzymes and inhibitors Drugs acting on the gastrointestinal system Drugs acting on the blood and cardiovascular system Drugs acting on the immune system Drugs acting on the muscular system Anticancer drugs and carcinogens Drugs acting on the nervous system Psychotropic agents Drugs acting on the respiratory system Drugs acting on the skin Vitamins and antagonists Miscellaneous activity terms New activity terms

4. CHEMISTRY 4.1 4.2 4.3 4.4 4.5 4.6 4.7 4.8 4.9 4.10 4.11 4.12 4.13 4.14 4.15 4.16 4.17 4.18 4.19 4.20 4.21 4.22 4.23 4.24 Alicycles (in groups of increasing ring size) Aminoacids and peptides Arenes and other benzenoids Functions connected to a benzene ring Carboxylic acids and derivatives Charged functions Carbohydrates Carbamates, Ureas, etc. Heterocycles (in groups of increasing ring size, subdivided by heteroatom) Halogen-containing functions Aldehydes and ketones Complexes Salts Monovalent N-containing functions Polyvalent N-containing functions Monovalent O-containing functions P-containing functions Functions within rings Ring-linked terms Monovalent S-containing functions Polyvalent S-containing functions Steroids Unsaturated functions Miscellaneous

2. ORGANISMS 2.1 2.2 2.3 2.4 Animals Microorganisms Plants Viruses

3. OTHER BIOLOGICAL/PHYSICAL AREAS 3.1 3.2 3.3 3.4 3.5 3.6 3.7 3.8 3.9 3.10 Diseases Galenics and biopharmaceutics Metabolism Organs and cells Physical and analytical terms General medical terms Nutrition Physiological processes Physical processes Miscellaneous

1030 APPENDIX C 1. BIOLOGICAL ACTIVITIES 1.1 Pesticides and plant hormones ACARICIDES ALGICIDES ATTRACTANTS FUNGICIDES HERBICIDES INSECT-HORMONES INSECTICIDES MOLLUSCICIDES PLANT-GROWTH-FACTORS REPELLENT RODENTICIDES 1.2 Anesthetics and drugs relieving fever, inflammation and pain ANALGESICS ANTIGOUTS ANTIINFLAMMATORIES ANTIPYRETICS ANTIRHEUMATICS CASPASE-1-INHIBITORS CASPASE-3-INHIBITORS CASPASE-9-INHIBITORS CASPASE-INHIBITORS COLLAGENASE-= INHIBITORS CORTICOSTEROIDS CYCLOOXYGENASE-1-= INHIBITORS CYCLOOXYGENASE-2-= INHIBITORS CYCLOOXYGENASEINHIBITORS GELATINASE-A-INHIBITORS GELATINASE-B-INHIBITORS GELATINASE-INHIBITORS GEN.ANESTHETICS HISTAMINERGICS INTERLEUKIN-= CONVERTING-= ENZYME-INHIBITORS LOCAL-ANESTHETICS MATRIX-= METALLOPROTEINASE-= INHIBITORS MORPHINE-ANTAGONISTS NARCOTICS OPIOIDS OPIOID-ANTAGONIST PROSTAGLANDIN-= ANTAGONISTS RUBEFACIENTS STROMELYSIN-1-= INHIBITORS STROMELYSIN-2-= INHIBITORS 1.3 STROMELYSIN-INHIBITORS TACE-INHIBITORS XANTHINE-OXIDASE-= INHIBITORS Antimicrobials and chemotherapeutics ALGICIDES AMEBICIDES ANTHELMINTICS ANTIBIOTICS ANTILEPROTICS ANTISEPTICS COCCIDIOSTATICS FUNGICIDES HIV-INTEGRASE-= INHIBITORS HIV-PROTEASE-INHIBITORS INOSINE-= MONOPHOSPHATE-= DEHYDROGENASE-= INHIBITORS INTERFERON-INDUCERS PHYTONCIDES PROTOZOACIDES RAS-INHIBITORS TUBERCULOSTATICS TYROSINE-KINASE-= INHIBITORS VIRUCIDES 1.4 Hormones and antagonists ACE-INHIBITORS ACTH-AGONISTS ACTH-ANTAGONISTS ALDOSTERONE-= ANTAGONISTS ANABOLICS ANDROGENANTAGONISTS ANDROGENS ANGIOTENSIN-AGONISTS ANGIOTENSIN-2-= ANTAGONISTS ANGIOTENSIN-= ANTAGONISTS ANTIDIABETICS ANTITHYROIDS AROMATASE-INHIBITORS BRADYKININ-= ANTAGONISTS CONTRACEPTIVES CORTICOLIBERIN-= AGONISTS CORTICOLIBERIN-= ANTAGONISTS CORTICOSTEROID-= ANTAGONISTS CORTICOSTEROIDS CYCLOOXYGENASE-1-= INHIBITORS CYCLOOXYGENASE-2-= INHIBITORS CYCLOOXYGENASE-= INHIBITORS ESTROGEN-ANTAGONISTS ESTROGENS FOLLIBERIN-AGONISTS FOLLIBERIN-ANTAGONISTS GASTRIN-ANTAGONISTS GASTROINTEST.HORMONES GLUCAGON-AGONISTS GLUCAGON-= ANTAGONISTS GLUCOSIDASE-INHIBITORS GONADOLIBERIN-= AGONISTS GONADOLIBERIN-= ANTAGONISTS GONADOTROPIN-= ANTAGONISTS GONADOTROPINS GROWTH-FACTOR INSULIN-AGONISTS INSULIN-ANTAGONISTS INTERMEDIN-AGONISTS INTERMEDIN-= ANTAGONISTS KININS LEUKOTRIENE-= ANTAGONISTS LIPOXYGENASE-= INHIBITORS LULIBERIN-AGONISTS LULIBERIN-ANTAGONISTS MELANOLIBERIN-= AGONISTS MELANOSTATIN-= AGONISTS MELATONIN-AGONISTS MELATONIN-= ANTAGONISTS MINERALOCORTICOIDS OXYTOCIN-AGONISTS OXYTOCIN-ANTAGONISTS PAF-ANTAGONISTS PANCREAS-HORMONES PANCREOZYMIN-= AGONISTS PANCREOZYMIN-= ANTAGONISTS PITUITARY-HORMONES PROGESTOGENS PROLACTIN-AGONISTS PROLACTIN-ANTAGONISTS PROLACTOLIBERIN-= AGONISTS PROSTACYCLIN-AGONISTS PROSTAGLANDIN-= ANTAGONISTS PROSTAGLANDINS RELEASING-FACTOR-= INHIBITORS RELEASING-FACTORS RENIN-INHIBITORS SELECTIVE-ESTROGEN-= RECEPTOR-= MODULATORS SOMATOLIBERIN-= AGONISTS SOMATOSTATIN-= AGONISTS SOMATOTROPIN-= AGONISTS SOMATOTROPIN-= ANTAGONISTS SUBSTANCE-P-AGONISTS SUBSTANCE-P-= ANTAGONISTS THROMBOXANE-= AGONISTS THROMBOXANE-= ANTAGONISTS THYMUS-HORMONES THYROID-HORMONES THYROLIBERIN-AGONISTS THYROMIMETICS THYROTROPIN-AGONISTS VASOPRESSIN-AGONISTS VASOPRESSIN-= ANTAGONISTS 1.5 Enzymes and inhibitors ACAT-INHIBITORS ACE-INHIBITORS ACETYL-COA-= CARBOXYLASE-= INHIBITORS ADENOSINE-= DEAMINASE-INHIBITORS ADENOSINE-KINASE-= INHIBITORS ADENYLATE-CYCLASE-= INHIBITORS AGE-INHIBITOR AKT-INHIBITOR ALCOHOL-= DEHYDROGENASE-= INHIBITORS ALDOSE-REDUCTASE-= INHIBITORS ALKALINE-= PHOSPHATASE-= INHIBITORS ALKYLGUANINE-DNA-= TRANSFERASE-= INHIBITORS ALPHA-GLUCOSIDASE-= INHIBITORS

Derwent Drug File 1031 Thesaurus ANTICHOLINESTERASES ARGINASE-INHIBITORS AROMATASE-INHIBITORS BACE-INHIBITOR BETA-GLUCOSIDASE-= INHIBITORS BETA-LACTAMASE-= INHIBITORS CARBONIC-ANHYDRASE-= INHIBITORS CASPASE-1-INHIBITORS CASPASE-3-INHIBITORS CASPASE-9-INHIBITORS CASPASE-INHIBITORS CATHEPSIN-INHIBITORS CHOLINESTERASE-= REACTIVATORS CHYMOTRYPSIN-= INHIBITORS CLOTTING-FACTOR-XA-= INHIBITORS COENZYME COLLAGENASE-= INHIBITORS COMT-INHIBITOR CYCLIN-DEPENDENT-= KINASE-INHIBITORS CYCLOOXYGENASE-1-= INHIBITORS CYCLOOXYGENASE-2-= INHIBITORS CYCLOOXYGENASE-= INHIBITORS DNA-DIRECTED-DNA-= POLYMERASE-= INHIBITORS DNA-DIRECTED-RNA-= POLYMERASE-= INHIBITORS DOPA-DECARBOXYLASE-= INHIBITORS ENDOTHELIN-= CONVERTING-= ENZYME-INHIBITORS ENZYMES ERK-INHIBITOR FARNESYL-PROTEIN-= TRANSFERASE-= INHIBITORS GARFT-INHIBITORS GELATINASE-A-INHIBITORS GELATINASE-B-INHIBITORS GELATINASE-INHIBITORS GERANYLGERANYL-= PROTEIN-= TRANSFERASE-= INHIBITORS GLUCOSIDASE-INHIBITORS GLUCOSYL-= TRANSFERASE-= INHIBITORS GLUTAMATE-= DECARBOXYLASE-= INHIBITORS GLUTATHIONE-= TRANSFERASE-= INHIBITORS GLYCOSIDASE-INHIBITORS GUANINE-DEAMINASE-= INHIBITORS GUANYLATE-CYCLASE-= INHIBITORS HISTIDINE-= DECARBOXYLASE-= INHIBITORS HISTONE-DEACETYLASE-= INHIBITORS HIV-INTEGRASE-= INHIBITORS HIV-PROTEASE-INHIBITORS H-K-ATPASE-INHIBITORS HMG-COA-REDUCTASE-= INHIBITORS HMG-COA-SYNTHASE-= INHIBITORS INOSINE-= MONOPHOSPHATE-= DEHYDROGENASE-= INHIBITORS INTERLEUKIN-= CONVERTING-= ENZYME-INHIBITORS LIPOXYGENASE-= INHIBITORS MAO-INHIBITORS MAP-KINASE-INHIBITORS MATRIX-= METALLOPROTEINASE-= INHIBITORS MYOSIN-LIGHT-CHAIN-= KINASE-INHIBITORS NA-CA-ATPASE-INHIBITOR NA-H-EXCHANGE-= INHIBITORS NA-K-ATPASE-INHIBITORS NEURAMINIDASE-= INHIBITORS NEUTRAL-= ENDOPEPTIDASE-= INHIBITORS NEUTROPHIL-ELASTASE-= INHIBITORS NF-KAPPA-B-INHIBITORS NITRIC-OXIDE-= SYNTHASE-INDUCERS NITRIC-OXIDE-= SYNTHASE-INHIBITORS ORNITHINE-= DECARBOXYLASE-= INHIBITORS PANREATIC-ELASTASE-= INHIBITORS PARP-INHIBITORS PEPTIDE-HYDROLASE-= INHIBITORS P-GLYCOPROTEIN-= INHIBITORS PHOSPHODIESTERASE-= INHIBITORS PHOSPHOLIPASE-= INHIBITORS PROTEASOME-INHIBITOR PROTEIN-KINASE-C-= INHIBITORS PROTEIN-= PHOSPHORYLASE-= INHIBITORS RAS-INHIBITORS RENIN-INHIBITORS REVERSE-= TRANSCRIPTASE-= INHIBITORS RHO-KINASE-INHIBITORS SQUALENE-SYNTHASE-= INHIBITORS STROMELYSIN-1-= INHIBITORS STROMELYSIN-2-= INHIBITORS STROMELYSIN-INHIBITORS TACE-INHIBITORS TELOMERASE-INHIBITORS THROMBIN-INHIBITORS THYMIDINE-KINASE-= INHIBITORS THYMIDYLATE-= SYNTHASE-INHIBITORS TOPOISOMERASE-II-= INHIBITORS TOPOISOMERASE-I-= INHIBITORS TOPOISOMERASE-= INHIBITORS TYROSINASE-INHIBITORS TYROSINE-KINASE-= INHIBITORS UREASE-INHIBITOR XANTHINE-OXIDASE-= INHIBITORS 1.6 Drugs acting on the gastrointestinal system ANTACIDS ANTIDIARRHEICS ANTIEMETICS ANTIFLATULENTS ANTIHISTAMINES ANTIHISTAMINES-H2 ANTIULCERS CHOLAGOGUES DIGESTANTS EMETIC GASTRIC-SECRETION-= INHIBITORS HEPATOTROPICS LAXATIVES 1.7 Drugs acting on the blood and cardiovascular system ACE-INHIBITORS ADENOSINE-AGONISTS ADENOSINE-= ANTAGONISTS ANGIOTENSIN-2-= ANTAGONISTS ANGIOTENSIN-= ANTAGONISTS ANTIAGGREGANTS ANTIANEMICS ANTIARRHYTHMICS ANTIARTERIOSCLEROTICS ANTICOAGULANTS ANTIFIBRINOLYTICS ANTISICKLINGS BIOFLAVONOIDS BLOOD-CLOTTING-= FACTOR BLOOD-SUBSTITUTES C5-ANTAGONISTS CALCIUM-AGONISTS CALCIUM-ANTAGONISTS CARDIANTS CARDIOGLYCOSIDES CLOTTING-FACTOR-XA-= INHIBITORS ENDOTHELIN-= ANTAGONISTS ENDOTHELIN-= CONVERTING-= ENZYME-INHIBITORS FIBRINOGEN-= ANTAGONISTS GPIIB-IIIA-ANTAGONISTS HEMOSTATICS HEPARINOIDS HMG-COA-REDUCTASE-= INHIBITORS HYPERTENSIVES HYPOTENSIVES NA-H-EXCHANGE-= INHIBITORS NEUTRAL-= ENDOPEPTIDASE-= INHIBITORS NITRIC-OXIDE-= ANTAGONISTS NITRIC-OXIDE-= SYNTHASE-INDUCERS NITRIC-OXIDE-= SYNTHASE-INHIBITORS POTASSIUM-= ANTAGONISTS RENIN-INHIBITORS RHO-KINASE-INHIBITORS

1032 APPENDIX C SYMPATHOLYTICS SYMPATHOLYTICS-ALPHA SYMPATHOLYTICS-BETA THROMBIN-INHIBITORS THROMBOLYTICS VASOCONSTRICTORS VASODILATORS VASOTROPICS 1.8 Drugs acting on the immune system ADJUVANTS ANTIANAPHYLACTICS ANTIHISTAMINES ANTIHISTAMINES-H1 DESENSITIZERS IMMUNOMODULATOR IMMUNOSTIMULANTS IMMUNOSUPPRESSIVES INTERFERON-INDUCERS VACCINES 1.9 Drugs acting on the muscular system CURARE-ANTAGONISTS NEUROMUSC.BLOCKER-= ANTAGONISTS NEUROMUSC.BLOCKERS RELAXANTS 1.10 Anticancer drugs and carcinogens ADENOSINE-= DEAMINASE-INHIBITORS AKT-INHIBITOR ALKYLGUANINE-DNA-= TRANSFERASE-= INHIBITORS ANGIOGENESIS-= INHIBITORS ANTICARCINOGEN ANTIMUTAGEN APOPTOSIS-INDUCERS CARCINOGEN COCARCINOGEN CYTOSTATICS EPIDERMAL-GROWTH-= FACTOR-ANTAGONIST DNA-INTERCALATORS ERK-INHIBITOR FOLATE-ANTAGONISTS HISTONE-= DEACETYLASE-= INHIBITORS IMMUNOSTIMULANTS IMMUNOSUPPRESSIVES INTERFERON-INDUCERS MUTAGEN P-GLYCOPROTEIN-= INHIBITORS PROTEASOME-INHIBITOR RHO-KINASE-INHIBITORS TELOMERASE-INHIBITORS TOPOISOMERASE-I-= INHIBITORS TOPOISOMERASE-II-= INHIBITORS TOPOISOMERASE-= INHIBITORS TYROSINE-KINASE-= INHIBITORS VEGF-ANTAGONIST 1.11 Drugs acting on the nervous system AMPA-AGONISTS AMPA-ANTAGONISTS ANALEPTICS ANTICHOLINESTERASES ANTICONVULSANTS ANTIPARKINSONIANS ANTISEROTONINS BACE-INHIBITOR BENZODIAZEPINE-= ANTAGONISTS CANNABINOID-AGONICTS CANNABINOID-= ANTAGONISTS CEREBROPROTECTIVE CHOLINESTERASE-= REACTIVATORS COMT-INHIBITOR CONVULSANTS CURARE-ANTAGONISTS DOPA-DECARBOXYLASE-= INHIBITORS DOPAMINE-ANTAGONISTS DOPAMINERGICS GABA-ANTAGONISTS GABAMINERGICS GANGLION-STIMULANTS GANGLIONOPLEGICS GLUTAMATE-AGONISTS GLUTAMATE-ANTAGONIST GLYCINE-ANTAGONIST IMIDAZOLINE-AGONISTS IMIDAZOLINE-= ANTAGONISTS KAINATE-AGONISTS KAINATE-ANTAGONISTS MAO-INHIBITORS METHYLASPARTATE-N-= ANTAGONISTS MYDRIATICS NEUROMEDIC-AGONISTS NEUROMEDIN-= ANTAGONISTS NEUROMUSC.BLOCKER-= ANTAGONISTS NEUROMUSC.BLOCKERS NEUROPEPTIDE-Y-= AGONISTS NEUROPEPTIDE-Y-= ANTAGONISTS NEUROPROTECTIVE NEUROTROPHIC OPIOIDS OPIOID-ANTAGONIST PARASYMPATHOLYTICS PARASYMPATHOMIMETICS PURINE-ANTAGONISTS PURINERGICS QUISQUALATE-= ANTAGONISTS RELAXANTS SEROTONINERGICS SPASMOLYTICS SUBSTANCE-K-AGONISTS SUBSTANCE-K-= ANTAGONISTS SYMPATHOLYTICS SYMPATHOLYTICS-ALPHA SYMPATHOLYTICS-BETA SYMPATHOMIMETICS SYMPATHOMIMETICS-= ALPHA SYMPATHOMIMETICS-= BETA 1.12 Psychotropic agents ANTIMANICS ANORECTICS ANTIDEPRESSANTS BENZODIAZEPINE-= AGONISTS BENZODIAZEPINE-= ANTAGONISTS MAO-INHIBITORS NEUROLEPTICS NOOTROPICS PSYCHOSEDATIVES PSYCHOSTIMULANTS PSYCHOTOMIMETICS PSYCHOTONICS SEDATIVES TRANQUILIZERS 1.13 Drugs acting on the respiratory system ANALEPTICS ANTIANAPHYLACTICS ANTIASTHMATICS ANTIHISTAMINES ANTIHISTAMINES-H1 ANTITUSSIVES BRONCHOCONSTRICTOR BRONCHODILATORS EXPECTORANTS MUCOLYTICS 1.14 Drugs acting on the skin ANTIPERSPIRANTS ANTIPRURITICS ANTIPSORIATICS ANTISEBORRHEICS ASTRINGENT DEODORANTS DEPILATORY DERMATOLOGICAL KERATOLYTICS RADIOPROTECTIVES SUNTAN-ACCELERATOR TYROSINASE-INHIBITORS VULNERARIES 1.15 Vitamins and antagonists ANTIVITAMINS BIOFLAVONOIDS FOLATE-ANTAGONISTS VITAMINS VITAMINS-A VITAMINS-B VITAMINS-B1 VITAMINS-B2 VITAMINS-B6 VITAMINS-B12 VITAMINS-C VITAMINS-D VITAMINS-E VITAMINS-K VITAMINS-K1 VITAMINS-K2 VITAMINS-K3 VITAMINS-K4 1.16 Activity terms, miscellaneous ABORTIFACIENT ADSORBENT ALLOSTERIC-ENHANCERS ANGIOGENESIS-= STIMULATORS ANTAGONIST ANTIALCOHOLICS ANTIBODY ANTIDIURETICS ANTIDOTES ANTIHISTAMINES-H1 ANTIHISTAMINES-H3 ANTIOXIDANTS ANTISMOKING APHRODISIAC APOPTOSIS-INHIBITORS CALMODULIN-= ANTAGONISTS CCR2-ANTAGONISTS CCR2B-ANTAGONISTS CCR5-ANTAGONISTS

Derwent Drug File 1033 Thesaurus CELL-ADHESION-= INHIBITORS CHELATORS DIAGNOSTICS DIURETICS DYE EMULSIFIER GLOBULIN HYPERGLYCEMICS ICAM-ANTAGONISTS IMAGING-AGENTS IMMUNOGLOBULIN INHIBIN-ANTAGONISTS INTEGRIN-ANTAGONISTS INVERSE-AGONIST IONEXCHANGERS IONOPHORES LITHOLYTICS LIVER-OIL OPHTHALMOLOGICAL NEPHROTROPIC PARTIAL-AGONIST PDGF-ANTAGONISTS PENETRATION-= ENHANCERS PHYTOTOXINS POTASSIUM-AGONIST PPAR-AGONISTS PPAR-ANTAGONISTS RADIOPAQUES RADIOSENSITIZERS SELECTIN-ANTAGONISTS SPERMATOCIDES SURFACTANTS SYNERGISTS TERATOGEN TOCOLYTICS TONICS TOXINS URICOSURICS UTEROTONICS VCAM-ANTAGONISTS VITRONECTIN-= ANTAGONISTS VLA4-ANTAGONISTS ZOOTOXINS 1.17 New activity terms ACAT-INHIBITORS ADENOSINE-AGONISTS ADENOSINE-= ANTAGONISTS ADENOSINE-KINASE-= INHIBITORS AGE-INHIBITOR AKT-INHIBITOR ALLOSTERIC-ENHANCERS ALPHA-GLUCOSIDASE-= INHIBITORS APOPTOSIS-INHIBITORS ARGINASE-INHIBITORS BACE-INHIBITOR BETA-GLUCOSIDASE-= INHIBITORS CANNABINOID-AGONISTS CANNABINOID-= ANTAGONISTS CASPASE-1-INHIBITORS CASPASE-3-INHIBITORS CASPASE-9-INHIBITORS CASPASE-INHIBITORS CATHEPSIN-INHIBITORS CCR2-ANTAGONISTS CCR2B-ANTAGONISTS CCR5-ANTAGONISTS CLOTTING-FACTOR-XA-= INHIBITORS COMT-INHIBITOR CYCLIN-DEPENDENT-= KINASE-INHIBITORS EPIDERMAL-GROWTH-= FACTOR-ANTAGONIST ERK-INHIBITOR GLUTAMATE-AGONISTS GLUTATHIONE-= TRANSFERASE-= INHIBITORS GLYCOSIDASE-INHIBITORS HISTONE-DEACETYLASE-= INHIBITORS IMIDAZOLINE-AGONISTS IMIDAZOLINE-= ANTAGONISTS INOSINE-= MONOPHOSPHATE-= DEHYDROGENASE-= INHIBITORS MAP-KINASE-INHIBITORS MELATONIN-AGONISTS MELATONIN-= ANTAGONISTS METHYLASPARTATE-N-= ANTAGONISTS NA-H-EXCHANGE-= INHIBITORS NEURAMINIDASE-= INHIBITORS NEUROMEDIN-AGONISTS NEUROMEDIN-= ANTAGONISTS NEUROPEPTIDE-Y-= AGONISTS NEUROPEPTIDE-Y-= ANTAGONISTS NEUROTROPHIC NEUTROPHIL-ELASTASE-= INHIBITORS NF-KAPPA-B-INHIBITORS NITRIC-OXIDE-= SYNTHASE-INDUCERS PANCREOZYMIN-= AGONISTS PANREATIC-ELASTASE-= INHIBITORS PARP-INHIBITORS POTASSIUM-= ANTAGONISTS PROTEASOME-INHIBITOR RAS-INHIBITORS RHO-KINASE-INHIBITORS SELECTIVE-ESTROGEN-= RECEPTOR-= MODULATORS SUBSTANCE-K-AGONISTS TACE-INHIBITORS TYROSINASE-INHIBITORS VEGF-ANTAGONIST VLA4-ANTAGONISTS 2. ORGANISMS 2.1 Animals ARTHROPOD CASES CESTODE FISH FLY GERIATRICS HUMAN INFANT LAB.ANIMAL MAMMAL MITE MOLLUSC MOSQUITO NEMATODE PEDIATRICS REPTILE TICK TREMATODE ZOOLOGY 2.2 Microorganisms ALGA AMEBA BACT. FUNGUS GRAM-NEG. GRAM-POS. PROTOZOON RICKETTSIALES SPIROCHAETALES YEAST 2.3 Plants ALGA BOTANY FRUIT LICHEN MUSHROOM NUT POTATO VEGETABLE 2.4 Viruses ADENOVIRUS ARBOVIRUS ARENAVIRUS CALICIVIRUS CORONAVIRUS HERPESVIRUS IRIDOVIRUS LEUKOVIRUS MYXOVIRUS ONCOVIRUS PAPOVAVIRUS PARVOVIRUS PICORNAVIRUS POXVIRUS REOVIRUS RHABDOVIRUS VIRUS 3. OTHER BIOLOGICAL/ PHYSICAL AREAS 3.1 Disease terms ADDICTION ADRENOPATHY ALLERGY AMINOACID-= METAB.DISORDER ANEMIA ANIMAL-NEOPLASM ANXIETY-DISORDER ARRHYTHMIA AUTOIMMUNE-DISEASE BILIARY-TRACT-DISEASE BIPOLAR-DISORDER BLADDER-DISEASE BURN CARBOHYDRATE-= METAB.DISORDER CARDIOPATHY CARTILAGE-DISEASE CEREBROVASCULAR-= DISEASE CESTODIASIS COLLAGENOSIS CONGENITAL-DISEASE CORONARY-DISEASE DEMENTIA DEMYELINATING-DISEASE DELUSIONAL-DISORDER DERMATOLOGY EATING-DISORDER EDEMA ELECTROLYTE-= METAB.DISORDER ENCEPHALOPATHY

1034 APPENDIX C ESOPHAGUS-DISEASE EYE-DISEASE FACTITIOUS-DISORDER GASTROENTEROPATHY GRANULOMA GRANULOMATOUS-= DISEASE GYNECOLOGY HAIR HEADACHE HEM.DIATHESIS HEMORRHAGE HEPATOPATHY HERNIA HYPERVITAMINOSIS HYPOCHONDRIA HYPOGONADISM HYPOTHALAMUS-DISEASE HYPOVITAMINOSIS IMMUNODEFICIENCY-= DISEASE INFECTION,ALGA INFECTION,BACT. INFECTION,FUNGUS INFECTION,PROTOZOON INFECTION,RICKETTSIALES INFECTION,VIRUS INFERTILITY INFESTATION,ECTOPARASITE INTERSEX INTOXICATION JOINT-DISEASE KINETOSIS LEUKOCYTE-DISORDER LEUKOSIS-COMPLEX LIPID-METAB.DISORDER LITHIASIS LYMPH-DISEASE LYMPHOPROLIFERATIVE-= DISEASE MALABSORPTION MALNUTRITION MAMMA-DISEASE MARROW-DISEASE MENSTRUATION MENTAL-DISORDER MOOD-DISORDER MUCOPOLYSACCHARIDOSIS MULTI-INFARCT-DEMENTIA MYOPATHY NAIL NEMATODIASIS NEOPLASM NEPHROPATHY NEUROMUSC.DISEASE OBESITY OBSTETRICS OCCUPATIONAL-DISEASE ODONTOLOGY OLIGOPHRENIA ORL-DISEASE OSTEOPATHY OVARY-DISEASE PANCREOPATHY PARANOIA PARAPROTEINEMIA PARATHYROID-DISEASE PENIS-DISEASE PERIPHERAL-NERVE-= DISEASE PIGMENTATION PITUITARY-DISEASE PNEUMOPATHY PERSONALITY-DISORDER PORPHYRIA PROSTATE-DISEASE PROTEIN-= METAB.DISORDER PSYCHOTIC-DISORDER PURINE-METAB.DISORDER RADIOLESION RESPIRATION-DISORDER SLEEP SMELL SPINAL-CORD-DISEASE SPLEEN-DISEASE STOMATOLOGY SWEAT SYNDROME TERATOGENESIS TESTIS-DISEASE THIRST THROMBOSIS THYMUS-DISEASE THYROID-DISEASE TRANSPLANTATION TREMATODIASIS ULCER URINARY-TRACT-DISEASE UTERUS-DISEASE VAGINA-DISEASE VASCULAR-DISEASE VENEREAL-DISEASE ZOONOSIS 3.2 Galenics and biopharmaceutics AUXILIARY-INGREDIENT BIOADHESIVE BIOAVAILABILITY BIOPHARM. CONTAINER DESICCANT DISPERSION DRESSING DRUG-DELIVERY FLOCCULANT HUMECTANT LUBRICANT PACKAGING PENETRATION-= ENHANCERS PHARM.PREP. PHARMACEUTICS PHARMACOKINETICS PLASTICIZER PRESERVATION PRESERVATIVE PROPELLANT QUALITY-CONTROL STABILITY STABILIZER STERILIZATION SWEETENER 3.3 Metabolism AMINOACID-METAB. AMINOACID-= METAB.DISORDER BILE-ACID-METAB. CARBOHYDRATE-METAB. CARBOHYDRATE-= METAB.DISORDER CELL-RESPIRATION CORTICOSTEROID-METAB. ELECTROLYTE-METAB. ELECTROLYTE-= METAB.DISORDER ENERGY-METAB. ESTROGEN-METAB. GASTROINTEST.= HORMONE-METAB. GONADOTROPIN-METAB. HORMONE-METAB. KININ-METAB. LEUKOTRIENE-METAB. LIPID-METAB. LIPID-METAB.DISORDER MICROSOME-DRUG-= METAB. MINERALOCORTICOID-= METAB. N-METAB. NUCLEIC-ACID-METAB. OPIOID-METAB. PANCREAS-HORMONE-= METAB. PITUITARY-HORMONE-= METAB. PORPHYRIN-METAB. PROGESTOGEN-METAB. PROSTAGLANDIN-METAB. PROTEIN-METAB. PROTEIN-= METAB.DISORDER PURINE-METAB. PURINE-METAB.DISORDER THYMUS-HORMONE-= METAB. THYROID-HORMONE-= METAB. VITAMIN-METAB. 3.4 Organs and cells ABDOMEN ADRENAL BILE-DUCT BLOOD BONE BRAIN CARTILAGE CONN.TISSUE EAR ERYTHROCYTE ESOPHAGUS EXTREMITY EYE G.U.TRACT GALLBLADDER HAIR HEART HYPOTHALAMUS INTESTINE JOINT KIDNEY LEUKOCYTE LIVER LUNG LYMPH-NODE LYMPHOCYTE MAMMA MARROW MUSCLE NAIL NERVE NEUROMUSC. ORL OVARY PENIS PITUITARY PLACENTA PLATELET PROSTATE RES RESPIRAT.TRACT SALIVA SKIN SMOOTH-MUSCLE SPERM SPINAL-CORD SPINAL-FLUID SPLEEN STOMACH TESTIS THYMUS TISSUE-CULTURE

Derwent Drug File 1035 Thesaurus TOOTH TUMOR-CELL UTERUS VAGINA VESSEL 3.5 Physical and analytical terms ANALYSIS BIOASSAY CHROMATOGRAPHY CRYSTALLOGRAPHY ELECTROCHEM. ELECTROPHORESIS ENZYME-IMMUNODET. IMMUNODET. PHOTOCHEM. PHYS.CHEM. RADIOACTIVITY SEROLOGY SPECTROMETRY SPECTROSCOPY 3.6 General medical terms DIAGNOSIS FORENSIC-MED. GERIATRICS HOMEOPATHY HYGIENE IND.MED. ISOTOPIC-THERAPY MILIT.MED. OCCUPATIONAL-DISEASE OCCUPATIONAL-MED. PEDIATRICS PHYSICOTHERAPY RADIOTHERAPY SEROTHERAPY SPORTS-MED. SURGERY TROP.MED. VET.MED. ZOONOSIS 3.7 Nutrition BEVERAGE DIET FEED-ADDITIVE FEEDING FEEDSTUFF FLAVOR MEAT MILK MILK-FOOD NUTRIENT-TECHNOLOGY NUTRITION PERFORMANCE SPICE SWEETENER TRACE-ELEMENT 3.8 Physiological processes ACT.TRANSPORT BLOOD-CLOTTING BODY-TEMPERATURE BODY-WEIGHT ELECTROPHYSIOL. ESTRUS GASTRIC-SECRETION GROWTH HEMODYNAMICS IMMUNITY INTELLIGENCE LACTATION MENSTRUAL-CYCLE PSYCHOLOGY RESPIRATION 3.9 Physical Processes FILTRATION KINETICS MANOMETRY MICROSCOPY OPT.ROTATION OSMOSIS OXIDATION REDUCTION RHEOLOGY SEDIMENTATION TEMPERATURE THERMODYNAMICS ULTRASONICS 3.10 Miscellaneous ANIMAL-BEHAVIOR ANTIBODY ANTIGEN APPARATUS ART.PANCREAS BIOMETRICS BLOOD-GROUP BREEDING CASTRATION CATALYST CLIMATE COLLOID COMB. COMPLEX COSMETICS CYTOCHROME CYTOLOGY DOSAGE DYE ECONOMICS EGG EMBRYO ESS.OIL GENETICS GLOBULIN GLYCOLIPID GLYCOPROTEIN GNOTOBIOTICS HEMOGLOBIN HISTOCOMPATIBILITY HISTOLOGY HISTONE IMMUNOGLOBULIN INTRAUTERINE-DEVICE MATHEMATICS MEMBRANE NEUROLEPTANALGESIA NOMENCLATURE OIL PH-PK PHOSPHOLIPID PHOTOSYNTH. PLANT-SUBSTANCE PLASMA-LIPID PLASMA-PROTEIN RACE RAY REAGENT RECEPTOR REFLEX RESISTANCE SEX SKIN-TEST SOLVENT STEREOCHEM. STRESS STRUCT.ACT. SUBCELL.STRUCT. SUBSTRATE TAXONOMY TIME TOX. TUBERCULIN VICE WOOL ZOOTECHNICS 4. CHEMISTRY 4.1 Alicycles General AA-LINKED AH-LINKED-CC AH-LINKED-CX BA-LINKED 3-membered CYCLOPROPANE 4-membered CYCLOBUTANE 5-membered AZULENE CYCLOPENTANE FLUORENE INDENE 6-membered ADAMANTANE AMINOCYCLITOL ANTHRACYCLINES CANNABINOIDS CAROTENOID CYCLITOL CYCLOHEXANE QUINONE RETINOID TETRACYCLINES 7-membered AZULENE CYCLOHEPTANE DIBENZOCYCLO= HEPTADIENE TROPANE 8-membered CYCLOOCTANE 9-membered CYCLONONANE 10-membered CYCLODECANE 11-membered CYCLOUNDECANE 12-membered CYCLODODECANE 13-membered CYCLOTRIDECANE 14-membered CYCLOTETRADECANE 15-membered CYCLOPENTADECANE 16-membered CYCLOHEXADECANE 17-membered CYCLOHEPTADECANE 24-membered CYCLOTETRACOSANE

1036 APPENDIX C 4.2 Aminoacids and Peptides AMINOACID BETAINE CEPHALOSPORINS DEPSIPEPTIDE GLYCOPROTEIN LIPOPROTEIN PENICILLINS PEPTIDE PEPTIDE,CYCLIC PROTEIN 4.3 Arenes and other benzenoids ANTHRACENE ARENE BA-LINKED BB-LINKED BENZENE BH-LINKED-CC BH-LINKED-CX BIPHENYL CANNABINOIDS DIPHENYLMETHANE NAPHTHALENE PHENANTHRENE STILBENE 4.4 Functions connected to a benzene ring ARALKYLAMINE ARYL-C-ACID ARYL-C-AMIDE ARYL-C-ESTER ARYLALDEHYDE ARYLAMINE ARYLBROMIDE ARYLCHLORIDE ARYLFLUORIDE ARYLIODIDE ARYLKETONE ARYLSULFIDE BUTYROPHENONE CHALCONE DEPSIDE NITROARENE PHENOL PHENOL-ETHER POLYPHENOL SALICYLIC-ACID THIOPHENOL THYRO-C-ACID 4.5 Carboxylic acids and derivatives ACYLHALIDE AMINOACID ANHYDRIDE ANHYDRIDE,CYCLIC ARYL-C-ACID ARYL-C-AMIDE ARYL-C-ESTER BARBITURATES BILE-ACID C-ACID C-AMIDE C-ESTER CEPHALOSPORINS COUMARIN CS-ACID CS-ESTER DEPSIDE DEPSIPEPTIDE FATTY-ACID GLYCERIDE HAL.FATTY-ACID HYDANTOIN HYDROXAMIC-ACID HYDROXYACID IMIDE,CYCLIC KETOACID LACTAM LACTONE ONIC-ACID PENICILLINS PHOSPHOLIPID PHTHALIMIDE POLY-C-ACID SALICYLIC-ACID THIOBARBITURATES THIOHYDANTOIN THIOHYDROXAMIC-ACID THIOLACTAM THIOLACTONE THYRO-C-ACID UNSAT.FATTY-ACID URONIC-ACID 4.6 Charged functions BETAINE ONIUM PHOSPHONIUM QUAT.AMINE SULFONIUM YLIDE 4.7 Carbohydrates AMINOSUGAR GLYCOPROTEIN GLYCOSIDE NUCLEOSIDE NUCLEOTIDE ONIC-ACID POLYSACCHARIDE SUGAR THIOSUGAR URONIC-ACID 4.8 Carbamates, Ureas, etc. BARBITURATES CARBAMATE CARBAMATE,CYCLIC CARBONATE DITHIOCARBAMATE HYDANTOIN SEMICARBAZIDE SEMICARBAZIDE,CYCLIC THIOBARBITURATES THIOCARBAMATE THIOCARBAMATE,CYCLIC THIOHYDANTOIN THIOSEMICARBAZIDE THIOSEMICARBAZIDE,CYCLIC THIOUREA THIOUREA,CYCLIC THIURAM UREA UREA,CYCLIC XANTHOGENATE 4.9 Heterocycles General AH-LINKED-CC AH-LINKED-CX BH-LINKED-CC BH-LINKED-CX HH-LINKED-CC HH-LINKED-CX HH-LINKED-XX 3-membered with N AZIRIDINE DIAZIRIDINE OXAZIRIDINE 3-membered with O OXAZIRIDINE OXIRANE 3-membered with S THIIRANE 4-membered with N AZETIDINE CEPHALOSPORINS DIAZETIDINE PENICILLINS 4-membered with O DIOXETANE OXAMERCURETANE OXETANE 4-membered with S DITHIETANE 4-membered with X OXAMERCURETANE 5-membered with N AZAPHOSPHOLE BENZIMIDAZOLE CARBAZOLE CARBOLINE CORRINOID DIAZAPHOSPHOLE DITHIAZOLE HYDANTOIN IMIDAZOLE INDAZOLE INDOLE INDOLIZINE ISOINDOLE ISOTHIAZOLE ISOXAZOLE OXADIAZOLE OXATRIAZOLE OXAZOLE PENICILLINS PHTHALIMIDE PORPHYRIN PURINE PYRAZOLE PYRROLE PYRROLIDINE PYRROLIZINE SELENADIAZOLE SELENAZOLE TETRAZOLE THIADIAZOLE THIAZAGERMOLANE THIAZASILACYCLO= PENTANE THIAZOLE THIOHYDANTOIN TRIAZOLE TROPANE 5-membered with O AMINOSUGAR BENZOFURAN DIOXAPHOSPHOLANE DIOXARSOLE DIOXASTANNOLE DIOXATHIOLANE DIOXOLE FURAN GLYCOSIDE ISOBENZOFURAN ISOXAZOLE NITROFURAN ONIC-ACID OXADIAZOLE OXAPHOSPHOLE OXASELENOLE OXATHIOLE OXATRIAZOLE

Derwent Drug File 1037 Thesaurus OXAZOLE SUGAR THIOSUGAR URONIC-ACID 5-membered with S DIOXATHIOLANE DITHIARSOLE DITHIASTIBOLE DITHIAZOLE DITHIOLE ISOTHIAZOLE OXATHIOLE PENICILLINS THIADIAZOLE THIASELENOLE THIAZAGERMOLANE THIAZASILACYCLO= PENTANE THIAZOLE THIOPHENE 5-membered with X AZAPHOSPHOLE DIAZAPHOSPHOLE DIOXAPHOSPHOLANE DIOXARSOLE DIOXASTANNOLE DITHIARSOLE DITHIASTIBOLE OXAPHOSPHOLE OXASELENOLE PHOSPHOLE SELENADIAZOLE SELENAZOLE SILACYCLOPENTANE THIASELENOLE THIAZAGERMOLANE THIAZASILACYCLO= PENTANE 6-membered with N ACRIDINE AZAPHENOTHIAZINE AZAPHOSPHORINE BARBITURATES BENZOQUINOLIZINE CEPHALOSPORINS CINNOLINE DIAZAPHOSPHORANE DIOXAZINE DITHIAZINE INDOLIZINE ISOQUINOLINE MORPHINAN MORPHOLINE NAPHTHYRIDINE OXADIAZAPHOSPHORINE OXADIAZINE OXATHIAZINE OXAZADISILACYCLO= HEXANE OXAZAPHOSPHORINE OXAZINE PHENANTHRIDINE PHENAZINE PHENOTHIAZINE PHENOXAZINE PHTHALAZINE PIPERAZINE PIPERIDINE PTERIDINE PURINE PYRAZINE PYRIDAZINE PYRIDINE PYRIMIDINE QUINAZOLINE QUINOLINE QUINOLIZINE QUINOXALINE QUINUCLIDINE SELENAZINE TELLURAZINE TETRAZINE THIADIAZINE THIATRIAZA= DIPHOSPHORANE THIATRIAZINE THIAZINE THIOBARBITURATES TRIAZATRIPHOSPHORINE TRIAZINE TROPANE 6-membered with O AMINOSUGAR BENZOPYRAN CANNABINOIDS COUMARIN DIOXABORIN DIOXANE DIOXAPHOSPHABORIN DIOXAPHOSPHORINANE DIOXASTANNIN DIOXATHIANE DIOXAZINE FLAVONOID GLYCOSIDE ISOBENZOPYRAN MORPHOLINE NUCLEOSIDE NUCLEOTIDE ONIC-ACID OXADIAZINE OXADIAZAPHOSPHORINE OXAZADISILACYCLO= HEXANE OXAPHOSPHORIN OXATHIANE OXATHIAZINE OXAZAPHOSPHORINE OXAZINE PHENOXAZINE PYRAN SUGAR TETRAOXANE THIOSUGAR TRIOXANE URONIC-ACID XANTHENE 6-membered with S AZAPHENOTHIAZINE CEPHALOSPORINS DIOXATHIANE DITHIANE DITHIAZINE OXATHIANE OXATHIAZINE PHENOTHIAZINE THIADIAZINE THIAPYRAN THIATRIAZA= DIPHOSPHORANE THIATRIAZINE THIAXANTHENE THIAZINE 6-membered with X AZAPHOSPHORINE DIOXABORIN DIAZAPHOSPHORANE DIOXAPHOSPHABORIN DIOXAPHOSPHORINANE DIOXASTANNIN GERMANIN OXADIAZAPHOSPHORINE OXAPHOSPHORIN OXAZADISILACYCLO= HEXANE OXAZAPHOSPHORINE SELENAZINE SELENIN SILACYCLOHEXANE TELLURAPYRAN TELLURAZINE THIATRIAZA= DIPHOSPHORANE TRIAZATRIPHOSPHORINE 7-membered with N AZEPINE BENZODIAZEPINE DIAZAPHOSPHEPINE DIAZEPINE DIBENZAZEPINE DIOXAZEPINE DITHIADIAZEPINE DITHIAZEPINE OXADIAZEPINE OXATHIAZEPINE OXAZAPHOSPHEPINE OXAZEPINE THIADIAZEPINE THIAZEPINE TRIAZEPINE TRITHIAZEPINE 7-membered with O DIOXADITHIEPIN DIOXAPHOSPHEPIN DIOXATHIEPIN DIOXAZEPINE DIOXEPIN OXADIAZEPINE OXATHIAZEPINE OXATHIEPIN OXAZAPHOSPHEPINE OXAZEPINE OXEPIN TRIOXEPIN 7-membered with S DIOXADITHIEPIN DIOXATHIEPIN DITHIADIAZEPINE DITHIATETRASTANNEPIN DITHIAZEPINE OXATHIAZEPINE OXATHIEPIN THIADIAZEPINE THIAZEPINE THIEPIN TRITHIAZEPINE 7-membered with X DIAZAPHOSPHEPINE DIOXAPHOSPHEPIN DITHIATETRASTANNEPIN OXAZAPHOSPHEPINE SELENEPIN 8-membered with N AZOCINE DIAZADIPHOSPHOCINE DIAZAPHOSPHOCINE DIAZOCINE DIOXADIAZOCINE DIOXAZAPHOSPHOCIN DIOXAZOCINE DITHIAZOCINE OXADIAZOCINE OXAZOCINE SELENAZOCINE

1038 APPENDIX C TETRAAZATETRA= PHOSPHOCINE TETRATHIAZOCINE TETRAZOCINE THIADIAZOCINE THIAZOCINE TRIAZOCINE 8-membered with O DIOXADIAZOCINE DIOXADITHIOCIN DIOXAZAPHOSPHOCIN DIOXAZASILACYCLO= OCTANE DIOXAZOCINE DIOXOCIN OXADIAZOCINE OXAZOCINE OXOCIN TETRAOXATETRASILA= CYCLOOCTANE TRIOXADISILACYCLO= OCTANE 8-membered with S DIOXADITHIOCIN DITHIAZOCINE TETRATHIAZOCINE THIADIAZOCINE THIAZOCINE THIOCIN 8-membered with X DIAZADIPHOSPHOCINE DIAZAPHOSPHOCINE DIOXAZAPHOSPHOCINE DIOXAZASILACYCLOOCTANE SELENAZOCINE TETRAAZATETRA= PHOSPHOCINE TETRAOXATETRASILA= CYCLOOCTANE TRIOXADISILACYCLO= OCTANE 9-membered with N AZONINE DIAZONINE OXADIAZONINE OXATHIAZABORONINE OXATHIAZONINE OXAZONINE TRIAZONINE 9-membered with O DIOXADITHIONIN DIOXONIN OXADIAZONINE OXATHIAZABORONINE OXATHIAZONINE OXAZONINE TRIOXONIN 9-membered with S DIOXADITHIONIN OXATHIAZABORONINE OXATHIAZONINE 9-membered with X OXATHIAZABORONINE 10-membered with N AZECINE DIOXAZASTANNECINE DITHIADIAZECINE OXADIAZECINE OXATHIAZECINE OXAZECINE TETRAOXADIAZECINE TETRAZECINE 10-membered with O DIOXAZASTANNECINE DIOXECIN OXADIAZECINE OXATHIAZECINE OXATHIECIN OXAZECINE OXECIN TETRAOXADIAZECINE 10-membered with S DITHIADIAZECINE OXATHIAZECINE OXATHIECIN 10-membered with X DIOXAZASTANNECINE 11-membered with N AZACYCLOUNDECANE DIAZACYCLOUNDECANE DIOXATHIADIAZACYCLO= UNDECANE 11-membered with O DIOXACYCLOUNDECANE DIOXATHIADIAZA= CYCLOUNDECANE OXACYCLOUNDECANE TETRAOXASILA= CYCLOUNDECANE 11-membered with S DIOXATHIADIAZA= CYCLOUNDECANE 11-membered with X TETRAOXASILA= CYCLOUNDECANE 12-membered with N AZACYCLODODECANE DIAZACYCLODODECANE OXADIAZACYCLO= DODECANE TETRAAZACYCLO= DODECANE THIATRIAZACYCLO= DODECANE 12-membered with O DIOXACYCLODODECANE OXACYCLODODECANE OXADIAZACYCLO= DODECANE TETRAOXACYCLO= DODECANE TRIOXACYCLODODECANE 12-membered with S TETRATHIACYCLO= DODECANE THIATRIAZACYCLO= DODECANE 13-membered with N AZACYCLOTRIDECANE DIAZACYCLOTRIDECANE OXADIAZACYCLO= TRIDECANE TETRAAZACYCLO= TRIDECANE THIATRIAZACYCLO= TRIDECANE TRIOXAZACYCLO= TRIDECANE 13-membered with O DIOXACYCLOTRIDECANE OXACYCLOTRIDECANE OXADIAZACYCLO= TRIDECANE TRIOXAZACYCLO= TRIDECANE 13-membered with S THIATRIAZACYCLO= TRIDECANE 14-membered with N AZACYCLOTETRADECANE DIAZACYCLOTETRADECANE OXADIAZACYCLOTETRA= DECANE OXAZACYCLOTETRA= DECANE TETRAAZACYCLOTETRA= DECANE 14-membered with O DIOXACYCLOTETRA= DECANE OXACYCLOTETRA= DECANE OXADIAZACYCLOTETRA= DECANE OXAZACYCLOTETRA= DECANE TRIOXACYCLOTETRA= DECANE 15-membered with N AZACYCLOPENTADECANE AZATETRAOXACYCLO= PENTADECANE DIOXADIAZACYCLO= PENTADECANE DIOXAZACYCLO= PENTADECANE CORRINOID DIAZACYCLOPENTADECANE OXADIAZACYCLO= PENTADECANE OXAZACYCLOPENTA= DECANE PENTAAZACYCLO= PENTADECANE TETRAAZACYCLO= PENTADECANE TRIOXADIAZACYCLO= PENTADECANE 15-membered with O AZATETRAOXACYCLO= PENTADECANE DIOXACYCLOPENTA= DECANE DIOXADIAZACYCLO= PENTADECANE DIOXAZACYCLOPENTA= DECANE OXACYCLOPENTADECANE OXADIAZACYCLOPENTA= DECANE OXAZACYCLOPENTA= DECANE PENTAOXACYCLOPENTA= DECANE TRIOXACYCLOPENTA= DECANE TRIOXADIAZACYCLOPENTA= DECANE 16-membered with N AZAPENTAOXACYCLO= HEXADECANE DIOXAZACYCLOHEXA= DECANE OCTAAZACYCLOHEXA= DECANE OXADIAZACYCLOHEXA= DECANE OXAZACYCLOHEXADECANE

Derwent Drug File 1039 Thesaurus PENTAAZACYCLOHEXA= DECANE PORPHYRIN TETRAAZACYCLOHEXA= DECANE THIATETRAAZACYCLO= HEXADECANE 16-membered with O AZAPENTAOXACYCLO= HEXADECANE DIOXACYCLOHEXADECANE DIOXAZACYCLOHEXA= DECANE OXACYCLOHEXADECANE OXADIAZACYCLOHEXA= DECANE OXAZACYCLOHEXADECANE TETRAOXACYCLOHEXA= DECANE TRIOXACYCLOHEXADECANE 16-membered with S THIATETRAAZACYCLO= HEXADECANE 17-membered with N DITHIATETRAAZACYCLO= HEPTADECANE OXADIAZACYCLO= HEPTADECANE 17-membered with O DIOXACYCLOHEPTADECANE OXACYCLOHEPTADECANE OXADIAZACYCLO= HEPTADECANE 17-membered with S DITHIATETRAAZACYCLO= HEPTADECANE 18-membered with N DIAZACYCLOOCTADECANE DIOXAZASILACYCLOOCTA= DECANE HEXAAZACYCLOOCTA= DECANE OXADIAZACYCLOOCTA= DECANE OXAPENTAAZACYCLO= OCTADECANE PENTAOXAZACYCLO= OCTADECANE TETRAOXADIAZACYCLO= OCTADECANE 18-membered with O DIOXACYCLOOCTADECANE DIOXAZASILACYCLOOCTA= DECANE HEXAOXACYCLOOCTA= DECANE OXACYCLOOCTADECANE OXADIAZACYCLOOCTA= DECANE OXAPENTAAZACYCLO= OCTADECANE PENTAOXACYCLOOCTA= DECANE PENTAOXAZACYCLOOCTA= DECANE TETRAOXACYCLOOCTA= DECANE TETRAOXADIAZACYCLO= OCTADECANE TRIOXACYCLOOCTA= DECANE 18-membered with S HEXATHIACYCLOOCTA= DECANE 18-membered with X DIOXAZASILACYCLOOCTA= DECANE 19-membered with N AZACYCLONONADECANE DIAZACYCLONONADECANE OXADIAZACYCLO= NONADECANE OXATRIAZACYCLO= NONADECANE OXATRITHIADIAZACYCLO= NONADECANE OXAZACYCLONONADECANE THIADIAZACYCLO= NONADECANE 19-membered with O DIOXACYCLONONADECANE OXADIAZACYCLONONA= DECANE OXATRIAZACYCLO= NONADECANE OXATRITHIADIAZACYCLO= NONADECANE OXAZACYCLONONADECANE TETRAOXACYCLONONA= DECANE TRIOXACYCLONONADECANE 19-membered with S OXATRITHIADIAZACYCLO= NONADECANE THIADIAZACYCLO= NONADECANE 20-membered with N OXAZACYCLOEICOSANE TETRAAZACYCLOEICOSANE THIATRIAZACYCLO= EICOSANE 20-membered with O DIOXACYCLOEICOSANE HEXAOXACYCLOEICOSANE OXACYCLOEICOSANE OXAZACYCLOEICOSANE TETRAOXACYCLOEICOSANE TRIOXACYCLOEICOSANE 20-membered with S THIATRIAZACYCLO= EICOSANE 21-membered with N AZACYCLOHENEICOSANE DIOXAZACYCLOHEN= EICOSANE HEXAOXAZACYCLO= HENEICOSANE PENTAOXADIAZACYCLO= HENEICOSANE 21-membered with O DIOXACYCLOHENEICOSANE DIOXAZACYCLOHEN= EICOSANE HEXAOXACYCLO= HENEICOSANE HEXAOXAZACYCLO= HENEICOSANE PENTAOXADIAZACYCLO= HENEICOSANE TETRAOXACYCLO= HENEICOSANE TRIOXACYCLO= HENEICOSANE 21-membered with S THIACYCLOHENEICOSANE 22-membered with N DIAZACYCLODOCOSANE TETRATHIATETRAAZA= CYCLODOCOSANE 22-membered with O HEXAOXACYCLODOCOSANE OXACYCLODOCOSANE PENTAOXACYCLODOCOSANE TETRAOXACYCLODOCOSANE 22-membered with S TETRATHIATETRAAZA= CYCLODOCOSANE 23-membered with N AZACYCLOTRICOSANE OXADIAZACYCLOTRI= COSANE OXATRIAZACYCLOTRI= COSANE OXAZACYCLOTRICOSANE 23-membered with O HEXAOXACYCLOTRI= COSANE OXADIAZACYCLOTRI= COSANE OXATRIAZACYCLOTRI= COSANE OXAZACYCLOTRICOSANE TRIOXACYCLOTRICOSANE 24-membered with N DIOXADIAZACYCLO= TETRACOSANE DIOXAHEXAAZACYCLO= TETRCOSANE HEXAAZACYCLO= TETRACOSANE OCTAAZACYCLO= TETRACOSANE OXADIAZACYCLO= TETRACOSANE OXAZACYCLO= TETRACOSANE 24-membered with O DIOXACYCLOTETRACOSANE DIOXADIAZACYCLO= TETRACOSANE DIOXAHEXAAZACYCLO= TETRCOSANE HEPTAOXACYCLO= TETRACOSANE OCTAOXACYCLO= TETRACOSANE OXACYCLOTETRACOSANE OXADIAZACYCLO= TETRACOSANE OXAZACYCLO= TETRACOSANE TRIOXACYCLO= TETRACOSANE 25-membered with N DIOXADIAZACYCLO= PENTACOSANE DIOXAZACYCLO= PENTACOSANE OXAZACYCLO= PENTACOSANE 25-membered with O DIOXACYCLOPENTACOSANE DIOXADIAZACYCLO= PENTACOSANE DIOXAZACYCLO= PENTACOSANE OXACYCLOPENTACOSANE OXAZACYCLOPENTA= COSANE TRIOXACYCLOPENTA= COSANE

1040 APPENDIX C 26-membered with N DIOXAZACYCLO= HEXACOSANE OCTAAZACYCLO= HEXACOSANE OXAPENTAAZACYCLO= HEXACOSANE 26-membered with O DIOXAZACYCLO= HEXACOSANE OCTAOXACYCLO= HEXACOSANE OXACYCLOHEXACOSANE OXAPENTAAZACYCLO= HEXACOSANE 27-membered with N DIOXAZACYCLO= HEPTACOSANE NONAOXAZACYCLO= HEPTACOSANE OCTAOXAAZACYCLO= HEPTACOSANE OXATRIAZACYCLO= HEPTACOSANE 27-membered with O DIOXACYCLOHEPTACOSANE DIOXAZACYCLO= HEPTACOSANE NONAOXACYCLO= HEPTACOSANE NONAOXAZACYCLO= HEPTACOSANE OCTAOXAAZACYCLO= HEPTACOSANE OCTAOXACYCLO= HEPTACOSANE OXATRIAZACYCLO= HEPTACOSANE 28-membered with N DIOXADIAZACYCLO= OCTACOSANE DIOXADITHIATETRA= AZACYCLOOCTACOSANE OXAPENTAAZACYCLO-= OCTACOSANE OXAZACYCLOOCTACOSANE 28-membered with O DIOXACYCLOOCTACOSANE DIOXADIAZACYCLO= OCTACOSANE DIOXADITHIATETRA= AZACYCLOOCTACOSANE OCTAOXACYCLO-= OCTACOSANE OXACYCLOOCTACOSANE OXAPENTAAZACYCLO= OCTACOSANE OXAZACYCLOOCTACOSANE TETRAOXACYCLO= OCTACOSANE 28-membered with S DIOXADITHIATETRA= AZACYCLOOCTACOSANE 29-membered with N AZACYCLONONACOSANE DIOXAZACYCLO= NONACOSANE 29-membered with O DIOXAZACYCLO= NONACOSANE 30-membered with N DIOXADIAZACYCLO= TRIACONTANE NONAOXAZACYCLO= TRIACONTANE TETRATHIAHEPTA= AZACYCLOTRIACONTANE 30-membered with O DIOXACYCLOTRIACONTANE DIOXADIAZACYCLO= TRIACONTANE NONAOXACYCLO= TRIACONTANE NONAOXAZACYCLO= TRIACONTANE OXACYCLOTRIACONTANE TRIOXACYCLOTRIACONTANE 30-membered with S TETRATHIAHEPTAAZA= CYCLOTRIACONTANE 31-membered with N AZACYCLOUNTRIA= CONTANE 31-membered with O TETRAOXACYCLOHEN= TRIACONTANE TRIOXACYCLOHEN= TRIACONTANE 32-membered with N DIOXADIAZACYCLODO= TRIACONTANE HEXAAZACYCLODO= TRIACONTANE OCTAAZACYCLODO= TRIACONTANE 32-membered with O DIOXACYCLODO= TRIACONTANE DIOXADIAZACYCLODO= TRIACONTANE OCTAOXACYCLODO= TRIACONTANE OXACYCLODOTRIA= CONTANE 33-membered with N DECAOXAZACYCLO= TRITRIACONTANE 33-membered with O DECAOXAZACYCLO= TRITRIACONTANE UNDECAOXACYCLO= TRITRIACONTANE 34-membered with O DIOXACYCLOTETRA= TRIACONTANE HEPTAOXACYCLOTETRA= TRIACONTANE HEXAOXACYCLOTETRA= TRIACONTANE TETRAOXACYCLOTETRA= TRIACONTANE OCTAOXACYCLOTETRA= TRIACONTANE OXACYCLOTETRA= TRIACONTANE 35-membered with N UNDECAAZACYCLOPENTA= TRIACONTANE 35-membered with O OXACYCLOPENTA= TRIACONTANE 36-membered with O DIOXACYCLOHEXA= TRIACONTANE OXACYCLOHEXA= TRIACONTANE TETRAOXACYCLOHEXA= TRIACONTANE 38-membered with N HEXAAZACYCLOOCTA= TRIACONTANE 38-membered with O OXACYCLOOCTA= TRIACONTANE 40-membered with N DIOXATRITHIAHEXAAZA= CYCLOTETRACONTANE 40-membered with O DIOXATRITHIAHEXAAZA= CYCLOTETRACONTANE DIOXACYCLOTETRA= CONTANE 40-membered with S DIOXATRITHIAHEXAAZA= CYCLOTETRACONTANE 42-membered with O OXACYCLODOTETRA= CONTANE 44-membered with O OXACYCLOTETRATETRA= CONTANE 4.10 Halogen-containing functions ACYLHALIDE ALKYLBROMIDE ALKYLCHLORIDE ALKYLFLUORIDE ALKYLIODIDE ARYLBROMIDE ARYLCHLORIDE ARYLFLUORIDE ARYLIODIDE BROMINE CHLORINE FLUORINE HAL.FATTY-ACID IODINE N-MUSTARD SEMI-N-MUSTARD SULFONYL-HALIDE THYRO-C-ACID 4.11 Aldehydes and Ketones ALDEHYDE ANTHRACYCLINES ARYLALDEHYDE ARYLKETONE BUTYROPHENONE CHALCONE FLAVONOID KETENE KETOACID KETONE KETONE,CYCLIC POLYALDEHYDE POLYKETONE QUINONE THIOALDEHYDE THIOKETONE 4.12 Complexes ALUMINUM-COMPLEX ANTIMONY-COMPLEX BARIUM-COMPLEX BERYLLIUM-COMPLEX BISMUTH-COMPLEX BORON-COMPLEX CADMIUM-COMPLEX

Derwent Drug File 1041 Thesaurus CALCIUM-COMPLEX CESIUM-COMPLEX CHROMIUM-COMPLEX COBALT-COMPLEX COMPLEX COPPER-COMPLEX DYSPROSIUM-COMPLEX EUROPIUM-COMPLEX GADOLINIUM-COMPLEX GALLIUM-COMPLEX GOLD-COMPLEX HAFNIUM-COMPLEX HOLMIUM-COMPLEX INDIUM-COMPLEX IODINE-COMPLEX IRIDIUM-COMPLEX IRON-COMPLEX LANTHANUM-COMPLEX LEAD-COMPLEX LITHIUM-COMPLEX MAGNESIUM-COMPLEX MANGANESE-COMPLEX MERCURY-COMPLEX MOLYBDENUM-COMPLEX NEODYMIUM-COMPLEX NICKEL-COMPLEX OSMIUM-COMPLEX PALLADIUM-COMPLEX PLATINUM-COMPLEX POTASSIUM-COMPLEX PRASEODYMIUM-= COMPLEX RHENIUM-COMPLEX RHODIUM-COMPLEX RUBIDIUM-COMPLEX RUTHENIUM-COMPLEX SCANDIUM-COMPLEX SILVER-COMPLEX SODIUM-COMPLEX STRONTIUM-COMPLEX TECHNETIUM-COMPLEX TELLURIUM-COMPLEX TERBIUM-COMPLEX THORIUM-COMPLEX THULIUM-COMPLEX TIN-COMPLEX TITANIUM-COMPLEX TUNGSTEN-COMPLEX URANIUM-COMPLEX VANADIUM-COMPLEX YTTERBIUM-COMPLEX YTTRIUM-COMPLEX ZINC-COMPLEX ZIRCONIUM-COMPLEX 4.13 Salts ALUMINUM-SALT ANTIMONY-SALT BARIUM-SALT BISMUTH-SALT CADMIUM-SALT CALCIUM-SALT CERIUM-SALT CHROMIUM-SALT COBALT-SALT COPPER-SALT DYSPROSIUM-SALT ERBIUM-SALT EUROPIUM-SALT GADOLINIUM-SALT GALLIUM-SALT GOLD-SALT INDIUM-SALT IRON-SALT LANTHANUM-SALT LEAD-SALT LITHIUM-SALT LUTETIUM-SALT MAGNESIUM-SALT MANGANESE-SALT MERCURY-SALT NEODYMIUM-SALT NICKEL-SALT PALLADIUM-SALT PLATINUM-SALT PLUTONIUM-SALT POTASSIUM-SALT PRASEODYMIUM-SALT RHODIUM-SALT SAMARIUM-SALT SILVER-SALT SODIUM-SALT TERBIUM-SALT THALLIUM-SALT THULIUM-SALT TITANIUM-SALT TUNGSTEN-SALT URANIUM-SALT YTTERBIUM-SALT YTTRIUM-SALT ZINC-SALT 4.14 Monovalent N-containing functions AMIDINE AMIDINE,CYCLIC AMIDRAZONE AMINE AMINOACID AMINOALCOHOL AMINOCYCLITOL AMINOSUGAR ARALKYLAMINE ARYLAMINE CEPHALOSPORINS FORMAZAN GUANIDINE GUANIDINE,CYCLIC HYDRAZINE HYDROXAMIC-ACID HYDROXYLAMINE IMIDATE ISOCYANATE LACTAM MUSTARD-OIL N-ACID N-ESTER N-MUSTARD NITRO NITROARENE NITROFURAN NITROSO PENICILLINS POLYAMINE QUAT.AMINE SEMI-N-MUSTARD SEMICARBAZIDE SEMICARBAZIDE,CYCLIC SULFENAMIDE SULFINAMIDE SULFONAMIDE SULTAM THIOHYDROXAMIC-ACID THIOIMIDATE THIOSEMICARBAZIDE THIOSEMICARBAZIDE,= CYCLIC TRIAZENE 4.15 Polyvalent N-containing functions ALDIMINE AMIDINE AMIDINE,CYCLIC AMIDRAZONE AZIDE AZO CARBODIIMIDE CYANATE DIAZONIUM FORMAZAN GUANIDINE GUANIDINE,CYCLIC IMIDATE ISOCYANATE KETIMINE MUSTARD-OIL N-ACID N-ESTER N-OXIDE N-OXIDE,CYCLIC NITRILE OXIME SULFOXIMIDE THIOCYANATE THIOIMIDATE TRIAZENE 4.16 Monovalent O-containing functions ACETAL ALCOHOL AMINOALCOHOL AMINOCYCLITOL AMINOSUGAR CYANATE CYCLITOL DEPSIDE ENOL ETHER GLYCOSIDE HYDROXAMIC-ACID HYDROXYACID HYDROXYLAMINE IMIDATE KETAL N-ACID N-ESTER ONIC-ACID ONIUM ORTHO-C-ESTER OXIME PEROXIDE PHENOL PHENOL-ETHER POLYALCOHOL POLYPHENOL SALICYLIC-ACID SUGAR THIOSUGAR THIOHYDROXAMIC-ACID THYRO-C-ACID URONIC-ACID 4.17 P-containing functions NUCLEOTIDE P-ACID P-AMIDE P-ESTER PHOSPHINE PHOSPHOLIPID PHOSPHONIC-ACID PHOSPHONIUM PS-ACID 4.18 Functions within rings AMIDINE,CYCLIC ANHYDRIDE,CYCLIC ANTHRACYCLINES BARBITURATES CARBAMATE,CYCLIC CEPHALOSPORINS COUMARIN FLAVONOID

1042 APPENDIX C GUANIDINE,CYCLIC HYDANTOIN IMIDE,CYCLIC KETONE,CYCLIC LACTAM LACTONE N-OXIDE,CYCLIC PENICILLINS PEPTIDE,CYCLIC PHTHALIMIDE QUINONE SEMICARBAZIDE,CYCLIC SULFONE,CYCLIC SULFOXIDE,CYCLIC SULTAM SULTONE THIOBARBITURATES THIOCARBAMATE,CYCLIC THIOHYDANTOIN THIOLACTAM THIOLACTONE THIOSEMICARBAZIDE,= CYCLIC THIOUREA,CYCLIC UREA,CYCLIC 4.19 Ring-linked terms AA-LINKED AH-LINKED-CC AH-LINKED-CX BA-LINKED BB-LINKED BH-LINKED-CC BH-LINKED-CX HH-LINKED-CC HH-LINKED-CX HH-LINKED-XX 4.20 Monovalent S-containing functions ARYLSULFIDE CS-ACID CS-ESTER DISULFIDE DITHIOCARBAMATE MERCAPTAN S-ACID S-ESTER SULFENAMIDE SULFIDE SULFONIUM THIOACETAL THIOCYANATE THIOHYDROXAMIC-ACID THIOIMIDATE THIOKETAL THIOPHENOL THIOSUGAR THIURAM 4.21 Polyvalent S-containing functions CS-ACID CS-ESTER DITHIOCARBAMATE MUSTARD-OIL S-ACID S-ESTER SULFINAMIDE SULFONAMIDE SULFONE SULFONE,CYCLIC SULFONIC-ACID SULFONYL-HALIDE SULFOXIDE SULFOXIDE,CYCLIC SULFOXIMIDE SULTAM SULTONE THIOALDEHYDE THIOBARBITURATES THIOCARBAMATE THIOCARBAMATE,CYCLIC THIOHYDANTOIN THIOKETONE THIOLACTAM THIOLACTONE THIOSEMICARBAZIDE THIOSEMICARBAZIDE,= CYCLIC THIOUREA THIOUREA,CYCLIC XANTHOGENATE 4.22 Steroids ANDROSTANE BILE-ACID CHOLESTANE CYCLOSTEROID ESTRANE HETEROSTEROID HOMOSTEROID ISOSTEROID NORSTEROID PREGNANE SECOSTEROID STEROID TRITERPENE 17-BETA-ALKYLSTEROID 4.23 Unsaturated functions ACETYLENE CAROTENOID CHALCONE ENOL KETENE OLEFIN POLYOLEFIN RETINOID STILBENE UNSAT.FATTY-ACID 4.24 Miscellaneous ALKALOID ALKANE AMMONIA BRIDGE-STRUCT. COND.RING HYDRIDE MACROCYCLE ORGANOMETALLIC PLANT-SUBSTANCE POLYMER SPIRO TERPENE

Derwent Drug File 1043 Thesaurus

APPENDIX D
KWOC LISTING
INTRODUCTION This KWOC (KeyWord Out of Context) listing is simply an inversion of the Thesaurus terms in which all specific keywords (lower terms) are collated under the corresponding generic keywords (higher terms). The listing includes appropriate keywords for all the entries contained in the seventh edition of the Thesaurus. The major use of the KWOC is to identify those lower terms which will be retrieved when a higher term is used in a strategy. It may also be used to establish how a strategy may be made more precise by using one or more of the lower terms listed. Furthermore, it indicates our policy on terminology; this might be useful if a searcher wishes to know how Derwent would index, say, a new vaccine which did not appear in the Thesaurus. It should be noted that some specific keywords appear in the list in lower case letters. These are not directly retrievable in this form; please consult the Thesaurus itself for instructions on how they should be entered in a search. ABDOMEN OMENTUM PERITONEUM ACARICIDES ABAMECTIN ALDICARB ALDICARB-SULFONE ALDICARB-SULFOXIDE ALTEMICIDIN AMITRAZ ARAMITE BALSAM-PERU BENOXAFOS BENZYLBENZOATE BROMOCICLEN BROMOFOS-ETHYL BROMOPROPYLATE CARBOPHENOTHION CHLORACETOPHOS CHLORBENSIDE

CHLORFENETHOL CHLORFENSON CHLOROBENZILATE CHLOROPROPYLATE CHLORPHENAMIDINE CROTAMITON CYCLOPRATE CYHALOTHRIN CYMIAZOLE CYPERMETHRIN CYPERMETHRIN-ALPHA DERMOCEPT DICOFOL DINOBUTON DINOCAP DIOXATION DIXANTHOGEN DORAMECTIN FENAZAFLOR FENPROPATHRIN FENSON FIPRONIL FLUMETHRIN FLUVALINATE FOLBEX-VA FORMOTHION GOMELIN ISOFEN IVERMECTIN KAS-81 MALATHION MESULFEN METHAMIDOPHOS METRIFONATE-ACETATE MILBEMYCIN-A MILBEMYCIN-B-41D MILBEMYCIN-BETA-1 MILBEMYCIN-BETA-3 MILBEMYCIN-D MILBEMYCIN-E MILBEMYCIN-G MILBEMYCIN-OXIME MOXIDECTIN NAPHTHALENE (Drug) NIMIDANE OXYDEMETON-METHYL PESTOBAN PHENKAPTON PHOSMET PIPERONYL-BUTOXIDE PIQUEROL-A PIRIMIPHOS-ETHYL PLIZON PROCLONOL PROMACYL PROPETAMPHOS PYRIMITATE RESMETHRIN

SELAMECTIN SULFIRAM TEPP TETRADIFON TIBENZATE TIOCTILATE TRIAZOPHOS TRICYCLOHEXYLHYDROXYTIN VARROXAN-T-1 VJ-45 VJ-52 VJ-53 VJ-58 VJ-60 ACAT-INHIBITORS 447-C-88 57-118 AVASIMIBE BEZAFIBRATE CI-1011 CI-976 CL-277082 CL-283546 CL-283796 COLESTYRAMINE CP-113818 CRILVASTATIN E-5324 F-1394 FCE-27677 FR-145237 GERI-BP-001-M HL-004 KW-3033 MELINAMIDE NTE-122 PD-138142 PYRIPYROPENE-A RP-64477 RP-73163 SC-435 SCH-48461 TMP-153 YM-17E ACE-INHIBITORS A-58365A A-58365B AB-47 ALACEPRIL ALATRIOPRIL ALTIOPRIL CALCIUM ANCOVENIN BAY-O-6997 BAY-Q-1313 BENAZEPRIL BENAZEPRILAT BENZOYLCAPTOPRIL

BMS-182657 BPP-9A BRL-36378 BW-A575C BW-B385C CAPTOPRIL CAPTOPRIL-CYSTEINE CAPTOPRIL-DISULFIDE CAPTOPRIL-GLUTATHIONE CERONAPRIL CGS-13928C CGS-26582 CGS-26670 CGS-28106 CGS-30440 CI-925 CILAZAPRIL CILAZAPRILAT CL-242817 CONVERSTATIN CV-5975 DEACETYLALACEPRIL DELAPRIL DELAPRIL-DIACID DU-1227 DU-1777 ENALAPRIL ENALAPRILAT EPICAPTOPRIL ER-32935 EU-4867 EU-5476 FOROXYMITHINE FOSINOPRIL FOSINOPRILAT GEMOPATRILAT H-76 HEMORPHIN-4 HOE-065 HOE-288 IMIDAPRIL IMIDAPRILAT INDOLAPRIL INDOLAPRILAT K-13 L-155212 L-681176 LACTORPHIN-ALPHA LACTORPHIN-BETA LIBENZAPRIL LISINOPRIL LYCIUMIN-A LYCIUMIN-B MDL-100173 MDL-27088 MDL-27210 METIAPRIL METIOPRIL

1044 APPENDIX D MIXANPRIL MK-351A MOEXIPRIL MOEXIPRILAT MURACEIN-A MURACEIN-B MURACEIN-C NITROSOCAPTOPRIL OMAPATRILAT PENTOPRIL PENTOPRILAT PERINDOPRIL PERINDOPRILAT PIVOPRIL PROCYANIDIN-B2-DIGALLATE QUINAPRIL QUINAPRILAT RAMIPRIL RAMIPRILAT RB-105 RENTIAPRIL REV-6207 RHC-3454 RO-31-8472 SA-291 SA-7090 SCH-54470 SPIRAPRIL SPIRAPRILAT SQ-13297 SQ-13863 SQ-14102 SQ-14551 SQ-20475 SQ-27786 SQ-28370 TEMOCAPRIL TEMOCAPRILAT TEPROTIDE TRANDOLAPRIL TRANDOLAPRILAT UTIBAPRIL WY-44221 YS-980 Z-13752-A ZABICIPRIL ZABICIPRILAT ZOFENOPRILAT ZOFENOPRILAT-ARGININE-= SALT ACETYL-COA-CARBOXYLASEINHIBITORS AICA-RIBOTIDE ACIDOSIS LACTIC-ACIDOSIS ACT.TRANSPORT SODIUM-PUMP ACTH-AGONISTS ACTH ACTH-1-10 ACTH-1-13 ACTH-1-13-AMIDE ACTH-1-14 ACTH-1-16 ACTH-1-16-AMIDE ACTH-1-18 ACTH-1-4 ACTH-11-24 ACTH-4-10 ACTH-4-10,7-D-PHE ACTH-4-11 ACTH-4-7 ACTH-5-10 ACTH-5-24 ACTH-6-9 ACTH-7-24 ACTH-7-38 ACTH-CATTLE ACTH-HUMAN ACTH-PIG-A ACTH-PIG-BETA ACTH-SHEEP ALSACTIDE BA-44680 BETA-CELL-TROPIN CLIP CODACTIDE EBIRATIDE GIRACTIDE NORLEUSACTIDE ORG-2766 SEMAX SERACTIDE TETRACOSACTIDE TOSACTIDE TRICOSACTIDE ACTH-ANTAGONISTS LIPOCORTIN-1-188 LIPOCORTIN-1-HUMAN ACTION-POTENTIAL MIGRATING-MYOELECTRIC-= COMPLEX ADDICTION ALCOHOLISM DELIRIUM-TREMENS WITHDRAWAL-SYNDROME ADENOCARCINOMA A427-CELL A549-CELL CACO2-CELL CC531 CC531-CELL DU145-CELL DUNNING-R3327H DUNNING-R3327H-CELL HCCL-CELL HCT8-CELL HEY-CELL HOC1-CELL HOC7-CELL HT29-CELL HUTU80-CELL MCF7-CELL ME180-CELL MKN1-CELL MKN28-CELL R3230AC-CELL RAG-CELL TA3-CELL WALKER-256-= ADENOCARCINOMA WALKER-256-CELL ADENOMA MA160-CELL ADENOSINE-AGONISTS ATL-193 CVT-3033 CVT-3146 CVT-510 DWH-146-E GR-190178 MRE-0470 MRS-1760 PD-125944 RPR-100579 WRC-470 XYLOADENINE ADENOSINE-ANTAGONISTS ADENOSINE ARC-69931-MX CS-747 KW-6002 MRS-1754 R-99224 VUF-8501 VUF-8504 VUF-8505 VUF-8507 ADENOSINE-DEAMINASEINHIBITORS ADECHLORIN ADECYPENOL AZACOFORMYCIN-2 COFORMYCIN COFORMYCIN-= MONOPHOSPHATE DIHYDROROBINETIN PENTOSTATIN ADENOVIRUS CELO-VIRUS HEM.ANEMIA-SYNDROME-= VIRUS HEM.ENTERITIS-VIRUS ICH-VIRUS INCLUSION-BODY-HEPATITIS-= VIRUS MARBLE-SPLEEN-DISEASE-= VIRUS ADENYLATE-CYCLASEINHIBITORS BRL-35135 DIAZEPAM IODOAMINOFLISOPOLOL KHELLIN LITHIUM-CHLORIDE PD-81723 RO-5-4864 SQ-22536 ADJUVANTS ALGAMMULIN ARABINOGALACTAN BERYLLIUM-HYDROXIDE BORDETELLA PERTUSSIS CDRI-84-201 CGP-11637 CGP-19835 CGP-19835A CHACONINE-ALPHA CORYNEBACT.CUTIS CRL-1005 CRP-HUMAN DETOX DIMETHYLDIOCTADECYL= AMMONIUM BROMIDE DJ-7041 EMI-1 EMI-2 EMI-3 ENTEROTOXIN-HEAT-LABILE-= E.COLI ENTEROTOXIN-HEAT-LABILE-= E.COLI-LTK63 ENTEROTOXIN-HEAT-LABILE-= E.COLI-LTR72 FREUND-ADJUVANT GPI-0100

Derwent Drug File 1045 Thesaurus IMMTHER INTERLEUKIN-1-BETA-SHEEP ISA-70 L-101 L-121 L-644257 LA-18-PP LIPID-A MARCOL-52 MEDICAGENATE MONTANIDE-103 MONTANIDE-ISA-25 MONTANIDE-ISA-720 MURABUTIDE MURAMETIDE MURAMYL-DIPEPTIDE MURAMYL-DIPEPTIDE-B30 MURAMYL-DIPEPTIDE-= DIPALMITOYL-GLYCEROL MURAMYL-TRIPEPTIDE MYCOBACT.TUBERCULOSIS P-1005 PARAFFIN-LIQUID PIMELAUTIDE POLYADENYLATE POLYADENYLATE-URIDYLATE POLYURIDYLATE QUIL-A QUILLAJA-SAPONIN RANTES RESIQUIMOD RIBI-ADJUVANT ROMURTIDE SAF-M SDZ-280-636 SPECOL STEARYL-PHENYLALANINE STEARYL-TYROSINE SYNTEX-ADJUVANT-= FORMULATION-1 T150R1 TITERMAX TRIMETHYLCHITOSAN-N-= CHLORIDE VC-1052 VILOZEN ADRENAL ADRENAL-CORTEX ADRENAL-MEDULLA ZONA-FASCICULATA ZONA-GLOMERULOSA ZONA-RETICULARIS ADRENAL-CORTEX ZONA-FASCICULATA ZONA-GLOMERULOSA ZONA-RETICULARIS ADRENOPATHY ACHARD-THIERS-SYNDROME ADDISON-DISEASE adrenal-virilism ADRENOGENITAL-SYNDROME ADRENOLEUKODYSTROPHY ALDOSTERONISM ALDOSTERONOMA BARTTER-SYNDROME congenital-adrenal-= hyperplasia CUSHING-SYNDROME HYPERADRENALISM hyperadrenocorticism HYPOADRENALISM hypoadrenocorticism hypoadrenocorticism HYPOALDOSTERONISM LIDDLE-SYNDROME WATERHOUSE-= FRIDERICHSEN-SYNDROME AFFINITY-LABELED PHOTOAFFINITY-LABELED ALCOHOL-DEHYDROGENASEINHIBITORS CIMETIDINE DEXTRAN-SULFATE FOMEPIZOLE PENTOSAN-POLYSULFATE ALCOHOLISM alcoholic-cirrhosis DELIRIUM-TREMENS KORSAKOFF-SYNDROME laennec-cirrhosis ZIEVE-SYNDROME ALDOSE-REDUCTASEINHIBITORS A-1576 ACARBOSE ADN-138 AL-01766 AL-03077 AL-03150 AL-03152 AL-03153 AL-1567 AL-3152 AL-4114 ALO-3363 ALRESTATIN CT-112 DANSHENOL-A DANSHENOL-B EPALRESTAT GP-1447 ICI-215918 IMIRESTAT ISODIBUT ISOLIQUIRITIN LIQUIRITIN M-16049 MINALRESTAT NEOMANOALIDE NZ-314 PONALRESTAT SNK-860 SORBINIL SPR-210 TOLRESTAT WAY-121509 WF-3681 ZD-5522 ZENARESTAT ZOPOLRESTAT ALDOSTERONE-ANTAGONISTS CANRENOATE CANRENOATE POTASSIUM CANRENONE DEOXYALDOSTERONE-18 DICIRENONE DIHYDROSPIRORENONE EPLERENONE ETHINYLPROGESTERONE-18 L-632481 MESPIRENONE METYRAPOL METYRAPONE MEXRENOATE POTASSIUM OXPRENOATE POTASSIUM PRORENOATE POTASSIUM PRORENONE RO-14-9012 RU-26752 SC-11927 SC-19886 SC-24813 SC-25152 SC-26519 SC-27169 SC-5233 SC-8109 SPIRONOLACTONE SPIRORENONE SPIROXASONE SU-10603 SU-9055 VINYLPROGESTERONE-18 ZK-30595 ZK-91587 ZK-97894 ALGA ANACYSTIS CHLAMYDOMONAS CHLORELLA CLADOPHORA COELASTRUM CYANOPHYCEAE CYMPOLIA DICTYOTA EUGLENA FUCUS FURCELLARIA GAURENCIA GRATELOUPIA HALIMEDA LAMINARIA LAURENCIA MICROCYSTIS NEMALION OCHROMONAS ODONTHALIA OSCILLATORIA PHAEODACTYLUM PHYLLOPHORA PLUMARIA POLYSIPHONIA PROTOTHECA RHODOGLOSSUM RHODOMELA SARGASSUM SCENEDESMUS SEAWEED TICHOCARPUS TRIBONEMA TURNERELLA ULVA ALGICIDES CYANOBACTERIN EPIPOLYGODIAL ISOISOVELLERAL LANOSOL VELLERAL ALKALINE-PHOSPHATASEINHIBITORS CHLORPROMAZINE CROMOLYN SODIUM TRETINOIN ALLERGY allergic-alveolitis ALLERGIC-GRANULOMATOSIS ANAPHYLAXIS ANGIONEUROTIC-EDEMA ARTHUS-REACTION atopic-dermatitis

1046 APPENDIX D atopic-eczema CALCIPHYLAXIS CHINESE-RESTAURANT-= SYNDROME contact-dermatitis DERMATOGRAPHIA farmers-lung FIXED-ERUPTION HAY-FEVER HYPERERGIA HYPERSENSITIVITY JARISCH-HERXHEIMER-= REACTION MAZZOTTI-REACTION mesnier-prurigo neurodermatitis RED-MAN-SYNDROME SERUM-SICKNESS SHWARTZMAN-= PHENOMENON SWEET-ITCH WISSLER-FANCONI-= SYNDROME ALOPECIA congenital-hypotrichosis HYPOTRICHOSIS unna-syndrome ALPHA-GLUCOSIDASEINHIBITORS ACARBOSE AMEBA ACANTHAMOEBA ENTAMOEBA HARTMANELLA NAEGLERIA AMEBICIDES AMOPYROQUINE BTI-2286E CAERULOMYCIN-A CEPHAELINE CHLORBETAMIDE CHLOROQUINE CHONEMORPHINE CINCHONAMINE CLAMOXYQUINE CLEFAMIDE CONESSINE DEHYDROEMETINE DIFETARSONE DILOXANIDE DILOXANIDE-FUROATE EMETINE ETOFAMIDE GLAUCARUBIN HYDROXYVERNOLIDE INSULARINE METRONIDAZOLE MK-910 MSI-103 MSI-94 NIRIDAZOLE NITROPHENIDE ORNIDAZOLE PANIDAZOLE PHANQUINONE PHENARSONE-SULFOXYLATE PIRINIDAZOLE POLYBENZARSOL QUINFAMIDE QUINIDINONE RAPANONE SATRANIDAZOLE SECNIDAZOLE STEVALADIL STIRIMAZOLE SYMETINE TECLOZAN USAMBARENSINE USAMBARINE VERNOLIDE AMINOACID-METAB. TRANSAMINATION AMINOACID-METAB.DISORDER ALKAPTONURIA CITRULLINURIA CYSTATHIONINURIA CYSTINE-STORAGE-DISEASE CYSTINURIA HARTNUP-DISEASE HISTIDINEMIA HOMOCYSTEINEMIA HOMOCYSTINEMIA HOMOCYSTINURIA HYPERARGININEMIA HYPERGLYCINEMIA HYPERPHENYLALANINEMIA HYPOMETHIONINEMIA MAPLE-SYRUP-DISEASE METHYLMALONICACIDEMIA METHYLMALONICACIDURIA OCHRONOSIS OCULOCEREBRORENAL-= SYNDROME PHENYLKETONURIA PROPIONICACIDEMIA TYROSINEMIA TYROSINOSIS AMPA-AGONISTS AMINOPHOSPHONOCAPROATE ANIRACETAM FG-9065 LY-404187 OXIRACETAM AMPA-ANTAGONISTS ACEA-1021 ACEA-1031 ACEA-1328 CP-465022 EGIS-8332 FG-9041 FG-9202 GYKI-52466 KAITOCEPHALIN KAITOCEPHALIN LY-215490 LY-293558 PD-152247 S-17625 YM-900 ANABOLICS ALVESIN-NEW ANDROSTANOLONE ANDROSTANOLONEPROPIONATE ANDROSTENEDIOL-= DIPROPIONATE BA-36644 BOLANDIOL BOLANDIOL-DIPROPIONATE BOLASTERONE BOLAZINE BOLAZINE-CAPROATE BOLDENONE BOLDENONE-UNDECYLENATE BOLENOL BOLMANTALATE CLOSTEBOL CLOSTEBOL-ACETATE CLOSTEBOL-CAPROATE CLOSTEBOL-PROPIONATE DEHYDROCHLORMETHYL= TESTOSTERONE DROSTANOLONE DROSTANOLONEPROPIONATE ENESTEBOL ETHYLESTRENOL FORMEBOLONE FURAZABOL HEAD-ACTIVATOR IPRIFLAVONE MEBOLAZINE MESABOLONE MESTANOLONE METANDIENONE METENOLONE METENOLONE-ACETATE METENOLONE-ENANTHATE METHANDRIOL METRIBOLONE MIBOLERONE NANDROLONE NANDROLONE-17-ALPHA NANDROLONE-= CYCLOHEXYLPROPIONATE NANDROLONE-CYCLOTATE NANDROLONE-DECANOATE NANDROLONE-HEXYLOXY= PHENYLPROPIONATE NANDROLONE-LAURATE NANDROLONE-= PHENYLPROPIONATE NANDROLONE-PROPIONATE NANDROLONE-SULFATE SODIUM NANDROLONE-= UNDECYLENATE NORBOLETONE NORCLOSTEBOL NORETHANDROLONE OXABOLONE-CIPIONATE OXANDROLONE OXYMESTERONE OXYMETHOLONE PROPETANDROL PS-179 QUINBOLONE RO-4-8932 SILABOLIN STANOZOLOL STENBOLONE STENBOLONE-ACETATE TESTOSTERONE TESTOSTERONE-= GLUCURONIDE TESTOSTERONE-NICOTINATE TESTOSTERONE-SULFATE TIBOLONE TIOMESTERONE TRENBOLONE TRENBOLONE-ACETATE ZEARALANONE ZEARALENONE ZERANOL ANALEPTICS ALMITRINE AMINOPICOLINE AMIPHENAZOLE ANIBINE ASPIDOSPERMINE AZABON BEMEGRIDE BUFOGENIN CAFEDRINE CAFFEINE CAFFEINE-SODIUM-= BENZOATE

Derwent Drug File 1047 Thesaurus CAFFEINE-SODIUM-= SALICYLATE CAMPHOR CAMPHOSTYL CAMPHOTAMIDE CENTPHENAQUIN CROPROPAMIDE CROTETAMIDE DECLOXIZINE DIETHADIONE DIHYDROACTINIDIOLIDE DIMEFLINE DIMETOFRINE DIMORPHOLAMINE DOXAPRAM ENDOMIDE ETAMIVAN ETHYLNORANTIFEINE ETILEFRINE F-1459 FENMETOZOLE FOMINOBEN GALANTAMINE HEPTAMINOLACEFYLLINE HPT-430 HYDROXYAMPHETAMINE HYDROXYEPHEDRINE KOLA LEPTACLINE LOBELINE MEPIXANOX METAMFEPRAMONE NICOTINOYL-PROCAINE NIKETHAMIDE NORFENEFRINE OCTOPAMINE OSTOL PENTETRAZOL PHOLEDRINE PHTHALETHAMIDE PICROTOXIN PIMECLONE PRETHCAMIDE PROLINTANE PYROVALERONE S-9581 SAH-41-178 SOBREROL STRYCHNINE TALOXIMINE TAUREMESIN THEOBROMINE THEOBROMINE-= SALICYLATE-SODIUM THEOBROMINE-SODIUM-= ACETATE THEODRENALINE TOLDIMFOS WIN-8626 ANALGESICS 156-S 4030-W-92 66A-078 AA-2379 AA-501 AAL-13 ABBOTT-41988 ABT-594 ABT-702 ACEA-0593 ACEBURATE ACECLOFENAC ACEFURTIAMINE ACEMETACIN ACEQUINOLINE ACETANILIDE ACETIAMINE ACETORPHAN ACETORPHINE ACETYLDIHYDROCODEINE ACETYLMETHADOL ACETYLMORPHINE ACETYLMORPHINE-3 ACONITINE AD-1211 AF-2259 AG-246 AG-310 AGATOXIN-ALPHA-489 AGNUSIDE AGR-614 AH-7921 AJULEMATE ALCLOFENAC ALFENTANIL ALFETAMINE ALIMADOL ALLETORPHINE ALLYLCINCHOPHEN ALLYLNORPETHIDINE ALLYLPRODINE ALMINOPROFEN ALOXIPRIN ALPHAMEPRODINE ALPHAMETHADOL ALPHAPRODINE AM-404 AMBREIN AMINOANTIPYRINE AMINOCHLORTHENOXAZINE AMINODEOXYADENOSINE-= 5+,5+ AMINOPHENAZONE AMINOPHENAZONE = CYCLAMATE AMINOPHENAZONE-= BUTYLCHORAL-HYDRATE AMINOPICOLINE AMINOPROPYLONE ANALGEN ANAZOCINE ANIDOXIME ANILERIDINE ANILOPAM ANIROLAC ANPIRTOLINE ANTRAFENINE AP-237 APHANORPHINE APRONALIDE APYRAMIDE ARA-3000-BETA ARACHIDONYLGLYCINE-N ARVANIL ASIMADOLINE ASPIRIN ASPIRIN-LYSINE-SALT ATRASENTAN AU-8001 AY-30068 AZAPROCIN AZAPROPAZONE AZIDOMORPHINE AZIDOTHIORPHAN B-777-81 BENFOTIAMINE BENHEPAZONE BENORILATE BENOXAPROFEN BENTIAMINE BENZASAL BENZETHIDINE BENZOFUROCAINE BENZOSALIN BENZYDAMINE BENZYDAMINE SALICYLATE BENZYLMORPHINE BERMOPROFEN BETACETYLMETHADOL BETAMEPRODINE BETAMETHADOL BETAPRODINE BETOL BEZITRAMIDE BICIFADINE BIPHALIN BISBENTIAMINE BISFENAZONE BN-80933 BOA BP-2-94 BRADYZIDE BREMAZOCINE BRIFENTANIL BRL-53001A BROMADOLINE BROMAMID BROMFENAC BROMOPRIDE BROPERAMOLE BUCETIN BUCLOXATE BUCOLOME BUFEXAMAC BUFEZOLAC BUPRENORPHINE BUTACETIN BUTANIXIN BUTANOYLMORPHINE-6 BUTIBUFEN BUTOPYRAMMONIUM IODIDE BUTORPHANOL CAMPHOR CAPPORPHIN CARBAMOYLPHENOXYACETATE CARBASALATE CALCIUM CARBAZOCINE CARBIFENE CARFENTANIL CARISOPRODOL CARPERIDINE CARPROFEN CARSALAM CAUSYTH CDRI-82-205 CELECOXIB CENTCHROMANE CEP-701 CERM-10194 CERPEGIN CESEDON CETOTIAMINE CGP-29030-A CGP-44532 CH-150 CHIMAPHILIN CHINOIN-127 CHLORBICYCLEN CHLORDIMORINE CHLORPHENESIN-= CARBAMATE CHLORTHENOXAZINE CHLORZACETAMOL CHOLINE-MAGNESIUM-= TRISALICYLATE CICLOPROFEN CIHEPTOLANE CINCHOPHEN CINNAMEDRINE CINNOFURADIONE CINNOPENTAZONE

1048 APPENDIX D CIPREFADOL CIPROQUAZONE CIRAMADOL CLANTIFEN CLIDAFIDINE CLOFURAC CLOMETACIN CLONITAZENE CLONIXERIL CLONIXIN CLONIXIN-LYSINE-SALT CLORACETADOL CLOXIMATE CNS-5788 COCAINE-METHIODIDE CODEINE CODEINE-EPOXIDE COGAZOCINE COLFENAMATE CONIINE CONORFONE CORYTUBERINE CP-0494 CP-0499 CP-331 CP-55244 CP-55940 CP-56667 CRESOTAMIDE CRYOFLUORANE CYCLAZOCINE CYCLOHEXAMINE CYCLORPHAN CYCOTIAMINE D-13223 D-15917 D-16120 D-675 DA-5018 DARBUFELONE DBO-11 DBO-83 DELFANTRINE DELMETACIN DEMETHYLNEFOPAM DEMETHYLTRAMADOL-O DERMORPHIN,2-D-ARG DERMORPHIN,7-LYS DESMETHYLMORAMIDE DESOMORPHINE DETOMIDINE DEXINDOPROFEN DEXKETOPROFEN DEXPROXIBUTENE DEXTILIDINE DEXTROMORAMIDE DEXTROPROPOXYPHENE DEXTRORPHAN DEZOCINE DIACEREIN DIACETAMATE DIACETYLMORPHINE DIAMPROMIDE DIANOSIDE-A DIANOSIDE-B DIBEMETHINE DIBUPYRONE DIBUSADOL DIBUTANOYLMORPHINE DICLOFENAC DICLOFENAC HYDROXY= ETHYLPYRROLIDINE DICLONIXIN DIETHYLTHIAMBUTENE DIFENAMIZOLE DIFENPIRAMIDE DIFLUNISAL DIHYDROCAPSAICIN DIHYDROETORPHINE DIHYDROMORPHINE DIMEFADANE DIMENOXADOL DIMEPHEPTANOL DIMETHYLSULFOXIDE DIMETHYLTHIAMBUTENE DIOXAPHETYL-BUTYRATE DIPIPANONE DIPROQUALONE DIPROXADOL DISALICYLSUCCINATE DIZATRIFONE DM-235 DOXPICOMINE DRINIDENE DROTEBANOL DROXICAM DROXYPROPINE DUOMETACIN DUP-747 DYNORPHIN-1-13 DYNORPHIN-1-9 E-5110 E-6087 EDRONOCAINE EGIS-5645 EK-209 ELTENAC EM-405 EMBUTRAMIDE EMD-60400 EMORFAZONE ENALLYPROPYMAL ENDOMORPHIN-1 ENDOMORPHIN-2 ENKEPHALIN,2-D-ALA-5-= LEU-6-CYS ENKEPHALIN,2-D-ALA-5-= LEU-6-SER ENKEPHALIN-MET,6-ARG-= 7-PHE-AMIDE EPIBATIDINE EPIBOXIDINE EPIRIZOLE EPS-4032 EPTAZOCINE ES-52 ESEROLINE ESEROLINE-SALICYLATE ETERSALATE ETHENZAMIDE ETHOHEPTAZINE ETHYLKETAZOCINE ETHYLMETHYLTHIAMBUTENE ETHYLMORPHINE ETOFENAMATE ETONITAZENE ETORICOXIB ETORPHINE ETOSALAMIDE ETOXAZENE ETOXERIDINE F-1044 F-1067 F-13714 FAMPROFAZONE FECLOBUZONE FELBINAC FENACETINOL FENARIDINE FENBUFEN FENCHONE FENCLORAC FENCLOZATE FENDOSAL FENFLUMIZOLE FENOPROFEN FENTANYL FENYRAMIDOL FEPRAZONE FI-302 FK-33-824 FK-3311 FLOCTAFENINE FLOSULIDE FLUCARBRIL FLUFENISAL FLUMEXADOL FLUNIXIN FLUNIXIN MEGLUMINE FLUPIRTINE FLUPROFEN FLUPROQUAZONE FLURADOLINE FLURBIPROFEN FLURBIPROFEN-ETHYL-ESTER FLURETOFEN FOPIRTOLINE FOSFOSAL FPP-028 FR-123826 FR-140423 FR-172357 FR-64822 FS-205-397 FUMARILINE FUNALTREXAMINE-ALPHA FUNALTREXAMINE-BETA FURAPROFEN FURETHIDINE FUROFENAC FURSULTIAMINE FX-205-754 G-264 GELSEMINE GENTISATE GI-90291 GIAREG GINGEROL-6 GLAFENINE GLAUCOLIDE-A GLUCAMETACIN GP-53633 GPA-1657 GPA-1658 GR-103545 GR-190178 GR-226206 GR-38414 GR-45809 GR-86014 GR-89696 GR-91272 GR-94839 GUAIMESAL GV-196771-A GW-274150 GX-258 HAEMANTHIDINE HAI-105 HCT-3012 HEMATEIN HENNOXAZOLE-A HEXAPROFEN HISTOGRANIN HISTORPHIN HOMOLAUDANOSINE HOMPRENORPHINE HP-573 HP-736 HYDROMORPHINOL HYDROMORPHONE HYDROXYETHYLSALICYLATE

Derwent Drug File 1049 Thesaurus HYDROXYFLAVONE-7 HYDROXYPETHIDINE HYDROXYPHENYLALANINE-= BETA HYDROXYQUINOLINE= SULFONATE-PARA HYDROXYTOLUATE HYPOXOSIDE HZ-2 IBAZOCINE IBUPROFEN ARGININE IBUPROFEN LYSINE IBUPROXAM ICI-120518 ICI-197067 ICI-199441 ICI-49455 ICILIN ID-1229 IMIDAZOLE SALICYLATE IMPROGAN INCARVILLATEINE INDOPINE INDOPROFEN IODOPHENAZONE ISOFEZOLAC ISOMETHADONE ISONIXIN ISOPROFEN ISOSULFORPHANOL = PERCHLORATE ISOTETRANDRINE ISOXEPAC ISOXICAM ISPIRIN J-113397 JESACONITINE JMV-390-1 JMV-449 JTE-522 KELATORPHAN KENTSIN KETAMINE KETAZOCINE KETOBEMIDONE KETOPROFEN KETOPROFEN LYSINE KETOROLAC KT-90 KT-95 KYOTORPHIN-D L-651896 L-652343 L-689660 L-733060 L-745337 L-761066 LACTYLPHENETIDINE LANEPITANT LAS-333 LEFETAMINE LEIOCARPOSIDE LETIMIDE LEVACETYLMETHADOL LEVOMETHADONE LEVOMETHORPHAN LEVOMORAMIDE LEVONANTRADOL LEVOPHENACYLMORPHAN LEVOPROPOXYPHENE LEVORPHANOL LEXOFENAC LICOFELONE LIPOMESACONITINE LOFENTANIL LONAZOLAC LORCINADOL LOXOPROFEN LUMIRACOXIB LUPENYL-ACETATE LY-136596 LY-297802 LY-300164 LY-303870 LY-316108 LY-379268 LY-393053 M-320 M-5011 M-6007 MANOALIDE MB-432 MCN-5195 MCN-5195-11 MEDETOMIDINE MEFENAMATE MENABITAN MEPTAZINOL MESACONITINE MESECLAZONE METACETAMOL METAMFAZONE METAMIZOLE SODIUM METANIXIN METAZAMIDE METAZOCINE METETHOHEPTAZINE METHADONE METHAMILANE METHEPTAZINE METHYLDESORPHINE METHYLDIHYDROMORPHINE METHYLFENTANYL-4 METHYLFENTANYL-ALPHA METHYLHOMOEPIBATIDINE-N METHYLMEPTAZINOL-N METHYLMORPHINE-N METHYLNALOXONE-N METHYLNIPHENAZINE METHYLPHENOBARBITAL METKEFAMIDE METOFOLINE METOMIDATE METOPON METOXIBUTROPATE MIMBANE MIRFENTANIL MITRAGYNINE MITRAGYNINE-= PSEUDOINDOXYL MK-1-203 MK-1-907 MK-966 MM-218 MOFEBUTAZONE MOFEZOLAC MOL-5210 MOLINAZONE MOLINDONE MORAZONE MORNIFLUMATE MORPHERIDINE MORPHICEPTIN MORPHINE MORPHINE-EPOXIDE MORPHINE-HEXANOATE-3 MORPHINE-= MONONICOTINATE-3 MORPHINE-= MONONICOTINATE-6 MORPHINE-PROPIONATE-3 MORPHINE-SULFATE-3 MORPHINE-SULFATE-6 MORPHINONE MOXADOLEN MOXAZOCINE MP-2001 MPV-2426 MR-1268 MR-1353 MR-2033 MR-2034 MR-2096-CL MR-2261 MR-2264-CL MR-2549 MR-714 MRZ-2-576 MYFADOL MYROPHINE MZ-108 NABITAN NALBUPHINE NALBUPHINE-= ACETYLSALICYLATE-3 NALMEXONE NALORPHINE-6GLUCURONIDE NALORPHINE-6-SULFATE NALOXONAZINE NALTREXONE NALTREXONE-= METHOBROMIDE NAMOXYRATE NANTRADOL NAPROXEN NAPROXOL NARCEINE NARCOBARBITAL NARCYL NCX-701 NE-21610 NE-28345 NEFOPAM NERAMEXANE NEUROTROPIN NEXERIDINE NICAFENINE NICOMORPHINE NICOTINOYLTRYPTAMINE-N NIFENAZONE NIFLUMATE NIH-10741 NIOMETACIN NITRAQUAZONE NITROACETYLSALICYLATE NMI-377 NONIVAMIDE-ACETATE NORACYMETHADOL NORBUTORPHANOL NORCODEINE NORKETAMINE NORLEVORPHANOL NORMETAZOCINE NORMETHADONE NORMORPHINE NORMORPHINE-= GLUCURONIDE-3 NORMORPHINE-= GLUCURONIDE-6 NORPETHIDINE NORPIPANONE NOTOPTEROL NPC-18521 NPC-18688 NPC-567 NPC-573 NS-398 OCFENTANIL OCILTIDE OCTAZAMIDE

1050 APPENDIX D OHM-3295 OHM-3463 OLVANIL ONO-9902 ONO-NT-012 OPIUM OREXIN-A ORIPAVINE OT-7100 OXAPADOL OXEPINAC OXETORONE OXINDANAC OXPHENERIDINE OXYBATE SODIUM OXYCINCHOPHEN OXYCODONE OXYMORPHAZONE OXYMORPHONAZINE OXYMORPHONE PAPAVERETUM PARACETAMOL PARADOL-8 PARAPROPAMOL PARECOXIB PARSALMIDE PAXISTEROL PD-117302 PD-164387 PEMEDOLAC PENTAMORPHONE PENTAZOCINE PERISOXAL PETASIN PETHIDINATE PETHIDINE PEUDOPTEROSINE-B PHELORPHAN PHENACETIN PHENADOXONE PHENAMPROMIDE PHENAZOCINE PHENAZONE PHENCYCLIDINE PHENERIDINE PHENICARBAZIDE PHENOMORPHAN PHENOPERIDINE PHENYL-SALICYLATE PHENYLETHANOLAMINE PHETHARBITAL PHLEBODRIL PHOLCODINE PICENADOL PICOLAMINE-SALICYLATE PIFENATE PIMINODINE PINADOLINE PIPERIDOLATE PIPERYLONE PIPRAMADOL PIRFENIDONE PIRITRAMIDE PK-14068 PL-017 PRANOPROFEN PRANOSAL PRAVADOLINE PRAXADINE PREFENAMATE PRINOMIDE PROCAINE PRODILIDINE PROFADOL PROGLUMETACIN PROHEPTAZINE PROPACETAMOL PROPERIDINE PROPETAMIDE PROPIRAM PROPOXYPHENE PROPYPHENAZONE PROQUAZONE PROSULTIAMINE PROXAZOLE PROXIBARBAL PROXIBUTENE PROXIFEZONE PROXORPHAN PSEUDOPTEROSIN-A PSEUDOPTEROSIN-B PSEUDOPTEROSIN-C PSEUDOPTEROSIN-D PYRROLIFENE QUILLIFOLINE QUININE SALICYLATE R-84760 RACEMETHORPHAN RACEMORAMIDE RACEMORPHAN RB-1000 RB-101 RB-120 REMIFENTANIL RETROTHIORPHAN RHEIN RIMAZOLIUM-METILSULFATE RO-03-4661 RO-15-8081 ROFECOXIB ROHITUKINE ROHITUKINE RP-60180 RP-67580 RS-2131 RS-37619 RU-29693 RU-43526 RUVAZONE RWJ-20142 RX-336M RX-77989 RX-783030 S-12813-4 S-14080 S-16474 S-2474 S-6907 SALACETAMIDE SALAMIDACETATE SODIUM SALCOLEX SALETAMIDE SALICIN SALICYLAMIDE SALICYLATE DIETHYLAMINE SALICYLATE MORPHOLINE SALICYLATE SODIUM SALICYLATE-CHOLINE SALICYLATE-MEGLUMINE SALPROTOSIDE SALSALATE SAMERIDINE SANTALOL-ALPHA SB-227122 SC-17599 SC-236 SC-39566 SC-51089 SC-51234A SC-560 SC-58125 SCH-32615 SCH-34826 SD-62 SDZ-NKT-343 SH-254 SHOGAOL-6 SIMETRIDE SINOMENINE SK-9709 SKF-10047 SKF-26070 SNC-121 SNC-162 SNC-243-A SNF-9007 SPIROXATRINE ST-4250 STAMPYRINE STRINOLINE SUFENTANIL SULINDAC SULINDAC-SULFIDE SULPROSAL SUMACETAMOL SUPROFEN SY-6001 SYNDYPHALIN-25 SYNDYPHALIN-33 SYNDYPHALIN-49 SYNDYPHALIN-62 T-614 TA-404 TA-60 TALMETACIN TALNIFLUMATE TALOSALATE TAURINAMINOPYRIDINE TAZADOLENE TENOXICAM TETRIDAMINE TETRIPROFEN THEBACON THEBAINE THIAMINE-DISULFIDE THIOCOLCHICOSIDE THIORPHAN TIAPROFENATE TIARAMIDE TIEMONIUM IODIDE TIEMONIUM METILSULFATE TIFEMOXONE TIFLUADOM TIFURAC TILIDINE TINORIDINE TIOPINAC TIROPRAMIDE TOFETRIDINE TOLFENAMATE TOLFETRIDINE TOLMETIN-PARACETAMOL-= ESTER TOLPRONINE TOMOXIPROLE TONAZOCINE TRAMADOL TREFENTANIL TRICHLOROETHYLENE TRICLACETAMOL TRIFEZOLAC TRIMEPERIDINE TRK-820 TZI-615 U-50488 U-50488E U-50488H U-53455E U-63640 UM-1250 UM-747 UP-20232

Derwent Drug File 1051 Thesaurus UP-20256 UPF-523 V-33 VALDECOXIB VAPREOTIDE VERILOPAM VIMINOL VINTIAMOL VOLAZOCINE WIN-42610 WIN-55212 WIN-55212-2 WY-41770 XC-386 XORPHANOL XYLAZINE XYLOPROPAMINE Y-23023 ZICONOTIDE ZK-48491 ZOLIPROFEN ZOMEPIRAC ANALYSIS AMPEROMETRY BIOASSAY CALORIMETRY CONDUCTIMETRY COULOMETRY DTA ELISA EMIT ENZYME-IMMUNODET. ENZYME-RECEPTOR-DET. FLUORIMETRY FLUORIMETRY fpia GONOZYME GRAVIMETRY IMMUNODET. NEPHELOMETRY OSMOMETRY PETINIA PHOTOMETRY POTENTIOMETRY RADIOENZYME-DET. RADIOENZYME-IMMUNODET. RADIOIMMUNODET. RADIORECEPTOR-DET. THERMAL-ANALYSIS THERMOGRAVIMETRY TITRATION ANAPHYLAXIS MAZZOTTI-REACTION ANDROGEN-ANTAGONISTS ABIRATERONE AS-601811 AS-602240 BENORTERONE BICALUTAMIDE CB-7630 CB-7645 CHLOROPHORIN CIOTERONEL CURBICIN CYPROTERONE CYPROTERONE-ACETATE DELANTERONE DELMADINONE DELMADINONE-ACETATE DUTASTERIDE EB-40 ETHOCYN FINASTERIDE FK-143 FLUTAMIDE GG-745 GYKI-24479 HYDROXYCYPROTERONE-= ACETATE-15-BETA KF-20405 L-39 L-636028 L-651580 L-733692 LY-191704 LY-266111 LY-300502 LY-300503 MDL-18341 METOGEST MK-0963 MK-316 MK-386 MK-434 NILUTAMIDE NORDINONE NORETHISTERONE-= ENANTHATE OXENDOLONE PINOBANKSIN PROPYLTESTOSTERONE-17-= ALPHA R-2956 RO-2-7239 RO-5-2537 RU-38882 RU-56187 RU-58841 SCH-16423 SHL-434A SKF-105657 SKF-22340 TOPTERONE TRILOSTANE TZP-4238 VN-85-1 VN-87-1 WS-9659A WS-9659B WS-9761-A WS-9761-B ZANOTERONE ZK-136799 ZK-30595 ANDROGENS 20-AET-1 8354 8356 ADRENOSTERONE ANDROSTANEDIOL ANDROSTANEDIONE ANDROSTANOLONE ANDROSTANOLONE-5-BETA ANDROSTANOLONE-= BENZOATE ANDROSTANOLONE-= HEPTANOATE ANDROSTANOLONE-= PROPIONATE ANDROSTENEDIOL ANDROSTENEDIOL-= DIPROPIONATE ANDROSTENEDIONE ANDROSTENONE ANDROSTERONE BROMOEPIANDROSTERONE-= 16-ALPHA CLOXOTESTOSTERONE CLOXOTESTOSTERONE-= ACETATE DROSTANOLONE DROSTANOLONE-PROPIONATE EPIANDROSTERONE EPITESTOSTERONE EPITIOSTANOL ETIOCHOLANEDIONE ETIOCHOLANOLONE ETIOCHOLANOLONE-BETA-3 FLUOXYMESTERONE HYDROXYSTENOZOLE MESABOLONE MESTANOLONE MESTEROLONE METHANDRIOL METHYLTESTOSTERONE MIBOLERONE NBO-6 NORANDROSTENEDIONE-19 OXYMETHOLONE PENMESTEROL PRASTERONE PRASTERONE-ACETATE PRASTERONE-ENANTHATE PRASTERONE-SULFATE SC-12790 SILABOLIN SILANDRONE TESTOSTERONE TESTOSTERONE-ACETATE TESTOSTERONE-BENZOATE TESTOSTERONE-= CYCLOHEXANOATE TESTOSTERONE-= CYCLOHEXYLPROPIONATE TESTOSTERONE-CYPIONATE TESTOSTERONE-DECANOATE TESTOSTERONE-ENANTHATE TESTOSTERONE-= GLUCURONIDE TESTOSTERONE-= HEXAHYDROBENZYL-= CARBONATE TESTOSTERONE-= ISOBUTYRATE TESTOSTERONE-= ISOCAPROATE TESTOSTERONE-= KETOLAURATE TESTOSTERONE-= PHENYLACETATE TESTOSTERONE-= PHENYLPROPIONATE TESTOSTERONE-PROPIONATE TESTOSTERONE-SUCCINATE TESTOSTERONE-SULFATE TESTOSTERONE-= UNDECANOATE TESTOSTERONE-= UNDECENOATE TESTOSTERONE-= UNDECYLENATE TESTOSTERONE-VALERATE TRESTOLONE TRESTOLONE-ACETATE U-13851 U-30684A ANEMIA AGNOGENIC-MYELOID-= METAPLASIA asymptomatic-thalassemia COMLY-SYNDROME CROSBY-SYNDROME DANA-SYNDROME ECKLIN-SYNDROME ELLIPTOCYTOSIS ERYTHROBLASTOPENIA FANCONI-PETRASSI-= SYNDROME GASSER-KARRER-SYNDROME GERBASI-SYNDROME HEM.ANEMIA-SYNDROME

1052 APPENDIX D HEMOGLOBINOPATHY HEMOLYTIC-DISEASE-OF-= NEONATE HEMOLYTIC-UREMIC-= SYNDROME HYPOCHROMASIA IMERSLUND-GRASBECK-= SYNDROME marchiafava-micheli-= syndrome MOSCHOWITZ-SYNDROME paroxysmal-nocturnal-= hemoglobinuria PLUMMER-VINSON-= SYNDROME rietti-greffi-micheli-syndrome RUNDLES-FALLS-SYNDROME SCHISTOCYTOSIS SIDEROPENIA silvestroni-bianco-syndrome SPHEROCYTOSIS STRANSKY-REGALA-= SYNDROME THALASSEMIA thalassemia-minor ZUELZER-KAPLAN-= SYNDROME ZUELZER-OGDEN-SYNDROME ANGIOGENESIS-INHIBITORS ABT-510 ABT-526 ACHARAN-SULFATE AE-941 AGM-1470 ANGINEX ANGIOSTATIN ANGIOZYME ANTITHROMBIN-LATENT AW-464 BATIMASTAT BAY-12-9566 BEVACIZUMAB BLEOMYCIN BMS-275291 BORRELIDIN BUFALIN CALCITRIOL CAPTOPRIL CC-5013 CEP-5214 CGP-53716 CLOMIFENE CM-101 COLECALCIFEROL COMBRESTATIN-A4-= PHOSPHATE COMBRETASTATIN-A-4 CP-547632 DC-101 DEAZAXANTHINE-7 DECORIN DEPUDECIN DICLOFENAC DIHYDROXYFLAVONE-3+,4+ DOXYCYCLINE DS-4152 EMD-121974 EMD-66203 ENDOSTATIN-HUMAN ENDOSTATIN-MOUSE ER-68203-00 EVEROLIMUS FR-118487 FULVESTRANT FUMAGILLIN HEPATOCYTE-GROWTH-= FACTOR-NK4 HRK-055512 HRK-429 HYDROXYCINNAM= ALDEHYDE-2+ ICI-164384 IDN-5390 IM-862 INTERFERON-ALPHA INTERFERON-BETA IRSOGLADINE ISOSORBIDE-DINITRATE ISOSORBIDE-MONONITRATE ISOTRETINOIN KR-31372 LACTOFERRIN-CATTLE LAF-389 LAVENDUSTIN-A LM-609 LY-317615 MASPIN METHOXYCINNAM= ALDEHYDE-ORTHO METHOXYESTRADIOL-2 METHYLSELENOL MINOCYCLINE MMI-166 MOTUPORAMINE-C NAFOXIDINE NF-326 OCTREOTIDE OVALICIN OXI-4503 PD-173074 PEX PI-88 PIGMENT-EPITHELIUM-= DERIVED-FACTOR PKI-166 PNU-145156-E RAZOXANE RETINAL RETINOL RO-28-2653 RO-31-7453 ROQUINIMEX S-137 SCH-66336 SEMAXANIB SJ-749 SOMATOMEDIN-C-BINDING-= PROTEIN-3 SPIRONOLACTONE ST-1646 SU-6668 SULINDAC SURAMIN TAMOXIFEN THALIDOMIDE TOCOPHEROL-ALPHA TRANILAST TRAPYMINE TRETINOIN TUMSTATIN TZ-93 TZT-1027 UROKINASE VAPREOTIDE VATALANIB VINCRISTINE VINFLUNINE WX-360 XR-5967 YLL-224 ZD-4190 ZD-6126 ANGIOGENESIS-STIMULATORS MCI-154 ANGIOTENSIN-2-ANTAGONISTS 606-A ABBOTT-81282 BAY-10-6734 BIBS-222 BIBS-39 CANDESARTAN CANDESARTAN-CILEXETIL CGP-42112A CL-329167 CP-191166 DUP-532 EPROSARTAN EXP-3174 EXP-3312 EXP-3892 EXP-597 EXP-6155 EXP-6159 EXP-6803 EXP-7711 EXP-9270 FK-739 GR-117289 GR-138950-C HN-65021 HR-720 ICI-D-6888 IRBESARTAN KT-3-671 L-158809 L-159913 L-162223 L-162313 L-162389 L-163017 L-163491 LOSARTAN LR-B-081 LY-301875 ME-3221 MK-996 OLMESARTAN-MEDOXOMIL PD-123177 PD-123319 RNH-6270 S-8307 S-8308 SARALASIN SARILESIN SARLEUSIN SARMESIN SARTHRAN SC-51316 TA-606 TAK-536 TH-142177 U-97018 UR-7280 WK-1492 WL-19 ANGIOTENSIN-AGONISTS ANGIOTENSIN ANGIOTENSIN-1 ANGIOTENSIN-1-7 ANGIOTENSIN-1-CATTLE ANGIOTENSIN-1-HORSE ANGIOTENSIN-1-SAR-1 ANGIOTENSIN-2 ANGIOTENSIN-2-(1-6) ANGIOTENSIN-2-(3-7) ANGIOTENSIN-2-CATTLE ANGIOTENSIN-2-DE-ASP-= 1,DE-ARG-2 ANGIOTENSIN-2-HORSE

Derwent Drug File 1053 Thesaurus ANGIOTENSIN-2-SAR-1 ANGIOTENSIN-3 ANGIOTENSIN-3-CATTLE ANGIOTENSIN-3-HORSE ANGIOTENSINAMIDE L-163491 RENIN-SUBSTRATE-= TETRADECAPEPTIDE (Drug) ANGIOTENSIN-ANTAGONIST ACE-INHIBITOR ANGIOTENSIN-2-ANTAGONIST RENIN-INHIBITOR ANGIOTENSIN-ANTAGONISTS 351-A 606-A A-58365A A-58365B A-65317 A-68064 A-72517 A-74273 A-779 A-81988 AB-47 ABBOTT-81282 ACE-INHIBITORS ALACEPRIL ALATRIOPRIL ALISMOL ALTIOPRIL CALCIUM ANCOVENIN ANGIOTENSIN-2-= ANTAGONISTS ANGIOTENSIN-3,ILE-7 ARFALASIN BAY-10-6734 BAY-O-6997 BAY-Q-1313 BENAZEPRIL BENAZEPRILAT BENZOYLCAPTOPRIL BIBS-222 BIBS-39 BILA-2157-BS BMS-180560 BMS-182657 BMS-183920 BMS-184698 BPP-9A BRL-36378 BW-A575C BW-B385C CANDESARTAN CANDESARTAN-CILEXETIL CANDOXATRIL CAPTOPRIL CAPTOPRIL-CYSTEINE CAPTOPRIL-DISULFIDE CAPTOPRIL-GLUTATHIONE CERONAPRIL CGP-29287 CGP-38560 CGP-38560A CGP-42112A CGP-42112B CGP-44099A CGS-13928C CGS-28106 CGS-30440 CI-925 CI-996 CILAZAPRIL CILAZAPRILAT CL-242817 CL-329167 CONVERSTATIN CP-191166 CP-71362 CP-80794 CV-11194 CV-5975 CYCLOTHIAZOMYCIN DEACETYLALACEPRIL DELAPRIL DELAPRIL-DIACID DITEKIREN DMP-581 DMP-811 DU-1227 DU-1777 DUP-532 E-4177 EMD-56133 ENALAPRIL ENALAPRILAT ENALKIREN EPICAPTOPRIL EPROSARTAN ER-32935 ES-1005 ES-295 ES-300 ES-305 ES-313 ES-316 ES-317 ES-6864 ES-8891 EU-4867 EU-5476 EX-89 EXP-063 EXP-132 EXP-3174 EXP-3312 EXP-3892 EXP-597 EXP-6155 EXP-6159 EXP-6803 EXP-7711 EXP-9270 FK-739 FK-906 FOROXYMITHINE FOSINOPRIL FOSINOPRILAT GA-0056 GEMOPATRILAT GR-117289 GR-117289-C GR-138950 GR-138950-C H-113 H-256 H-261 H-76 HEMORPHIN-4 HN-65021 HOE-065 HOE-288 HR-720 ICI-D-6888 ICI-D-8731 IDRAPRIL IMIDAPRIL IMIDAPRILAT INDOLAPRIL INDOLAPRILAT IRBESARTAN JTP-2724 K-13 KR-30988 KR-31372 KRH-594 KRI-1177 KRI-1314 KT-3-671 KT-3-671 L-155212 L-158338 L-158809 L-159689 L-159913 L-161177 L-162223 L-162313 L-162389 L-162441 L-163017 L-163491 L-681176 LABEDIPINEDILOL-A LACTORPHIN-ALPHA LACTORPHIN-BETA LIBENZAPRIL LISINOPRIL LOSARTAN LR-B-057 LR-B-081 LY-301875 LYCIUMIN-A LYCIUMIN-B MDL-100173 MDL-100240 MDL-27088 MDL-27210 ME-3221 METIAPRIL METIOPRIL MIXANPRIL MK-351A MK-954 MK-996 MOEXIPRIL MOEXIPRILAT MURACEIN-A MURACEIN-B MURACEIN-C NITROSOCAPTOPRIL-S OLMESARTAN-MEDOXOMIL OMAPATRILAT PD-123177 PD-123319 PD-132002 PD-134672 PD-98059 PENTOPRIL PENTOPRILAT PERINDOPRIL PERINDOPRILAT PHENACEIN PIVOPRIL POMISARTAN PROCYANIDIN-B2-DIGALLATE QUINAPRIL QUINAPRILAT RAMIPRIL RAMIPRILAT RB-105 RENIN-INHIBITORS RENTIAPRIL REV-6207 RHC-3454 RNH-6270 RO-31-8472 RO-42-5892 RWJ-46458 S-2864 S-8307

1054 APPENDIX D S-8308 SA-291 SA-7090 SARALASIN SARILESIN SARLEUSIN SARMESIN SARTHRAN SB-203220 SC-45075 SC-46507 SC-46944 SC-51316 SC-52458 SC-54628 SC-54629 SCH-54470 SCRIP SPIRAPRIL SPIRAPRILAT SPP-100 SQ-13297 SQ-13863 SQ-14102 SQ-14551 SQ-20475 SQ-20661 SQ-20718 SQ-20858 SQ-20859 SQ-20861 SQ-27786 SQ-28370 SQ-33800 SR-42128 SR-42128A SR-43845 TA-606 TAK-536 TELMISARTAN TEMOCAPRIL TEMOCAPRILAT TEPROTIDE TH-142177 TRANDOLAPRIL TRANDOLAPRILAT U-62168-E U-62168E U-71909E U-72407-E U-72407E U-72408-E U-72408E U-72409-E U-72409E U-73777-E U-77451-E U-77451E U-77455-E U-77646-E U-77646E U-77647E U-80215-E U-80215E U-97018 UP-269-6 UR-7280 UTIBAPRIL VALSARTAN WAY-126227 WF-10129 WK-1492 WL-19 WY-44221 XR-510 YM-21095 YM-358 YS-980 Z-13752-A ZABICIPRIL ZABICIPRILAT ZD-7155 ZOFENOPRIL ZOFENOPRILAT ZOFENOPRILAT-ARGININE-= SALT ANGIOTENSIN-RECEPTOR ANGIOTENSIN-2-RECEPTOR ANIMAL-BEHAVIOR AVOIDANCE CLIMBING CONDITIONED-AVOIDANCE CONDITIONED-REFLEX DISCRIMINATION GNAWING GROOMING HEAD-SHAKE HEAD-TURNING HEAD-TWITCHING IMPRINTING JUMPING MATING MURICIDAL REARING SELF-STIMULATION SHAM-RAGE SNIFFING STARTLE-REFLEX STEREOTYPY WET-DOG-SHAKE ANIMAL-NEOPLASM 9L-GLIOSARCOMA B16-MELANOMA CC531 CENTROCYTOMA CG-GLIOMA CLOUDMAN-MELANOMA CT26 DUNNING-R3327H EB-LYMPHOMA EHRLICH-ASCITES ERYTHROLEUKOSIS ESB-LYMPHOMA FRIEND-LEUKEMIA GROSS-LEUKEMIA HARDING-PASSEY-= MELANOMA HCT116 IMMUNOBLASTOMA KIRKMAN-ROBBINS-= HEPATOMA L1210 L40 L5222 leukemia,bovine LEUKOSIS LEUKOSIS-COMPLEX LEWIS-LUNG-CARCINOMA LIPOMYXOSARCOMA M5076-SARCOMA mareks-disease mareks-disease MBL2-ASCITES MELANOMA METH-A MORRIS-HEPATOMA NEMETH-KELLNER-= LYMPHOMA NOVIKOFF-HEPATOMA P1798 P388 P815 P815Y PULMONARY-= ADENOMATOSIS RIF1 SARCOMA-180 SARCOMA-37 SARCOMA-45 SOMATOLIBERINOMA TLX5 WALKER-256-= ADENOCARCINOMA YOSHIDA-ASCITES YOSHIDA-SARCOMA ANORECTICS 1229-U-91 ACRIDOREX AMFECLORAL AMFEPENTOREX AMFEPRAMONE AMINOREX AMLINTIDE ANISACRIL AO-124 ARL-15849-XX AY-14948 AY-18672 AY-20213 AY-20214 BENFLUOREX BENZPHETAMINE BISPHENOL-A-DIGLYCIDYL-= ETHER BMS-210285 BRL-26830-A BRL-26830A BRL-35135A BUTABINDIDE CGP-71683-A CHLOROCITRATE-THREO CHLORPHENTERMINE CL-316243 CLOBENZOREX CLOFOREX CLOMINOREX CLORTERMINE CM-57373 CP-114271 CP-94253 CROTONOLACTONE DEETHYLAMFEPRAMONE DEXAMPHETAMINE DEXFENFLURAMINE DIFEMETOREX ENTEROSTATIN ETILAMFETAMINE ETIOCHOLANEDIONE ETOLOREX FENBUTRAZATE FENFLURAMINE FENISOREX FENPROPOREX FLUCETOREX FLUDOREX FLUMINOREX FLUTIOREX FORMETOREX FURFENOREX GUANIDINOPROPIONATE-3 GW-5823 GYKI-13380 HYDROXYPHENTERMINE ICI-198157 ICI-D-7114 INDANOREX J-104870 JPC-6036 L-783281 L-796568

Derwent Drug File 1055 Thesaurus LEVOFACETOPERANE LY-106737 LY-117413 LY-377604 LY-79771 LY-88329 MAZINDOL MEFENOREX METAMFEPRAMONE METHAMPHETAMINE METHYLAMPHETAMINE-PARA MK-212 MORFOREX MSI-1436 NN-2211 NORDEXFENFLURAMINE NORFENFLURAMINE NORPSEUDOEPHEDRINE ORTETAMINE OXIFENTOREX PENTOREX PHENATINE PHENDIMETRAZINE PHENMETRAZINE PHENTERMINE PICILOREX PM-170 PN-2034 PROPYLHEXEDRINE RO-16-8714 RO-22-0654 RO-23-7637 S-422 SATIETIN SB-334867 SELEGILINE SETAZINDOL SHU-9119 SKF-L-39728-A TIFLOREX U-16178F ANTACIDS ACEGLUTAMIDE-ALUMINUM ALCLOXA ALDIOXA ALEXITOL SODIUM ALGELDRATE ALMADRATE-SULFATE ALMAGATE ALMAGCIT ALMASILATE ALUMINUM-CARBONATE ALUMINUM-GLYCINATE ALUMINUM-HYDROXIDE ALUMINUM-HYDROXY= CARBONATE ALUMINUM-PHOSPHATE ALUMINUM-SILICATE ALUSULF ATTAPULGITE BISMUTH-ALUMINATE BISMUTH-SUBCARBONATE BISMUTH-SUBNITRATE CALCIUM-HYDROXIDE CHLOROCAMPHAMIDE CMN-131 DE-NOL DIHYDROXYALUMINUM-= AMINOACETATE DIHYDROXYALUMINUM-= SODIUM-CARBONATE DQ-2511 GLUCALDRATE POTASSIUM GLUCALOX H-81-75 HYDROTALCITE MAALOXAN MAGALDRATE MAGNESIUM-ALUMINUM-= HYDROXIDE MAGNESIUM-ALUMINUM-= SILICATE MAGNESIUM-CARBONATE MAGNESIUM-HYDROXIDE MAGNESIUM-OXIDE MAGNESIUM-TRISILICATE POLYETADENE RANITIDINE-BISMUTH-= CITRATE SACCHARATE CALCIUM SODIUM-ALUMINOSILICATE SUCRALFATE SUCRALOX TROMETAMOL ANTHELMINTICS 153C51 72-70 ABAMECTIN ACRANIL ACRISORCIN ALAZANINE TRICLOFENATE ALBENDAZOLE ALBENDAZOLE-2-AMINO-= SULFONE ALBENDAZOLE-SULFOXIDE ALDICARB ALLOKAINATE-ALPHA ALLOSAMIDIN AMIDANTEL AMINOLEVAMISOLE-META AMOCARZINE AMOSCANATE AMPHOTALIDE ANTAFENITE ANTAZONITE ANTELMYCIN ANTHELVENCIN-A ANTHIOLIMINE ANTIENITE ANTIMONY-SODIUM-= TARTRATE ARECOLINE ASCARIDOLE ASPEROSIDE AVERMECTIN AVERMECTIN-A1A AVERMECTIN-A1B AVERMECTIN-A2A AVERMECTIN-A2B AVERMECTIN-B1A AVERMECTIN-B1A-EPI-13 AVERMECTIN-B1B AVERMECTIN-B2A AVERMECTIN-B2A-EPI-13 AVERMECTIN-B2B AVERMECTIN-H2B1B AZACOPROSTANE-25 AZADIRACHTIN BAC.THURINGIENSIS BECANTONE BEMOSAT BENACYL BENGAMIDE-A BENGAMIDE-B BENGAMIDE-C BENGAZOLE-A BENGAZOLE-B BEPHENIUM HYDROXY= NAPHTHOATE BIDIMAZIUM IODIDE BILHARCID BISBENDAZOLE BITHIONOLOXIDE BITOSCANATE BMK BROMOPHENOPHOS BROMOXANIDE BROTIANIDE BUNAMIDINE BUNAMIDINE HYDROXY= NAPHTHOATE BUTAMISOLE BUTONATE BUTYNORATE BW-61-435 BW-A-728C CAMBENDAZOLE CARBANTEL CARBENDAZIME CARDOL CDRI-77-6 CDRI-81-470 CDRI-82-437 CENTPERAZINE CETOVEX CGI-16343 CGI-17658 CGI-18041 CGP-13231 CGP-20308 CGP-20309 CGP-20376 CGP-20909 CGP-21306 CGP-21833 CGP-21835 CGP-23518 CGP-24589 CGP-26702 CGP-8065 CHERIMOLINE CICLOBENDAZOLE CLIOXANIDE CLONOSTACHYDIOL CLORSULON CLOSANTEL COLISTIN-A COSTUNOLIDE COUMAFOS CRUFOMATE CUCURBITINE CYACETACIDE CYMENE DAZOMET DBCP DESASPIDIN DESTOMYCIN-A DEXAMISOLE DIAMFENETIDE DICHLOROPHEN DICHLORVOS DIETHYLCARBAMAZINE DIETHYLCARBAMAZINE-N-= OXIDE DIMANTINE DIPHENAN DIPHEZYL DISOPHENOL DITHIAZANINE IODIDE DIUREDOSAN DOMOATE DORAMECTIN DROCARBIL EL-979 EMBELIN EMODEPSIDE EPSIPRANTEL EREMANTHINE ETHULIACOUMARIN-A ETHYL-CHLOROOXANILATE-= PARA

1056 APPENDIX D ETHYL-OXANILATE ETHYLENE-DIBROMIDE EUCALYPTOL FAMPHUR FEBANTEL FENBENDAZOLE FENIODIUM CHLORIDE FENSULFOTHION FKH-10 FLUBENDAZOLE FLURANTEL FOSPIRATE FTALOFYNE FURAPROMIDIUM FURAPYRIMIDONE FURODAZOLE G-1026 G-1460 G-185 G-476 G-545 G-937 GALOSFEN GAMMA-BHC GERANIOL GLYCARSAMATE SODIUM HALOXON HEDAQUINIUM CHLORIDE HEDERASAPONIN-B HEDERASAPONIN-C HEDERIN-ALPHA HELENIN HETOLIN HEXACHLOROETHANE HEXACHLOROPHENE HEXACHLORXYLOL HEXYLRESORCINOL HOE-S616 HOE-S688 HYCANTHONE HYDROXYMEBENDAZOLE HYDROXYVERNOLIDE HYGROMYCIN-B IA-3 IA-4 IA-5 IA-6 IMCARBOFOS IVERMECTIN IVERMECTIN-I IVERMECTIN-II JASPAMIDE JASPLAKINOLIDE JIETACIN-A JIETACIN-B KAINATE KALIHINOL-X KALIHINOL-Y KALIHINOL-Z KAMALA L-155175 L-631529 LACHNUMON-B1 LACHNUMON-B2 LEAD-ARSENATE LEUCANICIDIN LEVAMISOLE LL-F28249-BETA LL-F28249-GAMMA LL-F28249-LAMBDA LOBENDAZOLE LUCANTHONE LUXABENDAZOLE M-254 MALABARICONE-C MALACHITE-GREEN MEBENDAZOLE MEDAMINE MEL-AM MEL-GA MEL-GR MEL-NI MELARSOMINE METHYLROSANILINIUM = CHLORIDE METRIFONATE METYRIDINE MILBEMYCIN-A MILBEMYCIN-ALPHA-3 MILBEMYCIN-B-41D MILBEMYCIN-BETA-1 MILBEMYCIN-BETA-3 MILBEMYCIN-D MILBEMYCIN-E MILBEMYCIN-G MILBEMYCIN-OXIME MILBEMYCIN-OXIME-D MIRASAN MORANTEL MOXIDECTIN MURISOLIN MYCORRHIZIN-B1 MYCORRHIZIN-B2 NAFTALOFOS NEMADECTIN NEOAUREOTHIN NETOBIMIN NICLOFOLAN NICLOSAMIDE NICLOSAMIDE OLAMINE NICLOSAMIDE PIPERAZINE NIRIDAZOLE NITAZOXANIDE NITRAMISOLE NITRODAN NITROSCANATE NITROXINIL NOCODAZOLE OLTIPRAZ ONTIANIL OXAMNIQUINE OXANTEL OXFENDAZOLE OXIBENDAZOLE OXINIDE OXYCLOZANIDE P-903 PAPYRACON-A PAPYRACON-B PAPYRACON-C PARAHERQUAMIDE PARAHERQUAMIDE-B PARAHERQUAMIDE-C PARAHERQUAMIDE-D PARAHERQUAMIDE-E PARAHERQUAMIDE-F PARAHERQUAMIDE-G PARAROSANILINE EMBONATE PARBENDAZOLE PEXANTEL PF-1022A PHENACIZOLE PHENALIDONE PHENIODOL SODIUM PHENOSMOLIN PHENOTHIAZINE (Drug) PHENZIDOLE PHOXIM PIBENZIMOL PIERICIDIN-A PIPERAMIDE PIPERAZINE PLAKINIDINE-A PLAKINIDINE-B PLIZON PRAZIQUANTEL PRETAMAZIUM IODIDE PROFENOFOS PROPHOS PSORALEN PYRACLOFOS PYRANTEL PYRVINIUM CHLORIDE PYRVINIUM-EMBONATE RAFENDAZOLE RAFOXANIDE RALTITREXED RD-12869 RESORANTEL RO-11-3128 RO-15-5458 SALANTEL SANSHOOL-ALPHA SANTONIN SCH-18099 SELAMECTIN SPIRAZINE SPORANDOL SQ-18506 SQUAMOCIN STIBOCAPTATE SODIUM STIBOPHEN STILBAZIUM IODIDE STYRYLPYRIDINIUM SUBENDAZOLE SURAMIN SURAMIN SODIUM TARTAR-EMETIC TEGALID TEROXALENE TETRA TETRACHLOROETHYLENE TETRAMISOLE THENIUM CLOSILATE THIARUBRINE-A THIOFURADENE THIOPHANATE THIOPHANATE-METHYL THYSANOX TIABENDAZOLE TICARBODINE TIOXIDAZOLE TOLTRAZURIL TOOSENDANIN TRIBROMSALAN TRICLABENDAZOLE TRICLABENDAZOLE-= SULFOXIDE TRICLOFENOL-PIPERAZINE U-87407 U-88509 UK-3883 UMF-078 UMF-289 UREDOFOS VERNOLIDE VINCOFOS VM-44857 VM-44864 VM-44865 VM-44866 VUFB-14170 VUFB-15269 WR-129577 WR-175412 WR-190420 WR-251993 ZILANTEL ANTIAGGREGANTS 3178-AQ 48740-RP

Derwent Drug File 1057 Thesaurus 59227-RP ABCIXIMAB ABT-299 ACADESINE ACETYLEUGENOL ACTIVATED-PROTEIN-C-= HUMAN AFP-03 AG-34 AG-81 AGLAFOLINE AH-23848 AH-23848B AH-P-719 AJOENE ALBOLABRIN AMENTOFLAVONE-= HEXAACETATE AN-162 ANAGRELIDE ANEMARRHENASAPONIN-I ANEMARRHENASAPONIN-IA ANGELITRIOL ANGELOL-B ANGELOL-K ANISE-ALCOHOL ANTIARRHYTHMIC-PEPTIDE ANTITHROMBIN-III APAFANT APPLAGGIN APYRASE AQ-11 AR-12-456 ARC-69931-MX ARTOBILOXANTHONE AS-013 ASPALATONE ASPIRIN ASPIRIN ALUMINUM AT-1015 ATRINOSITOL AU-8001 AVELIZINE BARBOURIN BATROXOSTATIN BAY-U-3405 BCH-2763 BECLOBRIC-ACID BENZENESULFOHYDROXAMATE BENZOFENAC BERAPROST BG-8865 BIBU-104 BIBU-104-XX BIBU-52 BISCOUMACETATE-ETHYL BITISTATIN BL-3459 BM-14515 BM-500 BM-519 BM-531 BM-567 BM-573 BMS-180742 BMY-20844 BMY-21638 BMY-42393 BMY-43351 BMY-45778 BN-50341 BN-50726 BN-54062 BOTHROJARACIN BPAT-117 BPAT-143 BREVISCAPINE BROSIMONE-I BX-807834 C-18665 C-68-22 C-780698 C-801239 C-85 C-894095 C-894144 C-921-78 CCI-17810 CCT-62 CGS-22652 CH-102 CHF-2206 CILOSTAMIDE CILOSTAZOL CINNAMOPHILIN CIS-19 CK-53 CL-184005 CL-871502 CLOFIBRATE CLOFIBRATE CALCIUM CLOPIDOGREL CLORICROMEN COD-LIVER-OIL COLLAGEN-DERIVED-= OCTAPEPTIDE COLLININ CONFUSAMELINE CONIFERYL-ALCOHOL CRC-220 CREOSOTE CRL-42796 CS-747 CV-3988 CYCLOARTOMUNIN CYCLOCOMMUNOL CYCLOMORUSIN CYCLOMULBERRIN CYCLOTHEONAMIDE-A CYCLOTHEONAMIDE-B D-003 DAISAIKOTO DALTROBAN DANAPAROID SODIUM DAZMEGREL DAZOXIBEN DEFIBRINOTIDE DEMETHOXYANGONIN DEMETHOXYYANGONIN DH-6471 DIALLYL-TRISULFIDE DICRANIN DIHYDROISOCYCLOARTOMUNIN DIPETALIN DIPYRIDAMOLE DITAZOLE DIZATRIFONE DMP-754 DMP-757 DN-9693 DOCOSAHEXAENOATE-= ETHYL-ESTER DOMOXIN DT-TX-30 DT-TX-30-SE E-456 E-5510 ECHICETIN ECHISTATIN ECHISTATIN-GAMMA ELAROFIBAN ELEGANTIN EMD-122347 ENDOTHELIN-3 EP-092 EPIYANGAMBIN EPTIFIBATIDE ERISTOSTATIN ESTRAGOLE EVOLITRINE FAGARINE-GAMMA FCE-22178 FCE-27262 FK-409 FK-633 FLAVOCRISTAMIDE-B FLAVORIDIN FLUFOSAL FLUINDIONE FLUMIZOLE FLUOROADENOSINE-2 FLURBIPROFEN-NITROXY= BUTYLESTER FLURETOFEN FPL-66096 FPL-67085 FR-122047 FR-144420 FR-167653 FR-171113 FR-189419 FR-900359 FRAXINOL FRENOLICIN-B FUREGRELATE FUROFENAC G-25671 G-31442 G-33378 G-4120 G-619 G-6191 G-6249 G-6788 GALBANATE GANODERMATE-S GEA-3175 GINKGOLIDE-A GINKGOLIDE-B GINKGOLIDE-C GL-522 GLAUCOCALYXIN-A GR-144053 GR-36246 GT-12 HALYSIN HAPLOPINE HCL-31-D HELICHRYSETIN HEPE-12 HERNOVINE HFV-1017-C HIRUDIN-54-65 HISPANOLONE HMR-1794 HN-11500 HOLOTHURIANGLYCOSAMINOGLYCAN HPETE-12 HPETE-15 HUAJIAOSIMULINE IBI-P-05006 IFETROBAN INDOBUFEN INDOMETACIN-FARNESIL IQ-3-B ISOPSYCHOTRIDINE-C ISOTORACHRYSONE ITAZIGREL KB-3022 KBT-3022 KC-764

1058 APPENDIX D KDI-792 KF-4939 KISTRIN KME-4 KO-286011 KOKUSAGININE KP-10614 KT-2-962 KW-3635 L-367073 L-370518 L-372460 L-636499 L-640035 L-652343 L-652731 L-680573 L-703014 L-709780 L-734217 L-738167 L-762745 L-767685 LACHNUMON-B2 LCB-2853 LEECH-ANTIPLATELET-= PROTEIN LF-1351 LFM-A-13 LG-82-4-00 LG-82-4-01 LICOFELONE LINOTROBAN LIXAZINONE LOTRAFIBAN LU-58463 LY-214138 LY-806303 MARCHANTIQUINONE MB-3 ME-3229 ME-3277 MEDERMYCIN MELAGATRAN MELITERNATIN METHOXYCYPRO= HEPTADINE-3 METHYLACTINODAPHNINE-N METHYLBULBOCAPNINE-O MIDAZOGREL MILTIRONE MK-0852 MM-706 MOFEZOLAC MOLLUGIN MONAMIDOCIN MOPIDAMOLE MOTAPIZONE MY-5445 MYCORRHIZIN-B1 MYCORRHIZIN-B2 MYOINOSITOL-= TRIPHOSPHATE-1,2,6 MYRTOCYAN NAFAZATROM NAROPARCIL NCX-4016 NCX-4215 NITROACETYLSALICYLATE NITROSOHOMOCYSTEINE-S NORATHYRIOL NQ-Y-15 NSL-9403 OKY-1580 OKY-1581 OLIGVON ON-579 ONO-11120 ONO-1301 ONO-8809 ONO-AE-1-329 ONO-AP-227 ONO-AP-437 OPC-13135 OPC-33509 OPC-3911 ORBOFIBAN OROXYLIN-A OXAGRELATE OZAGREL P-280 PADMA-28 PAEONOL PALLIDIPIN PAPYRACON-A PCA-4230 PENTOXIFYLLINE PEROXYNITRITE PHOMACTIN-D PHOSPHOLIPASE-C PI-091 PI-201 PICOTAMIDE PIMILPROST PIRACETAM PIRMAGREL PIRSIDOMINE PLAFIBRIDE PODORHIZOL POLYDATIN PREDICENTRINE PS-028 PSEUDOSEMIGLABRIN PSYCHOTRIDINE PTERYXINE PUNICATE QUADRIGEMINE-A QUADRIGEMINE-B R-102444 R-99224 RC-39-2 RC-39II RE-1492 RE-2047 RG-12986 RG-2958 RHAPONTIGENIN RIDOGREL RK-286C RMI-7822 RO-09-0680 RO-15-2041 RO-19-1400 RO-19-3704 RO-24-4736 RO-43-5054 RO-43-8857 RO-44-3888 RO-44-9883 RO-48-3656 ROBUSTINE ROXIFIBAN RPR-109039 RPR-109891 RPR-110173 RS-93427 RUPATADINE RWJ-56110 RWJ-58259 RX-RE-92 S-1197 S-18204 S-18326 S-18886 SA-2572 SALMOSIN SANSHOOL-GAMMA SARPROGRELATE SB-214857 SC-38249 SC-42619 SC-46749 SC-47643 SC-52012 SC-54701 SC-54701-A SC-57101 SC-57101-A SCH-47918 SCH-59498 SDZ-216-744 SDZ-216-744 SDZ-217-766 SDZ-62-434 SDZ-62-694 SDZ-62-759 SDZ-62-826 SDZ-63-135 SDZ-MTH-958 SEL-2711 SEMIGLABRIN SK-549 SKF-107260 SKF-96365 SKF-96365 SKULLCAPFLAVONE-II SL-65-0472 SM-10906 SM-12502 SN-602 SQ-26536 SQ-27427 SQ-28668 SQ-28852 SQ-29535 SQ-29548 SQ-33261 SQ-33552 SQ-33961 SQ-80338 SR-121566 SR-121566-A SR-121787 SR-25990C SR-26334 SR-49059 SRI-63-072 SRI-63-119 SRI-63-675 SUBEROSIN SULEPAROIDE SULFINPYRAZONE SULFOBACIN-B SULOTROBAN SUN-9221 SUN-C-5174 SWIETEMAHONIN-D SWIETEMAHONIN-G SY-9215 T-250 TA-993 TAK-029 TAPP-BR TCV-309 TEI-4120 TER-930180 TERBOGREL TERRITREM-B TETRAFIBRICIN THALICMINE TICLOPIDINE TIMOSAPONIN-A-III

Derwent Drug File 1059 Thesaurus TIMOSAPONIN-B-I TIMOSAPONIN-B-II TIMOSAPONIN-B-III TIROFIBAN TJ-8014 TOLMETIN-PARACETAMOL-= ESTER TP-9201 TREQUINSIN TRI-11 TRI-25 TRI-59 TRIABIN TRIBAN TRIDEGIN TRIFENAGREL TRIFLAVIN TRIFLUSAL TRIGRAMIN TRILOBINE TYRPHOSTIN-A-48 U-73122 UK-34787 UK-74505 UP-116-77 UR-12460 UR-12592 UR-12670 UR-12947 VAPIPROST VASONIN VERAGUENSIN VINIGROL VINTOPEROL VON-WILLEBRAND-FACTOR-= 444-730 WEB-2347 WHI-P-131 WILD-20 WR-151326 XC-386 XEMILOFIBAN XJ-754 XJ-757 XU-063 XV-454 XV-459 Y-19018 Y-20811 Y-39241 Y-590 YANGAMBIN YC-1 YM-337 YM-461 YM-57029 YM-60828 Z-335 ZK-805412 ZK-805623 ANTIALCOHOLICS ACAMPROSATE ACETYLCYANAMIDE ACETYLTAURINE AMINOCYCLOPROPANOL-1 BENZOYLCYANAMIDE CALCIUM-BIS-ACETYL-= HOMOTAURINE CALCIUM-CARBIMIDE CALCIUM-CYANAMIDE-= CITRATED COPRINE DECZEIN DIETHYLTHIOCARBAMATE-= METHYL-ESTER DISULFIRAM HEPZEIN HEXZEIN HYDROXYMETRONIDAZOLE INMECARB LY-34580 LYCOPODINE METHOXYCORONARIDINE-18 METRONIDAZOLE METRONIDAZOLE-= PHOSPHATE METRONIDAZOLE-SUCCINATE NERAMEXANE NITREFAZOLE TERNIDAZOLE ZE-117 ANTIANAPHYLACTICS 48740-RP 59227-RP A-65260 AA-1777 AA-344 AB-23 AB-50 ABLUKAST ABT-080 ACETYL-ASPARTYL= GLUTAMATE-N AD-0261 AD-3264 AH-7725 AH-9679 AL-136 AM-682 AMENTOFLAVONE AMLEXANOX ANDOLAST ARNICOLIDE-C AS-35 BAICALEIN-PHOSPHATE BETOTASTINE BL-5255 BN-50069 BN-50090 BN-50125 BN-50726 BRYONOLATE BW-B70C C-4C CDP-840 CDRI-94-335 CGP-44826 CHELIDONATE CI-922 CI-949 CICLESONIDE COMPLESTATIN CROMITRILE CROMOLYN CROMOLYN SODIUM CROMPROXATE SODIUM CV-3988 D-58 DAMETRALAST DF-1111301 DOCEBENONE DOQUALAST DS-4574 E-6123 ECLAZOLAST EFLUMAST EMEDASTINE ENOXAMAST F-1322 FK-613 FPL-55618 FPL-55712 FPL-57231 FR-71021 GINKGOLIDE-A GINKGOLIDE-B GINKGOLIDE-C GLYTEER GMCHA-TBP HSR-6071 HSR-609 IPD-1151T KC-11404 KC-404 KF-17625 KF-19514 KW-4099 KW-4679 KW-4994 KY-556 KZ-111 L-648051 L-652731 L-657098 L-686708 LC-6 LCB-2183 LICORICIDIN LY-151364 LY-183001 LY-203647 LY-83583 MAR-99 MDL-26024-GO MDL-427 MINOCROMIL MIZOLASTINE MTB MY-1250 N-5+ NCO-650 NEDOCROMIL NEYDESIB NIGELLONE NZ-107 OXATOMIDE PAEONIFLORIN PAF-ACETYLHYDROLASE PCA-4248 PEMIROLAST PICUMAST PR-D-92-EA PROXICROMIL QUINOTOLAST REPIRINAST REV-3579 RG-12525 RG-7152 RHC-2851 RHC-3024 RHC-3164 RHC-3414 RHODIOCYANOSIDE-A RO-19-1400 RO-21-7634 RO-24-5913 ROFLUMILAST RWJ-50271 SANDOSAPONIN-A SANDOSAPONIN-B SAVENTOL SCH-37224 SENECIOYLPLENOLIN-O-6 SERINE-BORATE SF-2370 SKF-101132 SKF-102922 SKF-106203 SKF-78729-A SKF-84210 SKF-88046

1060 APPENDIX D SKF-S-106203 SL-85-0324 SOYASAPONIN-V SPAGLUMATE STEINAZIDE SUBMANDIBULAR-GLAND-= PEPTIDE-T SUPLATAST-TOSILATE SUPLATAST-TOSILATE TA-5707 TA-5707F TAZANOLAST TAZIFYLLINE TEI-9874 THEOPHYLLINE-SODIUM-= ANISATE THUNBERGINOL-A THUNBERGINOL-B THUNBERGINOL-F TIACRILAST TIOXAMAST TIPRINAST TJ-96 TOMELUKAST TRANILAST TYB-2285 VUF-K-8788 W-8011 WHI-P-131 WY-41195 WY-44329 Y-12141 Y-19432 YM-461 ZAFIRLUKAST ZAPRINAST ZCR-2060 ANTIANEMICS ACTIVIN-A CIDEFERRON COAMIDE DARBEPOETIN ALFA DIMETHYLADIPIMIDATE EDTA IRON FERAMID FEREDETATE SODIUM FERRIC-AMMONIUM-CITRATE FERRIC-CHONDROITINSULFATE FERRIC-CITRATE FERRIC-FRUCTOSE FERRIC-HYDROXIDE FERRIC-METHIONINE FERRIC-OXIDE FERRIC-OXIDE-SACCHARATED FERRIC-PYROPHOSPHATE FERRICLATE CALCIUM = SODIUM FERROCERON FERROCHOLINATE FERROGLUCIN-75 FERROPOLIMALER FERROTRENINE FERROUS-ASCORBATE FERROUS-ASPARTATE FERROUS-CHLORIDE FERROUS-CITRATE FERROUS-FUMARATE FERROUS-GLYCINE-SULFATE FERROUS-LACTATE FERROUS-OXALATE FERROUS-SUCCINATE FERROUS-SULFATE FERROUS-TARTRATE GLEPTOFERRON GLUCONATE FERRIC GLUCONATE FERROUS GLUSOFERRON HEMOFER IRON-CHONDROITINSULFATE IRON-DEXTRAN IRON-MALTOL IRON-PENTACARBONYL IRON-POLYMALTOSE IRON-SORBITEX ITF-282 LIXOTINIC PENTOKSIL THROMBOPOIETIN-MOUSE ANTIARRHYTHMICS 4595-RP 86017 A-2545 AC-623 ACC-9358 ACECAINIDE ACETYLSTROPHANTHIDIN ACTISOMIDE ADAPROLOL ADENOSINE AFD-19 AFD-21 AH-1058 AHR-12234C AJ-234 AJ-2615 AJMALINE ALINIDINE ALLOCRYPTOPINE ALLYLSECOBOLDINE-N ALMOKALANT ALPRAFENONE AMAFOLONE AMBASILIDE AMIDEPIN AMINOQUINOLINE-4 AMIODARONE AN-132 ANTAZOLINE ANTIARRHYTHMIC-PEPTIDE ANTIARRHYTHMIC-PEPTIDE-= 10 APRINDINE AR-12460 AR-12465 AR-LH-31 ARGININE-METHYL-ESTER ARK-5210 ARK-5211 ARK-5213 ARK-5310 ARK-5311 ARK-5312 ARTILIDE ASOCAINOL ATI-2001 AWD-160-275 AWD-19-166 AWD-23-111 AWD-G256 AZIMILIDE BARUCAINIDE BENDERIZINE BENRIXATE BERLAFENONE BERTOSAMIL BEVANTOLOL BIDISOMIDE BIIB-513 BISARAMIL BK-129 BRB-I-28 BREVICARINE BRL-31660A BRL-32872 BUCAINIDE BUCROMARONE BUFETOLOL BUNAFTINE BUPRANOLOL BUTAFENONE BUTIDRINE BUTOBENDINE BUTOPROZINE BW-A256C CAPSINOLOL CARCAINIUM CHLORIDE CARIPORIDE CAROCAINIDE CARYACHINE CCI-22277 CHANGROLIN CHROMANOL-293-B CIBENZOLINE CIPRAFAMIDE CK-1649 CK-3579 CL-284027 CLAMIKALANT CLOFILIUM CPU-23 CPU-57 CPU-86017 CRE-1087 CV-3611 CVT-510 CYCLOPROTOBUXINE-A CYCLOVIROBUXINE-D CYHEPTROPINE D-230 DA-1686 DAZOLICIN DC-015 DEETHYLACECAINIDE DEHYDROEVODIAMINE DEMETHYLENCAINIDE-N DEMETHYLIVABRADINE-N DENITRONIPRADILOL DEOXOAMIODARONE DEPROPYLPROPAFENONE-N DETAJMIUM BITARTRATE DEXPROPRANOLOL DIHYDROQUINIDINE DIOADIOLOL DIPRAFENONE DISOBUTAMIDE DISOPYRAMIDE DK-AH-269 DOFETILIDE DOPROPIDIL DRIDOCAINIDE DROBULINE DRONEDARONE DROXICAINIDE DYCLONINE E-0747 E-3753 E-4031 EDIFOLONE EGIS-7229 EGYT-1855 EMD-59730 EMD-60264 EMILIUM TOSILATE ENCAINIDE ENIPORIDE EO-122 EPICAINIDE EPROXINDINE EPS-2004 ESMOLOL ETACIZINE

Derwent Drug File 1061 Thesaurus ETAFENONE ETHAVERINE FALIPAMIL FALIRYTMIN FENETRADIL FEPROMIDE FLECAINIDE FLESTOLOL FLUZOPERINE FPL-13210 FR-168888 FR-183998 G-491 GALLANILIDE GE-430 GE-68 GE-70 GE-76 GLG-V-13 GLUTAPYRONE GUAFECAINOL GYKI-23107 H-2954 HEPTACAINE HEXACAINE HIGENAMINE HMR-1098 HMR-1372 HMR-1402 HMR-1556 HOE-694 HYDROXYCAPRATE-5 HYDROXYFENONE HYDROXYPIPERAQUINE HYDROXYPROPAFENONE-5 ICI-D-7288 IF-C-45 IHC-72 INDECAINIDE INDENOLOL IPAZILIDE IRFI-048 IVABRADINE K-953 KB-R-7943 KBR-9032 KC-12291 KC-8851 KCB-328 KETOCAINOL KLN-93 KW-3407 L-3937 L-691121 L-702958 L-706000 L-735821 L-768673 L-7810 LAPPACONITINE LB-32841 LG-6-101 LG-6-102 LG-83-6-05 LI-132 LIDOCAINE LL-115 LORAJMINE LORCAINIDE LY-190147 LY-97241 M-30 M-32 MCN-2165 MCN-4130 MEOBENTINE METHYLDEOXYMIDODRINE-N METIPRANOLOL MEXILETINE MG-1 MIBEFRADIL MJ-14030 MJ-9444 MK-142 MK-251 MONATEPIL MORACIZINE MOXAPRINDINE MS-551 N-3601 NADOLOL NADOXOLOL NAFENODONE NE-10133 NIBENTAN NICAINOPROL NIFEKALANT NIPRADILOL NISOLDIPINE-META NOFECAINIDE NORLORCAINIDE NOVDIMAL OLEUROPEIN OPC-88117 ORG-7797 OXIRAMIDE OXYBATE LITHIUM OXYBATELITHIUM PENTISOMIDE PERAKINE PH-776-141 PHENICARBERAN PILSICAINIDE PINCAINIDE PIRMENOL PIROLAZAMIDE POTASSIUM-GLUTAMATE POTASSIUM-MAGNESIUM-= ASPARTATE PRAJMALIUM BITARTRATE PRAJMALIUM BROMIDE PRANOLIUM CHLORIDE PRIMIDOLOL PROCAINAMIDE PROLEKOFEN PROPAFENONE PROPIONYLPROCAINAMIDE-N PROPRANOLOL PROPRANOLOL-CLOFIBRATE PROPRANOLOL-DIBUDINATE PYRINOLINE QUINACAINOL QUINIDINE QUINIDINE PHENOBARBITAL QUININE QUININE-ETHYLCARBONATE R-56865 R-70608 R-83572 RAUNATIN RECAINAM RESTACORIN RG-16 RG-25 RHINOCAINE RITMIDAZOL RO-22-9194 RO-5-5340 ROM-126 ROM-131 ROPITOIN RP-58866 RS-2135 RS-67333 RS-67506 RS-87337 RSD-1000 RSD-1019 RSD-1070 RSD-1235 RWJ-28810 S-16257 S-16257-2 S-16260-2 S-2150 S-24623 S-26191 SA-3212 SAZ-VII-22 SAZ-VII-23 SD-3212 SEA-ANEMONE-TOXIN-II SEMATILIDE SIMENDAN SKF-101055 SM-20550 SM-266 SM-345 SMP-300 SOLPECAINOL SOTAHEXAL SPARTEINE STENOPRIL STH-2148 STIROCAINIDE SURICAINIDE T-162559 TAXINE-II TE-176 TEDISAMIL TERIKALANT TH-91-21 TH-92-20 TH-92-4 TIAPAMIL TJN-505 TK-620-9 TMB-5 TMB-6 TOCAINIDE TOLAMOLOL TOSIFEN TRANSCAINIDE TRECETILIDE TY-12533 TZ-50-2 U-82208E U-82209E U-88943E UBISINDINE UK-1745 UK-66914 ULFS-49 UM-424 USVC-6524 VULM-411 WAY-123398 WY-48986 XIPRANOLOL Y-27632 Z-13752-A ZATEBRADINE ANTIARTERIOSCLEROTICS 447-C-88 A-87049 ACA-147 ACETIROMATE ACIFRAN ACIPIMOX AD-5075 AG-1295

1062 APPENDIX D AHR-16303B AL-294 ALUFIBRATE AMEU ANISACRIL ANNA-PAVALA-SINDHOORAM APOLIPOPROTEIN-A1-MILANO APOLIPOPROTEIN-A1-= MILANO-HUMAN AR-12-456 AR-12455 AR-12463 AR-12464 AR-12465 ASCOFURANONE ATORVASTATIN ATORVASTATIN-METHYL-= ESTER ATRASENTAN ATZ-1993 AVASIMIBE AVI-4126 AY-9944 AZ-242 AZACOSTEROL BAY-02752 BECLOBRATE BECLOBRIC-ACID BELOXAMIDE BENFLUOREX BEZAFIBRATE BF-759 BIBX-79 BICLOFIBRATE BINIFIBRATE BM-130907 BM-15766 BMS-187745 BMS-188494 BMY-21950 BMY-22089 BO-653 BOXIDINE BP-42 BRAZILIN BREYNIN-A BREYNIN-B BRL-26314 BUTHIOBATE BUTOXAMINE BUTYLPHTHALIDE-3 CERIVASTATIN CETABEN CGP-43371 CGS-23425 CGS-26214 CHINOIN-123 CHIRO-INOSITOL CHOLINE-ALFOSCERATE CI-1011 CI-924 CI-976 CIGLITAZONE CIPROFIBRATE CK-3368 CL-274471 CL-277082 CL-283546 CL-283796 CLIMIQUALINE CLINOFIBRATE CLINOLAMIDE CLOBUZARIT CLOFENAPATE CLOFIBRATE CLOFIBRATE CALCIUM CLOFIBRIC-ACID CLOFIBRIDE CLOMESTRONE CLORIDAROL CLX-0901 COLESEVELAM COLESTIPOL CONFERIN CP-105191 CP-113818 CP-148623 CP-230821 CP-340868 CRILVASTATIN CT-052923 CYCLOARTENOL CYCLOARTENOL-FERULATE CYNARINE D-003 DALVASTATIN DARGLITAZONE DECARESTRICTINE-B DECARESTRICTINE-D DH-990 DIACETYLCYSTINE-N,N+ DIHYDROMEVASTATIN DIHYDROMEVINOLIN DIMETHYLPYRAZOLE-3,5 DIOSPONIN DIPROGULATE DISOGLUSIDE DIVERSIN DMP-565 DRF-2189 DRF-2725 DROSTANOLONE DULOFIBRATE DUP-128 E-5050 E-5324 EICOSAPENTAENOATE-= ETHYL-ESTER EM-652 ENICLOBRATE EPISESAMIN ER-27856 ETHOXYSILATRANE-1 ETHYLCYSTEINE-S ETIROXATE ETOFIBRATE ETOFYLLINE-CLOFIBRATE EZETIMIBE F-10863-C F-10863-D F-12511 F-1394 F-1839-B F-1839-E FARGLITAZAR FCE-27677 FENBUTYRAMIDE FENERITROL FENIROFIBRATE FENOFIBRATE FENOFIBRIC-ACID FILICOL FL-386 FLUVASTATIN FOMESAFEN FR-145237 FR-186054 FURANACRYLATE-2 FURAZABOL FUROATE-2 GALBANATE GAMOLENATE GARLIC-EXTRACT GEMCADIOL GEMFIBROZIL GLISOPRENIN-A GLISOPRENIN-B GLUCOMANNAN GLUNICATE GLYCITEIN GM-1077 GP-45699 GUGULIPID GW-1929 GW-510516 GW-7647 GW-7845 HALOFENATE HEMATEIN HEXANOYLTAXOL-7 HL-004 HR-780 HYDROXYMEVASTATIN-3-= BETA ICI-53072 IMPLITAPIDE ITANOXONE J-104118 J-104132 JTT-705 KARATAVATE KC-515 KCD-232 KF-1492 KW-3033 L-154819 L-157012 L-44-0 L-645164 L-647318 L-654969 L-659699 L-660281 L-660343 L-660347 L-679336 L-796449 L-805645 LFA-703 LG-101305 LIFIBRATE LIFIBROL LIPAMIDE LK-903 LODAZECAR LOVASTATIN LU-224332 LY-290181 LY-290293 LY-295427 M+B-30227 M+B-31426 MCI-196 MDL-14514 MDL-28815 MDL-29311 MEGLUTOL MELINAMIDE MEPIROXOL MESOGLYCAN MET-RANTES METHYLCYSTEINE-= SULFOXIDE-S METHYLENECYCLO= ARTANOL-24 METIBRIDE MEVASTATIN MEVINOLINATE MIFOBATE ML-236A MLM-160 MOCTAMIDE

Derwent Drug File 1063 Thesaurus MONACOLIN-J MONACOLIN-K MONACOLIN-L MONACOLIN-X MOQUIZONE MRZ-3-124 MRZ-3124 N-4472 N-4909 NAFENOPIN NB-598 NEOGRIFOLIN NIADENATE NICERITROL NICOCLONATE NICOFIBRATE NICOFURATE NICOMOL NIP-200 NITROACETYLSALICYLATE NO-1886 NS-1 NTE-122 OCTIMIBATE SODIUM OLIFEN OLIGVON OXANDROLONE OXFENICINE OXINIACATE P-0654 PADMA-28 PANAXYDIOL PANTENICATE PANTETHINE PD-132301-2 PD-134965 PD-135022 PD-138142 PD-138142-15 PD-146176 PD-69405 PD-72953 PERFLUOROOCTANE-= SULFONATE PERFLUOROROOCTANOATE PHEPRACET PHLORACETOPHENONE PICAFIBRATE PIMETINE PIOGLITAZONE PIRIFIBRATE PIRINIXATE PIRINIXIL PLAFIBRIDE PM-170 POLIDEXIDE POLYDATIN POLYSPONINE PONFIBRATE POTASSIUM-CHROMATE PRAVASTATIN PRAVASTATIN SODIUM PROBUCOL PROMEGA PROPYLCYSTEINE-S PURPACTIN-A PURPACTIN-B PURPACTIN-C PYRIDINOL-CARBAMATE PYRIDOXAL-PHOSPHATE-= GLUTAMATE PYRIPYROPENE-A PYRIPYROPENE-B PYRIPYROPENE-C PYRIPYROPENE-D RAWSONOL RESVERATROL RG-50858 RG-50875 RO-12-1989 RO-16-6532 RO-20-1724 RO-22-0654 RO-48-8071 ROSUVASTATIN RP-54275 RP-64477 RP-70676 RPR-101821 RPR-107393 S-1321 S-1322 S-20478 S-422 SALAFIBRATE SB-204990 SB-435495 SC-37111 SC-435 SC-68693 SCH-48461 SCH-58053 SCH-58235 SCH-60663 SCH-9122 SDZ-267-489 SE-1475 SERFIBRATE SF-482 SIM-6080 SIMFIBRATE SIMVASTATIN SIMVASTATIN SITOFIBRATE SKF-16467-A SKF-2314 SKF-7732-A3 SKF-97426A SKF-99085 SKF-L-94901 SORBINICATE SQ-10591 SQ-31360 SQ-31906 SQ-33600 SQUALESTATIN-1 SR-12813 SR-9223-I SR-9223I SSF-109 SUCROSE-POLYESTER SULODEXIDE SULTOSILATE SURFOMER SY-9215 T-686 TA-1801 TA-7552 TA-993 TAD-235 TAK-636 TAZASUBRATE TERBUFIBROL TERBUFICIN TIADENOL TIADENOL-NICOTINATE TIAFIBRATE TIBRATE TIGOGENIN-CELLOBIOSIDE TIMEFURONE TIMOFIBRATE TIRATRICOL TISOQUONE TIZOPROLATE TMP-153 TOCOFIBRATE TORILIN TRELOXINATE TRETHOCANATE TRIACSIN-A TRIACSIN-B TRIACSIN-C TRIACSIN-D TRIEICOSAPENTAENIN TRIPARANOL TROGLITAZONE U-22105 U-25030 UCF-1-C UREFIBRATE W-2531 W-398 WY-3457 X-50 XD-793 XENALIPIN XENBUCIN XENTHIORATE XENYHEXENATE XIMEDONE XT-199 Y-27632 Y-9738 YM-17E YM-53601 YM-95831 ZARAGOZATE-A ZARAGOZATE-B ZARAGOZATE-C ZM-250462 ZM-97480 ANTIASTHMATICS 48740-RP A-249377 A-277323 A-93178 AA-344 AB-23 AB-50 ABC-99 ABLUKAST ABT-080 ABT-761 AC-119 ACETOSYRINGENIN ADRENALINE AFORMOTEROL AH-7725 ALOE-EXTRACT AMBROXOL = THEOPHYLLINATE AMBUPHYLLINE AMITEROL AMLEXANOX ANDOLAST ANDROSIN AP-0341 APC-2059 APC-366 AR-C-68397-AA ARPENAL AS-35 ASTHMA-TROPON AWD-12-281 AZANATOR AZASPIRIUM CHLORIDE BAMBUTEROL BAMIFYLLINE BAY-U-9773 BAY-X-7195 BAY-Y-1015

1064 APPENDIX D BB-1502 BI-RM-270 BITOLTEROL BL-5255 BM-531 BN-50726 BQ-123 BROXATEROL BUFROLIN BUTYLETHARINE BW-B218C CARBUTEROL CDP-840 CGP-44826 CGP-45715A CGP-57698 CHAMAZULENE CHOLINE-THEOPHYLLINATE CI-1018 CI-922 CILOMILAST CLENBUTEROL CLORPRENALINE COLTEROL CONOPHYLLINE CONTIGNASTEROL CP-199331 CROMITRILE CROMOLYN CROMOLYN SODIUM CROMPROXATE SODIUM CV-3988 D-18024 D-22888 D-2343 D-4026 D-4030 DAMETRALAST DECLOXIZINE DEPTROPINE DIBUNATE SODIUM DIMABEFYLLINE DINIPROFYLLINE DIOXETHEDRIN DIPHENYLTHIOSULFINATE DIPROPHYLLINE DOCEBENONE DOQUALAST DOXANTRAZOLE DOXOFYLLINE EFLUMAST EMEDASTINE ENOFELAST ENPROFYLLINE EPHEDRINE EPRAZINONE EPROZINOL ETAFEDRINE ETANTEROL ETHYLNORADRENALINE F-1322 FENOTEROL FENPIPRANE FENSPIRIDE FLEZELASTINE FLUTROPIUM BROMIDE FORMOTEROL FPL-52694 FPL-52757 FR-71021 FUPRAZOLE GEA-3175 GINKGOLIDE-A GINKGOLIDE-B GINKGOLIDE-C GUAIFYLLINE HEXOPRENALINE HOQUIZIL HSR-284 HSR-609 HWA-214 IBUDILAST IBUTEROL ICI-58301 ICI-61129 ICI-63197 ICI-D-2138 IG-10 IPRATROPIUM BROMIDE ISAMOXOLE ISOETARINE ISOPRENALINE KAA-276 KC-404 KF-15570 KF-17625 KF-19514 KW-4099 KWD-2131 KZ-111 L-670630 L-686708 L-691816 L-739010 L-746530 LCB-2183 LEVOSALBUTAMOL LM-1453 LM-1468 LODOXAMIDE LY-163443 LY-280810 M-711 MABUTEROL MAR-99 MDL-26024-GO MEQUITAMIUM IODIDE METHOXYPHENAMINE METHYLEPHEDRINE MINOCROMIL MKS-492 MONTELUKAST NAMINTEROL NCX-1020 NEDOCROMIL NIAPRAZINE NISBUTEROL NORBUDRINE OMALIZUMAB ONO-RS-347 ORCIPRENALINE OXARBAZOLE OXATOMIDE OXITROPIUM BROMIDE PEGANIN PF-904 PICUMAST PICUMETEROL PIMETHIXENE PIPERLONGUMINE PIPOXIZINE PIQUIZIL PIRBUTEROL PIROLATE PIRQUINOZOL PROCATEROL PROTOKYLOL PROXICROMIL PSEUDOEPHEDRINE QH-25 QUAZOLAST QUINETALATE QUINOTOLAST QUINPRENALINE REPROTEROL REVENAST RG-12553 RG-7152 RHC-3164 RIMITEROL RITOLUKAST RO-24-4736 RO-24-5913 ROFLUMILAST RP-73401 RS-91309 RU-42173 RWJ-22108 S-16474 S-9795 SALBUTAMOL SALMEFAMOL SALMETEROL SB-207499 SB-210396 SC-37872 SCH-351591 SCH-37224 SDZ-217-744 SERATRODAST SKF-104353 SKF-107310 SKF-78729-A SM-10661 SM-11044 SOTERENOL SP-600125 SPIRGETINE SQ-33961 SR-27417 SUDEXANOX SULFONTEROL SULOXIFEN T-440 TA-073 TA-5707 TAK-225 TAZANOLAST TEI-9874 TERBUTALINE TERFENADINE TETRAGALLOYLQUINATE THEOPHYLLINE THEOPHYLLINE-LYSINE THEOPHYLLINE-SODIUM-= GLYCINATE THIAZINAMIUM IODIDE THIAZINAMIUM-SULFOXIDE = IODIDE TIACRILAST TJ-96 TOLIMIDONE TOMELUKAST TRANILAST TRETOQUINOL TRIACANTHINE TRICLOFYLLINE TROPINE-BENZILATE TROPIRINE TROVENTOL TULOBUTEROL U-101033-E UCB-JO28 UROGUANYLIN VASICINONE VEPHYLLINE VERLUKAST VEROFYLLINE VILOZEN VUF-K-8788 W-8011 WY-44329

Derwent Drug File 1065 Thesaurus WY-50295-T XANOXATE Y-12141 YM-461 YM-57158 YM-934 Z-335 ZAFIRLUKAST ZD-6021 ZILEUTON ZINDOTRINE ZINTEROL ANTIBIOTICS 2355-S 6643-X A-16686 A-16686-A1 A-16686-A2 A-16686-A3 A-16886A A-16886B A-19009 A-204A A-21459-A A-21459-B A-21978-C1 A-21978-C2 A-21978-C3 A-25822-A A-25822-B A-25822-D A-25822-L A-25822-M A-25822-N A-26771B A-32390-A A-35512B A-40926-PA A-41030A A-41030C A-41030D A-41030E A-41030F A-41030G A-477 A-47934 A-54145A A-54145A1 A-54145B A-54145B1 A-54145C A-54145D A-54145E A-54145F A-62514 A-62671 A-66005 A-66173 A-69334 A-80915A A-83586-C ABAMECTIN ABIERIXIN ABIKOVIROMYCIN ABT-773 ACETOMYCIN ACETOPYRROTHINE ACETOXYCYCLOHEXIMIDE ACETYLARANOTIN ACETYLDAUNORUBICIN-N ACETYLDOXORUBICIN-N ACETYLPHOMALACTONE ACIVICIN ACLACINOMYCIN ACLACINOMYCIN-B ACLACINOMYCIN-S ACLACINOMYCIN-T ACLARUBICIN ACTAGARDIN ACTAMYCIN ACTAPLANIN-A ACTAPLANIN-B1 ACTAPLANIN-B2 ACTAPLANIN-B3 ACTAPLANIN-C1 ACTAPLANIN-C2 ACTAPLANIN-G ACTINOBOLIN ACTINOHIVIN ACTINOIDIN ACTINOIDIN-A ACTINOIDIN-A2 ACTINOIDIN-B ACTINOMYCIN ACTINOMYCIN-C2 ACTINOMYCIN-C3 ACTINOMYCIN-D ACTINOMYCIN-K2T ACTINOMYCIN-V ACTINOMYCIN-Z5 ACTINONIN ACTINOPLANONE-A ACTINOPYRONE-A ACTINORHODINE ACTITHIAZATE ACULEACIN-A ACULEXIMYCIN AD-143 AD-198 AD-199 AD-280 AD-32 ADICILLIN ADIPOSIN ADIPOSIN-2 ADOZELESIN AEROCYANIDIN AF-013 AF-05 AF-150 AF-ABDMP AF-ABDP AF-ABP AGELASIDINE-A AGELASIDINE-C AGELINE-A AGGLOMERIN-A AGGLOMERIN-B AGGLOMERIN-C AGGLOMERIN-D AK-165-3 AKLAVIN AKROBOMYCIN AL-87 ALAHOPCIN ALAMETHICIN ALAMETHICIN-I ALAMETHICIN-II ALANOSINE ALAZOPEPTIN ALBIDIN ALBOCYCLINE ALBOFUNGIN ALBOMITOMYCIN-A ALBOMYCIN ALBOMYCIN-DELTA-1 ALBOMYCIN-DELTA-2 ALBONOURSIN ALBORIXIN ALCINDOROMYCIN ALDECALMYCIN ALISAMYCIN ALKANNIN ALLDIMYCIN-A ALLIACOLIDE ALLICIN ALLOSAMIDIN ALMECILLIN ALTEMICIDIN ALTERSOLANOL-A ALTERSOLANOL-B ALTHIOMYCIN ALTROMYCIN-A ALTROMYCIN-B ALTROMYCIN-C ALTROMYCIN-D ALTROMYCIN-H ALTROMYCIN-I AMA-1294 AMA-3176 AMANTOCILLIN AMFOMYCIN AMICETIN AMICLENOMYCIN AMICYCLINE AMIDINOMYCIN AMIDOMYCIN AMIJITRIENOL AMIKACIN AMINOCEPHALOSPORANATE AMINOPENICILLANATE AMOXICILLIN AMPHOGLUCAMINE AMPHOTERICIN-A AMPHOTERICIN-B AMPHOTERICIN-B-= METHYLESTER AMPHOTERICIN-X AMPICILLIN AMQ-2 AMRUBICIN AN-201I AN-201II ANDRASTIN-A ANDRIMID ANDROCTONIN ANGELMICIN-B ANGIOLAM-A ANGOLAMYCIN ANGOLAMYCIN-P1 ANGUIDIN ANGUSTMYCIN-A ANHYDROFRUCTOSE-1,5 ANHYDROFUSARUBIN ANHYDROJAVANICIN ANISOMYCIN ANKINOMYCIN ANNAMYCIN ANSAMITOCIN-P3 ANTELMYCIN ANTHELVENCIN-A ANTIBIOTIC-273A2 ANTIBIOTIC-273A2-ALPHA ANTIBIOTIC-273A2-BETA ANTICAPSINE ANTIMYCIN-A ANTIMYCIN-A1 ANTIMYCIN-A1A ANTIMYCIN-A1B ANTIMYCIN-A2 ANTIMYCIN-A2A ANTIMYCIN-A2B ANTIMYCIN-A3 ANTIMYCIN-A3A ANTIMYCIN-A3B ANTIMYCIN-A4 ANTIMYCIN-A4A ANTIMYCIN-A4B ANTRAFORMIN ANTRAMYCIN AO-1100

1066 APPENDIX D APALCILLIN APHE-1 APHE-2 APHIDICOLINE APICYCLINE APLASMOMYCIN APRAMYCIN AQUAYAMYCIN ARANCIAMYCIN ARANOROSIN ARANOTIN ARBEKACIN ARBUTIN ARDACIN ARENARIN ARENOMYCIN-B ARGINOMYCIN ARGYRIN-B ARIDICIN-A ARIDICIN-B ARIDICIN-C ARISTEROMYCIN ARISTOLOCHATE-I ARISTOLOCHATE-IA ARISTOLOCHATE-II ARIZONIN-A1 ARIZONIN-B1 ARMENTOMYCIN ARPHAMENINE-A ARPHAMENINE-B ARUGOMYCIN AS-48 AS-924 ASCAMYCIN ASCOCHITAL ASCOCHLORIN ASCOFURANOL ASCOFURANONE ASCOMYCIN ASCOSFEROL ASCOSIN ASPARENOMYCIN-A ASPARENOMYCIN-B ASPARENOMYCIN-C ASPARTOCIN ASPERENTIN ASPERLIN ASPIROCHLORINE ASPOCHALASINE-A ASPOCHALASINE-B ASPOCHALASINE-C ASPOXICILLIN ASPYRONE ASTROMICIN ASUKAMYCIN AT-2433-A1 AT-2433-A2 AT-2433-B1 AT-2433-B2 AT-265 ATPENIN-A4 ATPENIN-A4 ATPENIN-A5 ATPENIN-B ATRANORATE ATRANORIN AURAMYCIN-A AURAMYCIN-B AURAMYCINONE AURANTININ-B AUREOBASIDIN-B AUREOBASIDIN-C AUREOBASIDIN-D AUREOBASIDIN-E AUREOBASIDIN-F AUREOBASIDIN-G AUREOBASIDIN-H AUREOBASIDIN-I AUREOBASIDIN-J AUREOBASIDIN-K AUREOBASIDIN-L AUREOBASIDIN-M AUREOBASIDIN-N AUREOBASIDIN-O AUREOBASIDIN-P AUREOBASIDIN-Q AUREOBASIDIN-R AUREOFACIN AUREOFUNGIN AUREOTHIN AUREOTHRICIN AUROCITRIN AUROMOMYCIN AUROVERTIN-B AVELLANEOL AVENACIOLIDE AVERMECTIN AVERMECTIN-A1A AVERMECTIN-A1B AVERMECTIN-A2A AVERMECTIN-A2B AVERMECTIN-B1A AVERMECTIN-B1B AVERMECTIN-B2A AVERMECTIN-B2B AVERMECTIN-H2B1B AVILAMYCIN AVILAMYCIN-A AVILAMYCIN-B AVILAMYCIN-C AVILAMYCIN-D1 AVILAMYCIN-D2 AVILAMYCIN-E AVOPARCIN AVOPARCIN-ALPHA AVOPARCIN-BETA AWAMYCIN AY-24668 AZACYTIDINE AZAHYPOXANTHINE-8 AZALOMYCIN-F AZALOMYCIN-F4 AZASERINE AZATYROSINE AZAXANTHINE-8 AZEPINOMYCIN AZETOMYCIN-I AZETOMYCIN-II AZICEMICIN-A AZICEMICIN-B AZIDAMFENICOL AZIDOCILLIN AZINOMYCIN-A AZINOMYCIN-B AZITHROMYCIN AZLOCILLIN AZOMYCIN AZOTOMYCIN AZTREONAM BAC-1829 BACAMPICILLIN BACILLOMYCIN-D BACILLOMYCIN-F BACILLOMYCIN-L BACITRACIN BACITRACIN-A BACITRACIN-F BACITRACIN-METHYLENE= DISALICYLATE BACMECILLINAM BACTOBOLIN BACTROPONE BAFILOMYCIN BAFILOMYCIN-A BAFILOMYCIN-A1 BAFILOMYCIN-A2 BAFILOMYCIN-B1 BAFILOMYCIN-B2 BAFILOMYCIN-C1 BAFILOMYCIN-C2 BAFILOMYCIN-D BAL-9141 BALHIMYCIN BAMBERMYCIN BARMINOMYCIN-I BARMINOMYCIN-II BASIDALIN BASIFUNGIN BAUMYCIN-A1 BAUMYCIN-A2 BAUMYCIN-B2 BAUMYCIN-C1 BAY-3522 BAY-V-3522 BBK-29 BBR-2778 BBR-2828 BBR-2868 BE-12406A BE-12406B BE-18257A BE-18591 BEAUVERICIN BELLENAMINE BENANOMICIN-A BENANOMICIN-B BENASTATIN-A BENASTATIN-B BENETHAMINE-PENICILLIN BENGAMIDE-A BENGAMIDE-B BENGAMIDE-C BENZANTHRIN-A BENZANTHRIN-B BENZATHINEBENZYLPENICILLIN BENZATHINE-CEFAPIRIN BENZATHINE-CHLOR= TETRACYCLINE BENZATHINE-CLOXACILLIN BENZATHINE-PHENOXY= METHYLPENICILLIN BENZYLDAUNORUBICIN-N BENZYLPENICILLIN BENZYLSPARSOMYCIN BERYTHROMYCIN BETACLAMYCIN-A BETAMICIN BIAPENEM BICOZAMYCIN BILANAFOS BIOPOLYENE BIOXALOMYCIN-ALPHA-2 BIPHENOMYCIN-A BIPHENOMYCIN-B BISNORDIHYDROTOXIFERINE BISUCABERIN BIVITTOSIDE-A BIVITTOSIDE-B BIVITTOSIDE-C BIVITTOSIDE-D BIZELESIN BIZELESIN BL-6783 BL-P-875 BL-S-217 BL-S-339 BLASTICIDIN-S BLASTMYCINONE BLEOMYCIN BLEOMYCIN-A1 BLEOMYCIN-A2

Derwent Drug File 1067 Thesaurus BLEOMYCIN-A5 BLEOMYCIN-B2 BLEOMYCIN-B4 BLEOMYCINATE BLUENSOMYCIN BMS-180680 BMY-25067 BMY-25174 BMY-26107 BMY-28232 BMY-28251 BMY-28271 BMY-28864 BO-1165 BO-1166 BO-1236 BO-1341 BO-2727 BOHOLMYCIN BOLESATINE BONGKREKATE BOROMYCIN BORRELIDIN BOSTRYCIN BOSTRYCOIDIN BOTRYODIPLODIN BOTTROMYCIN-A2 BOUVARDIN BOXAZOMYCIN-B BRASILIQUINONE-A BREFELDIN-A BRL-41897A BRL-41897A BRL-44154 BROMAMPHENICOL BROMODAUNORUBICIN BROMOTETRACYCLINE BU-3129T BUCCINULIN BUTALACTIN BUTAMPICILLIN BUTIKACIN BUTIROSIN BUTIROSIN-A BUTIROSIN-B C-1027 C-19393-E5 C-27 C-2801-X CACTINOMYCIN CADEGUOMYCIN CAERULOMYCIN-A CAERULOMYCIN-C CAF-603 CAIROMYCIN-A CALBISTRIN-A CALBISTRIN-B CALCIMYCIN CALICHEAMICIN CALICHEAMICIN-ALPHA-2-I CALICHEAMICIN-ALPHA-3-I CALICHEAMICIN-BETA-1-BR CALICHEAMICIN-BETA-1-I CALICHEAMICIN-DELTA-1-I CALICHEAMICIN-GAMMA-= 1-BR CALICHEAMICIN-GAMMA-1-I CALOPOROSIDE CALPHOSTIN-A CALPHOSTIN-B CALPHOSTIN-C CALPHOSTIN-D CALPHOSTIN-I CALVATATE CANADENSOLIDE CANDICIDIN-D CANDIDIN CAP-18-HUMAN CAPOAMYCIN CAPREOMYCIN CAPREOMYCIN-IA CAPREOMYCIN-IB CAPREOMYCIN-IIA CAPREOMYCIN-IIB CAPTOCILLIN CAPURAMYCIN CARAMICILLIN CARAZOSTATIN CARBAZOMYCIN-A CARBAZOMYCIN-B CARBAZOMYCIN-C CARBAZOMYCIN-D CARBAZOMYCIN-G CARBAZOMYCINAL CARBENICILLIN CARBOMYCIN CARBOMYCIN-A CARBOMYCIN-A-P1 CARBOMYCIN-A-P2 CARBOMYCIN-A-P3 CARDAMONIN CARFECILLIN CARINDACILLIN CARMINAZONE CARMONAM CARPETIMYCIN-A CARPETIMYCIN-B CARQUINOSTATIN-A CARRIOMYCIN CARUBICIN CARUMONAM CARYOYNENCIN-A CARZELESIN CARZINOPHILIN CASPOFUNGIN CATIONOMYCIN CC-1065 CCI-779 CDP-1 CECROPIN-A CECROPIN-D CEFACETRILE CEFACLOR CEFADROXIL CEFALEXIN CEFALOGLYCIN CEFALONIUM CEFALORAM CEFALORIDINE CEFALOTIN CEFAMANDOLE CEFAMANDOLE-NAFATE CEFAPAROLE CEFAPIRIN CEFATHIAMIDINE CEFATRIZINE CEFAZAFLUR CEFAZEDONE CEFAZOLIN CEFBUPERAZONE CEFCAMATE-PIVOXIL CEFCANEL CEFCANEL-DALOXATE CEFCLIDIN CEFDALOXIME CEFDINIR CEFDITOREN CEFDITOREN-PIVOXIL CEFEMPIDONE CEFEPIME CEFETAMET CEFETAMET-PIVOXIL CEFETRIZOLE CEFIVITRIL CEFIXIME CEFMENOXIME CEFMETAZOLE CEFMINOX CEFODIZIME CEFONICID CEFOPERAZONE CEFORANIDE CEFOTAXIME CEFOTETAN CEFOTIAM CEFOTIAM-HEXETIL CEFOXAZOLE CEFOXITIN CEFOZOPRAN CEFPIMIZOLE CEFPIRAMIDE CEFPIROME CEFPODOXIME CEFPODOXIME-PROXETIL CEFPROZIL CEFQUINOME CEFRADINE CEFROTIL CEFROXADINE CEFSULODIN CEFSUMIDE CEFTAZIDIME CEFTERAM CEFTERAM-PIVOXIL CEFTEZOLE CEFTIBUTEN CEFTIOFUR CEFTIOLENE CEFTIOXIDE CEFTIZOXIME CEFTRIAXONE CEFURACETIME CEFUROXIME CEFUROXIME-AXETIL CEFUZONAM CEFUZONAME CELESTICETIN CELLOCIDIN CEPACIDINE-A1 CEPACIDINE-A2 CEPHABACIN-F1 CEPHABACIN-F2 CEPHABACIN-F3 CEPHABACIN-F4 CEPHABACIN-F5 CEPHABACIN-F6 CEPHABACIN-F7 CEPHABACIN-F8 CEPHABACIN-F9 CEPHABACIN-H1 CEPHABACIN-H2 CEPHABACIN-H3 CEPHABACIN-H4 CEPHABACIN-H5 CEPHABACIN-H6 CEPHABACIN-M1 CEPHABACIN-M2 CEPHABACIN-M3 CEPHABACIN-M4 CEPHABACIN-M5 CEPHABACIN-M6 CEPHALOCHROMIN CEPHALOSPORANATE CEPHALOSPORIN-C CEPHALOSPORIN-P1 CEPHAMYCIN CEPHAMYCIN-A CEPHAMYCIN-B CEPHAMYCIN-C CERCOSPORAMIDE CERULENIN CERVINOMYCIN-A1

1068 APPENDIX D CERVINOMYCIN-A2 CETOCYCLINE CETOFENICOL CEZOMYCIN CGP-17520 CGP-29861 CGP-31523A CGP-31608 CGP-4832 CGP-7040 CHAETIACANDIN CHAETOGLOBOSIN-A CHAETOGLOBOSIN-B CHAETOGLOBOSIN-C CHAETOGLOBOSIN-D CHAETOGLOBOSIN-E CHAETOGLOBOSIN-F CHAETOGLOBOSIN-J CHAETOGLOBOSIN-K CHALCOMYCIN CHARTREUSIN CHERIMOLINE CHETOMIN CHICAMYCIN-A CHITINOVORIN-A CHITINOVORIN-C CHLORAMPHENICOL CHLORAMPHENICOL-= PALMITATE CHLORAMPHENICOL-= STEARATE CHLORAMPHENICOL-= SUCCINATE SODIUM CHLOROBIOCIN CHLOROCARDICIN CHLOROEREMOMYCIN CHLOROORIENTICIN-A CHLOROORIENTICIN-B CHLOROORIENTICIN-C CHLOROPOLYSPORIN-A CHLOROPOLYSPORIN-B CHLOROPOLYSPORIN-C CHLOROTETAIN CHLOROTHRICIN CHLOROZOTOCIN CHLORPOLYSPORIN-C CHLORTETRACYCLINE CHOKOL-A CHONDRAMIDE-A CHONDRAMIDE-B CHONDRAMIDE-C CHONDRAMIDE-D CHONEMORPHINE CHROMOMYCIN-A3 CHROMOXYMYCIN CHRYSCANDIN CHRYSOMYCIN-A CHRYSOMYCIN-B CHUANGXINMYCIN CICLAMYCIN-0 CICLOSPORIN CILOFUNGIN CINCHOPHYLLINE CINERUBIN-A CINERUBIN-B CINNABARINATE CINNABARINE CINNAMYCIN CINODINE CIRCULIN CIRCULIN-A CIRCULIN-B CIROLEMYCIN CIRRAMYCIN-A CISPENTACIN CITREAMICIN-ALPHA CITREAMICIN-ETA CITREAMICIN-ZETA CITRININ CITROMYCETIN CITROMYCIN CITROPEPTIN CJ-12371 CL-329998 CL-331002 CL-331928 CL-344677 CLARITHROMYCIN CLARITHROMYCIN-= LACTOBIONATE CLAUSSEQUINONE CLAVALANINE CLAVARIOPSIN-A CLAVARIOPSIN-B CLAZAMYCIN CLAZAMYCIN-A CLAZAMYCIN-B CLEMIZOLE-PENICILLIN CLEROCIDIN CLINDAMYCIN CLINDAMYCIN-PALMITATE CLINDAMYCIN-PHOSPHATE CLOMETOCILLIN CLOMOCYCLINE CLOSTOMICIN-A CLOSTOMICIN-B2 CLOXACILLIN CLOXACILLIN-SULFONE CMT-1 CMT-3 CMT-5 CMT-8 COCHLEAMYCIN-A COCHLEAMYCIN-A2 COCHLEAMYCIN-B COCHLEAMYCIN-B2 COFORMYCIN COFORMYCIN-= MONOPHOSPHATE COL-3 COLABOMYCIN-A COLIMECYCLINE COLISTIMETHATE COLISTIN COLISTIN-A COLISTIN-NONAPEPTIDE COLLETALLOL COLLETODIOL COLLINEMYCIN COLLISMYCIN-A COLLISMYCIN-B COLORADOCIN COMPLICATATE CONCANAMYCIN-A CONCANAMYCIN-B CONCANAMYCIN-C CONCANAMYCIN-F COPIAMYCIN CORALLOPYRONIN-A CORALLOPYRONIN-A+ CORALLOPYRONIN-B CORALLOPYRONIN-C CORDIACHROMENE-A CORDYCEPIN CORTALCERONE CORYNETOXIN CORYNETOXIN-H17A COSMOCARCIN-A COSMOMYCIN-A COSMOMYCIN-B COSMOMYCIN-C COSMOMYCIN-D COUMAMIDINE-GAMMA-1 COUMAMYCIN CP-111905 CP-113056 CP-53607 CP-6162 CP-63956 CP-65207 CP-6679 CP-70429 CP-81054 CP-82009 CP-84657 CPW-86363 CRANOMYCIN CRINIPELLIN-A CRINIPELLIN-B CRINITOL CRISAMICIN-A CRYPTOSPORIN CRYPTOTANSHINONE CS-834 CUPRIMYXIN CURACIN-A CURACIN-B CURACIN-C CURROMYCIN-A CURROMYCIN-B CYANOBACTERIN CYANOCYCLINE-A CYANOMORPHOLINO= DAUNORUBICIN CYCLACILLIN CYCLAMIDOMYCIN CYCLOEUDESMOL CYCLOHEXIMIDE CYCLOSERINE CYCLOSERINE,LCYCLOSPORIN-B CYCLOSPORIN-C CYCLOSPORIN-D CYCLOSPORIN-H CYCLOSPORIN-K CYCLOSPORIN-M CYCLOSPORIN-O CYCLOSPORIN-Q CYCLOSPORIN-U CYCLOSPORIN-V CYCLOSPORIN-Z CYCLOTHIALIDINE CYCLOTHIALIDINE-B CYCLOTHIALIDINE-C CYCLOTHIALIDINE-D CYCLOTHIALIDINE-E CYCLOVIRACIN-B1 CYCLOVIRACIN-B2 CYTOCHALASINE-A CYTOCHALASINE-B CYTOCHALASINE-C CYTOCHALASINE-D CYTOCHALASINE-E CYTOCHALASINE-F CYTOCHALASINE-G CYTOCHALASINE-H CYTOCHALASINE-J CYTOCHALASINE-N CYTOCHALASINE-O CYTOCHALASINE-P CYTOCHALASINE-Q CYTOCHALASINE-R CYTOGENIN CYTORHODIN-A CYTORHODIN-D CYTOVARICIN D-788-1 DA-1131 DACTIMICIN DACTYLOCYCLINE-A DACTYLOCYCLINE-B DALFOPRISTIN

Derwent Drug File 1069 Thesaurus DAPTOMYCIN DAUNORUBICIN DAUNORUBICIN-CYCLO= HEXYLIDINEHYDRAZONE DAUNORUBICINOL DB-2073 DC-81 DC-92-B DC-92-D DEACETOXYCEFALOTIN DEACETOXYCEPHALO= SPORIN-C DEACETYLCEFOTAXIME DEACETYLCEFOTAXIME-= LACTONE DEACETYLRAVIDOMYCIN DEALANYLASCAMYCIN DEAMIDOBLEOMYCIN-A2 DEAMIDOBLEOMYCIN-B2 DECILORUBICIN DEETHYLPIPERACILLIN DEFUCOGILVOCARCIN-V DEFUROYLCEFTIOFUR DEHYDROALTENUSIN DEHYDROFALCARINDIOL DEHYDROXYASPOXICILLIN DEHYDROXYSPARSOMYCIN DELAMINOMYCIN-A DELAMINOMYCIN-B DELAMINOMYCIN-C DELTAMYCIN-A1 DELTAMYCIN-A1-P1 DELTAMYCIN-A2 DELTAMYCIN-A2-P1 DELTAMYCIN-A2-P2 DELTAMYCIN-A2-P3 DELTAMYCIN-A3 DEMECLOCYCLINE DEMECYCLINE DEMETHOXYFLOMOXEF DEMETHOXYVIRIDIN DEMETHYLALLOSAMIDIN DEMETHYLBLEOMYCIN-A2 DEMETHYLCHARTREUSIN-= 3++ DEMETHYLCHROMO= MYCIN-A2 DEMETHYLCHROMO= MYCIN-A3 DEMETHYLERYTHRO= MYCIN-N DEMETHYLGRISEOFULVIN-6 DEMETHYLLINCOMYCIN DEMETHYLMEROPENEM-1 DEMETHYLOLIVOMYCIN-A DEMETHYLOLIVOMYCIN-B DEMETHYLRAPAMYCIN-O-27 DEMETHYLVANCOMYCIN-N DEOXYAKLAVINONE-7 DEOXYCARUBICIN-13 DEOXYCARUBICIN-6 DEOXYDAUNORUBICIN-11 DEOXYDAUNORUBICINONE-= 11 DEOXYERYTHROMYCIN-A-6 DEOXYFRENOLICIN DEOXYGALACTOSTATIN-1 DEOXYGALACTOSTATIN-1 DEOXYNARGENICIN-A1-18 DEOXYNOGAROL-7 DEOXYNOJIRIMYCIN-1 DEOXYNOJIRIMYCIN-1-= METHYL-N DEOXYOXANOSINE-2+ DEOXYSALINOMYCIN DEOXYSANGIVAMYCIN-2+ DEOXYSPERGUALIN DEOXYTOYOCAMYCIN-2+ DEOXYTUBERCIDIN-2+ DERMASEPTIN DESERTOMYCIN DESMYCOSIN DESTOMYCIN-A DETALLIPTINIUM DETHIATHIENAMYCIN DETORUBICIN DF-100 DIALLYL-TRISULFIDE DIANEMYCIN DIAZAQUINOMYCIN-A DIAZAQUINOMYCIN-B DIBEKACIN DIBENZYLDAUNORUBICIN-N,N DICLOXACILLIN DIDEMNENONE-A DIDEMNENONE-B DIDEOXYGRISEORHODIN-C DIDEOXYKANAMYCIN-B-= 3+,4+ DIFFICIDIN DIHYDROCICLOSPORIN DIHYDROCYCLOSPORIN-C DIHYDROCYTOCHALASINE-B DIHYDROERYTHROMYCIN-9 DIHYDROFLUSTRAMINE-C DIHYDROGRANATICIN-B DIHYDROHALICHONDRAMIDE DIHYDROILLUDIN-M DIHYDRONEPLANOCIN-D DIHYDROROSARAMICIN DIHYDROSTREPTOMYCIN DIHYDROTANSHINONE-I DIMETHYL-FUMARATE DIMETHYLDAUNORUBICIN-= N,N DINACTIN DIPHENICILLIN DIPLOICIN DIPROLEANDOMYCIN DIRITHROMYCIN DISCODERMIN-A DISCORHABDIN-D DISTAMYCIN-2 DISTAMYCIN-5 DISTAMYCIN-A DITETRACYCLINE DITRISARUBICIN-A DITRISARUBICIN-B DIUMYCIN DN-9550 DNACIN-A1 DNACIN-B1 DOB-41 DOLABELLANIN-A DON DORRIGOCIN-A DORRIGOCIN-B DOXORUBICIN DOXYCYCLINE DOXYSEPTIN DQ-2556 DRIMENINE DU-6681-A DU-86 DUAZOMYCIN DUCLAUXIN DUNAIMYCIN-A1 DUNAIMYCIN-C2 DUNAIMYCIN-D2 DUNAIMYCIN-D2S DUNAIMYCIN-D3 DUNAIMYCIN-D4S DUOCARMYCIN-A DUOCARMYCIN-B1 DUOCARMYCIN-B2 DUOCARMYCIN-C1 DUOCARMYCIN-C2 DUOCARMYCIN-SA DURAMYCIN DURAMYCIN-B DURAMYCIN-C DX-52-1 DX-8739 DYNEMICIN-A DYNEMICIN-H DYNEMICIN-M DYNEMICIN-N DYSIDAZIRINE E-0702 E-1077 E-1100 E-1101 E-4868 ECHINOCANDIN-B ECHINOCANDIN-C ECHINOCANDIN-D ECHINOMYCIN ECHINOSIDE-B ECHINOSPORIN EDEINE EDEINE-A EDEINE-B EFRAPEPTIN-D EFRAPEPTIN-F EFROTOMYCIN ELACTOCIN ELAIOMYCIN ELAIOPHYLIN ELEUTHERIN ELLORAMYCIN ELLORAMYCIN-B ELLORAMYCIN-C ELLORAMYCIN-D ELLORAMYCIN-E ELSAMICIN ELSAMICIN-A ELSAMICIN-B EMERIMICIN EMERIMICIN-3 EMERIMICIN-4 EMESTRIN EMIMYCIN EMODINANTHRONE EMPEDOPEPTIN ENACTIN-IA ENACTIN-IB1 ENACTIN-IB2 ENACTIN-VA ENACYLOXIN-II ENDOMYCIN ENDURACIDIN ENDURACIDIN-A ENDURACIDIN-B ENNIATIN ENNIATIN-A ENNIATIN-B ENOPEPTIN-A ENTEROCIN ENVIOMYCIN EPELMYCIN-A EPELMYCIN-B EPELMYCIN-C EPELMYCIN-D EPIANHYDROTETRACYCLINE EPICILLIN EPIDERMIN EPIDERSTATIN EPIDOXYCYCLINE-4 EPIDOXYCYCLINE-6 EPINIGERICIN EPIPENTALENOLACTONE-F EPIPENTENOMYCIN-I EPIPOLASIN-A EPIRUBICIN

1070 APPENDIX D EPIRUBICINOL EPITHIENAMYCIN-6 EPITHIENAMYCIN-A EPITHIENAMYCIN-B EPITHIENAMYCIN-C EPITHIENAMYCIN-D EPITHIENAMYCIN-E EPONEMYCIN EPOXYQUINOMICIN-A EPOXYQUINOMICIN-B ER-35786 ER-42859 ERBSTATIN EREMOMYCIN EREMOMYCIN-PSI ERTAPENEM ERYCYCLINE ERYTHRALOSAMINE ERYTHROMYCIN ERYTHROMYCIN-ACETATE-2+ ERYTHROMYCIN-ACISTRATE ERYTHROMYCIN-BUTYRATE ERYTHROMYCIN-C ERYTHROMYCIN-= CARBONATE-CYCLIC-11,12 ERYTHROMYCIN-E ERYTHROMYCIN-ESTOLATE ERYTHROMYCIN-= ETHYLCARBONATE ERYTHROMYCIN-= ETHYLSUCCINATE ERYTHROMYCIN-= GLUCEPTATE ERYTHROMYCIN-= LACTOBIONATE ERYTHROMYCIN-= PROPIONATE ERYTHROMYCIN-STEARATE ERYTHROMYCIN-STINOPRATE ERYTHROMYCIN-SUCCINATE ERYTHROMYCIN-VALERATE ERYTHROMYCYLAMINE ESORUBICIN ESPERAMICIN ESPERAMICIN-A1 ESPERAMICIN-A1B ESPERAMICIN-A2 ESPERAMICIN-C ESPERAMICIN-D ESPERAMICIN-E ESPERAMICIN-X ESPERAMICIN-Z ESTERASTIN ETAMOCYCLINE ETAMYCIN ETAMYCIN-II ETHEROMYCIN ETHISOLIDE ETISOMICIN EUDISTOMIN-C EUDISTOMIN-D EUDISTOMIN-H EUDISTOMIN-I EUDISTOMIN-K EUDISTOMIN-L EUDISTOMIN-P EUDISTOMIN-Q EUDISTOMIN-T EUROPINE EVERNINOMICIN-D EVEROLIMUS FACTUMYCIN FAD-001 FAERIEFUNGIN-A FAERIEFUNGIN-A FAERIEFUNGIN-B FALCARINDIOL FALCARINOL FAROPENEM FASCAPLYSIN FATTIVIRACIN-FV-8 FCE-20635 FCE-22101 FCE-22250 FCE-22807 FCE-23762 FCE-24362 FCE-25199 FCE-25450-A FCE-28068 FD-594 FELDAMYCIN FENBENICILLIN FERENSIMYCIN-A FERENSIMYCIN-B FERVENULIN FEUDOMYCIN-B FEUDOMYCIN-D FIBRACILLIN FILIPIN FK-037 FK-041 FK-089 FL-120-A FL-120-B FL-120-B+ FL-120-C FL-120-C+ FL-120-D+ FL-120A FL-120B FL-120B+ FL-120C FL-120C+ FL-120D+ FLAVIDULOL-A FLAVIDULOL-B FLAVIDULOL-C FLAVIPIN FLAVIPUCINE FLAVOFUNGIN FLAVOPENTIN FLOMOXEF FLORFENICOL FLU-401 FLU-402 FLUCLOXACILLIN FLUDALANINE FLUORODAUNORUBICIN-2+ FLUOROFORMYCIN-2 FLUOROIDARUBICIN-2 FLUOROIDARUBICIN-3 FLURITHROMYCIN FLURITHROMYCIN-= ETHYLSUCCINATE FLUVIRUCIN-A1 FLUVIRUCIN-A2 FLUVIRUCIN-B1 FLUVIRUCIN-B2 FLUVIRUCIN-B3 FOMIDACILLIN FORMADICIN-A FORMADICIN-B FORMADICIN-C FORMADICIN-D FORMAMICIN FORMYCIN FORMYCIN-B FORMYLRIFAMYCIN-3 FORSYTHIASIDE FORTIMICIN-B FOSFOMYCIN FOSMIDOMYCIN FOSTRIECIN FR-10024 FR-131535 FR-17126 FR-182024 FR-21818 FR-66973 FR-66979 FR-66980 FR-900109 FR-900405 FR-900482 FR-900848 FR-901469 FRAMYCETIN FREDERICAMYCIN-A FRENOLICIN FRENOLICIN-B FRIDAMYCIN-E FRONTALIN FULVOPLUMIERIN FUMAGILLIN FUNGIMYCIN FUNICULOSIN FURAMPICILLIN FURANOMYCIN FURAQUINOCIN-A FURAQUINOCIN-B FURAQUINOCIN-C FURAQUINOCIN-D FURAQUINOCIN-E FURAQUINOCIN-F FURAQUINOCIN-G FURBENICILLIN FURBUCILLIN FUSACANDIN-A FUSACANDIN-B FUSAFUNGINE FUSARENONE FUSARUBIN FUSCIN FUSIDATE FUSIDATE SODIUM FUZLOCILLIN GALACTOSTATIN GALANTIN-I GALBONOLIDE-A GALBONOLIDE-B GALTAMYCIN GAR-936 GC-1993 GE-2270-A GE-2270A GE-3 GE-3-B GE-37468-A GECLOSPORIN GEDAMYCIN GELDANAMYCIN GEMTUZUMAB OZOGAMICIN GENETICIN GENTAMYCIN GENTAMYCIN-A GENTAMYCIN-B GENTAMYCIN-C1 GENTAMYCIN-C1A GENTAMYCIN-C2 GENTAMYCIN-C2A GILVOCARCIN-M GILVOCARCIN-V GIRINIMBINE GLADIOLATE GLIDOBACTIN-A GLIDOBACTIN-B GLIDOBACTIN-C GLIOTOXIN GLIOVIRIN GLOBOMYCIN GLOMOSPORIN GLUCOPIERICIDIN-A

Derwent Drug File 1071 Thesaurus GLUCOSONE GLUFOSINATE GLUTAMYCIN GLYCINMETHYLTETRACYCLINE GLYCOTHIOHEXIDE-ALPHA GLYCYCOUMARIN GLYKENIN-III-A GLYKENIN-III-B GLYKENIN-III-C GLYKENIN-IIIA GLYKENIN-IIIB GLYKENIN-IIIC GOLDINODOX GOUGEROTIN GR-122222-X GR-69153 GRAHAMIMYCIN-A1 GRAMICIDIN GRAMICIDIN-A GRAMICIDIN-D GRAMICIDIN-J2 GRAMICIDIN-NF GRAMICIDIN-S GRAMICIDIN-S-2 GRAMICIDIN-S-3 GRANATICIN GRANATICIN-A GRANATICIN-B GRANULYSIN GRIFOLIN GRISEOCHELIN GRISEOFULVIN GRISEORHODIN-C GRISEOVIRIDIN GRISEUSIN-A GRISEUSIN-B GRISORIXIN GUAMECYCLINE GUANIDYLFUNGIN-A GV-104326 GV-118819 GV-129606 HACHIMYCIN HADACIDIN HALENAQUINONE HALIMEDATRIAL HALISULFATE-1 HALOFUGINONE HAMYCIN HAPALINDOLE-E HAPALINDOLE-G HAPALINDOLE-H HAPALINDOLE-J HAPALINDOLE-M HAPALINDOLE-O HAPALINDOLE-U HAZIMYCIN-5 HAZIMYCIN-6 HEDAMYCIN HELIOMYCIN HELIQUINOMYCIN HELVECARDIN-A HELVECARDIN-B HELVOLATE HEPTAMYCIN HEPTELIDATE HEPTYLPENICILLIN HERBICOLIN-A HERBICOLIN-B HERBIMYCIN-A HERBIMYCIN-B HERBIMYCIN-C HETACILLIN HIBARIMICIN-A HIBARIMICIN-C HIBARIMICIN-D HIMASTATIN HINESOL HISTIDINOMYCIN HITACHIMYCIN HMR-3562 HMR-3787 HOLOTHURIN-B HOLOTOXIN-A1 HONGOQUERCIN-A HONGOQUERCIN-B HORMAOMYCIN HR-916-B HR-979 HRE-664 HUMULONE HYBRIMYCIN HYBRIMYCIN-A3 HYBRIMYCIN-B3 HYDROHEPTIN HYDROXYACIVICIN-4 HYDROXYACLARUBICIN-2 HYDROXYACLARUBICIN-II HYDROXYACTEOSIDE-BETA HYDROXYDOXORUBICIN-3+ HYDROXYETHYLCLAVAM HYDROXYFLUCLOXACILLIN HYDROXYMARASMATE-9-= BETA HYDROXYRUBICIN-D HYDROXYSTREPTOMYCIN HYDROXYUBENIMEX-PARA HYGROMYCIN-A HYGROMYCIN-B HYPELCIN-A HYPELCIN-A-III HYPERFORIN HYPNOPHILIN ICI-193428 ICI-194008 IDARUBICIN IKARUGAMYCIN IKD-8344 ILICICOLIN-C ILICICOLIN-H ILIMAQUINONE ILLUDIN ILLUDIN-C3 ILLUDIN-M ILLUDIN-S IMINODAUNORUBICIN-5 IMINODOXORUBICIN-5 IMIPENEM INDANOMYCIN INDISOCIN INDOLIZOMYCIN INDOLMYCIN INOSAMYCIN-A INOSAMYCIN-B INOSAMYCIN-C INOSAMYCIN-D INOSAMYCIN-E INOSTAMYCIN IODININ IODOAZOMYCIN-RIBOSIDE IODOPENICILLANATE IONOMYCIN IREMYCIN IRUMAMYCIN ISEPAMYCIN ISOAVENACIOLIDE ISOBLEOMYCIN-A2 ISOELEUTHERIN ISOGRISEOFULVIN ISOHEMATINATE ISOKIDAMYCIN ISOLASALOCID-A ISOMITOMYCIN-A ISONAPHTHOCYCLINONE-= GAMMA ISOPROPICILLIN ISOTRIKENTRIN-B-TRANS ISOVELLERAL ISTAMYCIN-A ISTAMYCIN-B IT-62-B ITURIN-A ITURIN-AL J-111225 J-114870 JAVANICIN JIETACIN-A JIETACIN-B JOSAMYCIN JOSAMYCIN-PROPIONATE JUGLOMYCIN-A JUGLOMYCIN-B JULIFLORINE JUNCUSOL K-4619 K-582-A KABIRAMIDE-C KALAFUNGIN KALIHINOL-A KALIHINOL-F KALIHINOL-X KALIHINOL-Y KALIHINOL-Z KALIMANTACIN-A KALIMANTACIN-B KALIMANTACIN-C KANAMYCIN KANAMYCIN-B KANAMYCIN-C KANAMYCIN-D KANCHANAMYCIN-A KANCHANAMYCIN-D KANOSAMINE KAPURIMYCIN-A1 KAPURIMYCIN-A2 KAPURIMYCIN-A3 KASUGAMYCIN KAZUSAMYCIN KAZUSAMYCIN-B KEDARCIDIN KELLETININ-I KENGSHENGMYCIN KERAMAMINE-B KERRIAMYCIN-A KERRIAMYCIN-B KERRIAMYCIN-C KETOMYCIN KIBDELIN-A KIBDELIN-B KIBDELIN-C1 KIBDELIN-C2 KIBDELLIN-D KIDAMYCIN KIJANIMICIN KINAMYCIN-C KINAMYCIN-D KISIMICIN KISTAMICIN-A KISTAMICIN-B KITASAMYCIN KJELLMANIANONE KOJATE KORBERIN-A KORBERIN-B KORMOGRISIN KORORMICIN KP-736 KRM-1648 KRM-1657 KRM-1668 KRM-1671 KRN-8602

1072 APPENDIX D KS-504A2 KS-504B KS-504D KS-504E KS-505A KT-3767 KT-3937 KT-4697 KT-4788 KW-2189 KY-106 KY-62 L-156602 L-62208 L-62211 L-640876 L-656575 L-659699 L-660631 L-683590 L-687781 L-688786 L-693989 L-694458 L-695256 L-696474 L-701677 L-733560 L-742728 L-749345 L-755805 L-786392 LABILOMYCIN LACHNELLULONE LACHNUMON-B1 LACHNUMON-B2 LACTENOCIN LACTIVICIN LACTOFERRICIN-B LACTOQUINOMYCIN LACTOQUINOMYCIN-A LAF-389 LAGOSIN LAGUNAMYCIN LAIDLOMYCIN LAIDLOMYCIN-BUTYRATE LAIDLOMYCIN-PROPIONATE LANDOMYCIN-A LANKACIDIN LANKACIDIN-A LANKACIDIN-C LANKACIDINOL-A LANKAMYCIN LANOMYCIN LANTHIOPEPTIN LARGOMYCIN LARGOMYCIN-F-II LASALOCID LASALOCID-A LASALOCID-B LASALOCID-C LASALOCID-D LASALOCID-E LASIOCARPINE-N-OXIDE LATAMOXEF LAVENDAMYCIN LAVENDAMYCIN-METHYL-= ESTER LAVENDOMYCIN LAVENDUSTIN-A LAXAPHYCIN-A LAXAPHYCIN-B LAXAPHYCIN-D LAXAPHYCIN-E LB-10827 LEINAMYCIN LENAMPICILLIN LENOREMYCIN LEPIOCHLORIN LEPTOMYCIN-A LEPTOMYCIN-B LEUCANICIDIN LEUCASCANDROLIDE-A LEUCINOSTATIN LEUCINOSTATIN-A LEUCINOSTATIN-B LEUCINOSTATIN-C LEUCINOSTATIN-D LEUCINOSTATIN-F LEUCINOSTATIN-H LEUCINOSTATIN-K LEUCOMYCIN-A1 LEUCOMYCIN-A5 LEUCOMYCIN-A7 LEUCOMYCIN-A9 LEUCOMYCIN-V LEUCYLNEGAMYCIN LEURUBICIN LEUSERAMYCIN LEVOERYTHROCYCLINE LEVOPROPICILLIN LEVORIN LEVOTETRASULFENE LIBLOMYCIN LICARIN-A LIDIMYCIN LIENOMYCIN LINCOMYCIN LINCOMYCIN-A LINCOMYCIN-B LINEARMYCIN-A LIPIARMYCIN LIPIARMYCIN-A3 LIPOSIDOMYCIN-A LIPOSIDOMYCIN-B LIPOSIDOMYCIN-C LIPOXAMYCIN LIRIODENINE LIVIDOMYCIN LL-14-I-352-ALPHA LL-AM-374 LL-AM374 LL-C10037-ALPHA LL-E-19020-ALPHA LL-E-19020-BETA LL-F28249-BETA LL-F28249-GAMMA LL-F28249-LAMBDA LL-S-491-BETA LL-Z-1271-ALPHA LL-Z-1272-EPSILON LOLOATIN-A LOLOATIN-B LOLOATIN-C LOMOFUNGIN LONOMYCIN LONOMYCIN-A LONOMYCIN-B LONOMYCIN-C LORACARBEF LUCIMYCIN LUCKNOMYCIN LUPULONE LUTEOSKYRIN LUZOPEPTIN LUZOPEPTIN-A LUZOPEPTIN-B LUZOPEPTIN-C LUZOPEPTIN-D LY-164846 LY-191145 LY-197221 LY-212556 LY-227409 LY-264656 LY-264826 LY-267108 LY-281389 LY-281980 LY-303366 LY-307599 LYDICAMYCIN LYMECYCLINE LYSINOMICIN LYSOBACTIN LYSOCELLIN LYSOLIPIN LYSOSTAPHIN M-14659 M-4365-G2 M-83 MA-144-M1 MA-144-N1 MACARBOMYCIN MACBECIN-I MACBECIN-II MACFARLANDIN-E MACLURAXANTHONE MACROCIN MACROLACTIN-A MACROLACTIN-B MACROLACTIN-E MACROLACTIN-F MACROLACTINATE MACROMOMYCIN MACROSPHELIDE-A MACROSPHELIDE-B MADUMYCIN-II MADURAMICIN MADURAMICIN-ALPHA MADUROPEPTIN MALEIMYCIN MALUCIDIN MALYNGOLIDE MANIWAMYCIN-A MANIWAMYCIN-B MANUMYCIN MANUMYCIN-G MANZAMINE-A MARASMATE MARCELLOMYCIN MARCHANTIN-A MARIDOMYCIN MARTINOMYCIN MASTOPARAN-17 MATLYSTATIN-A MATLYSTATIN-B MC-02479 MC-62 MC-77 MDL-19592 MDL-62208 MDL-62211 MDL-62873 MDL-63246 ME-1207 ME-1228 ME-2303 MECILLINAM MECILLINAM-ACETYL= METHYL-ESTER MECLOCYCLINE MEDERMYCIN MEDERRHODIN-A MEDERRHODIN-B MEDICAGENATE-= GLUCOSIDE-3 MEDIOCIDIN MEDORUBICIN MEGALOMICIN MEGALOMICIN-C MEGLUCYCLINE

Derwent Drug File 1073 Thesaurus MEGOVALICIN-A MEGOVALICIN-D MEGOVALICIN-G MEGOVALICIN-H MELANOCIDIN-A MELANOCIDIN-B MEN-10397 MEN-10400 MEN-10700 MENENSIN-B MEPARTRICIN MEPARTRICIN-A MEPARTRICIN-B MER-WF-3010 MEROPENEM MERSACIDIN MERULIDIAL METACYCLINE METACYCLOPRODIGIOSINE METAMPICILLIN METHOCIDIN METHOXYCARBAZO= MYCINAL-6 METHOXYHYGROMYCIN METHOXYSTROBILURIN-K-9 METHYL-ORSELLINATE-= ORTHO METHYLBETACLAMYCIN-= T,4-O METHYLENOLACTOCIN METHYLENOMYCIN-A METHYLENOMYCIN-B METHYLFORMYCIN-4 METHYLGLABRIDIN-4+-O METHYLIMIPENEM-1-BETA METHYLINDISOCIN-N METHYLTHIENAMYCIN-1-= BETA METHYMYCIN METICILLIN MEZLOCILLIN MICACOCIDIN MICACOCIDIN-A MICACOCIDIN-B MICACOCIDIN-C MICROCIN-7 MICROCIN-B17 MICROCIN-E492 MICROCIN-J25 MICROCOCCIN-P MICROCOCCIN-P1 MICRONOMICIN MICROTHECIN MIDECAMYCIN MIKAMYCIN MILBEMYCIN-A MILBEMYCIN-ALPHA-3 MILBEMYCIN-B-41D MILBEMYCIN-BETA-1 MILBEMYCIN-BETA-3 MILBEMYCIN-D MILBEMYCIN-E MILBEMYCIN-G MILDIOMYCIN MIMIMYCIN MIMOCIN MIMOSAMYCIN MINOCYCLINE MINOSAMINOMYCIN MIOKAMYCIN MIRINCAMYCIN MIROSAMICIN MITOGILLIN MITOMYCIN MITOMYCIN-A MITOMYCIN-B MITOMYCIN-D MITOMYCIN-F MITOMYCIN-G MITOMYCIN-H MITOMYCIN-K MITOSPER MIZORIBINE MM-17880 MM-22381 MM-22382 MM-44785 MM-44787 MM-4550 MM-46115 MOCIMYCIN MOENOMYCIN-A MONACTIN MONAMYCIN MONATE-A MONAZOMYCIN-A MONAZOMYCIN-B MONENSIN MONENSIN-A MONENSIN-B MONENSIN-C MONOGAGAINE MONOMYCIN MONORDEN MORPHOCYCLINE MORPHOLINODAUNORUBICIN MOYUKAMYCIN MS-8209 MSD-235-S2 MSD-819 MT-0703 MT-81 MULUNDOCANDIN MUPIROCIN MUREIDOMYCIN-A MUREIDOMYCIN-B MUREIDOMYCIN-C MUREIDOMYCIN-D MUREIDOMYCIN-F MUSCORIDE-A MUSETTAMYCIN MUTALOMYCIN MUTILIN MX MX-2 MY-5 MYCINAMICIN MYCINAMICIN-I MYCINAMICIN-III MYCINAMICIN-IV MYCINAMICIN-V MYCINAMICIN-VI MYCINAMICIN-VII MYCOBACILLIN MYCOBACTIN MYCOHEPTIN MYCOPENTEN MYCOPHENOLATE MYCOPLANECIN-A MYCORRHIZIN-B1 MYCORRHIZIN-B2 MYCOSUBTILIN MYCOTICIN-A MYCOTICIN-B MYCOTRIENIN-I MYCOTRIENIN-II MYCOVERSILIN MYOMYCIN MYRIOCIN MYROCIN-C MYRTUCOMMULONE-A MYRTUCOMMULONE-B MYXALAMIDE-A MYXALAMIDE-B MYXALAMIDE-C MYXALAMIDE-D MYXIN MYXOPYRONIN-A MYXOPYRONIN-B MYXOTHIAZOL MYXOVIRESCIN-A MYXOVIRESCIN-A1 MYXOVIRESCIN-A2 MYXOVIRESCIN-B NA-22598-A-1 NAFCILLIN NAFCILLIN-SULFONE NANAFROCIN NANAOMYCIN-D NANAOMYCIN-E NANNOCHELIN-A NAPHTHGERANINE-A NAPHTHOCYCLINONE-ALPHA NAPHTHOCYCLINONE-BETA NAPHTHOCYCLINONE-DELTA NAPHTHOCYCLINONE-= EPSILON NAPHTHOCYCLINONE-= GAMMA NAPHTHOMYCIN NAPHTHOMYCIN-A NAPHTHOMYCIN-B NAPHTHOMYCIN-C NAPHTHOMYCIN-H NAPHTHOPYRANOMYCIN NAPHTHYRIDINOMYCIN NAPYRADIOMYCIN-A1 NAPYRADIOMYCIN-A2 NAPYRADIOMYCIN-B1 NAPYRADIOMYCIN-C1 NAPYRADIOMYCIN-C2 NARASIN NARBOMYCIN NARGENICIN-A1 NATAMYCIN NEBRAMYCIN-4 NEBULARINE NEGAMYCIN NEIHUMICIN NEMADECTIN NEMOTIN NEO-ENACTIN-A NEO-ENACTIN-B1 NEO-ENACTIN-B2 NEO-ENACTIN-M2 NEO-ENACTIN-NL1 NEO-ENACTIN-NL2 NEOAUREOTHIN NEOCARZILIN-A NEOCRYPTOLEPINE NEOISOMIDECAMYCIN NEOMYCIN NEOMYCIN-A NEOMYCIN-C NEOOXAZOLOMYCIN NEOPYRROLOMYCIN NEOSIDOMYCIN NEOTHRAMYCIN NEOTHRAMYCIN-A NEOTHRAMYCIN-B NEOVIRIDOGRISEIN-II NEPLANOCIN-A NEPLANOCIN-C NEPLANOCIN-D NETILMICIN NETROPSIN NETZAHUALCOYONE NEUTRAMYCIN NIDDAMYCIN NIDULIN NIGERICIN NIKKOMYCIN-B

1074 APPENDIX D NIKKOMYCIN-BX NIKKOMYCIN-I NIKKOMYCIN-J NIKKOMYCIN-KX NIKKOMYCIN-KZ NIKKOMYCIN-OX NIKKOMYCIN-OZ NIKKOMYCIN-PSEUDO-J NIKKOMYCIN-PSEUDO-Z NIKKOMYCIN-WX NIKKOMYCIN-WZ NIKKOMYCIN-X NIKKOMYCIN-Z NIKKOMYCIN-ZH NIKKOMYCIN-ZT NIPHIMYCIN-I NISIN NITROCEFIN NITROCYCLINE NITROSOFUNGIN NIVALENOL NOBORITOMYCIN-A NOBORITOMYCIN-B NOCARDICIN-A NOCARDICIN-B NOCARDICIN-C NOCARDICIN-G NOCARDICYCLIN-A NODUSMICIN NOGALAMYCIN NOJIRIMYCIN NONACTIN NONYL-DEOXY= NOJIRIMYCIN-N NONYLOXYCARBONYL-= MITOMYCIN NORBORITOMYCIN-A NORBORITOMYCIN-B NORDENTATIN NORJAVANICIN NORPYRENOPHORIN NOSIHEPTIDE NOURSEOTHRICIN NOVOBIOCIN NSC-143414 NSC-255110 NSC-330507 NSC-354646 NSC-357704 NUCLEOCIDIN NUCLEOTICIDIN NYBOMYCIN NYSTATIN NYSTATIN-A1 NYSTATIN-A2 NYSTATIN-A3 OA-6129A OA-6129B1 OA-6129B2 OA-6129C OA-7653 OBAFLUORIN OBELMYCIN-A OBELMYCIN-B OBELMYCIN-C OBELMYCIN-D OBELMYCIN-E OBELMYCIN-F OBELMYCIN-G OCHROLIFURANINE-A OCTACIDOMYCIN OCTAPEPTIN OIDIOLACTONE-A OKILACTOMYCIN OLEANDOMYCIN OLIGOMYCIN OLIGOMYCIN-A OLIGOMYCIN-B OLIGOMYCIN-C OLIVOMYCIN OLIVOMYCIN-A OLIVOMYCIN-B OLIVOMYCIN-C OLIVOMYCIN-D OMOMYCIN OPHIOBOLIN-A OPHIOCORDIN ORIENTICIN-A ORITAVANCIN OSTHENOL OSTREOGRYCIN OSTREOGRYCIN-B3 OTIVARIN OUDEMANSIN OUDEMANSIN-A OUDEMANSIN-B OUDEMANSIN-X OVALICIN OXACILLIN OXANOSINE OXANTHROMICIN OXAUNOMYCIN OXAZINOMYCIN OXAZOLOMYCIN OXECLOSPORIN OXETACILLIN OXETANOCIN-A OXETIN OXIMONAM OXIRAPENTYN OXOFORMYCIN OXOFORMYCIN-B OXOSTAUROSPORINE-7 OXYDIFFICIDIN OXYTETRACYCLINE PACIDAMYCIN-1 PACIDAMYCIN-2 PACIDAMYCIN-3 PACIDAMYCIN-5 PACTAMYCIN PALDIMYCIN PALDIMYCIN-A PALDIMYCIN-B PALOMINOL PAMAMYCIN-607 PANIPENEM PAPUAMINE PAPULACANDIN PAPULACANDIN-A PAPULACANDIN-B PAPULACANDIN-C PAPULACANDIN-D PAPYRACON-A PARACELSIN PARACELSIN-A PARACELSIN-B PARACELSIN-C PARACELSIN-D PARADOL-6 PAROMAMINE PAROMOMYCIN PARTRICIN PARTRICIN-A PARTRICIN-B PARVISPORIN PARVODICIN-B2 PARVODICIN-C1 PARVODICIN-C3 PATRICIN PATRICIN-A PATRICIN-B PATULIN PATULOLIDE-A PATULOLIDE-B PATULOLIDE-C PAULOMYCIN PAULOMYCIN-A PAULOMYCIN-A2 PAULOMYCIN-B PAULOMYCIN-C PAULOMYCIN-D PAULOMYCIN-E PAULOMYCIN-F PC-766B PD-113270 PD-113271 PD-113876 PD-114027 PD-114631 PD-116152 PD-116198 PD-116250 PD-116740 PD-118309 PECILOCIN PECOCYCLINE PECTINATONE PELIOMYCIN PENAMECILLIN PENDOLMYCIN PENETHACILLIN PENICILLANATE PENICILLATE PENICILLIN-M PENICILLIN-X PENIMEPICYCLINE PENIMOCYCLINE PENITRICIN PENITRICIN-A PENITRICIN-B PENITRICIN-C PENTABROMOPSEUDILINE PENTALENOLACTONE PENTALENOLACTONE-E PENTALENOLACTONE-F PENTALENOLACTONE-G PENTALENOLACTONE-H PENTALENOLACTONE-O PENTALENOLACTONE-P PENTENOMYCIN PENTENOMYCIN-1 PENTENOMYCIN-2 PENTISOMICIN PENTIZIDONE PENTOSTATIN PENTYLSPARSOMYCIN PEP-5 PEPLOMYCIN PEPTICINNAMIN-E PERENIPORIN-A PERENIPORIN-B PERIMYCIN PERVICOSIDE-A PERVICOSIDE-B PERVICOSIDE-C PETROSYNOL PF-1163-A PHACIDIN PHAEANTHARINE PHENALAMIDE-A1 PHENAZINOMYCIN PHENCOMYCIN PHENELFAMYCIN-A PHENELFAMYCIN-B PHENELFAMYCIN-C PHENELFAMYCIN-E PHENELFAMYCIN-F PHENETICILLIN PHENOMYCIN PHENOXAN PHENOXYMETHYLPENICILLIN PHENYLAZOXYCYANIDE

Derwent Drug File 1075 Thesaurus PHENYRACILLIN PHLEOMYCIN PHLEOMYCIN-D1 PHLEOMYCIN-E PHLEOMYCIN-G PHOLIPOMYCIN PHOMALACTONE PHOMENOATE PHOSALACINE PHOSPHINOTHRICIN PHOSPHOLINE (antibiotic = cytostatic) PHTHIOCOL PICROMYCIN PIERICIDIN-A PILATIN PIPACYCLINE PIPERACILLIN PIPERAZINOMYCIN PIRARUBICIN PIRARUBICIN PIRAZMONAM PIRBENICILLIN PIRIDICILLIN PIRLIMYCIN PIRLIMYCIN-ADENYLATE PIROXICILLIN PISATIN PISIFERATE PIVAMPICILLIN PIVMECILLINAM PL-385 PLD-118 PLEUROMULIN PLEUROTIN PLICACETIN PLICAMYCIN PLUMERICIN PLURAMYCIN-A PLUSBACIN-A1 PLUSBACIN-A2 PLUSBACIN-A3 PLUSBACIN-A4 PLUSBACIN-B1 PLUSBACIN-B2 PLUSBACIN-B3 PLUSBACIN-B4 PNEUMOCANDIN-A0 PNEUMOCANDIN-A1 PNEUMOCANDIN-A2 PNEUMOCANDIN-A3 PNEUMOCANDIN-A4 PNEUMOCANDIN-B0 PNEUMOCANDIN-B2 PNEUMOCANDIN-C0 PNU-145156-E PODOSPORIN-A POLYMYXIN-B POLYMYXIN-B-NONAPEPTIDE POLYMYXIN-B1 POLYMYXIN-B2 POLYMYXIN-D POLYMYXIN-M POLYOXIN POLYOXIN-A POLYOXIN-B POLYOXIN-C POLYOXIN-D POLYOXIN-E POLYOXIN-F POLYOXIN-G POLYOXIN-H POLYOXIN-I POLYOXIN-J POLYOXIN-K POLYOXIN-L POLYOXIN-M POLYOXIN-N PORFIROMYCIN POROTHRAMYCIN-B PORTMICIN PR-19 PRADIMICIN-A PRADIMICIN-B PRADIMICIN-S PRADIMICIN-T1 PRADIMICIN-T2 PRAMANICIN PRASINOMYCIN PRAZOCILLIN PREUSSIN PREUSSOMERIN-D PREUSSOMERIN-E PREUSSOMERIN-F PREUSSOMERIN-G PREUSSOMERIN-H PREUSSOMERIN-I PRIMYCIN PRISTINAMYCIN PRISTINAMYCIN-IA PRISTINAMYCIN-IB PRISTINAMYCIN-IC PROCAINE-BENZYLPENICILLIN PRODIGIOSINE PROPICILLIN PROPIKACIN PROTEGRIN-1 PROTHRACARCIN PROTOANEMONIN PROTOLICHESTERATE PROTOMYCINOLIDE-IV PROTYLONOLIDE PRUMYCIN PS-5 PS-5-EPI-6 PS-6 PS-7 PS-990 PSAMMAPLIN-A PSAMMAPLYSIN-A PSAMMAPLYSIN-B PSEUDOMONATE PSEUDOMONATE-A PSEUDOMONATE-B PSEUDOMONATE-C PSEUDOMONATE-D PSEUDOMYCIN-C+ PSICOFURANINE PUNCTATIN-A PUNCTATIN-B PUNCTATIN-D PUROMYCIN PUROMYCIN-AMINO= NUCLEOSIDE PURPUROMYCIN PYLORICIDIN-A PYLORICIDIN-B PYLORICIDIN-C PYOLUTEORINE PYRAZOMYCIN PYRENOPHORIN PYRIDOMYCIN PYRIZINOSTATIN PYRROINDOMYCIN-A PYRROINDOMYCIN-B PYRROLNITRIN PYRROLOMYCIN-B PYRROLOMYCIN-C PYRROLOMYCIN-D PYRROLOMYCIN-E PYRROLOMYCIN-F1 PYRROLOSPORIN-A PYRROMYCIN PYRROXAMYCIN QUADRIGEMINE-C QUARTROMICIN-A1 QUARTROMICIN-A2 QUARTROMICIN-A3 QUARTROMICIN-D1 QUELAMYCIN QUINACILLIN QUINOCARCIN QUINOCARCINOL QUINOCARMYCIN QUINOLACTACIN-A QUINOLACTACIN-B QUINOMYCIN-C QUINUPRISTIN R-45656 R-95867 RABELOMYCIN RACEFENICOL RAMONTOSIDE RAMOPLANIN RAPAMYCIN RAPANONE RATANHIAPHENOL-I RATANHIAPHENOL-II RAVIDOMYCIN REBECCAMYCIN REDUCTIOMYCIN RELOMYCIN RENIERAMYCIN-A RENIERONE REPROMICIN RES-1149-1 RES-1149-2 RESISTOFLAVIN RESISTOMYCIN RESORCINOMYCIN-A RESORTHIOMYCIN RESPINOMYCIN-A1 RESPINOMYCIN-A2 RESPINOMYCIN-B RESPINOMYCIN-C RESPINOMYCIN-D RESTRICTICIN RESTRICTOCIN RETUSIN REUMYCIN REVEROMYCIN-A REVEROMYCIN-B REVEROMYCIN-C REVEROMYCIN-D RHIZOCHALIN RHIZOXIN RHIZOXIN-D RHODOMYCIN-A RHODOMYCIN-B RHODOMYCIN-I-BETA RHODOMYCINONE-BETA RI-331 RIBOSTAMYCIN RIFABUTIN RIFAMIDE RIFAMPICIN RIFAMPICIN-QUINONE RIFAMYCIN RIFAMYCIN-B RIFAMYCIN-O RIFAMYCIN-S RIFAMYCIN-W RIFAPENTINE RIFAXIMIN RIMOCIDIN RIPOSTATIN-A RIPOSTATIN-B RISTOCETIN RISTOCETIN-A RISTOCETIN-B RISTOCETIN-PSI RITIPENAM-ACOXIL

1076 APPENDIX D RITIPENEM RK-397 RMI-15307 RO-07-3149 RO-09-1428 RO-13-3892 RO-13-9259 RO-15-8074 RO-22-5851 RO-23-6829 RO-23-9424 RO-24-4383 RO-24-6392 RO-24-8138 RO-25-6833 RO-31-1215 RO-31-1740 RO-31-1741 RO-31-1749 RO-31-1966 RO-31-2035 RO-40-6890 RO-41-3399 RO-45-2081 RODAPLUTIN RODORUBICIN ROFLAMYCOIN ROKITAMYCIN ROLITETRACYCLINE RORITOXIN-A ROSAMICIN-P1 ROSARAMICIN ROSEOFUNGIN ROTAMICILLIN ROUTIENNOCIN ROXATICIN ROXITHROMYCIN RP-20132 RP-59500 RR-150 RS-22-A RS-22-B RS-22-C RU-004 RU-23345 RU-25159 RU-25328 RU-25519 RU-29065 RU-29702 RU-399 RU-44790 RU-469 RU-64004 RU-66647 RU-69874 RUBAMPICIN RUBEOMYCIN-A RUBEOMYCIN-A1 RUBEOMYCIN-B RUBICIN-1-ALPHA RUBICYCLAMIN RUBIFLAVIN RUBIFLAVIN RUBOMYCIN-F RUBOMYCIN-H RUBOXYL RUBRADIRIN RUDOLPHOMYCIN RUFOCROMOMYCIN RUTAMYCIN RUTAMYCIN-B S-1006 S-1090 S-4661 S-5556 S-810592 SACCHAROCIN SAFRACIN-A SAFRACIN-B SAFRAMYCIN-A SAFRAMYCIN-AD-1 SAFRAMYCIN-B SAFRAMYCIN-C SAFRAMYCIN-D SAFRAMYCIN-F SAFRAMYCIN-G SAFRAMYCIN-H SAFRAMYCIN-MX-1 SAFRAMYCIN-R SAFRAMYCIN-S SAFRAMYCIN-Y2B SAFRAMYCIN-Y2B-D SAFRAMYCIN-Y3 SAFRAMYCIN-YD-1 SAFRAMYCIN-YD-2 SAINTOPIN SAKYOMICIN-A SAKYOMICIN-B SAKYOMICIN-C SAKYOMICIN-D SALINOMYCIN SANCYCLINE SANDRAMYCIN SANGIVAMYCIN SANGUINARINE SAPHENAMYCIN SAPTOMYCIN-A SAPTOMYCIN-B SAPTOMYCIN-C1 SAPTOMYCIN-C2 SAPTOMYCIN-D SAPTOMYCIN-E SAPTOMYCIN-F SAPTOMYCIN-G SAPTOMYCIN-H SAPURIMYCIN SARCIN-ALPHA SARKOMYCIN SARKOMYCIN-A SARMOXICILLIN SARPICILLIN SARUBICIN-A SB-205952 SB-219383 SB-22484-1 SB-22484-2 SB-22484-3 SB-22484-4 SCE-20 SCH-21561 SCH-24893 SCH-25393 SCH-28191 SCH-29482 SCH-32260 SCH-33256 SCH-34164 SCH-34343 SCH-36606 SCH-37137 SCH-38518 SCH-38519 SCH-40873 SCH-50673 SCH-53174 SCYTOPHYCIN-B SCYTOPHYCIN-C SCYTOPHYCIN-D SCYTOPHYCIN-E SE-16 SELDOMYCIN SEMDURAMICIN SEPTAMYCIN SERRATAMOLIDE SETAMYCIN SF-2140 SF-2315-A SF-2315B SF-2324 SF-2361 SF-2370 SF-2446-A1 SF-2446-A2 SF-2446-A3 SF-2446-B1 SF-2446-B2 SF-2446-B3 SF-2487 SF-2575 SHOWDOMYCIN SIAMYCIN-I SIAMYCIN-II SIBIROMYCIN SICCANIN SIGMOIDIN-A SIGMOIDIN-B SIMAOMICIN-ALPHA SINEFUNGIN SISOMICIN SIWENMYCIN SKF-101542 SKF-102010 SKF-103658 SKF-104093 SKF-104214 SKF-104420 SKF-104421 SKF-104428 SKF-104662 SKF-105285 SKF-107647 SKF-88070 SMEGMATOCIN SMENOQUINONE SMENORTHOQUINONE SMENOSPONDIOL SMENOSPONGIARINE SMENOSPONGIDINE SMENOSPONGINE SN-38 SO-75R1 SORANGICIN-A SORANGICIN-B SORANGIOLIDE-A SORBISTIN-A1 SPA-S-565 SPA-S-717 SPA-S-753 SPA-S-843 SPARSOMYCIN SPECTINOMYCIN SPENOLIMYCIN SPERABILLIN-D SPERGUALIN SPHINGOFUNGIN-A SPHINGOFUNGIN-B SPHINGOFUNGIN-C SPHINGOFUNGIN-D SPICAMYCIN SPINAMYCIN SPIRAMYCIN SPIRAMYCIN-A SPIRAMYCIN-B SPIRAMYCIN-C SPIROTRYPROSTATIN-A SPIROTRYPROSTATIN-B SPORANGIOMYCIN SPORARICIN-A SPORAVIRIDIN SPORAVIRIDIN-A1 SPORAVIRIDIN-A2

Derwent Drug File 1077 Thesaurus SPORAVIRIDIN-B1 SPORAVIRIDIN-B2 SPORAVIRIDIN-C1 SPORAVIRIDIN-C2 SPOREAMICIN-A SQ-14359 SQ-26180 SQ-26324 SQ-26559 SQ-26630 SQ-26668 SQ-26917 SQ-27327 SQ-27629 SQ-27860 SQ-67590 SQ-81377 SQ-81387 SQ-81402 SQ-81427 SS-228-R SS-228-Y SS-56C STACHYBOTRIN-C STAUROSPORINE STEFFIMYCIN STEFFIMYCIN-D STEMPHOL STEMPHYPERYLENOL STICHOPOSIDE-A STIGMATELLIN STIGMATELLIN-A STRAVIDIN STRAVIDIN-S2 STRAVIDIN-S3 STREPTAZOLIN STREPTIMIDONE STREPTOGRAMIN STREPTOLYDIGIN STREPTOMYCIN STREPTOMYCIN-B STREPTOTHRICIN STREPTOTHRICIN-B STREPTOTHRICIN-C STREPTOTHRICIN-D STREPTOTHRICIN-E STREPTOTHRICIN-F STREPTOVARYCIN STREPTOVARYCIN-A STREPTOVARYCIN-B STREPTOVARYCIN-C STREPTOVARYCIN-D STREPTOVARYCIN-E STREPTOVARYCIN-F STREPTOVARYCIN-G STREPTOVARYCIN-I STREPTOVARYCIN-K STREPTOVIRUDIN STREPTOVITACIN-A STREPTOZOCIN STROBILURIN-A STROBILURIN-B STROBILURIN-E STROBILURIN-F STROBILURIN-G STROBILURIN-H STRONGYLOPHORINE-2 STRONGYLOPHORINE-3 SUBTILIN SULBENICILLIN SULBENICILLIN DISODIUM SULFAZECIN SULFOMYCIN-I SULFOMYXIN SULFONIDAZOLE SULFURMYCIN-A SULFURMYCIN-B SULTAMICILLIN SUN-5555 SUNCILLIN SURFACTANT-PROTEIN-B-= HUMAN SURGUMYCIN SUSPENSASIDE SUZUKACILLIN SWINHOLIDE-A SYRINGOMYCIN-E SYRINGOSTATIN-A T-1218 T-1221 T-1224 T-1982A T-1982B T-2525A T-2588A T-5575 TALAMPICILLIN TALAROMYCIN-A TALAROMYCIN-B TALAROMYCIN-C TALAROMYCIN-E TALISOMYCIN TALISOMYCIN-B TALISOMYCIN-S10B TALLIMUSTINE TAMETICILLIN TAN-1057-A TAN-1057-B TAN-1057-C TAN-1057-D TAN-1518-A TAN-950-A TAUTOMYCIN TEICOPLANIN TEICOPLANIN-A2 TEICOPLANIN-A2-1 TEICOPLANIN-A2-2 TEICOPLANIN-A2-3 TEICOPLANIN-A2-4 TEICOPLANIN-A2-5 TEICOPLANIN-A3 TEICOPLANIN-A3-1 TEICOPLANIN-A3-2 TEICOPLANIN-AGLYCONE TELITHROMYCIN TELOMYCIN TEMOCILLIN TENUAZONATE TERPENTECIN TERRECYCLATE-A TERREIN TETAINE TETRACENOMYCIN-C TETRACYCLINE TETRAHYDRO= DICRANENONE-B TETRAHYDROECHINO= CANDIN-B TETRANACTIN TETRANDRINE TETRAZOMINE TETROCARCIN-A TETRODECAMYCIN TETRONASIN TETRONOMYCIN TEVENEL THELEPHORATE THENOYL-HYDRAZIDE THERMORUBIN-A THERMOZYMOCIDIN THIACYCLINE THIAMPHENICOL THIAMPHENICOL-GLYCINATE THIAMPHENICOL-= GLYCINATE = ACETYLCYSTEINE THIANGAZOLE THIARUBRINE-A THIAZINOTRIENOMYCIN-B THIENAMYCIN THIOCORALINE THIOFORMYCIN-B THIOLACTOMYCIN THIOLUTIN THIOMARINOL THIOMARINOL-D THIOMARINOL-E THIOMARINOL-F THIOMARINOL-G THIOPEPTIN THIOPEPTIN-B THIOSANGIVAMYCIN THIOSTREPTON THIOTETROMYCIN THIOTROPOCIN THIOURIDINE-4 THIOXAMYCIN TIACUMICIN-A TIACUMICIN-D TIACUMICIN-E TIAMULIN TICARCILLIN TIFENCILLIN TIGEMONAM TILMICOSIN TIRANDALYDIGIN TIRANDAMYCIN TIRANDAMYCIN-A TIRANDAMYCIN-B TMC-016 TMC-151-A TMC-151-B TMC-151-C TMC-151-D TMC-151-F TMC-2-A TMC-2-B TMC-2-C TMC-69 TOBRAMYCIN TOC-39 TOC-50 TOLYPOMYCIN-Y TOLYTOXIN TOMATINE TOMAYMYCIN TOMICID TOTARADIOL TOTARAL TOXOFLAVIN TOYOCAMYCIN TRIACETYLDYNEMICIN-A TRICHODERMIN TRICHODERMOL TRICHOMYCIN-A TRICHOMYCIN-B TRICHORZIANINE-A1 TRICHOSETIN TRICHOSPORIN-B-III TRICHOSPORIN-B-V TRICHOSTATATE TRICHOSTATIN-A TRICHOSTATIN-C TRICHOTHECIN TRICHOTOXIN-A40 TRIENINE TRIENOMYCIN-A TRIENOMYCIN-B TRIENOMYCIN-C TRIKENTRIN-A-CIS TRIKENTRIN-A-TRANS TRIKENTRIN-B-CIS

1078 APPENDIX D TRIKENTRIN-B-TRANS TRIMETHYLELLAGATE-3,3+,4 TRINACTIN TRIOSTIN-A TRIOSTIN-C TRITRPTICIN TROLEANDOMYCIN TROSPECTOMYCIN TRYPTANTHRIN TU-1718B TUBERACTINOMYCIN-A TUBERACTINOMYCIN-O TUBERCIDIN TUBERCIDIN-= MONOPHOSPHATE TUBERIN TUBERMYCIN-B TULIPALIN-A TUNICAMYCIN TUNICAMYCIN-A TUNICAMYCIN-A2 TUNICAMYCIN-B TUNICAMYCIN-B2 TUNICAMYCIN-B3 TUNICAMYCIN-C TUNICAMYCIN-D TURIMYCIN TYLACTONE TYLOSIN TYROCIDINE TYROCIDINE-A TYROCIDINE-B TYROTHRICIN U-11921 U-11973 U-24 U-26727A U-43795 U-56407 U-62736 U-63360 U-66226 U-66664 U-66694 U-66866 U-67786 U-68819 U-70585 U-72799 U-75559 U-76074 U-76579 U-76915 U-78608 UBENIMEX UCE-1022 UCE-6 UCH-9 UCN-01 UCN-02 UCT-4B UK-2-A UK-3-A UK-63052 UK-65662 UK-69753 ULTRA-LEVURE UMBELLIFERONE UNCINATONE UNDECYLPRODIGIOSIN UNPHENELFAMYCIN URDAMYCIN-B URDAMYCIN-C URDAMYCIN-D URDAMYCIN-E URDAMYCIN-F URDAMYCINONE-B USNATE UVARETIN VA-2 VACIDIN-A VALANIMYCIN VALCLAVAM VALIDAMINE VALIDAMYCIN-A VALIDAMYCIN-B VALIENAMINE VALINOMYCIN VANCOMYCIN VARIAMYCIN VARIAPEPTIN VC-15-B VELLERAL VENTURICIDIN VENTURICIDIN-A VENTURIDICIN-B VERACTAMYCIN-A VERACTAMYCIN-B VERDAMICIN VERMICULINE VERMISTATIN VERMIXOCIN-A VERMIXOCIN-B VERNAMYCIN VERNAMYCIN-B-DELTA VERNAMYCIN-C VERRUCARIN-A VERRUCARIN-E VERRUCARIN-J VERRUCOSIDIN VERUCOPEPTIN VINEOMYCIN-A1 VIOLACEIN VIOLAMYCIN VIOLAMYCIN-B1 VIOLAMYCIN-B1-2 VIOLAMYCIN-B1-3 VIOMYCIN VIRANTMYCIN VIRGINIAMYCIN VIRGINIAMYCIN-M VIRGINIAMYCIN-M1 VIRGINIAMYCIN-M2 VIRGINIAMYCIN-S1 VIRGINIAMYCIN-S2 VIRGINIAMYCIN-S3 VIRGINIAMYCIN-S4 VIRGINIAMYCIN-S5 VIRIDOFULVIN VIRIDOFULVIN-A VIRIDOFULVIN-B VIRIPLANIN-A VIRUSTOMYCIN-A VM-44857 VM-44864 VM-44865 VM-44866 WB-608 WF-3161 WIN-35439 WP-401 WP-546 WP-549 WP-608 WP-631 WP-652 WS-5995A WS-5995B WS-5995C WS-79089-B WS-9659A WS-9659B WY-12556 WY-7953 WYERONE X-14667A X-14868A X-14868B X-14868C X-14868D X-14873A X-14881-E X-14885A X-14889A X-14889C X-14889D X-206 XANTHOCIDIN XANTHOQUINODIN-A1 XANTHOQUINODIN-A2 XANTHOQUINODIN-A3 XANTHOQUINODIN-B1 XANTHOQUINODIN-B2 XANTHOSTATIN XANTHOTHRICIN XANTOCILLIN XYLOSTASIN YELLAMYCIN-A YELLAMYCIN-B YELLAMYCIN-C YL-01869-P YM-13115 YM-30059 YM-47522 YM-75518 YOMOGIARTEMIN YS-822A ZG-1494-ALPHA ZINCOPHORIN ZINOSTATIN ZM-218463 ZORBAMYCIN ZORUBICIN ANTIBODY ABCIXIMAB ADALIMUMAB AGGLUTININ ALS ALS-ANTITHYMOCYTE ALS-ANTITHYMOCYTE-= GLOBULIN ALS-ANTITHYMOCYTE-= GLOBULIN-HORSE ALS-ANTITHYMOCYTE-= GLOBULIN-RABBIT ALS-GLOBULIN ALS-HORSE ALS-RABBIT ANTI-IDIOTYPE ANTINUCLEAR-FACTOR ANTITOXIN ANTIVENOM APOLIZUMAB AUNATIV AUTOANTIBODY BACTERIOLYSIN BASILIXIMAB BERIGLOBIN BEVACIZUMAB BM-01044 BT-563 BW-494 CAMPATH-1G CAMPATH-1H CAMPATH-1M CAMPATH-6 CDP-870 CENTOXIN CETUXIMAB CMV-IMMUNOGLOBULIN COLOSTRX CYTOGAM

Derwent Drug File 1079 Thesaurus CYTOTECT DACLIXIMAB DC-101 DIGIBIND DIGIDOT ECULIZUMAB EDRECOLOMAB EMD-55900 EMD-72000 ENDOBULIN EPRATUZUMAB FLEBOGAMMA GAMIMUNE GAMIMUNE-N GAMMA-16 GAMMA-VENIN GAMMAGARD GAMMAPROTECT GAMMAR-IV GAMMASTAN GAMMIMUNE-N GAMMONATIVE GEMTUZUMAB OZOGAMICIN GLOBULIN-N GLOBUMAN HEMAGGLUTININ HEP-B-GAMMAGEE HEPATECT HEPATITIS-B-= IMMUNOGLOBULIN HYPER-HEP IBRITUMOMAB-TIUXETAN ICI-D-0490 IDEC-131 IDEC-152 IMC-1C11 INTRAGLOBIN INTRAGLOBIN-F KELIXIMAB LACTOBIN LATS MDX-33 MDX-H-210 MUROMONAB-CD3 NATALIZUMAB OCTAGAM OMALIZUMAB OPSONIN PALIVIZUMAB PASCOLIZUMAB PENTAGLOBULIN POLYGAM POLYGLOBIN PRECIPITIN PSOMAGLOBIN PURIMMUN R3-36-16 RG-83852 SANDOGLOBULIN SB-249417 SC-72-14 SIPLIZUMAB SM-4300 TOSITUMOMAB VARITECT VEINOGLOBULIN VENILON VENIMMUN VENOGLOBULIN-I VENOGLOBULIN-S WINRHO ANTICHOLINESTERASES 217-AO 8203-HC AA-31 AMBENONIUM CHLORIDE AMINOSTIGMINE AMITON ARISUGACIN-A ARISUGACIN-B BUTACARB BUTONATE BW-284-C51 BW-62-C47 CARBARIL CARBOFURAN CHF-2819 CYCLOHEXYLSUBERO= GORGAMIDE-N DECADONIUM IODIDE DEHYDROEVODIAMINE DEMECARIUM BROMIDE DEOXYPEGANINE DFP DIAZINON DIMEFOX DIMETILAN DIOXACARB DONEPEZIL E-2030 ECOTHIOPATE IODIDE EDROPHONIUM CHLORIDE ESEROLINE ESEROLINE-SALICYLATE ETHION FENITROTHION FENTHION FONOFOS FONOFOS-OXON GA-102 GA-3 GA-95 GALANTAMINE GD-42 GD-7 GT-165 HEPTYLPHYSOSTIGMINE HSR-803 HUPERZINE-A HUPERZININE HUPRINE-X HUPRINE-Y ICOPEZIL ISOLAN KW-5092 LG-113 LG-114 LG-115 MALAOXON MALATHION MDL-73745 METHAMIDOPHOS METHANESULFONYL-= FLUORIDE METHIOCARB METHIOCARB-SULFOXIDE METHOXYTACRINE-7 METHYLTACRINE-9 METRIFONATE MF-268 MFS-3 MOBAM NAM-204 NAM-224 NEOSTIGMINE NEOSTIGMINE BROMIDE NEOSTIGMINE METHYLSULFATE NIBUFIN NORPHYSOSTIGMINE OXYDEMETON-METHYL P-10358 PARAOXON PARATHION PARATHION-METHYL PHENSERINE PHENYLMETHANE= SULFONYL-FLUORIDE PHOSPHAMIDON PHOSPHOSTIGMINE PHYSOSTIGMINE PIRIMICARB PROMECARB PYRAMAT PYRIDOSTIGMINE BROMIDE PYROLAN RA-7 RIVASTIGMINE RO-2-0683 RX-67668 SARIN SM-10888 SOMAN STEPHAGLABRINE STRYCHNINE SUBEROGORGIN SURONACRINE SUVANINE TABUN TAK-147 TEPP TERRITREM-B TETRACHLORVINPHOS THB-013 TL-363 TL-365 TOLSERINE TV-3326 VELNACRINE VX ANTICOAGULANT HEPARINOID ANTICOAGULANTS ACENOCOUMAROL ACETYLHEPARIN-N ACETYLTHROMBIN ACTIVATED-PROTEIN-C-= HUMAN AG-307 ANCROD ANCROD ANISINDIONE ANNEXIN-V ANTILIPOPOLYSACCHARIDE-= FACTOR-LIMULUS ANTISTASIN APOLATE SODIUM APROSULATE SODIUM ARC-69931-MX ARDEPARIN SODIUM ARGATROBAN ARMATAN ASTERRIQUINONE-CT-3 BEMIPARIN SODIUM BG-8865 BISCOUMACETATE-ETHYL BM-21-23 BMY-44621 BRODIFACOUM BROMADIOLONE BROMINDIONE BUFORIN-I BX-807834 C-921-78 CALPHOBINDIN-I CALRETICULIN CERANIL CERASTASE-F4 CERTOPARIN CHLOROPHACINONE

1080 APPENDIX D CHONDROITINSULFATE CHONDROITINSULFATE-A CHONDROITINSULFATE-C CITRATE SODIUM CLOCOUMAROL CLORINDIONE COUMACHLOR COUMATETRALYL COUMETAROL CUMARIN CX-397 CX-397R CY-222 CYCLOCOUMAROL DALTEPARIN SODIUM DANAPAROID SODIUM DIARBARONE DICOUMAROL DIFENACOUM DIHYDROXYPHENYLLACTATE DIOCOUMINE DIPETALIN DIPHENADIONE DOMOXIN DPC-423 DUP-714 DX-9065A E-456 ECOTIN EFEGATRAN ENOXAPARIN SODIUM ETABENZARONE ETHYLIDENEDICOUMAROL EXTRINSIC-PATHWAY-= INHIBITOR FEPROMARON FLUINDAROL FR-860 FXV-673 G-31150 GALACTAN-POLYSULFATE GC-94 GELIN GHILANTEN GLUCURONYLGLUCOS= AMINO-GLYCAN-SULFATE GLYCOSAMINOGLYCAN-= POLYSULFATE GM-1077 GS-522 GYKI-14166 GYKI-14451 GYKI-14451 GYKI-14766 HEMATIN HEMATIN-DERIVED-= ANTICOAGULANT HEMENTIN HEPARAN-SULFATE HEPARIN HEPARIN CALCIUM HEPARIN LITHIUM HEPARIN MAGNESIUM HEPARIN SODIUM HEPARIN-BETA HEPARIN-PENTASACCHARIDE HEPARINOIDS HEPARITIN HIRUDIN HIRUDIN-54-65 HIRUDIN-DESULFATED HIRUDIN-LYS-47 HIRUDOID HIRUGEN HIRULOG HIRULOG-1 HIRUNORM-IV HOLOTHURIAN-GLYCOS= AMINOGLYCAN IC-83-1423 INOGATRAN INTIMATAN ISOVALERYLINDANDIONE ITF-300 KC-6141 L-372460 L-374087 L-767679 LB-30057 LEPIRUDIN LONGOLYTIN LW-10078 LW-10079 LW-10086 LY-178207 M+B-4596 MALTOHEXOSE-SULFATE MDL-28050 MELAGATRAN MEPESULFATE MESOGLYCAN METHYLSULFINYLWARFARIN NADROPARIN CALCIUM NAP-5 NAP-C-2 NAPSAGATRAN NEMATODE-= ANTICOAGULANT-= PROTEIN-C2 NICOFURANOSE NITROFARIN OH-10172 ONO-3307 OP-2123 OP-386 OP-622 ORG-10172 ORG-31540 ORG-31550 ORG-34006 ORG-36764 OXYCOUMARIN P-532 P-8714 PARNAPARIN PEFA-1286 PENTOSAN-POLYSULFATE PHENINDIONE PHENPROCOUMON PHOSPHOLIPASE-C PI-88 PINDONE PLANCININ POLYANETHOLESULFONATE = SODIUM POLYPHEMUSIN-I POLYVINYLSULFATE PROLIXIN-S PROTEIN-C-HUMAN PROTEIN-C-INHIBITOR RATIBOL RD-11885 RE-1492 REVIPARINE RMI-10393 RMI-12366A RMI-14133A RO-1-8307 RO-12-1989 RO-2-7509 RPR-109891 RPR-128515 RPR-130737 RPR-208707 RWJ-56110 S-18326 S-2581 SALICYLALDOXIME SALVIANOLATE-A SANORG-32701 SB-249417 SC-59735 SDZ-217-766 SDZ-MTH-958 SEL-2711 SH-869 SK-549 SN-292 SOLULIN SPI-501 SQ-22536 SR-90107 SULEPAROIDE SULODEXIDE SURFACTIN TEDELPARIN THROMBOCID THROMBODYM THROMBOMODULIN TICK-ANTICOAGULANT-= PEPTIDE TINZAPARIN SODIUM TIOCLOMAROL TISSUE-FACTOR-PATHWAY-= INHIBITOR TISSUE-FACTOR-PATHWAY-= INHIBITOR-1-161 TRI-11 TRI-50-B TRI-59 TRIOLEIN VICASOL VK-744 VK-774 W-5 W-7 WARFARIN XR-334 XR-5118 XYLOCOUMAROL YAGIN YM-60828 YM-75466 ZK-805412 ZK-805623 ANTICONVULSANTS 2-170 43-U-87 A-134974 ABECARNIL ACEA-0762 ACEA-1011 ACEA-1021 ACEA-1328 ACEA-1416 ACETAZOLAMIDE ACETYLPHENETURIDE ACPD AD-11 ADD-17014 ADD-196022 ADD-213063 ADD-213066 ADD-219048 AF-CX-1325 AHR-11748 AHR-14042 ALBUTOIN ALLOMETHADIONE AMELTOLIDE AMINOBECLAMIDE-PARA AMINOGLUTETHIMIDE

Derwent Drug File 1081 Thesaurus AMINOOXYACETATE AMINOPHOSPHONO= HEPTANOATE AMINOPHOSPHONO= PROPIONATE AMINOPHOSPHONO= VALERATE AMINOVALERATE-DELTA AMOBARBITAL ANTIEPILEPSIRINE AQ-0145 AR-A-008055 ARFENDAZAM ARL-15895-AR ATOLIDE ATROLACTAMIDE AWD-131-138 AWD-140-076 AWD-140-190 AZETHYLNICOTINATE BARBEXACLONE BAU-426 BAY-36-7620 BECLAMIDE BENTAZEPAM BENZOBAMIL BENZOBARBITAL BENZOYLHETERATISINE-6 BIBO-3304 BM-11 BM-34 BRL-52537 BROFOXINE BROSOTAMIDE BROSUXIMIDE BTS-72664 BULBOCAPNINE BURAMATE BUTANEDIOL-DIVALPROATE-= 1,4 BW-534-U-87 BW-A78U CARBAMAZEPINE CARBAMAZEPINE-EPOXIDE CARBOCLORAL CARFEDONE CGP-33101 CGP-37849 CGP-39551 CGP-40116 CGP-43487 CGP-46381 CGP-56433 CGP-61334 CGS-17867A CGS-20625 CGS-9896 CHF-3381 CHLORPHENACEMIDE CI-953 CI-966 CINROMIDE CIPRAZAFONE CITENAMIDE CL-273547 CLOMETHIAZOLE CLONAZEPAM CLOTIAZEPAM CM-40142 CM-6 CNS-5788 CO-134444 CO-2-1068 CONANTOKIN-R CORYTUBERINE CP-14304 CP-465022 CYHEPTAMIDE D-20443 D-2916 D-3187 DECIMEMIDE DEHYDROVALPROATE-3 DENZIMOL DEZINAMIDE DICHLOROKYNURENATE-5,7 DIETHYLAMANTADINE-3,5 DIMETHADIONE DIMETHYLGLYCINE DIMETHYLPHENOBARBITAL DIOXAMATE DIPHENDIONE DIPHENYLBARBITURATE-5,5 DIZOCILPINE DM-44 DM-49 DOXENITOIN DULOZAFONE DYSIHERBAINE E-2050 EBORACIN EGIS-8332 ELTANOLONE ENOMELANIN ESTAZOLAM ETAZEPINE ETEROBARB ETHADIONE ETHOSUXIMIDE ETHOTOIN ETHYLPHENACEMIDE EX-10-542A FCE-26743 FEBARBAMATE FENACLON FG-8205 FG-9067 FG-9202 FLETAZEPAM FLUNITRAZEPAM FLUORESONE FLUZINAMIDE FOSENAZIDE FOSPHENYTOIN FPL-12495 FPL-12495-AA FPL-13950 FPL-15896-AR FUMARILINE GABA-ISOBUTYL GABAPENTIN GABOB GANAXOLONE GINGEROL-6 GLOBULIN-N GLUTAMATE-PALMITAMIDE GLUTAMYLAMINOMETHYL= SULFONATE-GAMMA GLUTAMYLASPARTATE-= GAMMA GLUTAMYLGLYCINE-= GAMMA-D GLUTAPYRONE GLYCINE-VALPROMIDE GP-47779 GP-683 GV-150526-A GV-213237-A GVS-111 GYKI-52466 GYKI-53784 HA-94 HALODIF HALONAL HEPTOBARBITAL HEXETHAL HISTOGRANIN HOPANTENATE CALCIUM HP-654 HYDROXYPYRIDINE-3 HYDROXYTRYPTOPHAN-= ETHYL-ESTER HYDROXYTRYPTOPHAN-= METHYL-ESTER IBMECA ICI-45337 IDPH-791 IEM-1460 IEM-1592 IEM-1754 IEM-1857 IL-40 IODOPROXYFAN ISOBUTYL-GABA ISONICOTINOYL-GABA ISOPROPYLAMANTADINE-3 KAINATE-BETA L-695902 L-698544 L-701252 L-701273 L-701324 L-703717 L-705022 L-708541 LAMOTRIGINE LEVETIRACETAM LODAXAPRINE LORECLEZOLE LOSIGAMONE LS-20 LU-2443 LY-156007 LY-163395 LY-201409 LY-201979 LY-227420 LY-300164 LY-302679 LY-354740 LY-81067 MAP-4 MDL-100453 MDL-104653 MDL-104653 MDL-105519 MDL-27192 MDL-27531 MDL-72483 MEPHENYTOIN MESUXIMIDE METAGLYCODOL METETOIN METHARBITAL METHINDIONE METHYLPHENOBARBITAL METHYLPHENYTOIN MEXILETINE MILACEMIDE MORSUXIMIDE MOTRAZEPAM MRZ-2-576 MY-103 NAFIMIDONE NCC-05-0711 NCS-382 NERAMEXANE NICOTINOYL-GABA NICOTINOYLALANINE NIMETAZEPAM NIRVANOL NNC-13-8119

1082 APPENDIX D NNC-14-0185 NNC-711 NNC-90-1515 NONAPYRIMINE NORANTOIN NPC-12626 NPC-17742 NPS-846 NSD-3004 ORG-6363 ORG-6370 OXCARBAZEPINE OXITRIPTAN OXITRIPTYLINE OXYFENAMATE PAEONIMETABOLINE-I PALMITONE PARAMETHADIONE PD-144550 PD-152247 PD-158473 PHENACEMIDE PHENAGLYCODOL PHENOBARBITAL PHENOBARBITAL SODIUM PHENSUXIMIDE PHENYLETHYLMALONDIAMIDE PHENYTOIN PHTHALOYL-GLYCINAMIDE PHTHALOYL-GLYCINE PIRIQUALONE PIVAGABINE PRIMIDONE PROGABIDE PUFEMIDE R-57720 RALITOLINE REMACEMIDE RETIGABINE RGH-4615 RILUZOLE RMI-71645 RO-11-6893 RO-11-6896 RO-24-6173 RO-41-7812 RO-42-8773 RO-5-5807 ROPIZINE RP-59037 RP-60503 RPR-104632 RU-31719 RU-32698 RU-32759 RU-33368 RU-33543 RWJ-37868 SABELUZOLE SB-204269 SB-271046 SC-12742 SC-12757 SCH-50911 SDZ-220-004 SDZ-220-040 SDZ-220-581 SH-3-24 SHOGAOL-6 SIB-1893 SKF-100330A SKF-100561 SKF-100591A SKF-100844A SKF-89976A SL-79-182 SM-13496 SM-31900 SNC-121 SR-41378 SRC-820 SUCLOFENIDE SULTIAME SUN-N-8075 TALTRIMIDE TEMAZEPAM THPO TILETAMINE TJ-960 TOPIRAMATE TRIMETHADIONE U-43465F U-54494A U-83892 U-83894 U-84042 VALPROATE VALPROATE CALCIUM VALPROATE MAGNESIUM VALPROATE SEMISODIUM VALPROATE SODIUM VALPROMIDE VALROCEMIDE VIGABATRIN YG-19256 ZK-91296 ZK-93423 ZONISAMIDE ANTIDEPRESSANTS 19148-RP 19749-RP 23669-RP 680-C-91 709-W-92 A-1866 A-80426 AB-15 ADEPREN ADINAZOLAM AGN-2979 ALAPROCLATE ALFETAMINE ALMOXATONE ALTINICLINE AMEDALIN AMIFLAMINE AMINEPTINE AMINOCYCLOPROPANE= CARBOXYLATE-1 AMITRIPTYLINE AMITRIPTYLINOXIDE AMIXETRINE AMOXAPINE AN-12 APTAZAPINE AS-8 AZ-16596 AZAPHEN AZEPINDOLE AZIPRAMINE B-193 B-777-81 BAZINAPRINE BEFLOXATONE BEFURALINE BENMOXIN BENZAPRINOXIDE BIFEMELANE BINEDALINE BMS-181101 BN-50043 BN-50156 BRL-14831 BRL-16644 BUDIPINE BUPROPION BUTACETIN BUTRIPTYLINE BW-1370U87 BW-1555-U-88 BW-17U BW-287U BW-306U BW-616U76 BW-A-494U C-153 C-307 C-383 C-394 C-395 CAPROXAMINE CARBENZIDE CAROXAZONE CARPIPRAMINE CARTAZOLATE CENTPROPAZINE CEPHEDRINE CERICLAMINE CGP-12104-A CGP-12104A CGP-22364A CHLORDESIPRAMINE CIANOPRAMINE CICLAZINDOL CICLINDOLE CICLOPRAMINE CIDOXEPIN CILOBAMINE CIMEMOXIN CIMOXATONE CINFENINE CIPROXIMIDE CITALOPRAM CL-255663 CLEMEPROL CLOCAPRAMINE CLODAZON CLOFENCICLAN CLOMIPRAMINE CLORGILINE CLOVOXAMINE COR-3224 COTININE COTRIPTYLINE CP-154526 CP-66713 CP-77059 CP-93393 CRA-1000 CRA-1001 CRL-40827 CYPENAMINE CYPROLIDOL DALEDALIN DANITRACEN DAPOXETINE DAZADROL DAZEPINIL DEMETHYLDOSULEPIN DEMETHYLDOXEPIN DESIPRAMINE DEXAMISOLE DEXIMAFEN DEXOXADROL DIBENZEPIN DICLOFENSINE DIMETACRINE DIOXADROL DITRAN DOSULEPIN DOXEPIN

Derwent Drug File 1083 Thesaurus DU-127090 DULOXETINE E-2011 E-6006 ECLANAMINE EGYT-2760 EGYT-3615 ELANZEPINE EMD-68843 ENCYPRATE ENPRAZEPINE EPROBEMIDE ESCITALOPRAM ETOPERIDONE EXP-561 F-13714 FA-37 FANTRIDONE FEMOXETINE FENGABINE FENMETOZOLE FENMETRAMIDE FENOXYPROPAZINE FENPENTADIOL FEZOLAMINE FI-4501 FI-4503 FIPEXIDE FLA-289 FLA-299 FLA-314 FLA-334 FLA-336 FLA-365 FLA-384 FLA-405 FLA-417 FLA-450 FLA-463 FLA-558 FLA-668 FLA-717 FLA-727 FLA-788 FLEROBUTEROL FLETAZEPAM FLUACIZINE FLUBANILATE FLUOROTRANYLCYPROMINE FLUOTRACEN FLUOXETINE FLUPERLAPINE FLURADOLINE FLUVOXAMINE FS-32 FTORMETAZINE FTORPROPAZINE GAMFEXINE GERFONAL GUANOXYFEN HEPZIDINE HEXACYCLONATE HEXACYCLONATE SODIUM HOMOPIPRAMOL HP-505 HT-90-B HYDROTHIADENE HYDROXYAMOXAPINE-7 HYDROXYAMOXAPINE-8 HYDROXYMAPROTILINE HYDROXYTRYPTOPHAN-= ETHYL-ESTER HYDROXYTRYPTOPHAN-= METHYL-ESTER HYPERICIN IF-C-45 IFOXETINE IMAFEN IMIPRAMINE IMIPRAMINE-METHIODIDE IMIPRAMINOXIDE INDALPINE INDATRALINE INDELOXAZINE INN-00835 INTRIPTYLINE IODOCLORGYLINE IPRINDOLE IPROCLOZIDE IPRONIAZID IRFI-165 ISOCARBOXAZID IVOQUALINE J-508 J-512 J-516 JL-3 KETIMIPRAMINE L-783281 LEVOFACETOPERANE LEVOPROTILINE LEVOSULPIRIDE LEVOXADROL LI-160 LILLY-51641 LIS-30 LITHIUM-ASPARTATE LITHIUM-CARBONATE LITHIUM-CHLORIDE LITHIUM-CITRATE LITHIUM-HYDROXYBUTYRATE LITHIUM-NITRATE LITHIUM-SALT (Drug) LITHIUM-SULFATE LITHIUM-TRYPTOPHANATE LITOXETINE LITRACEN LK-63 LOFEPRAMINE LORTALAMINE LOSINDOLE LU-10-134-C LU-11-109 LU-11-161 LU-11-305 LU-17-133 LU-43706 LY-113821 LY-227942 LY-51641 MAPROTILINE MAZINDOL MCN-4187 MCN-4612-Z MCN-5652-Z MCN-5707 MCN-5908 MD-240098 MD-240233 MD-760548 MDL-19660 MDL-26479 MDL-72394 MDL-72974 MEBANAZINE MEDIFOXAMINE MELITRACEN MEQUITAZINE MESEMBRINE METAPRAMINE METRALINDOLE MEZEPINE MIANSERIN MILNACIPRAN MIRTAZAPINE MK-0869 MK-306 (psychostimulant) MK-869 MKC-242 MOCLOBEMIDE MODALINE MONODEMETHYLDOXEPIN MONOMETACRINE NAFENODONE NAPACTADINE NAPAMEZOLE NBF-003 NBF-008 NBF-021 NDO-008 NEBRACETAM NEFAZODONE NEFOPAM NIALAMIDE NISOXETINE NITRAFUDAM NITROXAZEPINE NOMELIDINE NOMIFENSINE NORCLOMIPRAMINE NORFEMOXETINE NORFLUOXETINE NORTRIPTYLINE NOXIPTILINE NS-105 NUCLOTIXENE OCTAMOXIN OCTRIPTYLINE OI-77 OMILOXETINE OPC-14523 OPIPRAMOL ORG-4428 ORG-6582 ORG-6906 OXAPROTILINE OXITRIPTAN PANURAMINE PARAXAZONE PARGYLINE PAROXETINE PERAFENSINE PHENELZINE PHENIPRAZINE PIBERALINE PIM-35 PIPOFEZINE PIRANDAMINE PIRLINDOLE PIVAGABINE PIZOTIFEN PR-881-884A PRAZEPINE PRAZITONE PRIDEFINE PROPIZEPINE PROTRIPTYLINE PYRIDAZOLE QUINUPRAMINE RAN-113 REBOXETINE RO-60-0175 ROLICYPRINE RS-2232 RU-41656 SAFRAZINE SB-224289 SB-271046 SEPROXETINE SERTRALINE SETIPTILINE SIB-1508-Y

1084 APPENDIX D SIB-1553-A SIBUTRAMINE SPIROXEPIN SUCCINONITRILE SULPIRIDE SULTOPRIDE SUNEPITRON TALOPRAM TALSUPRAM TAMPRAMINE TANDAMINE TETRINDOLE THIONISOXETINE TIANEPTINE TIAZESIM TIENOPRAMINE TIFEMOXONE TIFLUCARBINE TIOMERGINE TISOCROMIDE TJS-010 TOFENACIN TOLOXATONE TOLQUINZOLE TOMOXETINE TOZALINONE TRACAZOLATE TRANYLCYPROMINE TRAZODONE TREBENZOMINE TRELIBET TRIMIPRAMINE TRIZOXIME TROCIMINE TV-3326 TZ-650 U-1424 U-23807A U-48753E U-93385 UP-614-04 VENLAFAXINE VERATRYLHYDRAZINE VILOXAZINE VIQUALINE VUFB-15468 WF-31 WY-25093 WY-27587 WY-45233 YM-08054-1 YM-35992 ZAFULEPTINE ZE-117 ZIMELDINE ZOMETAPINE ANTIDIABETICS 53-540 68-157 98-202 A-320454 A-3744 A-3787 ACARBOSE ACETOHEXAMIDE AD-4610 AD-5075 AG-EE-388-ZW AG-EE-623ZW AG-EE-624-ZW AG-EE-86 AGN-194204 ALT-4000 ALT-462 ALT-486 AMLINTIDE AO-128 AS-6 AY-31637 AZ-242 AZ-DF-265 BAY-1099 BAY-1248 BAY-M-1099 BDF-8933 BENFOSFORMIN BETACELLULIN BL-11778 BM-130907 BM-130913 BM-208 BM-42304 BMS-210285 BOUSSINGOSIDE-A1 BOUSSINGOSIDE-A2 BRL-48482 BTS-67-582 BUFORMIN BUTADIAZAMIDE BUTAGLYONAMIDE BUTOXAMINE CARBOXYTOLBUTAMIDE CARBUTAMIDE CGP-11112 CHIRO-INOSITOL CHLORHEXAMIDE CHLOROPROPIONATE-2 CHLORPROPAMIDE CIGLITAZONE CL-316243 CLOMOXIR CLX-0901 COLOSOLATE CP-316819 CP-92768 CP-92768 CS-261 CS-476 CT-112 DARGLITAZONE DC-23-99 DEHYDROCROTONIN-TRANS DEOXYNOJIRIMYCIN-1 DICHOL DIOSCORETINE DIPHENYLENEIODONIUM DRF-2189 DRF-2725 EMERIAMINE EMIGLITATE ENGLITAZONE EPALRESTAT ESCIN-II-A ESCIN-II-B ETOFORMIN ETOMOXIR FARGLITAZAR FENBUTAMIDE GALEGINE GANODERAN-B GLIAMILIDE GLIBENCLAMIDE GLIBORNURIDE GLIBUTIMINE GLICARAMIDE GLICETANILE GLICLAZIDE GLICONDAMIDE GLIDAZAMIDE GLIFLUMIDE GLIMEPIRIDE GLIPALAMIDE GLIPIZIDE GLIQUIDONE GLISAMURIDE GLISENTIDE GLISINDAMIDE GLISOLAMIDE GLISOXEPIDE GLISULFAZID GLYBUTHIAZOL GLYBUZOLE GLYCLOPYRAMIDE GLYCYCLAMIDE GLYHEXAMIDE GLYMIDINE GLYOCTAMIDE GLYPARAMIDE GLYPINAMIDE GLYPROTHIAZOL GLYSOBUZOLE GP-1447 GR-92132-X GR-92132-X GW-0072 GW-1929 GW-409544 GW-510516 GW-7845 GYMNEMATE-III GYMNEMATE-IV GYMNEMATE-V GYMNEMATE-VII GYMNEMOSIDE-B HEPTOLAMIDE HYDROXYHEXAMIDE HYDROXYISOLEUCINE-4 HYDROXYTOLBUTAMIDE INSULIN-DETEMIR INSULIN-GLARGINE ISOAMYLENEGUANIDINE KAD-1229 KGR-1380 KGR-1421 KOLAVIRON L-165041 L-165461 L-783281 L-796449 LINOGLIRIDE LN-5330 LY-177507 LY-275585 LY-307161 M+B-39890A M-16049 MARSUPSIN MCC-555 MDL-25637 MDL-73945 MEGLITINIDE METAHEXAMIDE METASULFANILYLBUTYL= CARBAMIDE METFORMIN METHYL-PALMOXIRATE METHYLBELLIDIFOLIN METHYLCYSTEINE-= SULFOXIDE-S MIDAGLIZOLE MIGLITOL MITIGLINIDE MK-467 MTP-1307

Derwent Drug File 1085 Thesaurus NATEGLINIDE NC-8-12 NN-2211 NNC-25-2504 NVP-DPP-728 NZ-314 ONO-1714 P-32-98 PALMOXIRATE PENTAGALLOYLGLUCOSE PERVANADATE PHENFORMIN PHENSUCCINAL PINITOL PIOGLITAZONE PIROGLIRIDE PJ-34 PMS-812 PN-2034 PNU-106817 PNU-140975 PRAMLINTIDE PROTOTIMOSAPONIN-A-III PSEUDOPROTOTIMO= SAPONIN-A-III PYRUVATE-METHYL-ESTER RMI-10026 RMI-11894 RO-16-8714 ROSIGLITAZONE RX-871024 S-22068 S-3075 S-33113 S-4048 SALACINOL SALVIFOLIN SARI-59801 SAUDIN SB-213068 SDZ-51-641 SDZ-CPI-975 SDZ-FOX-988 SDZ-PGU-693 SECOISOLARICIRESINOL-= DIGLUCOSIDE SECOMANOALIDE SKF-34288 SL-840418 SL-860714 SL-860715 SPC-5002 ST-1326 SWERCHIRIN SYNTHALIN-A SYNTHALIN-B T-1095 T-174 TA-078 TA-174 TARASAPONIN-VI TECOMINE THIOHEXAMIDE TIFORMIN TIMOSAPONIN-B-I TOLAZAMIDE TOLBUTAMIDE TOLPENTAMIDE TOLPYRRAMIDE TOLRESTAT TORMENTATE TRESTATIN TRESTATIN-A TRESTATIN-B TRESTATIN-C TROGLITAZONE U-19425 UL-DF-9 VALINE-PYRROLIDIDE VANADYL DIPICOLINATE Y-3310 ZD-5522 ANTIDIARRHEICS AGIOCUR ALKOFANONE BENZETIMIDE BERBERINE BIM-4004-1 BIOFLORIN BIOLFORIN BISMUTH-SUBGALLATE BISMUTH-SUBSALICYLATE BISNORDIHYDROTOXIFERINE BUTOXYLATE BW-942C CADINOL-T CHLOROXINE CI-750 CICARPERONE COLOPTEN DIFENOXIMIDE DIFENOXIN DIPHENOXYLATE FETOXILATE FLUPERAMIDE FTORASOL GR-C-507-75 GUARANA KF-18259 KF-20170 LIDAMIDINE LOCUST-BEAN LOPERAMIDE LOPERAMIDE-N-OXIDE MALETAMER MEBIQUINE MM-218 NC-8-12 NIFALATIDE NITROVIN NUFENOXOLE PERENTEROL POLYCARBOPHIL ROLGAMIDINE SACCH. BOULARDII SACOLENE SKF-35886 STULLMISAN THIHEXINOL-METHYL= BROMIDE TJ-14 UZARIN WHR-1049 WHR-1049A WILD-20 ZY-17617B ANTIDIURETICS CARINAMIDE EX-4877 FL-155 MJ-9465-2 SR-58539B SR-58572A ANTIDOTES ACETYLPENICILLAMINE ACTIVATED-CHARCOAL ALLOXIME AMINOACETONITRILE AMINOPROPIOPHENONE-= PARA ANTAMANIDE BDB-106 BDB-108 BDB-27 BDB-39 BDB-91 BM-01014 BUTYRYLCHOLINESTERASE CARBOXIME CARBOXYPEPTIDASE-G2 CDTA-DISODIUM-CALCIUM CONGO-RED DA-10 DIACETYL-MONOXIME DIACETYLNALORPHINE DICOBALT-EDETATE DIETHYXIME DIMERCAPROL DIMETHYLAMINOPHENOL EDTA-COBALT FOMEPIZOLE GLUTATHIONE-MONO= ETHYL-ESTER HGA-1 HGG-12 HGG-21 HGG-42 HGG-52 HGG-65 HGG-70 HH-38 HI-6 HI-7 HS-12 HS-14 HS-3 HS-4 HS-6 ISONITROSINE METHYLTHIONINIUM = CHLORIDE MMB-4 OBIDOXIME CHLORIDE ORGANOPHOSPHATE-= ANHYDRASE OXOTHIAZOLIDINE-2-= CARBOXYLATE-4 P-65 PARATHION-HYDROLASE PHENETHYL-ISOTHIO= CYANATE PHOSPHOTRIESTERASE PRALIDOXIME IODIDE PRALIDOXIME MESILATE PYRIMIDOXIME R-665 RHODANESE RMI-71626 SAD-128 SUCCIMER-DIETHYL TACRINE THIONINE TRIMEDOXIME BROMIDE U-23223 UNITIOL UNO-3 W-84 ANTIEMETICS ABT-229 ACEPROMAZINE AD-8112 ADR-847

1086 APPENDIX D ADR-851 AL-1612 ALEPRIDE ALIZAPRIDE APREPITANT AS-5820 BATANOPRIDE BEMESETRON BENZQUINAMIDE BISMUTH-SUBSALICYLATE BROMOPRIDE BUFENADRINE BUTAPERAZINE CARPERONE CHLORFENETHAZINE CIPROPRIDE CITRATE SODIUM CLEBOPRIDE CYCLIZINE DAZOPRIDE DECLOXIZINE DIFENIDOL DIHYDROBENPERIDOL DIMENHYDRINATE DIMETPRAMIDE DOLASETRON DOMPERIDONE DRONABINOL DROPERIDOL E-3620 ETANAUTINE EXEPANOL FK-1052 FLUALAMIDE FLUBEPRIDE FLUDOREX GK-128 GR-125487 GR-203040 GR-205171 GR-65630A GR-C-507-75 GRANISETRON HSP-117 HYDROXYGRANISETRON-7 IPROZILAMINE ISOSULPRIDE KB-6933 KF-20170 L-646462 L-741671 L-742694 L-754030 L-758298 LERISETRON LEVOMETIOMEPRAZINE LEVONANTRADOL LEVOSULPIRIDE LUROSETRON MECLOZINE METADOXINE METHIOMEPRAZINE METOCLOPRAMIDE METOPIMAZINE METOXEPIN MEZILAMINE MK-0869 MK-869 MOCIPRAZINE MOLINDONE N-3256 N-3389 NABOCTATE NK-422 NONABINE ONDANSETRON OXYPENDYL PANCOPRIDE PD-154075 PERPHENAZINE PERPHENAZINE-DECANOATE PERPHENAZINE-ENANTHATE PIPAMAZINE PIPRINHYDRINATE PIRENZEPINE POLYPORENATE-C PORICOATE-A POSKINE PROCHLORPERAZINE PYRICAPIRONE RAMOSETRON RENZAPRIDE RG-12915 RG-12915A RS-25259-197 SKF-103561 SULPIRIDE SULTOPRIDE THIETHYLPERAZINE THIOPROPERAZINE TIAPRIDE TRAZOLOPRIDE TRIFLUPROMAZINE TRIMETHOBENZAMIDE XANTHIOL Y-25130 ZACOPRIDE ZATOSETRON ANTIFIBRINOLYTICS ACEXAMATE AMINOCAPROATE-EPSILON CETRAXATE HISTIDINE-RICH-= GLYCOPROTEIN PAMBA PROTEIN-C-INHIBITOR TRANEXAMATE ANTIFLATULENTS AGALSIDASE-ALPHA ALPHA-D-GALACTOSIDASE CARVONE DIMETICONE ICI-111075 PEPPERMINT-OIL RITANSERIN SIMETHICONE ANTIGEN ALLERGEN AUTOANTIGEN FETOPROTEIN HAPTEN HLA IA-ANTIGEN ANTIGEN-PRESENTING-CELL DENDRITIC-CELL ANTIGOUTS ALLOPURINOL ALLYLCINCHOPHEN AMFLUTIZOLE BENZBROMARONE BENZIODARONE BOF-4269 BOF-4272 CIAPILOME CINCHOPHEN COLCHICEINE DITOLAMIDE ITANOXONE OSMADIZONE OXIPURINOL PROBENECID SECLAZONE SULFINPYRAZONE THIOPURINOL TRICLACETAMOL URATE-OXIDASE ANTIHISTAMINES AF-14 AWD-12-281 BM-113 DIAMIPHENE DIOXOPROMETHAZINE DISPACAMIDE-A ESCIN-I-B IEM-759 JUJUBOSIDE-A MAPINASTINE MAPINASTINE MALEATE METHAFURILENE NIGELLONE NSD-1034 PENASTEROL PROPIOMAZINE QURACOL-A QURACOL-B RHODIOCYANOSIDE-A SETASTINE SKF-91486 SKF-91606 SY-14 TESMILIFENE THIOPERAMIDE ANTIHISTAMINES-H1 ACETYLTYLOPHOROSIDE ACRIVASTINE AD-3264 AHR-5333 AIS-48 ALIMEMAZINE ALOENIN AMLEXANOX ANTAZOLINE ANTIPARKIN ARNICOLIDE-C ARPROMIDINE ASTEMIZOLE AURANTIAMIDE-ACETATE AY-25674 AZATADINE AZELASTINE AZIDOKETANSERIN-7 BAMIPINE BENZMALECENE BEPIASTINE BERMASTINE BETOTASTINE BISULEPIN BISULEPINOXIDE BN-1267 BN-50069 BN-50090 BN-50125 BROCRESINE BROMAZINE BROMOPYRAMINE BROMOPYRILENE BROMPHENIRAMINE BU-E-75 BU-E-76 BUCLIZINE BUFENADRINE BUFROLIN CABASTINE CARBINOXAMINE CAREBASTINE CETIRIZINE CETOXIME CHLORCYCLIZINE

Derwent Drug File 1087 Thesaurus CHLOROPYRAMINE CHLOROPYRILENE CHLORPHENAMINE CHLORPHENOXAMINE CI-959 CINNARIZINE CLEMIZOLE CLOBENZEPAM CLOBENZTROPINE CLOCINIZINE CLOSIRAMINE CROMPROXATE SODIUM CYAMEMAZINE CYCLIRAMINE CYCLIZINE CYPROHEPTADINE D-18024 DAMETRALAST DECARBETHOXYLORATADINE DECLOXIZINE DEPTROPINE DEXBROMPHENIRAMINE DEXCHLORPHENIRAMINE DEXTROCABASTINE DF-1111301 DIETHAZINE DIFENIDOL DIFETEROL DIMEBON DIMENHYDRINATE DIMETHOLIZINE DIMETHYLGLYCYLPHENO= THIAZINE DIMETHYLGLYCYLPHENO= THIAZINE DIMETINDENE DIMETOTIAZINE DIPHENHYDRAMINE DIPHENHYDRAMINE-= METHIODIDE DIPHENHYDRAMINE-= METHYLBROMIDE DIPHENYLPYRALINE DIXYRAZINE DORASTINE DOXANTRAZOLE DOXYLAMINE EBASTINE EMBRAMINE EMEDASTINE EMETHALLICIN-A EMETHALLICIN-B EMETHALLICIN-C EPINASTINE ETANAUTINE ETOLOXAMINE ETYMEMAZINE F-1322 FCC-13 FCC-5 FENETHAZINE FENPIPRANE FEXOFENADINE FLEZELASTINE FLUNARIZINE FRAN-12 GANODERATE-A GANODERATE-B GANODERATE-D HISTAPYRRODINE HOMOCHLORCYCLIZINE HQL-79 HSR-609 HWA-214 IPD-1151T IPROHEPTINE ISOTHIPENDYL K-4300 KAA-276 KC-11404 KETOTIFEN KW-4099 KW-4679 LEVOCABASTINE LEVOCETIRIZINE LEVOPROTILINE LIBECILLIDE LISURIDE LODOXAMIDE LORATADINE LORATADINE M-711 MAGNOSALICIN MDL-16455-A MDL-427 MEBHYDROLIN MECLASTINE MECLOZINE MEDRYLAMINE MEPYRAMINE MEQUITAMIUM IODIDE MEQUITAZINE METHAPHENILENE METHAPYRILENE METHDILAZINE METHOXYDEOXYVASICINONE METIPRENALINE METOXEPIN MIANSERIN MIZOLASTINE MOXASTINE MYOSTIMIN NCO-650 NIAPRAZINE NIPROFAZONE NIVIMEDONE NOBERASTINE OCTASTINE ORG-2305 OXADIMEDINE OXOMEMAZINE PARATHIAZINE PENASTERONE PERASTINE PHENBENZAMINE PHENINDAMINE PHENIRAMINE PHENIRAMINE PAS PHENYLTOLOXAMINE PICLOPASTINE PIMETHIXENE PIPERACETAZINE PIPETHIADENE PIPOXIZINE PIPRINHYDRINATE PIRDONIUM BROMIDE PROMETHAZINE PYRABROM PYROXAMINE PYRROBUTAMINE QUIFENADINE QUINOTOLAST R-44271 REVENAST RHC-3024 ROCASTINE ROTOXAMINE RUPATADINE S-9795 SCH-37370 SENECIOYLPLENOLIN-O-6 SEQUIFENADINE SGB-1534 SKF-93319 SL-85-0324 SUPLATAST-TOSILATE SUPLATAST-TOSILATE TALASTINE TAZIFYLLINE TEMELASTINE TERBUCROMIL TERFENADINE THENALIDINE THENYLDIAMINE THIAZINAMIUM IODIDE THIAZINAMIUM-CHLORIDE THIAZINAMIUM-= METILSULFATE THIAZINAMIUM-SULFOXIDE THIAZINAMIUM-SULFOXIDE = IODIDE THONZYLAMINE THYRONAMINE TIXANOX TMK-688 TOLPROPAMINE TRAZITILINE TRIPELENNAMINE TRIPROLIDINE TRITOQUALINE UCB-28557 UCB-JO28 UR-12592 VUF-8401 VUF-8532 VUF-K-8788 WY-49051 XANOXATE Y-19432 ZCR-2060 ZEPASTINE ZOLAMINE ANTIHISTAMINES-H2 ACEROXATIDINE AD-2646 AH-22216 AMINOINDAZOLE-6 AY-29315 BL-6341A BMY-25271 BMY-25368 BMY-25405 BURIMAMIDE CIMETIDINE CRC-1970 DA-4626 DA-4643 DEMETHYLNIZATIDINE-N2 DONETIDINE E-1309 EBROTIDINE ETINTIDINE FAMOTIDINE FR-145715 FR-A-19 FRG-8813 H-335-25 ICI-162846 ICI-A-5165 IGN-2098 IK-82029 IMPROGAN IT-066 KU-1257 L-643411 L-643441 LAMTIDINE LOXTIDINE METIAMIDE MIFENTIDINE NIPEROTIDINE NIZATIDINE

1088 APPENDIX D NO-794 NORBURIMAMIDE ORF-17578 ORF-17910 OXABURIMAMIDE OXMETIDINE RAMIXOTIDINE RANITIDINE RANITIDINE-BISMUTH-CITRATE ROXATIDINE SKF-92373 SKF-92408 SKF-92540 SKF-92629 SKF-93241 SKF-93319 SKF-93479 SKF-94674 SKF-95083 SKF-95299 SKF-95456 SKF-95495 SKF-95565 SKF-95601 SUFOTIDINE T-593 THIABURIMAMIDE TIOTIDINE TRM-115 TUVATIDINE VUF-8294 VUF-8296 VUF-8297 VUF-8298 VUF-8403 VUF-8406 WHR-2568 WY-45086 WY-45662 WY-45727 YM-14471 Z-300 ZALTIDINE ZOLANTIDINE ANTIHISTAMINES-H3 AQ-0145 BETAHISTINE BURIMAMIDE CIPROXIFAN CLOBENPROPIT CLOPHENPROPIT FUB-181 FUB-360 FUB-451 GR-168320 GT-2227 GT-2331 IMPROMIDINE IODOPHENPROPIT IODOPROXYFAN PROXYFAN THIOPERAMIDE UCL-1199 VUF-4613 ANTIHYPOXICS OLIFEN ANTIINFLAMMATORIES 156-S 230-A 4030-W-92 7351 A-137491 A-192621 A-249377 A-277323 A-771726 A-85783 A-93178 AA-231-1 AA-2379 AAL-13 ABBOTT-29590 ABT-080 ABT-702 ACECLOFENAC ACEMETACIN ACEQUINOLINE ACETAMINOSALOL ACETYL-PAS-N ACLANTATE AD-0261 AE-1734 AE-941 AEOL-11201 AETHIOPINONE AF-150 AF-2259 AGN-190742 AGN-190744 AH-2835 AHR-1911 AJULEMATE AKI-1 ALCLOFENAC ALKANNIN ALLYLCINCHOPHEN ALNUSTONE ALOENIN AMBREIN AMFENAC AMIXETRINE AMPIROXICAM AMTOLMETIN GUACIL ANACROTINE ANAKINRA ANDALUSOL ANGIOSTATIN ANILAMATE ANIROLAC ANITRAZAFEN ANTIFLAMMIN-1 ANTIFLAMMIN-2 ANTRAFENINE APC-366 APREPITANT APYRAMIDE ARA-3000-BETA ARC-69931-MX ARISTOLOCHATE ARISTOLOCHATE-I ARISTOLOCHATE-IA ARISTOLOCHATE-II ARNIDIOL ARTOBILOXANTHONE ARVENSOSIDE-B AS-601811 AS-602240 ASPIRIN ASPIRIN ALUMINUM ASPIRIN MAGNESIUM ASPIRIN SODIUM ASPIRIN-COPPER ASPIRIN-LYSINE-SALT AU-8001 AWD-12-281 AZAPROPAZONE AZIDOPROFEN B-9430 BAY-11-7821 BAY-Y-1015 BB-1101 BB-16 BB-2275 BDH-7538 BENDAZAC BENDAZAC-LYSINE-SALT BENHEPAZONE BENOXAPROFEN BENZASAL BENZOFENAC BENZOFUROCAINE BENZOPYRAZONE BENZOSALIN BENZYDAMINE BENZYDAMINE SALICYLATE BERGENIN BERMOPROFEN BETOL BF-389 BI-L-226XX BI-L-45XX BI-RM-270 BINDARIT BIRB-796 BL-2338 BL-2365 BM-16-2353 BM-16-2354 BM-16-2374 BMS-181162 BMY-30094 BN-063 BORJATRIOL BORNYL-COUMARATE BP-2-94 BRADYZIDE BREIN BRL-10720 BRL-20459 BROFEZIL BROMAMID BROMFENAC BROMOPHENAZONE-4 BROPERAMOLE BUCLOXATE BUCOLOME BUFEXAMAC BUFEZOLAC BUMADIZONE BUTAGLYONAMIDE BUTANIXIN BUTIBUFEN BW-540C BW-755C BX-471 BXT-51072 C-5720 CACOSPONGIONOLIDE-B CAFESTOL CALENDULADIOL CARBAMOYLPHENOXY= ACETATE CARPROFEN CASSUMUNARIN-A CASSUMUNARIN-B CASSUMUNARIN-C CASSUMUNIN-A CASSUMUNIN-B CBS-1108 CBS-113A CCI-779 CDP-571 CDP-870 CELECOXIB CENTAUREIDIN CENTCHROMANE CEREBROCRAST CGP-28237 CGP-47969-A

Derwent Drug File 1089 Thesaurus CGP-8716 CGS-15529 CGS-22745 CGS-23885 CGS-25019-C CGS-25019C CGS-27023-A CH-127 CHAMAZULENE CHF-1194 CHIMAPHILIN CHLORTHENOXAZINE CHLOTAZOLE CHOLINE-MAGNESIUM-= TRISALICYLATE CI-1004 CI-986 CICLOPROFEN CID-85 CINCHOPHEN CINFENOAC CINMETACIN CINNOPENTAZONE CIPROQUAZONE CIS-19 CK-101-A CK-102 CK-103-A CK-113 CK-123 CK-17 CL-306293 CLAMIDOXATE CLANTIFEN CLETOQUINE CLIDANAC CLIPROFEN CLOBENOSIDE CLOFENAMATE CLOFEZONE CLOMETACIN CLONIXERIL CLONIXIN CLONIXIN-LYSINE-SALT CLOPIRAC CLOXIMATE CMI-206 CMI-392 CMT-1 CN-100 CNI-1493 CO-1828 COLFENAMATE COLOSOLATE COMMUNATE-CIS COMPLEMENT-RECEPTOR-= 1-RELATED-GENE-PR.Y CORDIACHROMENE-A CP-0597 CP-105696 CP-122288 CP-14304 CP-195543 CP-331 CP-77059 CROTOXIN-A CS-670 CT-2251 CUPARENE CURCUMENE-ALPHA CURCUMIN CX-659-S CYLEXIN CYTOGENIN D-58 DA-1529 DA-5018 DAISAIKOTO DAK-16 DARBUFELONE DEHYDROPROLINE-3,4 DEHYDROTUMULOSATE DEHYDROZINGERONE DELFANTRINE DELMETACIN DEOXYCHOLATE DEXINDOPROFEN DEXKETOPROFEN DIACEREIN DICLOFENAC DICLOFENAC HYDROXY= ETHYLPYRROLIDINE DICLONIXIN DIFENAMIDE DIFENAMIZOLE DIFENPIRAMIDE DIFLUMIDONE DIFLUNISAL DIFTALONE DIMETHYLSULFOXIDE DIPROSPIDIUM BROMIDE DITAZOLE DKA-9 DORIDOSINE DOTAP DROXICAM DULCEROZINE DUOMETACIN DUP-630 DUP-654 DUP-983 DWH-146-E E-3040 E-5090 E-5110 E-6087 EBSELEN EGIS-5645 ELTENAC EM-405 EMD-66203 EMORFAZONE ENFENAMATE ENKAD EPI-LIPOXIN-B4-15 EPIAFZELECHIN EPIRIZOLE EPOXOMICIN EPOXYQUINOMICIN-D ERMANIN ESCIN-BETA ESCIN-I-B ETABENZARONE ETANERCEPT ETERSALATE ETODOLAC ETOFENAMATE ETOPRINDOLE ETORICOXIB F-1044 F-1067 FARADIOL FC-3280 FECLOBUZONE FELBINAC FELIPYRINE FENAMIFURIL FENAMOLE FENBUFEN FENCHONE FENCLOFENAC FENCLORAC FENCLOZATE FENDOSAL FENFLUMIZOLE FENOPROFEN FENPIPALONE FENSPIRIDE FENTIAZAC FENTIN-CHLORIDE FEPRADINOL FEPRAZONE FEVICORDIN-A FEVICORDIN-A-GLUCOSIDE-2 FI-302 FITOSTIMOLINE FK-3311 FK-706 FLAZALONE FLOBUFEN FLORIPAVINE FLOSULIDE FLUFENAMATE FLUFENISAL FLUMIZOLE FLUNIXIN FLUNIXIN MEGLUMINE FLUNOXAPROFEN FLUPROFEN FLUPROQUAZONE FLUQUAZONE FLURBIPROFEN FLURBIPROFEN-ETHYL-ESTER FLURBIPROFEN-NITROXY= BUTYLESTER FLURETOFEN FLUTIAZIN FPL-62064 FPL-64170-XX FPL-67047-XX FPP-028 FR-110302 FR-123826 FR-133605 FR-134043 FR-140423 FR-167344 FR-173657 FRIEDELANOL FTAXILIDE FURAPROFEN FUROBUFEN FUROFENAC FUSCOSIDE-B GALECTIN-1 GALOSEMIDE GEA-3162 GEA-5024 GF-109203X GLAFENINE GLUCAMETACIN GLYCOSAMINOGLYCAN-= POLYSULFATE GLYCYRAM GLYCYRRHIZATE GLYDERININE GLYTEER GOE-6983 GP-1-515 GP-53633 GPA-1851 GPI-6150 GSC-150 GUAIAZULENE GUAIMESAL GUALENATE SODIUM GUGGULSTERONE-E GUGGULSTERONE-Z GV-196771-A GW-274150 GW-4459 GW-92527

1090 APPENDIX D GX-258 GY-97 GYKI-66114 H-88 HAI-105 HCT-3012 HELIANTRIOL-B2 HELIANTRIOL-C HEMATEIN HERACLENIN HERACLENOL HEXAPROFEN HIMACHALENE-BETA HOLAPHYLLINE HP-228 HP-466 HP-573 HWA-131 HYDROXYACECLOFENAC-4 HYDROXYACHILLIN-4 HYDROXYETHYLSALICYLATE HYRTIAL I-152 IBUFENAC IBUPROFEN IBUPROFEN LYSINE IBUPROXAM ICI-115432 ICI-216800 ICI-43823 ICI-D-2138 ID-955 IMBRICATOLATE IMIDAZOLE SALICYLATE INDOBUFEN INDOMETACIN INDOMETACIN MEGLUMINE INDOMETACIN-FARNESIL INDOPROFEN INDOXOLE INTERLEUKIN-13 INTERLEUKIN-18-BINDING-= PROTEIN-A-HUMAN INTRAZOLE INUVISCOLIDE IRCININ-1 IRCININ-2 IRFI-005 IRFI-016 ISAMFAZONE ISIS-2302 ISOCHLOROGENATE-A ISOCHLOROGENATE-C ISOCUPRESSATE ISOFEZOLAC ISOLARICIRESINOL ISONIXIN ISOPIMARATE ISOPLUMBAGIN ISOPROPYLAMINO= PHENAZONE ISOTETRANDRINE ISOXEPAC ISOXICAM ITANOXONE ITF-611 ITF-614 JM-34 JTE-522 K-1115-A K-76 KA-398 KB-1043 KB-2683 KEBUZONE KETOPROFEN KETOPROFEN LYSINE KF-24345 KL-11 KME-4 L-651392 L-651896 L-652343 L-674636 L-694458 L-745337 L-746483 L-746530 L-754030 L-761066 L-768277 L-8109 LABDANE-F2 LANEPITANT LEFLUNOMIDE LEIOCARPOSIDE LEVOMENOL LEX-032 LEXIPAFANT LEXOFENAC LG-101305 LICOFELONE LICORICIDIN LIGSTROSIDE LIPOMESACONITINE LIPOXIN-A4 LISOFYLLINE LM-1228 LOPIRINE LORNOXICAM LOXOPROFEN LU-20884 LUFFARIELLIN-A LUFFARIELLIN-B LUFFARIELLOLIDE LUMIRACOXIB LUPENYL-ACETATE LUPEOL-LINOLEATE LUPEOL-PALMITATE LY-178002 LY-221068 LY-256548 LY-269415 LY-293111 LY-334370 LY-393053 M-1704 M-40403 M-5011 MAGNOSALIN MAGNOSHININ MANOALIDE MANSUMBINOATE MANSUMBINONE MARIMASTAT MARMIN MASTICADIENONATE MB-432 MCD-PEPTIDE MCN-2891 MEBENOSIDE MECLOFENAMATE MEFENAMATE MELOXICAM MEPROTIXOL MERCAPTOETHYLGUANIDINE MESECLAZONE MET-RANTES METBUFEN METHYLCUMARIN-7 METHYLNIPHENAZINE METHYLSALICYLATE METIAZINATE METOXIBUTROPATE MEXOPROFEN MG-115 MG-132 MG-341 MILOXICAM MIROPROFEN MK-447 MK-715 MK-825 MK-966 MOFEBUTAZONE MOFEZOLAC MORAZONE MORELLOFLAVONE MORETENOL MORETENOL-ACETATE MORNIFLUMATE MR-714 MV-8608 MV-8610 MV-8612 MYTILAN NABUMETONE NAFTYPRAMIDE NAPROXEN NAPROXEN-LYSINE-SALT NAPROXOL NAT-02-677 NAT-06-097 NB-431 NC-1140 NCX-1015 NCX-4016 NCX-701 NCX-950 NE-28345 NEOLUPENOL NEPAFENAC NEUTROPHIL-INHIBITORY-= FACTOR NEYARTHROS NEYCHONDRIN NEYNORMIN NEYTHYMUN-F NEYTROPH NICHLOTEST NICOTINOYLTRYPTAMINE-N NICTINDOLE NIFENAZONE NIFLUMATE NIMAZONE NIMESULIDE NIMESULIDE-LYSINE-SALT NIOMETACIN NIPROFAZONE NITRAQUAZONE NITROACETYLSALICYLATE NITROFENAC NITROSALICYLATE-5 NITROSTANOLONE NIXYLATE NMI-377 NONIVAMIDE-ACETATE NPB-1 NPC-14692 NPC-15199 NPC-15669 NPC-18730 NR-583143 NS-398 OC-229-648 ONO-3144 ORGOTEIN ORIDINE ORPANOXIN OXACEPROL OXAMETACIN OXAPROZIN

Derwent Drug File 1091 Thesaurus OXEPINAC OXIFULVATE OXINDANAC OXOLAMINE OXPHAMAN OXYCINCHOPHEN OXYPHENBUTAZONE P-34081 P-8977 P-9782 P-SELECTIN-GLYCO= PROTEIN-LIGAND-1 PAEONIFLORIN PALAUOLOL PALMIDROL PARECOXIB PARSALMIDE PAXAMATE PC-796 PD-136095 PD-138387 PD-144795 PD-164387 PD-184352 PENICILLAMINE-COPPER PENTAGALLOYLGLUCOSE PEP-1261 PEUDOPTEROSINE-B PF-5901 PGV-20229 PH-163 PHENIDONE PHENYLBUTAZONE PHENYLBUTAZONE COPPER PHENYLBUTAZONE = PIPERAZINE PHILLYRIN PHLEBODRIL PHYCOCYANIN-C PICOBENZIDE PICROPOLYGAMAIN PICUMETEROL PIFOXIME PIMECROLIMUS PIMEPROFEN PIMETACIN PIPEBUZONE PIRAZOLAC PIRFENIDONE PIROXICAM PIROXICAM-CINNAMATE PIRPROFEN PJ-34 PKSI-527 PR-39 PRANOPROFEN PRANOSAL PRAXADINE PREFENAMATE PREPARATION-E PRINOMIDE PRODOLATE PROGLUMETACIN PROQUAZONE PROTIZINATE PROXAZOLE PROXIFEZONE PS-519 PSEUDOPTEROLIDE PSEUDOPTEROSIN-A PSEUDOPTEROSIN-B PSEUDOPTEROSIN-C PSEUDOPTEROSIN-D PSEUDOPTEROSIN-E PSEUDOPTEROSIN-F PSEUDOPTEROSIN-G PSEUDOPTEROSIN-H PSEUDOPTEROSIN-I PSEUDOPTEROSIN-J PYRUVATE-ETHYL-ESTER PZ-25 QUERCILICOSIDE-A QUINAZOPYRINE R-830 RDP-58 RENYTOLINE REV-5901 RHEIN RO-23-0238 RO-23-6457 RO-24-0238 RO-24-9981 RO-31-8425 RO-31-8830 RODAPLUTIN ROFECOXIB ROHITUKINE ROHITUKINE RP-61605 RP-62373 RP-63165 RP-63600 RP-67580 RPR-100893 RPR-130737 RS-2131 RS-37619 RS-504393 RU-29693 RU-43526 RUVAZONE RWJ-50271 RWJ-63556 S-16474 S-2474 S-6907 SAIKOSAPONIN-A SAIKOSAPONIN-D SALCOLEX SALICYLATE COPPER SALICYLATE DIETHYLAMINE SALICYLATE MORPHOLINE SALICYLATE-CHOLINE SALICYLATE-MEGLUMINE SALICYLATE-PROPYL SALPROTOSIDE SANDARACOPIMARATE SANTIN SB-202190 SB-203347 SB-203580 SB-206718 SB-220025 SB-239063 SC-41930 SC-50605 SC-51146 SC-52608 SC-53228 SC-57666 SC-58125 SC-8076 SC-8092 SCALARADIAL SCH-351591 SCH-40120 SCH-50971 SCHA-123 SCHA-395 SCHA-764 SCHA-87 SCYPHOSTATIN SDZ-224-015 SDZ-ASM-981 SECLAZONE SEK-1005 SERICATE SERICOSIDE SERMETACIN SF-2370 SHOSAIKO-TO SIDERITOFLAVONE SJC-13 SKF-104351 SKF-104493 SKF-105561 SKF-105809 SKF-106615 SKF-106978 SKF-26070 SKF-45905 SKF-86002 SKF-98625 SM-10661 SM-15178 SPINORPHIN SQ-29535 SR-31747 SR-31747-A ST-341 STAMPYRINE STRINOLINE SUBTILISIN SUDOXICAM SULINDAC SULINDAC-SULFIDE SULPROSAL SUPROFEN SY-6001 T-0757 T-3811-ME T-614 TA-60 TAI-908 TAK-603 TALMETACIN TALNIFLUMATE TALOSALATE TALSO TARAXASTEROL TARAXASTEROL-PSI TASPINE TAURINAMINOPYRIDINE TEBUFELONE TECTORIDIN TEI-1338 TEL-1338 TENIDAP TENOXICAM TEPOXALIN TEROFENAMATE TESICAM TESIMIDE TETRIDAMINE TETRIPROFEN THIELOCIN-B3 THIOCOLCHICOSIDE THYMOQUINONE TIANAFAC TIAPROFENATE TIARAMIDE TICLOPIDINE TIFLAMIZOLE TILOMISOLE TIMEGADINE TINORIDINE TIOPINAC TIOXAPROFEN TIZOPROLATE TOLFENAMATE TOLMETIN TOLMETIN-GLYCINE-AMIDE

1092 APPENDIX D TOLMETIN-PARACETAMOL-= ESTER TOMATINE TOMOXIPROLE TP-151 TP-72 TR-1722 TR-35 TRIACONTANOL TRIBUZONE TRICLACETAMOL TRIFEZOLAC TRIFLUMIDATE TROPESIN TUBERCULATIN TUMOR-NECROSIS-FACTOR-= RECEPTOR-I TYLOPHORINIDINE TZI-615 U-0126 U-101033-E U-24568 U-81581 U-82579 U-84849 U-91502 UFENAMATE UR-8880 V-33 VALDECOXIB VETIVAZULENE VICOLIDE-A VICOLIDE-C VICOLIDE-D VINIFERIN-ALPHA VUF-9019 VUF-9020 VUF-9045 WAY-121520 WILD-20 WIN-63759 WIN-64733 WIN-67694 WY-25110 WY-41770 WY-47288 WY-48090 WY-49232 XC-386 XIMOPROFEN XU-745 Y-23023 Y-24180 Y-39041 Y-5554 Y-9223 YAKUCHINONE-B YM-26567-1 YM-26734 YPE-01 YT-1 ZANHASAPONIN-A ZANHASAPONIN-B ZANHASAPONIN-C ZARDAVERINE ZCR-2060 ZIDOMETACIN ZK-158252 ZOLIPROFEN ZOMEPIRAC ANTILEPROTICS ACEDAPSONE ALDESULFONE SODIUM CLOFAZIMINE DAPSONE DIATHYMOSULFONE DIUCIPHON ETHIONAMIDE GLUCOSULFONE K-107 K-137 K-138 PROTIONAMIDE RIFAMPICIN SOLASULFONE SUCCISULFONE SULFADIASULFONE SODIUM THIAMBUTOSINE THIAZOSULFONE THIOACETAZONE ANTIMANICS CARBAMAZEPINE LITHIUM-CARBONATE LITHIUM-CITRATE RS-86 VALPROATE VALPROATE SODIUM ANTIOXIDANTS 116-L 129-L 764-3 AD-5 AEOL-10113 AEOL-11201 AK-135 AK-40 AK-49 ALLYLTHIOPYRAZINE-2 ALT-711 AM-36 AM-404 AMTIZOLE ANDRASTIN-A ANEMARRHENASAPONIN-IA ANHYDROFRUCTOSE-1,5 ANPHEN ASCORBATE ASCORBYL-STEARATE ASTAXANTHIN ASTRINGIN ATRACTYLOCHROMENE BCE-001 BCR-4 BENZALAZINE BENZASTATIN-A BENZASTATIN-B BENZASTATIN-C BENZASTATIN-D BGP-15 BISORBICILLINOL BLACK-TEA-EXTRACT BM-140830 BM-14686 BM-15-0639 BM-910183 BM-910228 BMS-182123 BN-80933 BO-653 BORNYL-COUMARATE BROUSSOCHALCONE-A BUTYLATED-HYDROXY= ANISOLE BUTYLATED-HYDROXY= TOLUENE CAFFEATE CARAZOSTATIN CARBAZOQUINOCIN-B CARBAZOQUINOCIN-C CARBAZOQUINOCIN-E CARBAZOQUINOCIN-F CARBOXYFULLERENE CASSUMUNARIN-A CASSUMUNARIN-B CASSUMUNARIN-C CASSUMUNIN-A CASSUMUNIN-B CBS-113A CDRI-82-437 CH-402 CHLORIN-E6-IRON CHLOROPHYLLIN-COPPER-= SODIUM CO-1828 CONJUGATED-LINOLEATE-= 10-TRANS-12-CIS CP-060 CP-130 CP-502 CP-511 CURVULATE CV-3611 CX-659-S CYANIDIN-3-GLUCOSIDE DEHYDROASCORBATE DEMETHOXYANGONIN DI-TERT-BUTYLPHENOL-2,6 DIALLYL-TETRASULFIDE DIHYDROTHIOCTATE DIHYDROXYFLAVONE-3+,4+ DIHYDROXYFLAVONE-6,7 DILUDINE DIPHENYL-PHENYLENE= DIAMINE-PARA DUOKVIN EBSELEN ECHINOCHROME EMQ EPC-K1 EPYGID ERIOCITRIN ETHOXYQUIN ETOMERSOL EUK-134 EUK-8 F-11344-A-1 FERULATE-ETHYL-ESTER FLAVANONE FORMALDEHYDE= SULFOXYLATE SODIUM FULLERENOL GACAVIT GALLATE-BUTYL GALLATE-DECYL GALLATE-DODECYL GALLATE-ETHYL GALLATE-HEPTADECYL GALLATE-METHYL GALLATE-OCTYL GALLATE-PROPYL GALLATE-TETRADECYL GARCINOL GEA-3162 GINKGO-BILOBA-EXTRACT GINSENOSIDE-RG5 GLABRENE GLABRIDIN H-290-51 H-2954 HAMAMELITANNIN HEMATEIN HERBERTENEDIOL HI-253 HISPIDIN HISTOCHROME HUMULONE HWA-131 HX-1171 HYDROXYCARVEDILOL-1 HYDROXYCHAVICOL HYDROXYINDAPAMIDE-5

Derwent Drug File 1093 Thesaurus HYDROXYPYRIDINE-3 I-152 IDEBENONE IH-636 IRFI-005 IRFI-016 IRFI-042 IRFI-048 ISALPININ ISOCHLOROGENATE-A ISOCHLOROGENATE-C ISOGINKGETIN ISOGUANOSINE ISOPROPOXYGERMATRANE ISORHAPONTIGENIN ISOTHIOBARBAMINE ISOTORACHRYSONE J-811 J-861 KB-5666 KR-31372 KR-31378 KS-79 LAVANDUQUINOCIN LEUCOSCEPTOSIDE-A LEX-032 LI-1370 LICOCHALCONE-A LICOCHALCONE-B LICOCHALCONE-D LICOCOUMARONE LITHOSPERMATE-B LOBENZARIT LUPULONE LY-213829 LY-221068 LY-231617 LY-294002 M-40401 M-40403 MAHARISHI-4 MANSONONE-F MDL-101002 MDL-102832 MDL-104342 MDL-105185 MDL-73404 MDL-74270 MDL-74366 MDL-74405 MEQUINOL MERCAPTODEXTRAN MERCAPTOETHYLGUANIDINE MESO-DIHYDRO= GUAIARETATE METHYLCATECHOL-4 MTDA-DA MTDQ-DA MYRIGALONE-A MYRIGALONE-B NAPHTHGERANINE-A NECTANDRIN-B NEOCARAZOSTATIN-B NORDIHYDROGUAIARETATE NXY-059 OCTADECADIENOATE-9-= CIS,11-TRANS OLEANOLATE-ACETATE OOLONG-TEA-EXTRACT OP-6 OPB-9195 OPC-14117 OPC-6535 OR-10141 P-1507 P-9782 PATULETIN PEP-1261 PHENOSAN PHENSUCCINAL PHYCOCYANIN-C PIFITHRIN-ALPHA PINOCEMBRIN POLAPREZINC PR-39 PROTOCATECHUALDEHYDE PROTOCATECHUATE PURPUREASIDE-A PYCNOGENOL PYRIDOXATIN PYRUVATE-ETHYL-ESTER PZ-25 QUERCETIN-GLUCURONIDE-3 R-830 REOFLUSINE RPR-100579 S-20478 S-2474 S-32502-1 S-33113 SALVIANOLATE-B SC-52608 SCHISANDRIN-A SCHIZANDRIN-B SECOISOLARICIRESINOL-= DIGLUCOSIDE SESAMOL SILIBOR SITOINDOSIDE-IX SITOINDOSIDE-X SODIUM-METABISULFITE SOPHORIDINE SOYASAPONIN-BETA-G SPINOCHROME-A SPINOCHROME-B SPINOCHROME-C SPINOCHROME-D SPINOCHROME-E SUN-N-8075 TAK-218 TENOX-TBHQ TETRAHYDROCURCUMIN TIOTRIAZOLIN TIRILAZAD MESILATE TOCOPHEROL-DELTA TOMERZOLE TR-1722 TRIHYDROXYBENZENE-1,2,4 TRIMETHYLELLAGATE-3,3+,4 TRIPTERIN TROGLITAZONE TROLOX TSITSIXENICIN-A TUBULOSIDE-B U-101033-E U-104067-F U-106311-E U-74389 U-74389F U-74389G U-74500-A U-75013 U-75014-E U-75412E U-78518-E U-78518F U-79206 U-83836 U-83836E U-87999 U-89843 U-89843-D U-89843-E U-94430-E VF-233 XAX-M ZAHAVIN-A ANTIPARKINSONIANS 1067-CERM A-77636 A-86929 ABT-431 ALAPTIDE ALTINICLINE AMANTADINE AMEDIN ANTIPARKIN BAM-1110 BENAPRIZINE BENSERAZIDE BENZATROPINE BIA-3-202 BIPERIDEN BN-80933 BORNAPRINE BOTIACRINE BROMOCRIPTINE BUDIPINE BUFENADRINE BUTYLSYMPATON CARAMIPHEN CARBIDOPA CARMANTADINE CGP-3466-B CGP-40116 CHLORPHENOXAMINE CILADOPA CITICOLINE CLOFENETAMINE CQA-206-291 CYCRIMINE DELERGOTRILE DEPRAMINE DEXETIMIDE DICARFEN DIETHAZINE DIPHENYLTROPINE DIPROBUTINE DOPA DOPAC DOPAMANTINE ELANTRINE ENTACAPONE ETANAUTINE ETISULERGINE ETYBENZATROPINE EUK-134 FLUNAMINE GLIAL-CELL-DERIVED-= NEUROTROPHIC-FAC.HUM GLIAL-CELL-DERIVED-= NEUROTROPHIC-FAC.RAT GLIAL-CELL-DERIVED-= NEUROTROPHIC-FACTOR HA-966 HALONAMINE HARMINE KW-6002 LEVODOPA LOMETRALINE MAZATICOL MEDIPINE MEMANTINE MESULERGINE METIXENE MINEPENTATE N-1199 NAXAGOLIDE NB-355 OMIDOLINE ORPHENADRINE

1094 APPENDIX D PAREPTIDE PHENGLUTARIMIDE PIROHEPTINE PIVAGABINE PR-000608 PRIDINOL PROCYCLIDINE PRODIPINE PROFENAMINE PROSAPTIDE-D-5 RASAGILINE ROMERGOLINE RS-1653 S-3473 S-584 SIB-1508-Y SIB-1553-A SIB-1765-F TIGLOIDINE TOFENACIN TOLCAPONE TOLPERISONE TRIHEXYPHENIDYL TRIPERIDEN TROPATEPINE TROPIGLINE U-91356 U-91356-A V-10367 WF-23 ANTIPERSPIRANTS GLUTARAL ANTIPRURITICS AZATADINE CALAMINE COLESTYRAMINE CROTAMITON DIMETINDENE DOXEPIN ISOPRENALINE JUNIPER-TAR MOMORDIN-IC MONODEMETHYLDOXEPIN OXOMEMAZINE PIMECROLIMUS POLIDOCANOL PURIGENS QUINISOCAINE SUCCINONITRILE TRK-820 ANTIPSORIATICS ACITRETIN ALOE-EMODIN-ANTHRONE AMEVIVE ANAPSOS APC-2059 AZARIBINE BEECH-TAR BMY-30123 BUTANTRONE CALCIPOTRIOL CGP-52411 CHLORANIL CHRYSAROBIN DIETHYL-FUMARATE DIMETHYL-FUMARATE DITHRANOL DUP-654 DUP-983 EB-1213 EFOMYCINE-M EMODINANTHRONE ETANERCEPT ETRETINATE FPL-62064 FUMADERM GS-1500 ISOACITRETIN ISOQUINOLINE (Drug) JUNIPER-TAR LONAPALENE LYSOPHOSPHATIDATE MONOETHYL-FUMARATE MONOMETHYL-FUMARATE MONOOCTYL-FUMARATE NDH-3080 NICOTINYL-AMINO= NICOTINATE-6 OLEOYLETHANOLAMINE-N P-9782 PIMECROLIMUS PS-519 SB-220025 SB-239063 SCH-40120 SDZ-281-240 SIPLIZUMAB SPC-103600 SULFUR-MUSTARD TACALCITOL TAZAROTENE ANTIPYRETICS AA-2379 ACETAMINOSALOL ACETANILIDE ACETYLPHENYLHYDRAZINE ACONITINE AF-2259 ALCLOFENAC ALLYLTHIOUREA AMINOANTIPYRINE AMINOCHLORTHENOXAZINE AMINOPHENAZONE AMINOPHENAZONE = CYCLAMATE ANALGEN APYRAMIDE ASPIRIN ASPIRIN ALUMINUM ASPIRIN MAGNESIUM ASPIRIN SODIUM ASPIRIN-COPPER AU-8001 BENHEPAZONE BENZYDAMINE BENZYDAMINE SALICYLATE BERMOPROFEN BOA BROPERAMOLE BUFEZOLAC BUMADIZONE CARBAMOYLPHENOXY= ACETATE CARPROFEN CAUSYTH CENTCHROMANE CHLORTHENOXAZINE CHLORZACETAMOL CLANTIFEN CLIPROFEN CRESOTAMIDE DETANOSAL DIBUPYRONE DIFENPIRAMIDE DIFLUNISAL DISALICYLSUCCINATE DROXICAM E-5110 EGIS-5645 ETERSALATE ETORICOXIB F-1044 FAMPROFAZONE FENCLORAC FENCLOZATE FENDOSAL FENFLUMIZOLE FENTIAZAC FI-302 FK-3311 FLURBIPROFEN FLURBIPROFEN-ETHYL-ESTER FOSFOSAL FPP-028 FS-205-397 FX-205-754 GINGEROL-6 GLUCAMETACIN GUAIMESAL GX-258 HCT-3012 HEXAPROFEN HYDROXYQUINOLINE= SULFONATE-PARA IBUPROXAM IMIDAZOLE SALICYLATE INDOMETACIN INDOMETACIN MEGLUMINE INDOXOLE IODOPHENAZONE ISOFEZOLAC ISOXICAM JTE-522 L-652343 L-745337 L-768277 LACTYLPHENETIDINE LICOFELONE LOPIRINE MESECLAZONE METAMIZOLE SODIUM METOXIBUTROPATE MOFEZOLAC NAPROXEN NAPROXOL NCX-701 NIOMETACIN NORAMIDOPYRINE NS-398 ORIDINE OXEPINAC OXYCINCHOPHEN PARACETAMOL PHENACETIN PHENAZONE PHENICARBAZIDE PHENYL-SALICYLATE PIMETACIN PIRFENIDONE PROPACETAMOL PROPYPHENAZONE QUININE QUININE SALICYLATE QUININE-ETHYLCARBONATE RS-2131 S-6907 SALACETAMIDE SALCOLEX SALICYLAMIDE SALICYLATE SALICYLATE MORPHOLINE SALICYLATE SODIUM SALICYLATE TROLAMINE SALICYLATE-CHOLINE SC-560 SHOGAOL-6 SKF-26070 SULINDAC SULINDAC-SULFIDE

Derwent Drug File 1095 Thesaurus SULPROSAL SUMACETAMOL SUPROFEN T-614 TIARAMIDE TIOPINAC TOLMETIN-PARACETAMOL-= ESTER TROPESIN TZI-615 V-33 VICOLIDE-A VICOLIDE-C VICOLIDE-D WY-41770 ZOLIPROFEN ANTIRHEUMATICS A-249377 A-277323 A-771726 ACARIT ACETAMINOSALOL ADALIMUMAB AF-2259 AG-4263 ALFLUTOP ALLOCUPREIDE SODIUM ALLOPURINOL ALLYLCINCHOPHEN ALOXIPRIN AMFLUTIZOLE ANAKINRA APYRAMIDE ARTEPARON ASPIRIN ASPIRIN ALUMINUM ASPIRIN MAGNESIUM ASPIRIN SODIUM ASPIRIN-COPPER AURANOFIN AUROCYANIDE AUROTHIOGLUCOSE AUROTHIOGLYCANIDE AUROTHIOMALATE SODIUM AUROTHIOSULFATE AUROTIOPROL BATIMASTAT BB-1101 BB-16 BENZOPYRAZONE BENZOSALIN BENZPIPERYLONE BENZYLNICOTINATE BETOL BI-L-45XX BINDARIT BIRB-796 BMS-224818 BUCILLAMINE BUCOLOME BUTOPYRAMMONIUM IODIDE CALCINAPHTHOL CAMPHOR CAUSYTH CBS-1114 CDP-571 CDP-870 CELECOXIB CGP-28237 CGP-29030-A CGP-47969-A CGS-27023-A CHLOROQUINE CHOLINE-MAGNESIUM-= TRISALICYLATE CI-1004 CI-987 CID-85 CINCHOPHEN CIPEMASTAT CL-306293 CLAMIDOXATE CLOFENAMATE CLOFEZONE CLORACETADOL COLCHICINE CP-105696 CPH-82 CUPROXOLINE CYTOGENIN DAK-16 DARBUFELONE DECLABEN DH-40J DIACEREIN DIFENPIRAMIDE DIFTALONE DIPYROCETYL DISALICYLSUCCINATE E-5110 EMD-66203 EPIAURANOFIN EPOXYQUINOMICIN-A EPOXYQUINOMICIN-B EPOXYQUINOMICIN-C EPOXYQUINOMICIN-D ETANERCEPT ETEBENECID ETORICOXIB FANETIZOLE FENAMIFURIL FENAMOLE FENCHONE FLOBUFEN GENTISATE GLUCURONYLGALACTOS= AMINO-GLYCAN-SULFATE GLYDERININE GOLD-CHLORIDE GOLD-CHLORIDE-TRIETHYL= PHOSPHINE GOLD-KERATINATE GOLD-SALT (Drug) GOLD-TRICHLORIDE-ACID GW-92527 HYDROXYACECLOFENAC-4 HYDROXYCHLOROQUINE IBUFENAC IBUPROFEN IBUPROFEN LYSINE INDOMETACIN INDOMETACIN MEGLUMINE INDOMETACIN-FARNESIL ISOPROPYLAMINO= PHENAZONE JTE-522 KE-298 KE-748 KEBUZONE L-758354 LACTYLPHENETIDINE LEFLUNOMIDE LOBENZARIT LOPIRINE MARIMASTAT MECLOFENAMATE MEFENAMATE METAMIZOLE SODIUM METBUFEN METHYLNIPHENAZINE METHYLSALICYLATE METOXIBUTROPATE MG-341 MNX-160 MOFEBUTAZONE MOLITRANS MR-714 MX-68 NB-431 NEOCINCHOPHEN NEYARTHROS NEYCHONDRIN NEYNEPHRIN NEYNORMIN NEYTHYMUN-F NEYTROPH NICOTINATE-BENZYL NIFENAZONE NIXYLATE NORLETIMOL OLETIMOL ORGOTEIN OXYCINCHOPHEN OXYPHENBUTAZONE PD-138387 PD-144795 PD-184352 PHENAZONE PHENIDONE PHENYL-SALICYLATE PHENYLBUTAZONE PHENYLBUTAZONE COPPER PHENYLBUTAZONE = PIPERAZINE PHYTODOLOR PIMETACIN PIPERAZINE PIRAZOLAC QUINATE R-830 RENYTOLINE RHEUMA-HEK RHEUMAJECTA RO-31-9790 RO-32-3555 ROMAZARIT RP-54745 RS-37619 RUMALON S-2474 S-6907 SA-679 SALACETAMIDE SALAMIDACETATE SODIUM SALICYLATE SALICYLATE COPPER SALICYLATE TROLAMINE SALICYLATE-MEGLUMINE SALOCOLUM SALSALATE SB-210396 SB-273005 SEATONE SINOMENINE SKF-101510 SKF-36914 SKF-40539 SKF-60817 SKF-80019 SKF-85626 SKF-85626 SKF-D-83940 SM-8849 SODIUM-TETRACHLORO= AURATE SR-31747-A SULFINPYRAZONE SUXIBUZONE T-72258 TAK-603 TEBUFELONE

1096 APPENDIX D TENIDAP TENOXICAM TIFLAMIZOLE TILOMISOLE TILUDRONATE TJ-114 TOK-8801 TOLFENAMATE TRIBUZONE TROPESIN U-11790 U-11866 U-18598 U-22312 U-22989 U-24278 U-24279 U-24522 U-24631 U-27391 U-81581 U-82579 U-84849 VALDECOXIB VASOLASTINE WY-41770 XIMOPROFEN Y-39041 ZINC-MONOGLYCEROLATE ZINC-SULFATE ZOXAZOLAMINE ANTISEBORRHEICS AS-601811 AS-602240 CHLOROXINE CLIMBAZOLE ISOTRETINOIN MK-386 PIROCTONE PROPYLTESTOSTERONE-17-= ALPHA PYRITHIONE ZINC RU-58841 STEINAZIDE TIOXOLONE XENYSALATE ANTISENSE ISIS-1082 ISIS-11061 ISIS-12449 ISIS-12959 ISIS-13650 ISIS-1570 ISIS-1751 ISIS-1753 ISIS-1755 ISIS-2105 ISIS-2302 ISIS-2503 ISIS-2922 ISIS-3082 ISIS-3521 ISIS-4015 ISIS-8005 ISIS-9044 ISIS-9047 ANTISEPTIC BACTERIOSTATIC ANTISEPTICS 216C 235C 272C 27753-RP 27753-RP A-56619 A-57274 A-62251 A-62824 A-86719-0 ACEDAPSONE ACEDIASULFONE SODIUM ACETYLISONIAZID ACETYLSULFADIAZINE ACETYLSULFAETHOXAZOLE ACETYLSULFAFURAZOLE ACETYLSULFAMETHOXAZOLE ACETYLSULFAMETHOXY= PYRAZINE ACETYLSULFAMETHOXY= PYRIDAZINE ACONIAZIDE ACRIFLAVINIUM CHLORIDE ACTINOQUINOL ACTOFURAN ADITOPRIM AG-1789 AGELIFERIN AKRITOIN ALAFOSFALIN ALCIDE ALDESULFONE SODIUM ALEXIDINE ALKONIUM BROMIDE ALLOCUPREIDE SODIUM AMANTANIUM BROMIDE AMBAZONE AMIFLOXACIN AMINOACRIDINE AMINOACRIQUINE AMINOQUINCARBAMIDE AMINOQUINURIDE AMINOSALICYLATE SODIUM AMQ-4 AMQ-5 AMUCHINA AMYLMETACRESOL ANTHRAROBIN APIDAECIN APIDAECIN-IB APLIDIASPHINGOSINE APLYSIANIN-E APLYVIOLENE ARSANILATE ARSANILATE SODIUM ARSPHENAMINE AUREOL AURINTRICARBOXYLATE AVAROL AVARONE AW-464 AXISONITRILE-3 AZAROLE AZD-2563 AZOSULFANILAMIDE B-1772 B-1865 B-1912 B-283 B-3640 B-3722 B-3770 B-3779 B-3785 B-3786 B-4019 B-4021 B-4076 B-4087 B-4100 B-4101 B-4154 B-4157 B-432 B-433 B-621 B-628 B-654 B-669 B-670 B-685 B-746 B-749 B-776 B-797 B-826 B-980 BA-30515 BA-32476 BA-32641 BA-34358 BA-35597 BA-35969 BA-36204 BA-36208 BA-36435 BA-37215 BA-40922 BA-42517 BACTENECIN BACTENECIN-5 BACTENECIN-7 BALOFLOXACIN BALSALAZIDE BALUDON BAQUILOPRIM BAS-118 BASTADIN-2 BASTADIN-6 BAY-P-9357 BAY-Q-3542 BAY-R-3964 BAY-S-9435 BAY-Y-3118 BAYCOVIN BENFLURON BENOFLOXACIN BENSALAN BENZALKONIUM BROMIDE BENZALKONIUM CHLORIDE BENZAMIDOSALICYLATE = CALCIUM BENZETHONIUM CHLORIDE BENZODODECINIUM = CHLORIDE BENZOXIQUINE BENZOXONIUM CHLORIDE BENZOYLPEROXIDE BENZYL-ALCOHOL BENZYLPARABEN BENZYLSULFAMIDE BETA-DEFENSIN-2-HUMAN BETA-DEFENSIN-3-HUMAN BETOL BIBROCATHOL BICLOTYMOL BIRCH-TAR BISMUTH SODIUM = TRIGLYCOLLAMATE BISMUTH-SODIUM-TARTRATE BISMUTH-TRIBROMPHENATE BITHIONOL BITIONOLATE SODIUM BKH-14 BMY-33315 BMY-40062 BMY-40124 BMY-40397 BMY-40662 BMY-41429 BMY-42230

Derwent Drug File 1097 Thesaurus BMY-43261 BRILLIANT-GREEN BRODIMOPRIM BROMCHLORENONE BROMCHLOROPHEN BRONIDIOL BRONOPOL BROQUINALDOL BROXALDINE BROXYQUINOLINE BT-402 BUFORIN-I BUFORIN-II BUTYLPARABEN C31G CACOSPONGIONOLIDE-B CADEXOMER-IODINE CAERIN-1.1 CALCINAPHTHOL CALCIUM-HYPOCHLORITE CANADALINE CAP-18-HUMAN CAPROCHLORONE CAPTAN CARBADOX CARBAMIDE-PEROXIDE CARBANILIDE CARBOXYFULLERENE CATAPOL CATIONIC-ANTIMICROBIAL-= PROTEIN-20-44 CECROPIN-B CECROPIN-B-1 CECROPIN-P-1 CETALKONIUM CHLORIDE CETHEXONIUM CHLORIDE CETRIMIDE CETRIMONIUM BROMIDE CETYLPYRIDINIUM BROMIDE CETYLPYRIDINIUM CHLORIDE CFC-222 CHAULMOSULFONE CHINIOFON CHLORAMINE-B CHLORAZODIN CHLORCARVACROL CHLORHEXIDINE CHLORHEXIDINE GLUCONATE CHLORHEXIDINEPHOSPHANILATE CHLORINE-DIOXIDE CHLOROBUTANOL CHLOROCRESOL CHLOROUS-ACID CHLOROXINE CHLOROXYLENOL CHLORPHENOCTIUM = AMSONATE CHLORQUINALDOL CHROMODOROLIDE-A CHRYSOIDINE CI-934 CIADOX CICLIOMENOL CINOQUIDOX CINOXACIN CIPROFLOXACIN CITENAZONE CL-64855 CLAVANIN-B CLAVANIN-C CLAVANIN-D CLEANUP CLINAFLOXACIN CLIOQUINOL CLOFAZIMINE CLOFOCTOL CLOGUANAMIL CLOPONONE CLORINDANOL CLOROFENE CLOXIQUINE CNV-9203 COMPOUND-1929 CP-67015 CREOLIN CRESOL CRESOL-META CRESOL-ORTHO CRESOL-PARA CRIBROSTATIN-2 CROTONIAZIDE CRYPTARGOL CS-61 CS-834 CS-940 CYACETACIDE CYCLO-PHE-PRO CYCLO-PRO-TRP CYCLOMENOL DA-3804 DA-3829 DA-3831 DA-3832 DA-3838 DA-3839 DA-3840 DA-3851 DA-3853 DA-3854 DA-3915 DANOFLOXACIN DAPSONE DEACETOXYOLEPUPUANE-7 DEDITONIUM BROMIDE DEGMIN DEHYDROACETATE DEHYDROPODOPHYLLOTOXIN DEMETHYLFLEROXACIN DEMETHYLOFLOXACIN-N DEOXYFRUCTO-SEROTONIN DEQUALINIUM CHLORIDE DERMACID DESOXYFUR DIATHYMOSULFONE DIBROMOAGELIFERIN DIBROMOHEXAMIDINE DIBROMPROPAMIDINE DIBROMSALAN DICHLORBENZALKONIUM DICHLOROBENZENE-ORTHO DICHLOROBENZYL= ALCOHOL-2,4 DICHLOROPHEN DICHLOROPHENARSINE DICHLOROXYLENOL DICYCLOHEXYLAMINE DIDECYLDIMETHYL= AMMONIUM CHLORIDE DIFLOXACIN DIFURACIL DIHYDROAMBAZONE DIHYDROFLUSTRAMINE-C DIHYDROGENISTEIN DIIODOHYDROXYQUINOLINE DIMETHYLDODECANAMINE DIOXIDINE DIPYRITHIONE DISULFANILAMIDE DITHRANOL DITHYRAL DITOPHAL DIXANTHOGEN DJ-6783 DODECLONIUM BROMIDE DODECYL-BENZENE-= SULFONATE DODECYLGLYCEROL DODECYLPYRIDINIUM DODICIN DOFAMIUM CHLORIDE DR-3862 DRAGMACIDIN-D DRAZIDOX DROSOCIN DROXACIN DS-4524 DU-6668 DU-6858 DUP-105 DUP-721 DV-7751 DV-7751-A DW-116 DWH-146-E E-3846 E-4441 E-4695 E-5065 E-5068 ECTEINASCIDIN-770 ECTERICIDE EKMOLIN ENDOFARM ENOXACIN ENROFLOXACIN EPEREZOLID EPI-OLEANOLATE ETHACRIDINE ETHAMBUTOL ETHIONAMIDE ETHONIUM ETHYLENEDIAMINE-= DIHYDROIODIDE ETHYLHYDROCUPREINE ETHYLPARABEN ETOCARLIDE EUCALYPTOL EUDISTOMIN-U EUGENOL FENAMISAL FERROCENE-A FLEROXACIN FLEROXACIN-N-OXIDE FLUDAZONIUM CHLORIDE FLUMEQUINE FLUORODEOXYCYTIDINE FLUOROSHIKIMATE-6 FLUROFAMIDE FLUSALAN FORMOPED FORMOSULFATHIAZOLE FORMYLSULFISOMIDINE FR-145715 FR-180102 FTIVAZIDE FURACRYLIN FURALAZINE FURALTADONE FURAZOLIDONE FURAZOLIUM CHLORIDE FURAZONAL FURMETHOXADONE FURSALAN FURYLFURAMIDE GALAPHENYLSULFONE GARCINOL GATIFLOXACIN GEMIFLOXACIN GENKWANIN GERMALL-115 GERMALL-II

1098 APPENDIX D GERMEX GLOXAZONE GLUCOSULFAMIDE GLUCOSULFONE GLUTARAL GLYCONIAZIDE GREPAFLOXACIN HALAZONE HALETAZOLE HALOCARBAN HALOPENIUM CHLORIDE HALOPROGIN HALQUINOL HEDAQUINIUM CHLORIDE HELMINTHOSPORIN HEXACHLOROPHENE HEXEDINE HEXETIDINE HEXYLPARABEN HEXYLRESORCINOL HSR-903 HYDRARGAPHEN HYDROGEN-PEROXIDE HYDROQUINONE HYDROXYCINNAM= ALDEHYDE-2+ HYDROXYCRYPTOLEPINE-11 HYDROXYFLUMEQUINE-7 HYDROXYMETRONIDAZOLE HYDROXYPIROMIDATE-BETA HYDROXYQUINOLINE HYDROXYSTILBAMIDINE HYDROXYSULFADIMIDINE-5 HYDROXYSULFA= METHOXAZOLE-5 HYDROXYSULFATR= OXAZOLE-5 HYDROXYTOLUATE ICHTHAMMOL IMBRICATOLATE INDOLEPROPIONATE INDOLICIDIN IODOBISMUTH-SULFAMIDE IODOFORM IODOGLYCOL IODOPHTHALEIN SODIUM IODOPYRON IPSALAZIDE IRIDOMYRMECIN IRLOXACIN ISLANDICIN ISOCONAZOLE ISOMETRONIDAZOLE ISONIAZID ISONIAZID-MESILATE ISOPULEGOL ISOTORALACTONE ITV-8912 K-107 K-120 K-122 K-137 K-138 K-150 K-96 KAPOSTAT KB-5246 KKM-43 KUBATOL LACTATE SODIUM LACTOFERRICIN LARUSAN LAURALKONIUM CHLORIDE LAURICIDIN LAUROGUADINE LAUROLINIUM ACETATE LAVASEPT LEVOFLOXACIN LEVOFURALTADONE LINEZOLID LISSOCLINOTOXIN-A LL-D-49194-ALPHA-1 LL-D49194-ALPHA-1 LOMADEN LOMBAZOLE LOMEFLOXACIN LORASOL-V LY-173013 LY-186826 LY-193239 LY-255262 LYSOVET LYSOVET-PA MACROCYCLON MAFENIDE MAGAININ-1 MAGAININ-2 MAGAININ-2-AMIDE MAGAININ-2-AMIDE-ALA-19 MAGAININ-A MAGAININ-B MAGAININ-G MAGAININ-H MALACHITE-GREEN MALEYLSULFATHIAZOLE MARBOFLOXACIN MBI-27 MBI-28 ME-93 MEDOL MELARSEN MELARSENOXIDE MELARSONYL POTASSIUM MELARSOPROL MENNO-QUAT-AR MENTHOL MEQUIDOX MERALEIN SODIUM MERBROMIN MERCUROBUTOL MESALAZINE METABROMSALAN METAZIDE METHANIAZIDE METHENAMINE METHYL-GREEN METHYLAL METHYLBENZETHONIUM = CHLORIDE METHYLPARABEN METHYLROSANILINIUM = CHLORIDE METHYLTHIONINIUM = CHLORIDE METIOPRIM METIOXATE METRONIDAZOLE METRONIDAZOLE-= PHOSPHATE METRONIDAZOLE-SUCCINATE MF-5137 MF-922 MF-961 MILD-SILVER-PROTEIN MILOXACIN MIRISTALKONIUM MONALAZONE SODIUM MONOFLUOROMETHYL= ORNITHINE-ALPHA MONTIPORATE-A MONTIPORATE-B MORINAMIDE MOXIFLOXACIN MSI-103 MSI-1436 MSI-30 MSI-78-A MSI-94 MSI-98 MY-40-20 MYCAPEROXIDE-A MYCAPEROXIDE-B MYRALACT MYRISTOYLCHOLINE = BROMIDE NALIDIXATE NAPHTHALAN-OIL ND-502 NEOARSPHENAMINE NEW-METHYLENE-BLUE NIBROXANE NICOTHIAZONE NIDROXYZONE NIFURADENE NIFURALDEZONE NIFURALIDE NIFURATEL NIFURATRONE NIFURDAZIL NIFURETHAZONE NIFURFOLINE NIFURIMIDE NIFURIZONE NIFURMAZOLE NIFUROQUINE NIFUROXAZIDE NIFUROXIME NIFURPIPONE NIFURPIRINOL NIFURPRAZINE NIFURQUINAZOL NIFURSTYRENATE SODIUM NIFURTHIAZOLE NIFURTOINOL NIFURVIDINE NIFURZIDE NIHYDRAZONE NITROAKRIDIN-3582 NITROFEN NITROFURAL NITROFURANTOIN NITROFURATHIAZIDE NITROMERSOL NITROSULFATHIAZOLE NITROVIN NITROXOLINE NM-394 NONOXINOL-15 NONOXINOL-30 NONOXINOL-4 NOPRYLSULFAMIDE NORFLOXACIN NORFLOXACIN-SUCCINIL NOXYTIOLIN NSC-87982 NSFQ-104 NSFQ-105 O-129 OBTUSIFOLIN OCTAFONIUM CHLORIDE OCTENIDINE OCTHILINONE OFLOXACIN OFLOXACIN-N-OXIDE OLAQUINDOX OLEANONATE OLSALAZINE ONO-1714 OPC-7251 OPINIAZIDE ORBIFLOXACIN ORCINOL OREGONIN

Derwent Drug File 1099 Thesaurus ORMETOPRIM ORTHOSAN OTIMERATE SODIUM OXIFULVATE OXO-ENOXACIN OXOLINATE OXOPHENARSINE OXYCHLOROSENE PAKOMA PARABEN PAS PAS SODIUM PASINIAZID PAZUFLOXACIN PAZUFLOXACIN MESILATE PD-111103 PD-115311 PD-116169 PD-116427 PD-117558 PD-117596 PD-119421 PD-122642 PD-123982 PD-124816 PD-125354 PD-125639 PD-126889 PD-131112 PD-131501-0 PD-131575 PD-131628 PD-131628-2B PD-135042 PD-135739 PD-137156 PD-138136 PD-138312 PD-138926 PD-139586 PD-140248 PD-143289 PD-158804 PD-160793 PD-161314 PD-164488 PEFLOXACIN PEFLOXACIN-N-OXIDE PELLITORINE PENOCTONIUM BROMIDE PERACETATE PGE-4175997 PGE-9262932 PGE-9509924 PGL-AMIDE PHANQUINONE PHENARSONE-SULFOXYLATE PHENAZOPYRIDINE PHENETHYL-ALCOHOL PHENODODECINIUM PHENOSMOLIN PHENOXETOL PHENYLMERCURIC-ACETATE PHENYLMERCURIC-BORATE PHENYLMERCURIC-NITRATE PHOSPHANILATE PHTHALYLSULFACETAMIDE PHTHALYLSULFAMETHIZOLE PHTHALYLSULFATHIAZOLE PICLOXYDINE PIPEMIDATE PIROMIDATE PIRRALKONIUM BROMIDE PIRTENIDINE PNU-171933 PNU-172576 POLIHEXANIDE POLYCRESOLSULFONATE POLYHEXAMETHYLENE-= BIGUANIDE POLYHYDROXYDINE POLYNOXYLIN POLYQUATERNIUM-1 POTASSIUM-HYPOCHLORITE POTASSIUM-TELLURITE POVIDONE-IODINE PR-39 PROFLAVINE PROPAMIDINE PROPHYL PROPIOLACTONE PROPIONATE SODIUM PROPYLPARABEN PROTIONAMIDE PURPURAMINE-H PYRAZINAMIDE PYRITHIONE PYRITHIONE ZINC PYROGALLOL-TRIACETATE PYRRHOCORICIN QR-2 QR-4 QR-5 QUESTIN QUINDECAMINE QUINDOXIN QUINIFUR QUINIFURIL QUINOXIDINE R-5144 R-6597 R-7000 R-7371 RANALEXIN RECTOSEPT RESIQUIMOD RESORCINOL RHODODENDROL RO-09-1168 RO-46-7864 RO-47-3359 RO-66-0376 RO-66-6976 ROMIFENONE ROSOXACIN ROXARSONE RU-64004 RUBROFUSARIN RUFLOXACIN RWJ-306490 RWJ-3981 RWJ-49815 S-25930 S-25932 S-28463 SALAZODIMETHOXINE SALAZODINE SALAZOPYRIDAZINE SALAZOSULFADIMIDINE SALAZOSULFAMIDE SALAZOSULFAPYRIDINE SALAZOSULFATHIAZOLE SALICYLATE SALICYLATE TROLAMINE SALINAZID SALSALATE SANGUIRITRINE SARAFLOXACIN SB-37 SC-28538 SCEPTRIN SEPAZONIUM CHLORIDE SHIVA-1 SILVER-PROTEIN SILVER-SULFACETAMIDE SILVER-SULFADIAZINE SILVER-SULFATHIAZOLE SILVER-SULFISOMIDINE SITAFLOXACIN SJ-749 SMAP-28 SMAP-29 SODIUM-CARBONATE SODIUM-HYDROXIDE SODIUM-HYPOCHLORITE SOLASULFONE SOLUPRONT SOZOLATE SPARFLOXACIN SQUALAMINE SRC-820 STEARYLSULFAMIDE STEINAZIDE STIBOSAMINE STILBAMIDINE ISETIONATE STREPTONIAZID SUBATHIZONE SUCCINYLSULFATHIAZOLE SUCCISULFONE SULBENTINE SULFABENZ SULFABENZAMIDE SULFABENZOYLAMIDE SULFABROMOMETHAZINE SULFACARBAMIDE SULFACECOLE SULFACETAMIDE SULFACHLORPYRIDAZINE SULFACHRYSOIDINE SULFACITINE SULFACLOMIDE SULFACLORAZOLE SULFACLOZINE SULFADIASULFONE SODIUM SULFADIAZINE SULFADIAZINE SODIUM SULFADICRAMIDE SULFADIMETHOXINE SULFADIMIDINE SULFAETHIDOLE SULFAETHOXYPYRIDAZINE SULFAFURAZOLE SULFAGUANIDINE SULFAGUANOLE SULFALENE SULFALOXATE SULFAMAZONE SULFAMERAZINE SULFAMERAZINE SODIUM SULFAMETHIZOLE SULFAMETHOXAZOLE SULFAMETHOXYPYRIDAZINE SULFAMETOMIDINE SULFAMETOXYDIAZINE SULFAMIDOCHRYSOIDINE SULFAMONOMETHOXINE SULFAMOXOLE SULFANILAMIDE SULFANILATE SULFANILATE ZINC SULFANITRAN SULFANTHROL SULFAPERIN SULFAPHENAZOLE SULFAPROXYLINE SULFAPYRAZINE SULFAPYRAZOLE SULFAPYRIDINE SULFAQUINOXALINE SULFARSPHENAMINE SULFASOMIZOLE SULFASUCCINAMIDE

1100 APPENDIX D SULFASYMAZINE SULFATHIAZOLE SULFATOLAMIDE SULFATRIAZINE SULFATROXAZOLE SULFATROZOLE SULFISOMIDINE SULFISOZOLE SULFONIAZIDE SULFORMETOXINE SULFOTIN SULPHIMIDAZOLE SYMCLOSENE T-283 T-3262A T-3262B T-3811-ME TACHYPLESIN-I TACHYPLESIN-II TALMETOPRIM TAURINAMIDE TAUROLIDINE TAURULTAM TEMAFLOXACIN TEMODOX TERIZIDONE TETRACHLORODECAOXIDE TETRADECYLTRIMETHYL= AMMONIUM BROMIDE TETRADONIUM BROMIDE TETROXOPRIM THALIDOMIDE THENOATE THIACETARSAMIDE SODIUM THIAMBUTOSINE THIAZOSULFONE THIOACETAZONE THIOCARBANIDIN THIOFURADENE THIOMERSAL THIONIUM THIRAM THYMOL TIBEZONIUM IODIDE TIBROFAN TICLATONE TIGERININ-1 TIMERFONATE SODIUM TIOCARLIDE TIODONIUM CHLORIDE TIOSALAN TIOXACIN TISOCARBAMIDE TN-121 TOLIODIUM CHLORIDE TOLOCONIUM-METILSULFATE TONZONIUM BROMIDE TORALACTONE TOROSACHRYSONE TOSUFLOXACIN TOSYLCHLORAMIDE SODIUM TRACHEAL-ANTIMICROBIAL-= PEPTIDE TRIBROMSALAN TRICHLOROPHENOL TRICLOBISONIUM CHLORIDE TRICLOCARBAN TRICLOSAN TRIETHYLENE-GLYCOL TRIFLUOROMETHYLHOMO= CYSTEINE TRIFLUOROMETHYLTHIO= RIBOSE-5 TRIMETHOPRIM TRM-115 TROCLOSENE TROCLOSENE POTASSIUM TROVAFLOXACIN TRYPAN-BLUE TRYPARSAMIDE UREA-HYDROGEN-PEROXIDE VANYLDISULFAMIDE VARIABILIN VERAZIDE VUF-8501 VUF-8514 VUF-8842 WAKAYIN WIN-57273 WIN-57294 XENYSALATE XIBORNOL Y-26611 Y-688 YOSHIXOL ANTISEROTONINS 1045-U-85 1192-U-90 ACC-7513 AD-5423 AD-8112 ADATANSERIN AGN-2979 AHR-16303B ALA-251 ALOSETRON ALTANSERIN AMESERGIDE AMINDOCATE AMINOKETANSERIN-7 AS-5370 AS-5820 ASIMILOBINE AT-1015 AWD-52-39 AZIDOKETANSERIN-7 BALAPERIDONE BEMESETRON BENANSERINE BIMU-0001 BIMU-1 BIMU-8 BMY-7378 BOL-148 BRL-15572 BRL-46470 BRL-46470A BROMERGURIDE BROMOERGOSINE BUTANSERIN BW-204-C67 BW-501 BW-501-C67 CANADALINE CGS-18102-A CILANSETRON CIMEPANOL CINANSERIN CONFUSAMELINE CP-88059 CV-5197 CYPROHEPTADINE DANITRACEN DAU-6215 DAU-6285 DEPTROPINE DIHYDROERGOCORNINE DIHYDROERGOCRISTINE DIHYDROERGOCRYPTINE DIHYDROERGOCRYPTINE-= ALPHA DIHYDROERGOCRYPTINE-= BETA DIHYDROERGOSINE DIHYDROERGOSININE DIHYDROERGOTAMINE DIHYDROERGOTOXINE DIMETOTIAZINE DOLASETRON DOMESTINE DU-125530 DV-7028 E-3620 EGIS-7056 EP-19-088 ERGOCORNINE ERGOCRISTINE ERGOCRYPTINE-ALPHA ERGOCRYPTINE-BETA ERGOSINE ERGOSININE ERGOTAMINE ESCIN-I-B FCC-13 FCC-5 FCE-22716 FENCLONINE FENCLONINE-ETHYL-ESTER FENCLONINE-METHYL-ESTER FG-5865 FG-5893 FG-5974 FK-1052 FLUFYLLINE FLUMEZAPINE FRAN-12 GK-128 GLEMANSERIN GMC-5032 GMC-5034 GR-113808 GR-125487 GR-125743 GR-127935 GR-65630 GR-65630A GR-C-507-75 GRANISETRON GYKI-32084 HW-13 HYDROXINDASATE HYDROXINDASOL HYDROXYAMESERGIDE-4 HYDROXYGRANISETRON-7 HYDROXYINDALPINE-5 ICI-169369 ICI-170809 ICI-205930 ILOPERIDONE INDOCATE IODOAMPHETAMINE-PARA IPRAZOCHROME IRINDALONE ISOLYSERGATE ITASETRON K-191 K-277 K-4300 KB-6933 KERAMADINE KETANSERIN KETANSERINOL KF-18259 KF-20170 KOKUSAGININE KW-4099 L-646462 L-683877 LE-300 LEK-8804 LEK-8829

Derwent Drug File 1101 Thesaurus LERISETRON LEVEMOPAMIL LEVODOPA-METHYL-ESTER LINTOPRIDE LISURIDE LU-21-099 LU-29024 LU-49938 LUROSETRON LY-108742 LY-165163 LY-193525 LY-197541 LY-206130 LY-211000 LY-214138 LY-215840 LY-225297 LY-254239 LY-258458 LY-278584 LY-278989 LY-333068 LY-353433 LY-53857 LY-86057 LYSERGAMIDE LYSERGATE M-840 MDL-100907 MDL-102382 MDL-26508 MDL-28133A MDL-72222EF MDL-72699 MDL-73147 MDL-73492 MDL-74156 MDL-74156EF MERREMOSIDE-B MERREMOSIDE-D METERGOLINE METERGOTAMINE METHOXYCHLOROETHYL= PROPYLAMINOTETRALIN-8 METHOXYCYPRO= HEPTADINE-3 METHYSERGIDE METRENPERONE MIANSERIN MK-711 MKC-242 ML-1035 ML-10375 MM-218 MP-3022 MS-377 N-3256 N-3389 NAN-190 NEXOPAMIL NK-122 NNC-22-0031 NRA-0045 NRA-0562 NSH-134 OCAPERIDONE ONDANSETRON ORG-2305 ORG-6997 ORG-GC-94 PALONOSETRON PANCOPRIDE PELANSERIN PERBUFYLLINE PIPETHIADENE PIPOXIZINE PIRENPERONE PIZOTIFEN PROPISERGIDE PTR-17402 QF-0307-B QF-0313-B QF-2004-B QF-503 QF-603 QF-607 R-102444 R-56413 RAMOSETRON RG-12718 RG-12915 RISPERIDONE RITANSERIN RK-153 RO-15-8081 RO-25-1553 RP-62203 RS-100235 RS-102221 RS-23597-190 RS-25259-197 RS-39604 RS-56532 RS-56812-197 RS-57639 RS-66331 S-11978 S-14063 S-14280 S-14489 S-14671 S-15535 S-15931 S-18327 S-21357 SARPROGRELATE SB-200646 SB-200646-A SB-203186 SB-204070 SB-204070-A SB-204741 SB-206553 SB-207266 SB-207266-A SB-207710 SB-216641 SB-219085 SB-220272 SB-224289 SB-228357 SB-258585 SB-258719 SB-271046 SB-357134 SC-49518 SC-52246 SC-53117 SC-53606 SDZ-205-557 SDZ-206-830 SDZ-216-525 SDZ-ICM-567 SDZ-ICT-322 SDZ-SER-082 SEGANSERIN SEQUIFENADINE SERGOLEXOLE SETOPERONE SGB-1534 SKF-83566 SL-65-0472 SM-13496 SN-307 SQ-11276 SR-46349B ST-1460 SUN-C-5174 THEANINE THIAZINAMIUM-CHLORIDE THIAZINAMIUM-SULFOXIDE TROPANSERIN TROPISETRON TROPOXIN TYPINDOLE UH-301 VA-21-B7 VALOFANE W-3795 W-4010 WAY-100135 WAY-100289 WAY-100579 WAY-100635 WB-4371 XYLAMIDINE TOSILATE Y-25130 Y-39241 YM-103 YM-108 YM-114 YM-35992 ZALOSPIRONE ZATOSETRON ZK-33839 ANTISICKLINGS BUTYLUREA BW-12C BW-A589C CEPHARANTHINE DIMETHYLADIPIMIDATE LYSYLPHENYLALANINE NS-1652 ZINC-ETHYLMALTOL ANTITHYROIDS AMINOTHIAZOLE BENZYLTHIOURACIL CARBIMAZOLE DIBROMOTYROSINE DIOBUTIL EMD-21388 EMD-49209 ETHYLENETHIOUREA GOITRIN IODOTHIOURACIL MERCAPTOTHIAZOLINE METHYLTHIOURACIL NPS-R-568 PROPYLTHIOURACIL THIAMAZOLE THIOBARBITAL THIOPHENOBARBITAL THIOURACIL TRICYANOAMINOPROPENE ANTITOXIN CENTOXIN ANTITUSSIVES 443-C ACEBROPHYLLINE ACEPROMETAZINE ACETYLCYSTEINE ADAMEXINE ALLOCLAMIDE AMBROXOL AMBROXOL = THEOPHYLLINATE AMICIBONE AMIFOSTINE

1102 APPENDIX D AMOXYDRAMINE CAMSILATE ANETHOLE APOMORPHINE AZEPEXOLE BENCISTEINE BENPROPERINE BENZOBUTAMINE BENZONATATE BEZITRAMIDE BIBENZONIUM BROMIDE BROMHEXINE BROMOPYRILENE BROVANEXINE BUCKTHORN-OIL BUTAMIRATE BUTETAMATE BUTOPIPRINE BUTORPHANOL CARAMIPHEN CARBOCISTEINE CARBOCISTEINE-LYSINE-SALT CARPERIDINE CEPHAELINE CG-37059 CHINOIN-170 CLOBUTINOL CLOFEDANOL CLOPERASTINE CLOROQUALONE CODEINE CODOXIME CYCLEXANONE DEMBREXINE DEXTROMETHORPHAN DEXTRORPHAN DEXTRORPHAN-= GLUCURONIDE DIBUNATE SODIUM DIBUNATE-ETHYL DIHYDROCODEINE DIHYPRYLONE DIMEMORFAN DIMETHOXANATE DIMETHYLGLYCYLPHENO= THIAZINE DIMETHYLGLYCYLPHENO= THIAZINE DIPHENHYDRAMINE-= METHYLBROMIDE DOMIODOL DROPROPIZINE DROTEBANOL DROXYPROPINE EMETINE EPRAZINONE ETAMINILE ETHYLMORPHINE ETOFURADINE EUCALYPTOL F-1459 FALIMINT FEDRILATE FLUALAMIDE FOMINOBEN GLAUCINE GLYCYRAM GLYCYRRHIZATE GUACETISAL GUAIAPATE GUAIETOLIN GUAIFENESIN GUAIMESAL HOMARYLAMINE HYDROCODONE IQUINDAMINE ISOAMINILE KHL-8425 LEDOL LETOSTEIN LEVODROPROPIZINE LEVOPROPOXYPHENE LIMONENE MECYSTEINE MEDAZOMIDE MENGLYTATE MEPROTIXOL MEQUITAZINE MESNA MITRAGYNINE MOFOXIME MOGUISTEINE MORCLOFONE MOXAZOCINE MYFADOL NAPHTHONONE NARCYL NICOCODINE NICODICODINE NORMETHADONE NOSCAPINE OMONASTEINE OXABREXINE OXELADIN OXOLAMINE OXOMEMAZINE PEMERID PENTOXYVERINE PHOLCODINE PICLOBETOL PICOPERINE PIPAZETATE PRENISTEINE PRENOXDIAZINE PROFADOL PROMOLATE PROPINETIDINE PROXAZOLE PROXORPHAN RACEMETHORPHAN REGENASOL SB-227122 SFERICASE SHOGAOL-6 SOBREROL SULFOGAIACOL SUXEMERID TAZIPRINONE TEREBINTH-OIL TERPIN-HYDRATE THALICMINE THEBACON TIOPRONIN TIPEPIDINE TRK-851 UBISINDINE VADOCAINE VIMINOL XYLOXEMINE ZIPEPROL ANTIULCERS ACEROXATIDINE AD-2646 AG-041-R AG-1777 AG-1789 AG-1812 AG-2000 AH-22216 AI-77-B AI-77-C AI-77-D AI-77-F AI-77-G ALCLOXA ALDIOXA ALE-36 ALGELDRATE ALGINOSIDE ALMADRATE-SULFATE ALMAGATE ALMASILATE ALUMINUM-HYDROXIDE ALUMINUM-SILICATE ALUSULF AMINOINDAZOLE-6 AMYLOSULFATE SODIUM ANTIGASTRIN APC-2059 ATTAPULGITE AWD-26-06 AWD-26-39 AY-28200 AY-29315 AY-31574 B-813-19 B-831-56 BAXITOZINE BENCYCLANE BENEXATE BENTIPIMINE BENZOHYDROXAMATE BENZOTRIPT BEPERIDIUM IODIDE BL-6341A BMY-25271 BMY-25368 BMY-26517-31 BTM-1041 BTM-1042 BTM-1086 BUPLEURAN-211C BURIMAMIDE BY-841 CARBENOXOLONE CASSIOL CASSIOSIDE CEREBROSIDE-B1B CETRAXATE CHLORBENZOXAMINE CHLOROCAMPHAMIDE CICLOXOLONE DISODIUM CIMETIDINE CINOXOLONE CINPRAZOLE CL-1700 CLIDINIUM BROMIDE CP-331 CRC-1970 CROTONIN D-51-9927 DBM-819 DE-NOL DECITROPINE DEHYDROCORYDALINE DEHYDROCROTONIN-TRANS DEPTROPINE-= METHOBROMIDE DICLOGUAMINE DICYCLOVERINE DIHYDROXYALUMINUM-= AMINOACETATE DONETIDINE DOSMALFATE DQ-2511 DROPEMPINE DS-4574 E-0711 EBROTIDINE ECABET SODIUM ELUCAINE ENOXOLONE

Derwent Drug File 1103 Thesaurus EPIPACHYSAMINE-A ESAPRAZOLE ETHADEN ETINTIDINE FAMOTIDINE FPL-52694 FR-145715 FRG-8813 FTAXILIDE FURANOGERMENONE GARCINOL GASTROZOL GEFARNATE GINGESULFONATE-6 GLUCALDRATE POTASSIUM GLUCALOX GLYCYRRHIZA-= DEGLYCYRRHINIZED GUALENATE SODIUM H-200-62 H-200-66 HEXAPRAZOL HEXOCYCLIUM = METILSULFATE HF-2035 HYDROTALCITE IBI-P-05006 ICI-162846 IDB-1027 IFETROBAN IGN-2098 IK-82029 INTEST.TREFOIL-FACTOR-RAT IO-21 IRSOGLADINE ISOPROPOXYGERMATRANE IT-066 IY-81149 K-1905 KB-5492 KELAMPAYOSIDE-A KERATINOCYTE-GROWTH-= FACTOR-2 KT-1-109 KU-1257 KW-5805 L-643411 LAMTIDINE LANSOPRAZOLE LEMINOPRAZOLE LEVOMENOL LOXTIDINE MAALOXAN MAGALDRATE MAGNESIUM-ALUMINUM-= HYDROXIDE MAGNESIUM-ALUMINUM-= SILICATE MAGNESIUM-CARBONATE MAGNESIUM-HYDROXIDE MAGNESIUM-OXIDE MASTIC MATRINE MAZ-525 MCI-727 MCN-A-1293 MECIADANOL METHANTHELINIUM = BROMIDE METHYLBENACTYZIUM = BROMIDE METIAMIDE METOQUIZINE MEZOLIDON MIFENTIDINE MUTAFLOR NC-1300 NC-1300-B NC-1300-SULFIDE NIK-228 NILPRAZOLE NITECAPONE NIZATIDINE NOLINIUM BROMIDE NORBERGENIN NORBURIMAMIDE NUVENZEPINE OF-743 OF-900 OF-900 OLEANOLATE-ACETATE OLEANOLATE-METHYL-ESTER OMEPRAZOLE OXOPROSTOL OXYFERRISCORBONE OXYMATRINE PANTOPRAZOLE PEPSTATIN PGJ2-DEOXY-15-DELTA-12,14 PGV-40350 PHENTHIMENTONIUM PICARTAMIDE PIFARNINE PIRENZEPINE PLAUNOTOL POLAPREZINC POLDINE-METILSULFATE POLIGEENAN POLIGNATE POLYETADENE PROGLUMIDE PROPANTHELINE PROPANTHELINE BROMIDE PYLORICIDIN-B QUIDITENE QUISULTAZINE RABEPRAZOLE RAMIXOTIDINE RANITIDINE RANITIDINE-BISMUTH-= CITRATE REBAMIPIDE RGH-5981 RHODODENDRIN RO-18-5362 RO-18-5364 ROSAPROSTOL ROSAVIN ROTRAXATE ROXATIDINE ROXOLONIUM-METILSULFATE RS-2039 RS-86505-007 RS-86505-008 RS-86812-007 S-0509 S-1924 S-4216 SAVIPRAZOLE SCH-28080 SCH-32651 SKF-93479 SL-81-0433 SMECTITE SODIUM-ALUMINOSILICATE SOFALCONE SOLCOSERYL SPI-447 SPIZOFURONE ST-341 SU-840 SUCRALFATE SUCRALOX SUCROSE-OCTASULFATE SUFOTIDINE SULGLICOTIDE T-330 T-593 TAMRABHASMA TELENZEPINE TEPRENONE THEASAPONIN-E1 TIMOPRAZOLE TIOPROPAMINE TIOTIDINE TIQUINAMIDE TOCORETINATE TOLIMIDONE TOQUIZINE TRILETIDE TRITIOZINE TRM-115 TROMETAMOL TROXIPIDE TRY-200 TU-199 TY-11345 UH-AH-37 URTIPHYLLIN VASCULAR-ENDOTHELIAL-= GROWTH-FACTOR-HUM VASCULAR-PERMEABILITY-= FACTOR WHR-1370A WHR-2568 WITHAFASTUOSIN-E WY-26769 WY-45662 WY-45727 YJA-20379-1 YJA-20379-8 YM-14471 Z-300 ZALTIDINE ZINC-ACEXAMATE ZINC-GLUTAMATE ZOLIMIDINE ANTIVITAMINS ACETYLPYRIDINE-3 AGN-193109 AMINONICOTINAMIDE AMINOTHIADIAZOLE AMINOTHIAMINE DEOXYPYRIDOXINE GALACTOFLAVIN MSD-235-S2 OXYTHIAMINE PIRITREXIM PT-441 PYRITHIAMINE RO-41-5253 STRAVIDIN STRAVIDIN-S2 STRAVIDIN-S3 TEI-9647 ZK-159222 ANXIETY-DISORDER ACUTE-STRESS-DISORDER AGORAPHOBIA ANXIETY BODY-DYSMORPHIC-= DISORDER cardiac-neurosis CLAUSTROPHOBIA da-costa-syndrome dysmorphophobia GENERALIZED-ANXIETY-= DISORDER HYPOCHONDRIA OBSESSIVE-COMPULSIVE-= DISORDER

1104 APPENDIX D PANIC-DISORDER PHOBIA POSTTRAUMATIC-STRESS-= DISORDER roemheld-syndrome SEPARATION-ANXIETY-= DISORDER SOCIAL-PHOBIA APOPTOSIS-INDUCERS A-151011 A-204197 ACETYLSPHINGOSINE-N ACYCLORETINOATE ADAPHOSTIN ALSTERPAULLONE AN-152 AN-207 AN-238 ANGINEX ANTITHROMBIN-LATENT AP-1903 APICULAREN-A APOLIZUMAB APOPTOLIDIN AVICIN-D AVICIN-G AW-464 B-201 B-327 B-429 BAL-9611 BAY-11-7085 BB-3103 BIBF-1000 BIM-46174 BMS-184476 BMS-214662 BMS-239091 BMS-247550 BMS-250749 BMS-250904 BN-80927 BOHEMINE BONE-MORPHOGENETIC-= PROTEIN-2 BROSTALLICIN BT-99-25 C-75 CANTHARIDATE CC-5013 CEP-5214 CEP-701 CETUXIMAB CP-248 CP-461 CV-787 CZ-48 DDE-131 DEOXYMETHYL= SPERGUALIN DIFLOMOTECAN EMD-121974 EMD-66203 EPI-OLEANOLATE ETHYLESTRONE-3-O-= SULFAMATE-2 EXISULIND FUB-407 GEMTUZUMAB OZOGAMICIN GRAPE-SEED-EXTRACT GW-8510 HA-14-1 HYDROXYVITAMIN-D5,1-= ALPHA IBANDRONATE IDEC-152 ILX-23-7553 IMATINIB INCADRONATE INDANOCINE JV-1-36 JWH-133 KF-25706 KF-58333 KW-2170 L-805645 LFM-A-13 METHYLSELENINATE MMI-166 MS-27-275 MZ-5-156 NCQ-344 NITROIBUPROFEN NSC-330507 ONO-8711 ORI-1313 ORI-1327 OXI-4503 PARADOL-6 PD-0183085 PD-180970 PD-98059 PEX PGJ2-DEOXY-15-DELTA-12,14 PKI-166 POLY-OXYPEPTIN PROLACTIN-HUMAN-G129R PROTEASOME-INHIBITOR-1 PXD-101 PYROXAMIDE RO-31-7453 S-23906-1 SALVICINE SB-T-1213 SB-T-12843 SC-58560 SCH-66336 SN-50 SPIKET-P1 STREPTOCOCCAL-= ANTITUMOR-= GLYCOPROTEIN SU-6668 SU-9516 SUBEROYLANILIDE-= HYDROXAMATE T-138067 T-900607 TACHPYRIDINE TIPIFARNIB TNF-RELATED-APOPTOSIS-= INDUCING-LIGAND TOSITUMOMAB TP-151 TUMSTATIN TX-1856 TYLOPHORINIDINE UROGUANYLIN VATDIOSPYROIDOL VINFLUNINE WHI-P-131 WHI-P-154 Y-27632 ZOLEDRONATE APOPTOSIS-INHIBITORS NN-2211 APPARATUS AEROCHAMBER APPLICATOR ART.PANCREAS ATOMIZER AUTOCLAVE AUTOMATIC-ANALYZER BIOSTATOR CALCULATOR CANNULA CATHETER CENTRIFUGE COMPUTER CONTACT-LENS DART DEFIBRILLATOR HEART-LUNG-MACHINE JET-INJECTOR METER MILL MOLD NEBUHALER NEBULIZER NEEDLE PACEMAKER PEAR-SPACER PHOTODETECTOR PROSTHESIS RESPIRATOR SPACER SPINHALER SYRINGE ULTRACENTRIFUGE VAPORIZER ARBOVIRUS AKABANE-DISEASE-VIRUS BORDER-DISEASE-VIRUS BUNYAMWERA-VIRUS BUSSUQUARA-VIRUS CALIFORNIA-VIRUS CALOVO-VIRUS CHIKUNGUNYA-VIRUS CONGO-VIRUS DENGUE-VIRUS EE-VIRUS ENCEPHALITIS-VIRUS GETAH-VIRUS JAPANESE-ENCEPHALITIS-= VIRUS LANGAT-VIRUS LOUPING-ILL-VIRUS MUCOSAL-DISEASE-VIRUS NAIROBI-SHEEP-DISEASE-= VIRUS POWASSAN-VIRUS PRRS-VIRUS PUNTA-TORO-VIRUS RIFT-VALLEY-FEVER-VIRUS SANDFLY-FEVER-VIRUS SEMLIKI-FOREST-VIRUS SINDBIS-VIRUS SNOWSHOE-HARE-VIRUS SPONDWENI-VIRUS ST.LOUIS-ENCEPHALITIS-= VIRUS TAHYNA-VIRUS WESSELSBRON-DISEASE-= VIRUS WEST-NILE-VIRUS YELLOW-FEVER-VIRUS ARENAVIRUS JUNIN-VIRUS LASSA-FEVER-VIRUS LYMPHOCYTIC-= CHORIOMENINGITIS-VIRUS MACHUPO-VIRUS PICHINDE-VIRUS TACARIBE-VIRUS AROMATASE-INHIBITORS AMINOGLUTETHIMIDE ANASTROZOLE CGP-47645 CGS-18320B EXEMESTANE

Derwent Drug File 1105 Thesaurus FADROZOLE FINROZOLE FORMESTANE FR-901537 HB-66 HYDROXYCHALCONE-4+ MINAMESTANE MPV-2213-AD MR-20492 NECTANDRIN-B R-76713 R-83842 SAE9 SEF-19 TAN-931 TESTOLACTONE VOROZOLE YM-31553 YM-511 ZK-138723 ARRHYTHMIA A.V.BLOCK ADAMS-STOKES-DISEASE ASYSTOLE atrial-fibrillation bouveret-syndrome BRADYCARDIA CARDIOAUDITORY-= SYNDROME ECTOPY EXTRASYSTOLE FIBRILLATION HEART-ARREST HEART-BLOCK LONG-QT-SYNDROME LOWN-GANONG-LEVINE-= SYNDROME PALPITATION PARASYSTOLE paroxysmal-tachycardia paroxysmal-ventricular-= tachycardia ROMANO-WARD-SYNDROME SICK-SINUS-SYNDROME SINOATRIAL-BLOCK TACHYCARDIA torsades-de-point ventricular-fibrillation WOLFF-PARKINSON-WHITE-= SYNDROME ART.PANCREAS BIOSTATOR ARTERIOSCLEROSIS ATHEROSCLEROSIS ARTERY AORTA ARTHRITIS FELTY-SYNDROME LYME-ARTHRITIS ARTHROPOD ACARAPIS ACARUS AEDES ANOPHELES ARGULUS ARTEMIA BATTUS BEE BOMBYX BOVICOLA CALLIPHORA CERATOPHYLLUS CHELOPISTES CHORIOPTES CNEMIDOCOPTES COCKROACH CTENOCEPHALIDES CULEX CYTODITES DEMODEX DERMACENTOR DERMANYSSUS DERMATOBIA DERMATOPHAGOIDES DROSOPHILA ECHIDNOPHAGA EPICAUTA EPILACHNA EUPROCTIS GASTEROPHILUS GLOSSINA GONIOCOTES GREEN-BOTTLE-FLY HAEMATOPINUS HAEMATOPOTA HELIOTHIS house-fly IXODES KERMES LERNAEA LIMULUS LINOGNATHUS LIPEURUS LOCUST LOXOSCELES LUCILIA lynxacarus-v MANSONIA MELOPHAGUS MENACANTHUS MONOPON MORELLIA MOSQUITO MUSCA musca-domestica MYOCOPTES MYRIAPODA NEOSCHOENGASTIA ONCOPELTUS OPHIONYSSUS ORNITHODORUS PANSTRONGYLUS PECTINOPYGUS PEDICULUS PERIPLANETA PHLEBOTOMUS PHTHIRUS PLUTELLA PNEUMONYSSUS POLYPLAX POPILLIA POROCEPHALUS PSOROPTES PULEX RHIPICEPHALUS RHODNIUS SARCOPTES SIMULIUM SOLENOPOTES SPILOPSYLLUS SPLENOPOTES TABANUS TETRANYCHUS TRIATOMA TRICHODECTES TROMBICULA TUNGA TYROGLYPHUS WASP XENOPSYLLA ASCOMYCOTINA SACCHAROMYCESCEREVISIAE ASTROCYTOMA 1321N1-CELL ATAXIA FRIEDREICH-ATAXIA ATTRACTANTS BOMBYKOL DICHLOROPHENOL-2,6 MUSCALURE PHENYLACETALDEHYDE AUTOANTIBODY ANTINUCLEAR-FACTOR LATS AUTOIMMUNE ANTINUCLEAR-FACTOR AUTOANTIBODY AUTOANTIGEN LATS AUTOIMMUNE-DISEASE ANTIPHOSPHOLIPID-= SYNDROME COLD-AGGLUTININ-DISEASE hashimoto-thyroiditis LUPUS-ERYTH. MYASTHENIA-GRAVIS SJOEGREN-SYNDROME sle systemic-lupus-eryth. AUXILIARY-INGREDIENT BINDER COATING DESICCANT DISINTEGRANT FILLER HUMECTANT B-CELL RPMI8422-CELL BACT. ACETOBACTER ACHOLEPLASMA ACHROMOBACTER ACIDAMINOCOCCUS ACINETOBACTER ACTINOBAC. ACTINOMADURA ACTINOMYCES ACTINOPLANES AEROBACTER AEROCOCCUS AEROMONAS AGROBACT. ALCALIGENES ALTEROMONAS AMPULLARIELLA ANAEROVIBRIO ARACHNIA ARTHROBACTER AZOTOBACTER BAC. BACTEROIDES BARTONELLA BIFIDOBACT. BORDETELLA BRANHAMELLA BREVIBACT. BRUC. BURKHOLDERIA BUTYRIVIBRIO CALYMMATOBACT. CAMPYLOBACTER

1106 APPENDIX D CAPNOCYTOPHAGA CARDIOBACT. CAULOBACTER CEDECEA CHROMOBACT. CITROBACTER CLOSTR. COMAMONAS CORYNEBACT. CYTOPHAGA DERMATOPHILUS DICHELOBACTER E.COLI EDWARDSIELLA EMPEDOBACTER ENTEROBACTER ENTEROCOCCUS ERWINIA ERYSIPELOTHRIX ESCHERICHIA EUBACT. FLAVOBACT. FLEXIBACTER FRANCISELLA FUSOBACT. GAFFKYA GARDNERELLA GEMELLA GLUCONOBACTER GRAM-NEG. GRAM-POS. HAEMOPHILUS HAFNIA HALOBACT. HELICOBACTER HISTOPHILUS KINGELLA KLEBS. LACTOBAC. LEGIONELLA LEPTOTRICHIA LEUC. LISTERIA LYSOBACTER MEGASPHAERA meningococcus MICROCOCCUS MICROMONOSPORA MOBILUNCUS MORAXELLA MORGANELLA MYCOBACT. MYCOPLASMA MYXOCOCCUS NEISSERIA neisseria-meningitidis NOCARDIA PAENIBAC. PAENIBACT. PARACOCCUS PASTEURELLA PEPTOCOCCUS PEPTOSTREPT. PHOTOBACT. PLESIOMONAS PROPIONIBACT. PROTEUS PROVIDENCIA PS. RAMIBACT. RENIBACT. RHODOCOCCUS RHODOPS. RHODOSPIRILLUM RUMINOBACTER RUMINOCOCCUS SALM. SAPROSPIRA SARCINA SELENOMONAS SERRATIA SHIGELLA SPHAEROTILUS SPIROPLASMA STAPH. STREPT. STREPTOBAC. STREPTOMYCES STREPTOSPORANGIUM STREPTOVERTICILLIUM SUCCINIVIBRIO SULFOLOBUS TAYLORELLA THERMOACTINOMYCES THERMOMONOSPORA THIOBAC. THIOBACT. UREAPLASMA VEILLONELLA VIBRIO WOLINELLA XANTHOMONAS YERSINIA ZOOGLOEA BENZODIAZEPINE-AGONISTS 340125 450247 450304 450789 450790 ADINAZOLAM ALPRAZOLAM ARFENDAZAM AWD-131-138 BAU-426 BROMAZEPAM CAMAZEPAM CARBURAZEPAM CB-34 CGS-8216 CHLORDIAZEPOXIDE CINOLAZEPAM CLAZOLAM CLIMAZOLAM CLOBAZAM CLONAZEPAM CLORAZEPATE CLOXAZOLAM CLOZAPINE CYPRAZEPAM DAA-1097 DAA-1106 DEALKYLFLURAZEPAM DELORAZEPAM DEMETHYLCLOBAZAM DEMETHYLFLUDIAZEPAM DEMOXEPAM DIAZEPAM DIHYDROFENAZEPAM DOXEFAZEPAM DTZ-323 ELFAZEPAM ESTAZOLAM FENAZEPAM FG-8205 FLETAZEPAM FLUDIAZEPAM FLUNITRAZEPAM FLURAZEPAM FLUTAZOLAM FLUTOPRAZEPAM FOSAZEPAM GIRISOPAM GYKI-52466 GYKI-53405 GYKI-53655 GYKI-53655 HALAZEPAM HALOXAZOLAM HYDROXYALPRAZOLAMALPHA HYDROXYCAMAZEPAM HYDROXYFENAZEPAM-3 ICLAZEPAM IRAZEPINE ISOCURCUMENOL KC-3756 KETAZOLAM LORAZEPAM LORMETAZEPAM MECLONAZEPAM MEDAZEPAM MENITRAZEPAM METACLAZEPAM MEXAZOLAM MIDAZOLAM MOTREZEPAM NERISOPAM NIMETAZEPAM NITRAZEPAM NITRAZEPATE NITRAZEPATE POTASSIUM NNC-13-8119 NNC-13-8199 NNC-13-8241 NORDAZEPAM NORTETRAZEPAM OXAZEPAM OXAZOLAM OXOQUAZEPAM-2 PINAZEPAM PIVOXAZEPAM PRAZEPAM PROFLAZEPAM QUAZEPAM RO-11-6893 RO-11-6896 RO-17-1812 RO-19-0528 RO-21-6347 RO-21-8384 RO-22-8349 RO-23-0364 RO-48-6791 RO-48-8684 RO-5-3590 RO-5-4864 RO-5-5115 RO-5-5807 RO-5-6669 RO-5-6945 RO-5-6993 RO-7-2750 RP-59037 RP-60503 SAS-646 SC-32855 SULAZEPAM SX-3228 TEMAZEPAM TETRAZEPAM TIMELOTEM TOFISOPAM TRIAZOLAM TRIFLUBAZAM TUCLAZEPAM U-43465F ULDAZEPAM XENOVULENE-A XR-7009 ZG-63

Derwent Drug File 1107 Thesaurus BENZODIAZEPINEANTAGONISTS AHR-11797 BRETAZENIL CGS-8216 CGS-9895 EMD-41717 FG-7098 FG-7106 FG-7142 FLUMAZENIL GYKI-53784 IMIDAZENIL IOMAZENIL PANADIPLON PK-11195 PK-14067 PK-14068 PK-14105 RO-14-7437 RO-15-3505 RO-15-3890 RO-17-1812 RO-19-4603 RO-19-8022 RO-21-7254 RO-21-8303 RO-23-0364 RO-41-7812 RO-42-8773 RO-5-3663 RU-33368 RU-34347 RU-40410 SR-25776 U-90042 U-97775 ZK-132553 ZK-93426 BETA-GLUCOSIDASEINHIBITORS CASTANOSPERMINE BETA-LACTAMASE-INHIBITORS BROBACTAM BROMOPENICILLANATE-6-= BETA CLAVULANATE MC-02479 PIVSULBACTAM R-95867 SB-214751 SULBACTAM SYN-2190 TAZOBACTAM BEVERAGE BEER COCOA COFFEE FRUIT-JUICE JUICE TEA BILE-DUCT sphincter-of-oddi BILIARY-TRACT-DISEASE biliary-calculi biliary-colic cholangiolitic-hepatitis CHOLANGITIS CHOLECYSTALGIA CHOLECYSTITIS CHOLEDOCHOLITHIASIS CHOLELITHIASIS CHOLESTASIS cholestatic-hepatitis cholestatic-icterus COURVOISIER-TERRIER-= SYNDROME crigler-najjar-disease familial-nonhemolytic-icterus GILBERT-SYNDROME hanot-macmahon-= tannhauser-syndrome HEPATOCHOLANGITIS HEPATOLITHIASIS HYDROCHOLECYSTITIS HYPERBILIRUBINEMIA ICTERUS idiopathic-icterus leptospiral-icterus weil-disease xanthomatous-biliary-cirrhosis BILOBA LI-1370 BINDING-PROTEIN PENICILLIN-BINDING-PROTEIN BIOAVAILABILITY BIOEQUIVALENCE BIOFLAVONOIDS ACACETIN AMENTOFLAVONE AMENTOFLAVONE-= HEXAACETATE BILOBETIN CIANIDANOL DIFRAREL DIHYDROFISETIN DIHYDROQUERCETIN DIOSMIN ENDOTELON ESCULIN ETHOXAZORUTOSIDE FLAVODATE GINKGETIN GOSSYPETIN GOSSYPIN GUAIJAVERIN HESPERIDIN HESPERIDIN-METHYL= CHALCONE ISALPININ ISOCRYPTOMERIN ISOQUERCITRIN ISORHAMNETIN JUGLANIN LEUCOCIANIDOL METHYLQUERCETIN-3 MONOXERUTIN MYRICETIN MYRICITRIN NARCISSIN NATSUDAIDAIN PINOBANKSIN PINOSTROBIN PRUNETIN QUERCETAGITRIN QUERCETIN QUERCIMERITRIN ROBINETIN RUTOSIDE SCIADOPITYSIN SINENSETIN TANGERETIN TAXIFOLIN TECTORIGENIN TECTORIGENIN-PSI TROXERUTIN VENORUTON-P4 Z-12000 Z-12001 Z-12007 BIOFUNGICIDES SACCHAROMYCES-= CEREVISIAE BIOL.CONTROL-AGENTS SACCHAROMYCES-= CEREVISIAE BIOMETRICS FIELD-ANALYSIS META-ANALYSIS NEURAL-NETWORKS REGRESSION-ANALYSIS BIOPHARM. PRODRUG BIPOLAR-DISORDER BIPOLAR-I-DISORDER BIPOLAR-II-DISORDER manic-depression BLADDER-DISEASE CYSTITIS CYSTOPYELITIS IRRITABLE-BLADDER BLOOD HEMATOPOIESIS HEMOCONCENTRATION BLOOD-CLOTTING BLEEDING-TIME CLOTTING-TIME PROTHROMBIN-TIME RECALCIFICATION-TIME THROMBIN-TIME THROMBOPLASTIN-= GENERATION-TEST THROMBOPLASTIN-TIME THROMBOTEST BLOOD-CLOTTING-FACTOR CLOTTING-FACTOR-IX CLOTTING-FACTOR-IX CLOTTING-FACTOR-IXAI CLOTTING-FACTOR-V CLOTTING-FACTOR-VII CLOTTING-FACTOR-VIIA CLOTTING-FACTOR-VIII CLOTTING-FACTOR-VIII-= DELTA-II CLOTTING-FACTOR-X CLOTTING-FACTOR-XI CLOTTING-FACTOR-XII CLOTTING-FACTOR-XII-A CLOTTING-FACTOR-XII-F clotting-factor-xiii COBYRATE CRYOPRECIPITATE FIBRIN-STABILIZING-FACTOR FIBRINOGEN GLUTAMYL-PLASMINOGEN KONYNE LYSYL-PLASMINOGEN PLASMINOGEN PLATELET-FACTOR-3 PLATELET-FACTOR-4 PLATELET-FACTOR-4-HUMAN PROTHROMBIN THROMBOPLASTIN VON-WILLEBRAND-FACTOR BLOOD-GROUP RH-FACTOR RH-NEG. RH-POS.

1108 APPENDIX D BLOOD-SUBSTITUTES ALBOSORB CITROGLUCOSALAN DEXTRAN-70 DUXON ELOHES FC-43 FC-80 GELAFUNDIN GELATINOL GLUCOSALAN HETASTARCH LACTASOL OXYPOLYGELATIN PENTASTARCH PERFLUAMINE PERFLUNAFENE POLYGELINE POLYVIDONE PYRIDOXALATED-= POLYHEMOGLOBIN QUARTASOL TRISOL BLOOD-SUGAR GLUCOSE-TOLERANCE BODY-TEMPERATURE HEAT-STROKE HYPERPYREXIA HYPERTHERMIA HYPOTHERMIA MALIGNANT-HYPERPYREXIA POIKILOTHERMY THERMOGENESIS BODY-WEIGHT metabolic-syndrome METABOLIC-SYNDROME-X OBESITY PICKWICK-SYNDROME WEIGHT-GAIN WEIGHT-LOSS BOLUS BULLET BONE DIAPHYSIS EPIPHYSIS FEMUR HUMERUS OSTEOBLAST OSTEOCLAST OSTEOPHYTE PATELLA RIB SCAPULA TIBIA BOTANY ACACIA ACHILLEA ACHYRANTHES ACHYROCLINE ACONITUM ACORUS ADATHODA ADENOPHORA ADIANTUM ADONIS AEGLE AESCULUS AGNUS AIZOON ALCHEMILLA ALEURITES ALFALFA ALISMA ALLIUM ALNUS ALOE ALPINIAE ALSTONIA AMARANTHUS AMARYLLIS AMBROSIA ANACARDIUM ANDROGRAPHIS ANEMARRHENA ANEMONE ANGELICA ANTHEMIS ANTHYLLIS APPLE ARACHIS ARALIA ARCTOSTAPHYLOS ARECA ARISTOLOCHIA ARNICA ARTEMISIA ASARUM ASPALATHUS ASPERULA ASPIDOSPERMA ASTRAGALI ASTRAGALUS ATHYLIUM ATRACTYLIS atractylodes ATROPA AURANTIUM AVENA AZADIRACHTA BALLOTA BAMBOO BAPTISIA BEAN BERBERIS BERRY beta-vulgaris BETULA BETULUS BIDENS BOERHAAVIA BORRAGO BOUGAINVILLEA BOUVARDIA BRASSICA BRUCEA BRUNELLA BRUNFELSIA BRUSSELS-SPROUT BRYONIA BRYOPHYLLUM BUPLEURUM CABBAGE CAESALPINIA CALAMUS CALENDULA CALLIGONUM CAMELLIA CAMPANULA CANNABIS CAPRICUM CAPSELLA CARALLUMA CARDIOSPERMUM CARROT CARTHAMUS CARUM CARYOPHYLLI CASEARIA CASIMIROA CASSIA CASSIPOUREA CATHARANTHUS CECROPIA CENTELLA CERATOCEPHALUS CESTRUM CHAEROPHYLLUM CHAMOMILLA CHELIDONIUM CHENOPODIUM CHINNAOMI CHRYSANTHEMUM CICUTA CIMICIFUGA CINCHONA CINNAMOMUM CIRSIUM CITRULLUS CITRUS CLUYTIA CNESTIS CNIDIUM COCCULUS COCONUT COCOS COIX COLCHICUM COMBRETUM COMMIPHORA CONDURANGO CONIUM CONVALLARIA CONVOLVULUS CONYZA CORN CORNUS CORONILLA CORYDALIS COTTON CRATAEGUS CREPIS CRINUM CROTOLARIA CROTON CUCUMBER CUCUMIS CUCURBITA CUPRESSUS CURCUMA CUSCUTA CUTANDEA CYMBOPOGON CYNARA CYNOGLOSSUM CYTISUS DALBERGIA DATURA DAUCUS DELPHINIUM DIANTHUS DIARTHRON DIEFFENBACHIA DIGITALIS DIOSCOREA DIOSPYROS DIPLOTAXIS DISTYLIUM DOLICHOS DORSTENIA DROSERA DRYOPTERIS DUCROSIA ECHINACEA ECHINOPS ECHIUM

Derwent Drug File 1109 Thesaurus ECLIPTA ELEPHANTOPUS ELEUTHEROCOCCUS EMEX EPHEDRA EPILOBIUM EPIMEDIUM EQUISETUM EREMOBIUM ERIGERON ERODIUM ERYTHROXYLUM EUCALYPTUS EUCOMMIA EUPATORIUM EUPHORBIA EURYOPS FERULA FESTUCA FICARIA FILIPENDULA FOENICULUM FRANCOEURIA FRANGULA FUMARIA GALIUM GELSEMIUM GENTIANA GERANIUM GINKGO GLOSSOSTEMON GLYCERIA GLYCYRRHIZA GNIDIA GOSSYPIUM GUETTARDA GYMNARRHENA GYMNEMA GYPSOPHILIA HALOXYLON HAMAMELIS HAMMADA HARPAGOPHYTUM HEDERA HEDYOTIS HELIOTROPIUM HERACLEUM HIBISCUS HOMERIA HORDEUM HUMULUS HYMENOXYS HYOSCYAMUS HYPERICUM HYPOXIS IFLOGA ILEX INDIGOFERA IPOMOEA ISOPLEXIS IXERIS JATROPHA JUGLANS JUJUBE JUNIPERUS JUSTICIA KALANCHOE KETJUBUNG KHAT KHAYA KRAMERIA LACHESIS LACTUCA LAGENARIA LANTANA LAUNAEA LAWSONIA LEDEBOURIELLA LEDUM LEONOTIS LEONTODON LEPIDIUM LESPEDEZA LETTUCE LEUCAENA LEUCOS LEUCOTHOE LIGUSTICUM LINARIA LINDERA LITHOSPERMUM LOLIUM LORANTHUS LOTUS LUPINUS LYCHNIS LYCOPERSICON LYCOPUS MACLEAYA MAGNOLIAE MAHONIA MAIZE MALLOTUS MALUS MALVAVISCUS MARSDENIA MATRICARIA MEDICAGO MELIA MELISSA MENTHA MERCURIALIS METASEQUOIA MILLETIA MITCHELLA MITELLA MOMORDICA MONTANOA MORAEA MORUS MOUTAN MUNRONIA MUSA MYOPORUM MYRISTICA NARTHECIUM NEURADA NICOTIANA NOTOCERAS OAT OCHROSIA OLEA OLEANDER OLIVE ONION ONONIDIS ONONIS OPHIOPOGON ORANGE ORTHOSIPHONIS ORYZA OSBECKIA OXYTROPIS PAEDERIA PAEONIA PANAX PANICUM PAPAVER PASSIFLORA PEA PEANUT PEAR PELTOPHORUM PENNISETUM PENTAS PEUCEDANUM PEUMUS PHALARIS PHASEOLUS PHILODENDRON PHYLLANTHUS PICNOMON PICRASMA PICRIS PICRORRHIZA PIMELEA PIMPINELLA PINELLIA PIPER PLAGIORHEGMA PLANTAGO PLATYCODI POINSETTIA POLYGONUM POPULUS PORIA PORTULACA POTATO POTENTILLA POUPARTIA PRIMULA PROSOPIS PRUNUS PSIDIUM PSORALEA PSOROSPERMUM PTERIDIUM PTEROCARPUS PTEROTABERNA PUERARIA PULSATILLA PUNICA PUREREA QUERCUS RADICULA RANUNCULUS RAPISTRUM RAUWOLFIA REHMANNIA RESEDA RHAMNUS RHEUM RHODODENDRON RHUS RIBES RICE RICINUS ROLLINIA ROSA ROSMARINUS RUBIA RUSCUS RYE SABAL SACCHARUM saccharum-officinarium SALACIA SALIX SALVIA SAMBUCUS SARACA SASSAFRAS SAUSSUREA SAVIGNYA SCHIMPERA SCHISANDRA SCHISMUS SCHIZANDRA SCILLA SCUTELLARIA SECALE SEDUM

1110 APPENDIX D SENECIO SENNA SEPIA SESBANIA SIDERITIS SILENE SILYBUM SINAPIS SOLANUM SOLENOSTEMMA SOLIDAGO SONCHUS SOPHORA SOULAMEA SOY-BEAN SPARGNIUM SPINACH SPINACIA STEGANOTAENIA STELLARIA STEVIA STREBLUS STRYCHNOS STYPANDRA SUAEDA SUGAR-BEET sugar-cane SWEETIA SWERTIA SYZIGIUM SYZYGIUM TABERNAEMONTANA TAMARIX TAMUS TANACETUM TAXUS TERMINALIA TETRAPANAX TETRAPLEURA TEUCRIUM THAMNOSMA THEOBROMA theobroma-cacao THUJA TINOSPORA TOMATO TREMA TRIBULUS TRIFOLIUM TRISETUM TUSSILAGO UNCARIA URTICA VACCINIUM VALERIANA VANDELLIA VERATRUM VERBASCUM VERBENA VERNONIA VETIVERIA VIBURNUM VICIA VINCA VIOLA VISCUM WERNERIA WHEAT WITHANIA XANTHOCERCIS YUCCA ZEA ZINGIBER ZIZYPHUS BRADYKININ-ANTAGONISTS B-1324 B-201 B-327 B-3814 B-3816 B-3820 B-3832 B-3878 B-3926 B-4144 B-4146 B-4148 B-429 B-4308 B-4310 B-9066 B-9340 B-9430 B-9436 B-9668 B-9812 B-9816 B-9858 B-9958 BRADYZIDE CP-0088 CP-0126 CP-0127 CP-0347 CP-0364 CP-0494 CP-0499 CP-0597 FR-167344 FR-172357 FR-173657 GR-100679 HOE-140-DE-ARG-10 ICATIBANT KALLIDIN-9-LEU-DE-ARG-10 MEN-11270 MV-8608 MV-8610 MV-8612 NEPADUTANT NPC-16731 NPC-17731 NPC-17761 NPC-18521 NPC-18688 NPC-414 NPC-567 NPC-573 PD-154075 PD-161182 R-715 S-16474 WIN-64338 WIN-64338 Y-23023 BRAIN AMYGDALA ARACHNOID ARCUATE-NUCLEUS AREA-POSTREMA ASTROCYTE AUDITORY-CORTEX BASAL-GANGLION BRAIN-STEM CAUDATE-NUCLEUS CAUDATE-PUTAMEN CENTRAL-GRAY CEREBELLUM CEREBRAL-CORTEX CEREBRUM CHOROID-PLEXUS CINGULATE-CORTEX CINGULATE-GYRUS CINGULUM-BUNDLE CISTERNA-MAGNA CLAUSTRUM CNS CORPUS-CALLOSUM CORPUS-STRIATUM CUNEATE-NUCLEUS DENTATE-GYRUS DIAGONAL-BAND-OF-BROCA DIENCEPHALON DORSOMEDIAL-NUCLEUS DURA-MATER ENTOPEDUNCULAR-NUCLEUS FIMBRIA-FORNIX FOREBRAIN FORNIX-CEREBRI FORNIX-FIMBRIA FRONTAL-CORTEX GENICULATE-BODY GLIACYTE GLOBUS-PALLIDUS HABENULA HIPPOCAMPUS INFERIOR-COLLICULUS INFERIOR-OLIVE INTERPEDUNCULAR-NUCLEUS LENTIFORM-NUCLEUS LEPTOMENINX LIMBIC-SYSTEM LOCUS-COERULEUS MEDULLA-OBLONGATA MENINGES MESENCEPHALON METENCEPHALON MICROGLIA MIDBRAIN MOTOR-CORTEX NEOCORTEX NEOSTRIATUM NUCLEUS-ACCUMBENS NUCLEUS-AMBIGUUS NUCLEUS-CENTRALIS-= SUPERIOR NUCLEUS-RETICULARIS-= GIGANTOCELLULARIS NUCLEUS-RETROAMBIGUALIS NUCLEUS-TRACTUS-SOLITARII NUCLEUS-VENTRALIS-= LATERALIS OCCIPITAL-CORTEX OLFACTORY-BULB OLFACTORY-CORTEX OLFACTORY-LOBE OLFACTORY-TRACT OLFACTORY-TUBERCLE OLIGODENDROGLIA OLIVARY-NUCLEUS OPTIC-TECTUM OPTIC-TRACT PALEOSTRIATUM PARIETAL-CORTEX PARS-COMPACTA PARS-RETICULATA PIA-ARACHNOID PIA-MATER PONS PONTO-CEREBELLAR-TRACT PREFRONTAL-CORTEX PREOPTIC-AREA PURKINJE-CELL PYRAMIDAL-CELL PYRAMIDAL-TRACT PYRIFORM-CORTEX RAPHE-NUCLEUS RETICULAR-FORMATION RHINENCEPHALON SENSORY-CORTEX

Derwent Drug File 1111 Thesaurus SEPTUM-PELLUCIDUM SUBFORNICAL-ORGAN SUBSTANTIA-INNOMINATA SUBSTANTIA-NIGRA SUBTHALAMIC-NUCLEUS SUPERIOR-COLLICULUS SYNAPTOSOME TEGMENTUM TELENCEPHALON THALAMUS TRIGEMINAL-NUCLEUS VENTROBASAL-COMPLEX VESTIBULAR-NUCLEUS VISUAL-CORTEX BRONCHODILATORS A-93178 ABC-99 ABLUKAST ABT-080 AC-119 ACEBROPHYLLINE ADRENALINE AFORMOTEROL AM-682 AMBROXOL THEOPHYLLINATE AMBUPHYLLINE AMITEROL ANDOLAST AR-C-68397-AA AS-35 AZANATOR AZASPIRIUM CHLORIDE B-9004-070 BAMBUTEROL BAMIFYLLINE BB-1502 BITOLTEROL BM-531 BMS-262084 BN-1267 BRAIN-NATRIURETIC-PEPTIDE BRL-55834 BROXATEROL CARBUTEROL CDP-840 CGP-57698 CHINOIN-170 CHOLINE-THEOPHYLLINATE CI-923 CILOMILAST CLENBUTEROL CLORPRENALINE COLTEROL CONOPHYLLINE CONTIGNASTEROL D-18024 D-2343 D-4030 DAC-5945 DAMETRALAST DECLOXIZINE DEPTROPINE DIBUNATE SODIUM DIMABEFYLLINE DINIPROFYLLINE DIOXETHEDRIN DIPROPHYLLINE EPHEDRINE EPRAZINONE ETAFEDRINE ETANTEROL ETHYLNORADRENALINE FENOTEROL FENSPIRIDE FKK FLUTROPIUM BROMIDE FORMOTEROL FR-113680 FR-167344 FUPRAZOLE FURAFYLLINE GEA-3175 GEA-3268 GEA-5145 HEPTAMINOLACEFYLLINE HEXOPRENALINE HOKU-81 HOQUIZIL HQL-79 HSR-284 IBUTEROL ICI-58301 ICI-61129 IPRATROPIUM BROMIDE ISAMOXOLE ISBUFYLLINE ISOETARINE ISOPRENALINE KC-11404 KC-399 KF-15570 KF-17625 KW-4099 KWD-2131 L-670630 L-686708 L-739010 L-826141 LEVOSALBUTAMOL M-711 MABUTEROL MEN-10376 MEQUITAMIUM IODIDE METHOXYPHENAMINE METHYLEPHEDRINE METHYLPROPYLXANTHINE1,3 MKS-492 MONTELUKAST MX-2-120 NAMINTEROL NCX-1020 NCX-950 NIAPRAZINE NISBUTEROL NORBUDRINE NZ-107 ORCIPRENALINE OXITROPIUM BROMIDE PAB-110 PAB-13 PAB-13 PAB-23 PAB-23 PEGANIN PF-904 PICUMETEROL PIMETHIXENE PIPERLONGUMINE PIPOXIZINE PIQUIZIL PIRBUTEROL PROCATEROL PROTOKYLOL PSEUDOEPHEDRINE QH-25 QUINETALATE QUINPRENALINE R-836 REPROTEROL RG-12553 RIMITEROL RLX RO-25-1553 RO-31-6930 RP-58802B RP-66471 RP-73401 RU-42173 RWJ-22108 S-9795 SALBUTAMOL SALMEFAMOL SALMETEROL SB-207499 SCA-40 SCA-41 SCH-351591 SDZ-217-744 SERINE-BORATE SIGUAZODAN SKF-102081 SKF-102922 SKF-104353 SOM-1397-CL SOTERENOL SQ-33961 SR-2640 SULFONTEROL SULOXIFEN T-0201 T-440 TA-073 TA-2005 TERBUTALINE TERFENADINE TETRAGALLOYLQUINATE THEOPHYLLINE THEOPHYLLINE-LYSINE THEOPHYLLINE-SODIUM-= ANISATE THEOPHYLLINE-SODIUM-= GLYCINATE THIAZINAMIUM IODIDE THIAZINAMIUM-CHLORIDE THIAZINAMIUM-SULFOXIDE THIAZINAMIUM-SULFOXIDE = IODIDE TIBENELAST TIOTROPIUM BROMIDE TOLIMIDONE TOMELUKAST TRETOQUINOL TULOBUTEROL UCB-JO28 UROGUANYLIN VASICINONE VEPHYLLINE VERLUKAST VEROFYLLINE XANOXATE YM-934 ZAFIRLUKAST ZARDAVERINE ZD-6021 ZINDOTRINE ZINTEROL BURN FROSTBITE C5-ANTAGONISTS L-164710 CALCINOSIS CHONDROCALCINOSIS CALCIUM-AGONISTS 202-791 202-791-(+) ADENOPHOSTIN-A ADENOPHOSTIN-B

1112 APPENDIX D BAY-K-8644 BAY-R-5417 BAY-T-5006 BAY-W-5035 BAY-W-5037 BAY-W-5434 BAY-Y-5959 CGP-28392 CGP-48506 FPL-64176 H-160-51 L-163191 NPS-R-568 RS-30026 XB-513 YC-170 ZOOXANTHELLATOXIN-A CALCIUM-ANTAGONISTS 130-B 202-791 202-791-(-) 233 8363-S AE-0047 AGATOXIN-OMEGA-IVA AGELASIMINE-A AGELASIMINE-B AH-1058 AHR-16303B AHR-5360 AHR-5360C AJ-2615 AJ-3941 ALISMOL AMAUROMINE AMINOPHYLLINE AMIODARONE AMLODIPINE ANIPAMIL ASPAMINOL ATHAMANTIN AZIDOPINE B-120 BAPTA BAPTA-AM BARNIDIPINE BAY-E-5759 BAY-E-6927 BAY-I-1441 BAY-K-9320 BAY-L-3505 BAY-L-8201 BAY-M-5579 BAY-N-5247 BAY-N-5248 BAY-N-6391 BAY-O-5572 BAY-P-8857 BAY-R-4407 BBR-2160 BBR-2196 BBR-2197 BELFOSDIL BENIDIPINE BENZOBENZAMIL BEPRIDIL BISARAMIL BM-20-1140 BMS-204352 BMY-20064 BRINAZARONE BRL-32872 BX-471 CADINOL-T CALCISEPTINE CALMIDAZOLIUM CARBOCROMEN CD-349 CD-832 CELTISINE CERM-11888 CERM-11956 CGS-10078B CILNIDIPINE CINNARIZINE CK-53 CLENTIAZEM CLOXACEPRIDE CNS-1237 CONOTOXIN-OMEGA CONOTOXIN-OMEGA-MVIIA CONOTOXIN-OMEGA-MVIIC CP-060 CP-060-S CP-1136S CP-894S CPU-23 CPU-57 CS-905 CULARIDINE CURINE CV-159 D-51-4700 D-528 D-557 D-559 D-595 D-617 D-620 D-784 D-792 D-846 D-890 DAPHNOLINE DARODIPINE DAURISOLINE DEACETYLDILTIAZEM DEMETHYLDILTIAZEM-N DEMETHYLNAFTOPIDIL DEVAPAMIL DEXNIGULDIPINE DEXVERAPAMIL DHP-218 DIAZOXIDE DICLOFURIME DILAZEP DILTIAZEM DIPERDIPINE DIPFLUZINE DIPROTEVERINE DIPYRIDAMOLE DOPROPIDIL DOTARIZINE DTZ-323 E-2050 EBASTINE ELGODIPINE EMOPAMIL EPERISONE ETACIZINE ETAFENONE EUGENOLOL EVOCARPINE FALIPAMIL FANTOFARONE FARGESIN FASUDIL FCE-24265 FELODIPINE FENDILINE FK-664 FLORDIPINE FOSTEDIL FPL-62129 FR-46171 FRAXINELLONE FTX-3.3 FURNIDIPINE GALLOPAMIL GOE-5438 GOE-5584-A GOE-5606 GOE-5806-A GOE-6070 GS-389 GYKI-12735 GYKI-12743 HA-1004 HE-30346 HERNANDEZINE HEXOBENDINE HIMBADINE HYDROXYINDAPAMIDE-5 I-65 IGANIDIPINE IODIPINE IOS-1-1212 IPROTIAZEM ISOCORYNOXEINE ISOCRASSIFOLINE ISOPERISONE ISRADIPINE KB-2796 KHL-8430 KP-840 KT-362 KV-1360 L-593754 L-648865 L-651525 LABEDIPINEDILOL-A LACIDIPINE LAS-30538 LERCANIDIPINE LEUALACIN LEVEMOPAMIL LF-20254 LIDOFLAZINE LIFARIZINE LOE-908 LU-48895 LU-49667 LU-49888 LU-49938 LU-49940 LU-51903 LUBELUZOLE MANIDIPINE MCI-154 MCI-176 MCN-5691 MCN-6186 MDL-72567 MEFLOQUINE-N-OXIDE MEPAMIL METHYLMEFLOQUIN-N METHYLRIPARIOCHROMENE MIBEFRADIL MONATEPIL MPC-2101 MRS-1754 N-3601 NC-1100 NEXOPAMIL NGP-1-01 NICARDIPINE NICTIAZEM NIFEDIPINE NIFEDIPINE-META NILUDIPINE NILVADIPINE

Derwent Drug File 1113 Thesaurus NIMODIPINE NISOLDIPINE NISOLDIPINE-META NITRENDIPINE NITROGLYCEROL NITROPRUSSIDE SODIUM NNC-09-0026 NORVERAPAMIL NP-252 NPK-1882 NPK-1886 NPS-2143 NS-21 NS-7 NSC-110333 OSTRUTHOL OXODIPINE OXYFEDRINE PAK-104 PAK-104-P PALONIDIPINE PAPAVERINE PCA-50938 PD-122860 PD-150606 PERHEXILINE PN-205033 PO-285 PR-22 PR-23 PRAERUPTORIN-C PRAERUPTORIN-E PRENYLAMINE PROPYLMETHYLENE= DIOXYINDENE R-4407 R-5417 R-56865 R-59494 R-70608 R-71811 R-83572 R-91154 RCC-36 REOFLUSINE RIODIPINE RK-30 RO-11-2933 RO-11-3651 RO-18-3981 RO-23-6152 RONIPAMIL RS-504393 RS-5773 RS-93522 RWJ-22108 S-11568 S-12967 S-12968 S-2150 S-247 S-312 S-312-(+) S-312-(-) SA-2572 SABELUZOLE SB-225002 SC-30552 SD-217595 SD-3212 SEMOTIADIL SFTX-3.3 SIM-6080 SIRATIAZEM SKF-96365 SKF-96365 SM-6586 SNX-111 SNX-239 SQ-31765 SQ-32547 SQ-33351 SR-33671 SR-33805 SR-45813 SULOCTIDIL SUN-N-8075 SZ-48 SZ-51 T-13 TA-993 TAK-779 TALUDIPINE TDN-345 TELUDIPINE TENUIPINE TERFLAVOXATE TERODILINE TIAMDIPINE TIAPAMIL TINCTORMINE TMB-8 TN-871 TRAPYMINE TRIPAMIDE U-92032 UK-52831 UK-84149 ULFS-49 VERAPAMIL VUF-4567 VUF-4568 Y-19638 YM-151 YM-16151-1 YM-430 YS-035 ZICONOTIDE CALICIVIRUS EBHS-VIRUS VE-VIRUS CALMODULIN-ANTAGONISTS BEPRIDIL CALMIDAZOLIUM CETIEDIL CHLORPROMAZINE CV-159 DIDEETHYLAMIODARONE DY-9760-E ELZIVERINE EUDISTOMIDIN-A FASCICULATE-A FELODIPINE FLUMERIDONE FLUPHENAZINE FLUPHENAZINE-DECANOATE FLUPHENAZINE-ENANTHATE J-8 KHL-8430 L-3937 NIGULDIPINE OPHIOBOLIN-A PENFLURIDOL PIMOZIDE PRENYLAMINE PSEUDODISTOMIN-A PSEUDODISTOMIN-B PYRIDINDOLOL QUIN-2-ACETOXYMETHY= LESTER RETICULOL RU-45144 S-728011 S-808314 S-811705 S-847445 SIM-6080 STELLETTAMIDE-A TH-1011 TH-1090 TH-1091 TH-1231 TH-1257 TH-1274 THIORIDAZINE TI-233 TRIFLUOPERAZINE W-13 W-5 W-66 W-7 W-77 ZALDARIDE CANNABINOID-AGONISTS ANANDAMIDE CP-55940 HU-210 METHANANDAMIDE-(R) WIN-55212-2 CANNABINOID-ANTAGONISTS AM-630 CARBOHYDRATE-METAB. BLOOD-SUGAR GLUCONEOGENESIS GLUCOSE-TOLERANCE GLYCOGENOLYSIS GLYCOLYSIS HMP-SHUNT STARCH-TOLERANCE CARBOHYDRATEMETAB.DISORDER ANDERSEN-DISEASE bronze-diabetes DAWN-PHENOMENON DEBRE-SYNDROME DIABETES diabetic-glomerulosclerosis diabetic-retinopathy FRUCTOSE-INTOLERANCE FUCOSIDOSIS GALACTOSEMIA GLYCOGENOSIS hepatorenal-glycogenosis HERS-DISEASE HYPERGLYCEMIA HYPERGLYCORRHACHIA HYPERINSULINISM HYPERLACTACIDEMIA HYPEROXALEMIA HYPEROXALURIA HYPOGLYCEMIA HYPOINSULINEMIA kimmelstiel-wilson-syndrome MANNOSIDOSIS MCARDLE-DISEASE metabolic-syndrome METABOLIC-SYNDROME-X POMPE-DISEASE troissier-hanot-chauffard-= syndrome von-gierke-syndrome CARBONIC-ANHYDRASEINHIBITORS ACETAZOLAMIDE AMINOZOLAMIDE BENDROFLUMETHIAZIDE BENZOLAMIDE BENZTHIAZIDE BUTAZOLAMIDE

1114 APPENDIX D CARZENIDE CHLOROTHIAZIDE CHLORTALIDONE CHLORZOLAMIDE DICLOFENAMIDE DORZOLAMIDE ETHOXYZOLAMIDE HYDROBENTIZIDE HYDROCHLOROTHIAZIDE HYDROFLUMETHIAZIDE L-643799 L-645151 L-662583 L-671152 L-693612 METHAZOLAMIDE METOLAZONE MK-927 POLYTHIAZIDE PROPAZOLAMIDE SEZOLAMIDE TRICHLORMETHIAZIDE TRIFLUORMETHAZOLAMIDE TRIFLUOROMETHANE= SULFONAMIDE CARCINOMA 3LL-CELL A15-CELL A1847-CELL A253-CELL A2780-CELL B4976-CELL BE-CELL BEN-CELL BT20-CELL BT474-CELL CAOV-CELL CASKI-CELL CO115-CELL CT26 CT26-CELL DETROIT-562-CELL DLD1-CELL EHRLICH-ASCITES EHRLICH-ASCITES-CELL ELCO2-CELL H157-CELL HBT3-CELL HCT-CELL HCT116 HCT116-CELL HELA-CELL HEP2-CELL HSO578-CELL HX13-CELL HX18-CELL HX29-CELL KB-CELL KPI-CELL KU1-CELL LEWIS-LUNG-CARCINOMA LEWIS-LUNG-CARCINOMA-= CELL LOVO-CELL M109-CELL MBT2-CELL MGH41-CELL MGHV1-CELL MKN45-CELL MOT-CELL NH1K-3025-CELL OVCAR2-CELL OVCAR3-CELL OVCAR4-CELL OVCAR5-CELL PC1-CELL PC10-CELL PC9-CELL POC-CELL QG56-CELL QG90-CELL RPMI2650-CELL RT112-CELL SH3-CELL SK-OV-CELL SW1271-CELL SW403-CELL SW48-CELL SW480-CELL SW620-CELL SW900-CELL T24-CELL T47D-CELL VX2-CELL WIDR-CELL CARDIANT CARDIOGLYCOSIDE CARDIANTS 201-106 202-791 202-791-(-) 349U85 606-A 661U88 8363-S A-2545 A-40557 AC-119 ACEFYLLINE ACEFYLLINE-PIPERAZINE ACETYLDIGITOXIN ACETYLDIGOXIN ACETYLDIGOXIN-12 ACETYLDIGOXIN-ALPHA ACETYLDIGOXIN-BETA ACETYLGITOXIN ACETYLSTROPHANTHIDIN ACETYLTYLOPHOROSIDE ACOVENOSIDE ACOVENOSIDE-A ACOVENOSIDE-B ACRIHELLIN ACTODIGIN ADIBENDAN ADONISIDE AFP-03 AFROGENIN AG-2H AGELASIMINE-A AGELASIMINE-B ALIFEDRINE ALLOPUMILIOTOXIN-339-A ALMOKALANT AMBUPHYLLINE AMIKHELLINE AMINOETHYL-NITRATE AMINOPHYLLINE AMINOXYTRIPHENE AMIODARONE AMLODIPINE AMOPROXAN AMRINONE AMYL-NITRITE ANIPAMIL ANTHOPLEURIN-A ANTHOPLEURIN-B APP-201-533 APRIKALIM AQ-AH-208 AQM-171 AR-L-100-BS AR-L-113-BS AR-L-57 AR-L-57-CL ARANIDIPINE ARENOBUFAGIN ARPROMIDINE ASCLEPOSIDE ASEBOTOXIN-X ASI-222 ASI-253 ASI-254 ATL-193 ATP-MAGNESIUM-CHLORIDE ATRASENTAN AY-22248 AZACLORZINE AZAFTOZINE B-744-96 B-744-98 B-744-99 BA-31531 BA-41899 BAMIFYLLINE BARNIDIPINE BAY-1518 BAY-I-1441 BAY-K-9320 BAY-L-3505 BAY-N-6391 BAY-O-5572 BAY-W-5035 BAY-Y-5959 BBR-2160 BDF-9148 BDF-9196 BDF-9198 BEMARINONE BEMORADAN BENDAZOL BENFURODIL-HEMISUCCINATE BENIDIPINE BENZIODARONE BEPRIDIL BERSALDEGENIN-= ORTHOACETATE BG-31 BG-32 BG-60 BGP-15 BM-121307 BM-500430 BMS-180448 BMS-182657 BMS-188797 BMS-189365 BMS-193884 BN-50417 BRAIN-NATRIURETIC-= PEPTIDE-HUMAN BU-E-75 BU-E-76 BUFALIN BUFOGENIN BUMEPIDIL BUQUINERAN BUTOPAMINE BUTOPROZINE BUTYLIDENEPHTHALIDE C-92-4609 CAMPHOTAMIDE CANARIGENIN CANDESARTAN-CILEXETIL CANDOXATRIL CAPOBENATE CAPSINOLOL CARBAZERAN CARBOCROMEN CARDIOGLYCOSIDES CARIPORIDE

Derwent Drug File 1115 Thesaurus CARSATRIN CARYACHINE CASSAINE CD-832 CEDO-8956 CELIPROLOL CERBERIOPSINE-2 CERBEROSIDE CERM-11956 CGP-28392 CGP-48506 CGS-5649B CH-102 CHLORACYZINE CHOLINE-THEOPHYLLINATE CI-930 CINECROMEN CINEPAXADIL CINEPAZATE CINEPAZET CINEPAZIDE CINOBUFAGIN CINPROPAZIDE CK-2130 CK-2289 CK-3197 CL-284027 CLAMIKALANT CLENTIAZEM CLONITRATE CLORICROMEN CLORIDAROL CONIVAPTAN CONVALLATOXIN CONVALLATOXOL CORCHOROSIDE-A CORDIALIN CORELBORIN-PI CORMINE CP-060 CP-060-S CPU-57 CRATAEGUTT CREATINOLFOSFATE CRYPTOSIN CS-747 CV-159 CV-1808 CVT-510 CYCLOVIROBUXINE-D CYMAROL D-477A D-4975 D-557 D-559 D-617 D-620 D-846 DAIGREMONTIANIN DANSHEN DARODIPINE DARUSENTAN DEACETYLDILTIAZEM DEETHYLACECAINIDE DEGLUCOCHEIROTOXIN DEGLUCOHYRCANOSIDE DEMETHYLDILTIAZEM-N DEMETHYLIVABRADINE-N DENDROASPIS-= NATRIURETIC-PEPTIDE DENOPAMINE DESLANOSIDE DEVAPAMIL DEXVERAPAMIL DIACETYLDIGOXIN-= ALPHA,BETA DIADENOSINE-= PENTAPHOSPHATE DIADENOSINE-= TETRAPHOSPHATE DICLOFURIME DIETHYLAMINOETHOXY= HEXESTROL DIGINATIN DIGITONIN DIGITOXIGENIN DIGITOXIGENIN-= BISDIGITOXOSIDE DIGITOXIGENIN-= DIGITOXOSIDE DIGITOXIN DIGOXIGENIN-DIGITOXOSIDE DIGOXIGENIN-RHAMNOSIDE DIGOXIN DIHYDROBUFALIN-22,23 DIHYDRODIGITOXIN DIHYDRODIGOXIGENIN DIHYDRODIGOXIN DIHYDROOUABAIN DIIODOTHYROPROPIONATE-= 3,5 DILAZEP DILMEFONE DILTIAZEM DIMABEFYLLINE DINECA DIPROTEVERINE DIPYRIDAMOLE DISOPYRAMIDE DK-AH-269 DOBUTAMINE DOPROPIDIL DOXAMINOL DPN-205-734 DROPRENILAMINE DS-201 DWH-146-E DY-9708 E-1020 E-4021 E-4080 E-4701 ECHINOSIDE-B EFLOXATE EGIS-9377 ELAEODENDROSIDE-A ELAEODENDROSIDE-B ELAEODENDROSIDE-C ELAEODENDROSIDE-D ELAEODENDROSIDE-E ELAEODENDROSIDE-J ELGODIPINE EMAKALIM EMD-41000 EMD-46512 EMD-53998 EMD-54622 EMD-54650 EMD-57033 EMD-60263 EMD-85131 ENIPORIDE ENOXIMONE EPC-K1 EPIDIGOXIGENIN ERITRITYL-TETRANITRATE ERYSIMOSIDE ETACIZINE ETAFENONE ETAMIPHYLLIN ETHYLCINEPAZATE ETOFYLLINE EVATROMONOSIDE EVODIAMINE FALIPAMIL FELODIPINE FENALCOMINE FENDILINE FENETRADIL FENOXIMONE FIBROBLAST-GROWTH-= FACTOR-ACIDIC FK-664 FKK FLOREDIL FOSTEDIL FPL-62129 FR-146801 FR-183998 FR-46171 FRUTISIN FURIDARONE FXV-673 GALLOPAMIL GAMABUFOTALIN GANGLEFENE GI-104313 GINGEROL-10 GINGEROL-8 GITALIN GITALOXIGENIN GITALOXIN GITOFORMATE GITOGENIN GITONIN GITOXIGENIN GITOXIN GITOXIN-EPI-16 GLIO-6 GLUCODIGIFUCOSIDE GLUCOEVATROMONOSIDE GLUCOGITOROSIDE GLYCEROL-MONONITRATE-1 GLYCEROL-MONONITRATE-2 GOE-5606 GOE-5806-A GOMPHOGENIN GOMPHOSIDE GP-1-531 GP-2-128 GYKI-12735 GYKI-52713 GYKI-52843 HA-1100 HALENOQUINOL HE-30346 HE-90481 HELLEBRIGENIN HELLEBRIN HELVETICOSIDE HELVETICOSOL HEPTAMINOL HEPTAMINOLACEFYLLINE HEXADILINE HEXOBENDINE HIGENAMINE HMR-1098 HMR-1372 HN-10200 HN-65021 HNS-32 HOE-694 HOE-782 HOLOTHURIN-B HYDROXYPROPAFENONE-5 HYDROXYTERODILINE-PARA IBMECA IBOPAMINE ICI-153110 ICI-170777 IDN-1965 IMAZODAN IMOLAMINE

1116 APPENDIX D INDOLIDAN INO-2628 INO-2628-CZ IPRAMIDIL IPS-1251 ISOBUTYL-NITRITE ISODIGITOXIN ISOIDIDE-DINITRATE ISOIDIDE-MONONITRATE ISOMANNIDE-DINITRATE ISOMANNIDE-MONONITRATE ISOMAZOLE ISOSORBIDE-DINITRATE ISOSORBIDE-MONONITRATE ISOSORBIDE-MONONITRATE-2 ISRADIPINE ITF-296 ITRAMIN TOSILATE IVABRADINE IWF-122-14 IWF-122-60 J-104132 JTV-506 JTV-519 KB-R-7943 KBR-9032 KC-116 KC-12291 KC-144 KC-146 KHELLIN KHELLOSIDE KHL-8430 KI-3315 KI-4032 KM-13 KP-403 KR-30450 KR-30818 KR-31378 KRN-2391 KW-3196 L-709780 L-738167 L-754142 L-8040 L-8412 L-9146 LANATOSIDE LANATOSIDE-A LANATOSIDE-B LANATOSIDE-C LANATOSIDE-D LANATOSIDE-E LASSBIO-294 LB-32841 LEVOSIMENDAN LEX-032 LI-132 LIDOFLAZINE LIGUSTILIDE LINSIDOMINE LIXAZINONE LND-369 LND-623 LND-796 LNF-209 LOTRAFIBAN LP-805 LU-49938 LY-137150 LY-163252 LY-181512 LY-186126 LY-186232 LY-195114 LY-197055 LY-197096 LY-206243 LY-249933 LY-256548 M-66 MAGNOFLORINE MALABEN MANIDIPINE MANNITOL-HEXANITRATE MARINOBUFAGIN MCI-154 MCI-176 MCN-6186 MDL-19438 MDL-73404 MDL-74270 MEDIBAZINE MEDIGOXIN MEDORINONE MEPRAMIDIL MEPROSCILLARIN MERIBENDAN METHYLCARBOXAMIDE-= ADENOSINE METRIFUDIL MF-10058 MIBEFRADIL MILDRONATE MILRINONE MIOFLAZINE MIROTON MITIPHYLLINE MIVAZEROL MIXIDINE MOLSIDOMINE MOROCROMEN MOTAPIZONE MPC-2101 MRE-0470 MS-857 N-3601 NATSUDAIDAIN NERIIFOLIN NEXOPAMIL NICEVERINE NICORANDIL NICOTAFURYL NICOTINOYLALANINE NICTIAZEM NIFEDIPINE NIFEDIPINE-META NILUDIPINE NILVADIPINE NISOLDIPINE NISOLDIPINE-META NITRENDIPINE NITROGLYCEROL NITROSOALBUMIN-S NITROSOGLUTATHIONE-S NORVERAPAMIL NPK-1867 NPK-1868 NPK-1882 NSP-804 NSP-805 OLEANDRIN OLEUROPEIN OLIGVON OLITORISIDE OPC-18790 OPC-6535 OPC-8490 OPHIOBOLIN-A OR-1896 ORG-10325 ORG-20494 ORG-30029 ORG-9731 ORG-9935 OUABAGENIN OUABAIN OXYBATE LITHIUM OXYBATELITHIUM OXYFEDRINE P-0160 P-87-7692 PANTETHINE PD-122860 PD-125944 PD-155080 PD-166793 PELRINONE PENGITOXIN PENTAERYTHRITYL-= TETRANITRATE PENTRINITROL PEPTIDE-6A PERHEXILINE PERUVOSIDE PIMEFYLLINE PIMETINE PIMOBENDAN PIRIDOXILATE PIROXIMONE PIROZADIL PIVAZIDE PLAKORTONE-D PR-22 PR-39 PRAERUPTORIN-C PRAERUPTORIN-E PRENALTEROL PRENYLAMINE PRETIADIL PROCAINAMIDE PROPAFENONE PROPATYLNITRATE PROPIONYLCARNITINE-= TAURINE PROSCILLARIDIN PROTHEOBROMINE PROXYPHYLLINE PS-519 PST-2107 PST-2744 PUMILIOTOXIN-A PUMILIOTOXIN-B PURLANOSIDE-A PURLANOSIDE-B PURPUREA-GLYCOSIDE-A PURPUREA-GLYCOSIDE-B PUWAINAPHYCIN-C PYRIDOFYLLINE QUAZINONE QUAZODINE QUINDONIUM BROMIDE R-80122 RA-159 RA-433 RAMNODIGIN RANOLAZINE RAZINODIL RB-105 RE-244 RE-61 REN-1053 RG-12152 RG-14202 RGW-2938 RIODIPINE RMI-82249 RO-18-3981 RO-23-6152 RO-47-8634 RO-7-2956

Derwent Drug File 1117 Thesaurus RONIPAMIL ROSEOTOXIN-B RPR-100579 RS-1893 RS-30026 RS-5773 RS-93522 S-15176 S-16257 S-312 SATERINONE SB-217242 SB-225002 SC-13173 SC-4453 SCH-00013 SCILLAREN-A SCILLARENIN SCILLIGLAUCOSIDE SCILLIROSIDE SENKYUNOLIDE SENKYUNOLIDE-H SEPARAN-AP-273 SF-43 SF-44 SG-209 SG-212 SG-89 SIGUAZODAN SIMENDAN SIN-1A SINORPHAN SIRATIAZEM SKF-94120 SKF-95654 SM-20550 SMP-300 SOLPECAINOL SOLUFLAZINE SORBINICATE SPARTEINE SPM-3672 SPM-4744 SPM-5185 SR-24870 STENOPRIL STROPHANTHIDIN STROPHANTHIDIN-ACETATE-3 STROPHANTHIN-H STROPHANTHIN-K-BETA STROPHANTHOSIDE-K STROSPESIDE SULMAZOLE SYNEPHRINE T-0201 T-1583 T-162559 TA-993 TAK-636 TALUDIPINE TAZOLOL TELOCINOBUFAGIN TENITRAMINE TEOPRANITOL TERODILINE TETRAMETHYLPYRAZINE TEZOSENTAN TH-1506 THALICMIDINE THEOBROMINE THEOBROMINE-= SALICYLATE-SODIUM THEOBROMINE-SODIUM-= ACETATE THEOPHYLLINE THEOPHYLLINE-LYSINE THEOPHYLLINE-SODIUM-= ANISATE THEOPHYLLINE-SODIUM-= GLYCINATE THEVETIN-A THURFYL-NICOTINATE THYRONAMINE TIAPAMIL TIGOGENIN TIGONIN TIXADIL TK-620-9 TOLAMOLOL TOSIFEN TRAPYMINE TRILLIN TROLNITRATE TY-12533 TYLOGENIN TZC-5665 UBIDECARENONE UCB-22073 UCB-L061 UD-CG-212 UK-14275 UK-1745 UK-36327 UK-52831 UK-61260 UK-69578 UZARIN VASONATRIN-PEPTIDE VERAPAMIL VERODOXIN VESNARINONE VISNADINE VISNAFYLLINE VITEXIN-RHAMNOSIDE VUF-5297 WK-1492 WRC-0342 WRC-0571 WRC-470 XB-513 XESTOQUINONE XJ-735 XJ-757 XT-199 Y-19638 Y-20487 Y-27632 YAKUCHINONE-A YM-430 YM-934 YT-1 YT-146 YT-146 Z-1046 Z-335 ZATEBRADINE ZSY-27 CARDIOGLYCOSIDES ACETYLDIGITOXIN ACETYLDIGOXIN ACETYLDIGOXIN-12 ACETYLDIGOXIN-ALPHA ACETYLDIGOXIN-BETA ACETYLGITOXIN ACETYLSTROPHANTHIDIN ACETYLTYLOPHOROSIDE ACOVENOSIDE ACOVENOSIDE-A ACOVENOSIDE-B ACRIHELLIN ACTODIGIN ADONISIDE AFROGENIN AQM-171 ARENOBUFAGIN ASCLEPOSIDE ASI-222 ASI-253 ASI-254 AY-22248 BERSALDEGENIN-= ORTHOACETATE BUFALIN CANARIGENIN CERBERIOPSINE-2 CERBEROSIDE CINOBUFAGIN CONVALLATOXIN CONVALLATOXOL CORCHOROSIDE-A CORELBORIN-PI CRATAEGUTT CRYPTOSIN CYMAROL DAIGREMONTIANIN DEGLUCOCHEIROTOXIN DEGLUCOHYRCANOSIDE DESLANOSIDE DIACETYLDIGOXIN-= ALPHA,BETA DIGINATIN DIGITONIN DIGITOXIGENIN DIGITOXIGENIN-= BISDIGITOXOSIDE DIGITOXIGENIN-= DIGITOXOSIDE DIGITOXIN DIGOXIGENIN-DIGITOXOSIDE DIGOXIGENIN-RHAMNOSIDE DIGOXIN DIHYDROBUFALIN-22,23 DIHYDRODIGITOXIN DIHYDRODIGOXIGENIN DIHYDRODIGOXIN DIHYDROOUABAIN ELAEODENDROSIDE-A ELAEODENDROSIDE-B ELAEODENDROSIDE-C ELAEODENDROSIDE-D ELAEODENDROSIDE-E ELAEODENDROSIDE-J EPIDIGOXIGENIN ERYSIMOSIDE EVATROMONOSIDE FRUTISIN GAMABUFOTALIN GITALIN GITALOXIGENIN GITALOXIN GITOFORMATE GITOGENIN GITONIN GITOXIGENIN GITOXIN GITOXIN-EPI-16 GLUCODIGIFUCOSIDE GLUCOEVATROMONOSIDE GLUCOGITOROSIDE GOMPHOGENIN GOMPHOSIDE HELLEBRIGENIN HELLEBRIN HELVETICOSIDE HELVETICOSOL ISODIGITOXIN KHELLOSIDE LANATOSIDE LANATOSIDE-A LANATOSIDE-B LANATOSIDE-C

1118 APPENDIX D LANATOSIDE-D LANATOSIDE-E LND-369 LND-623 MARINOBUFAGIN MEDIGOXIN MEPROSCILLARIN MIROTON MITIPHYLLINE NERIIFOLIN OLEANDRIN OLITORISIDE OUABAGENIN OUABAIN PENGITOXIN PERUVOSIDE PROSCILLARIDIN PURLANOSIDE-A PURLANOSIDE-B PURPUREA-GLYCOSIDE-A PURPUREA-GLYCOSIDE-B RAMNODIGIN SC-4453 SCILLAREN-A SCILLARENIN SCILLIGLAUCOSIDE SCILLIROSIDE STROPHANTHIDIN STROPHANTHIDIN-ACETATE-3 STROPHANTHIN-H STROPHANTHIN-K-BETA STROPHANTHOSIDE-K STROSPESIDE TELOCINOBUFAGIN THEVETIN-A TIGOGENIN TIGONIN TRILLIN TYLOGENIN UZARIN VERODOXIN CARDIOPATHY A.V.BLOCK ADAMS-STOKES-DISEASE angara-disease ANGINA-PECTORIS AORTIC-ARCH-ANOMALY AORTIC-STENOSIS ARRHYTHMIA ASYNERGY ASYSTOLE atrial-fibrillation AYERZA-SYNDROME bouveret-syndrome BRADYCARDIA BRISKET-DISEASE CARDIAC-ASTHMA CARDIALGIA CARDIOAUDITORY-= SYNDROME CARDIOMEGALY CARDIOMYOPATHY CARDIOSCLEROSIS CHYLOPERICARDITIS COR-PULMONALE DECOMPENSATION DRESSLER-SYNDROME EBSTEIN-ANOMALY ECTOPY EISENMENGER-SYNDROME ENCEPHALOMYOCARDITIS endocardial-fibroelastosis ENDOCARDITIS EXTRASYSTOLE HEART-ARREST HEART-BLOCK HEART-FAILURE HEGGLIN-SYNDROME HEMOPERICARDIUM HOLT-ORAM-SYNDROME hydropericardium-syndrome HYPERKINETIC-HEART-= SYNDROME HYPOSYSTOLE INCLUSION-BODY-HEPATITIS KUGEL-STOLOF-SYNDROME LONG-QT-SYNDROME LOWN-GANONG-LEVINE-= SYNDROME LUTEMBACHER-SYNDROME MYOCARD.INFARCT. MYOCARDITIS PALPITATION PARASYSTOLE paroxysmal-tachycardia paroxysmal-ventricular-= tachycardia PATENT-DUCTUSARTERIOSUS PATENT-FORAMEN-OVALE PERICARDITIS PLEUROPERICARDITIS PULMONARY-STENOSIS ROMANO-WARD-SYNDROME ROUND-HEART-DISEASE SICK-SINUS-SYNDROME SINOATRIAL-BLOCK TACHYCARDIA TAUSSIG-BING-SYNDROME TETRALOGY-OF-FALLOT THROMBOENDOCARDITIS torsades-de-point UHLENBRUCK-CONDORELLI-= SYNDROME ventricular-fibrillation ventricular-hypertrophy WOLFF-PARKINSON-WHITE-= SYNDROME CARTILAGE CHONDROCYTE FIBROCARTILAGE INTERVERTEBRAL-DISK PERICHONDRIUM CARTILAGE-DISEASE ACHONDROPLASIA CHONDRITIS CHONDRODYSTROPHY CHONDROMA CHONDROMALACIA costal-chondritis DISK-SYNDROME DYSCHONDROPLASIA DYSOSTOSIS MAFFUCI-SYNDROME meyenburg-altherr-= uehlinger-syndrome PERICHONDRITIS POLYCHONDRITIS QUITTOR systemic-chondromalacia tietze-syndrome CASES CASE-HISTORY CASPASE-INHIBITOR CASPASE-1-INHIBITOR CASPASE-3-INHIBITOR CASPASE-3-INHIBITOR CASPASE-9-INHIBITOR CASPASE-INHIBITORS CASPASE-1-INHIBITORS CASPASE-3-INHIBITORS CASPASE-3-INHIBITORS CASPASE-9-INHIBITORS CASTRATION ORCHIECTOMY OVARIECTOMY CCR5-ANTAGONISTS SCH-350634 SCH-351125 TAK-779 CELL-ADHESION-INHIBITOR ICAM-ANTAGONIST INTEGRIN-ANTAGONIST VCAM-ANTAGONIST VITRONECTIN-ANTAGONIST VLA-4-ANTAGONIST CELL-ADHESION-INHIBITORS A-286982 A-292949 ACETYLCYSTEINE ADXANTHROMYCIN ADXANTHROMYCIN-B CICLOSPORIN EMD-121974 EMD-270179 EMD-66203 F-4168 ICAM-ANTAGONISTS INTEGRIN-ANTAGONISTS LM-609 LOTRAFIBAN NEUTROPHIL-INHIBITORY-= FACTOR PD-117302 S-137 S-247 SB-265123 SB-273005 SH-306 SJ-749 SKF-107260 ST-1646 TOCOPHEROL-ALPHA VCAM-ANTAGONISTS VITRONECTIN-ANTAGONISTS VLA-4-ANTAGONISTS XT-199 CELL-RESPIRATION OXYGEN-CONSUMPTION CEREBRAL-CORTEX FORNIX-CEREBRI CEREBROVASCULAR-DISEASE APOPLEXY CEREBRAL-= ARTERIOSCLEROSIS CEREBRAL-VASOMOTOR-= SYNDROME cluster-headache cranial-arteritis-intracranial horton-disease-intracranial intracranial-hypertension MIGRAINE MOYAMOYA-DISEASE PERIVASCULITIS pseudotumor-cerebri SYNCOPE temporal-arteritis-intracranial THALAMIC-SYNDROME CESTODE ANOPLOCEPHALA AVITELLINA BERTIELLA BOTHRIOCEPHALUS CHOANOTAENIA

Derwent Drug File 1119 Thesaurus COENURUS COTUGNIA CYSTICERCUS DIPHYLLOBOTHRIUM DIPLOGONOPORUS DIPYLIDIUM ECHINOCOCCUS HYMENOLEPIS KHAVIA MESOCESTOIDES MONIEZIA PARANOPLOCEPHALA RAILLIETINA SPIROMETRA STILESIA TAENIA THYSANIEZIA CESTODIASIS COENUROSIS CHELATORS 309 ADR-925 ALENDRONATE AMINOHEXANE = DIPHOSPHONATE AMMONIUM-FERRIC-= FERROCYANIDE AMMONIUM-TETRATHIO= MOLYBDATE BAPTA BAPTA-AM BATHOCUPROINE-SULFONATE BATHOPHENANTHROLINE-= SULFONATE BM-210955 CARBONYL-SULFIDE CDTA CDTA-DISODIUM-CALCIUM CELLULOSE-PHOSPHATE CGP-41389 CGP-42166 CGP-43902B CGP-46360 CGP-47072 CGP-47875 CLODRONATE COLESEVELAM CP-02 CP-102 CP-106 CP-107 CP-110 CP-130 CP-21 CP-22 CP-24 CP-25 CP-26 CP-283 CP-38 CP-40 CP-41 CP-44 CP-502 CP-51 CP-511 CP-52 CP-93 CP-94 CP-96 CUPRIZONE CYCLAM CYCLEN DEFERIPRONE DEFEROXAMINE DESFERRITHIOCIN DIMERCAPTOPROPANE= SULFONATE-2,3 DOTA EDDA-N,N EDDHA EDITEMPA EDTA EDTA DIPOTASSIUM EDTA DISODIUM EDTA ZINC EDTA-COBALT EDTA-SODIUM-CALCIUM EDTA-ZINC-CALCIUM EGTA EGTA-DISODIUM-CALCIUM ENTEROBACTIN ETHYLMALTOL ETIDRONATE FOSFONET SODIUM FR-160 GADOLINIUM-EDTA HBED HBEDA HEDTA IBANDRONATE IBRITUMOMAB-TIUXETAN ICRF-192 ICRF-198 ICRF-226 IRC-11 ISA-13-1 LB-145 MALTOL MERCAPTODEXTRAN NE-10244 NE-58051 NERIDRONATE NITRILOTRIACETATE OCTANOHYDROXAMATE OLPADRONATE OR-10141 PAMIDRONATE PARABACTIN PENICILLAMINE PENICILLAMINE-CYSTEINE-= DISULFIDE PENTETATE PENTETATE CALCIUM PENTETATE ZINC PENTETATE-CALCIUM-= TRISODIUM PENTETATE-ZINC-TRISODIUM PHENANTHROLINE-O PHOSPHOCITRATE PHOSPHORIC-ACID POTASSIUM-FERRIC-= FERROCYANIDE PYRIDOXAL-BENZOYL-= HYDRAZONE PYRIDOXAL-= ISONICOTINOYL-= HYDRAZONE RHODOTORULATE RISEDRONATE SALICYLHYDROXAMATE SUCCIMER-DIETHYL TACHPYRIDINE TETRAMETHYLCYCLEN TETRATHIOMOLYBDATE THIOSALICYLATE TILUDRONATE TIRON TRIENTINE TRITHIOMOLYBDATE TTHA VF-233 ZINC-ETHYLMALTOL ZOLEDRONATE CHEMOKINE-RECEPTOR CXC-RECEPTOR CHOLAGOGUES AC-3092 ACETYLEUGENOL ALIBENDOL ANETHOLTRITHION ANETHOLTRITHIONE AZINTAMIDE BENZPYRINIUM BROMIDE BETAINE (Drug) BOLDINE C-29 CAPILLARTEMISIN-A CAPILLARTEMISIN-B CHENODEOXYCHOLATE CHOLATE CICLOXILATE CICROTOATE CIMEPANOL CINAMETATE CLANOBUTIN CLORINDANATE CYCLOBUTOATE CYCLOBUTYROL CYCLOHEXANE-= CARBOXYLATE CYCLOVALONE CYNARINE DA-1627 DEHYDROCHOLATE DEOXYCHOLATE DIBUPROL DIHYDROXYACETO= PHENONE-2,6 DIHYDROXYBUTYLETHER DIHYDROXYDIBUTYLETHER DIISOPROMINE DIMECROTATE EPOMEDIOL EXIPROBEN FEBUPROL FECLEMINE FELOGEN FENAFTATE FENCIBUTIROL FENIPENTOL FENOCINOL FEPENTOLATE FLAMIN FLORANTYRONE FLUOROURSODEOXY= CHOLATE-6-ALPHA GINGEROL-10 GLYCOURSODEOXYCHOLATE HEXACYPRONE HYDROXYACETOPHENONE-2 HYMECROMONE HYODEOXYCHOLATE ISOFRAXIDIN K-2234 LITHOCHOLATE-= GLUCURONIDE-3 MALOTILATE MENBUTONE METHONAPHTHONE SODIUM METHYLCHENODEOXY= CHOLATE-7-BETA METHYLCHOLATE-7-BETA METOCHALCONE MOQUIZONE NAFCAPROATE NICOTINYLMETHYLAMIDE NIKOMETAMIDE NORCHOLATE NORURSODEOXYCHOLATE

1120 APPENDIX D OSALMID OXAZORONE PIPROZOLIN PROZAPINE REGACHOLYL ROWACHOL SARCOURSODEOXYCHOLATE SC-2644 SF-482 TAUROCHENODEOXYCHOLATE TAURODEHYDROCHOLATE TAUROGLYCOCHOLATE TAUROHYOCHOLATE TAUROHYODEOXYCHOLATE TAUROURSOCHOLATE TAUROURSODEOXYCHOLATE TERBUPROL TOCAMPHYL TREPIBUTONE TRIXOLANE URSOCHOLATE URSODEOXYCHOLATE URSODEOXYCHOLATE-= GLUCURONIDE-3 URSULCHOLATE VANITIOLIDE CHOLINESTERASEREACTIVATORS BDB-106 BDB-108 BDB-27 BDB-37 BDB-91 CARBOXIME DEV-10 DEV-9 DIACETYL-MONOXIME DIETHYXIME HGA-1 HGG-12 HGG-21 HGG-42 HGG-52 HGG-65 HGG-70 HI-6 HI-7 HLOE-7 HS-12 HS-14 HS-3 HS-6 ICD-467 ISONITROSINE MMB-4 OBIDOXIME CHLORIDE P-65 PRALIDOXIME IODIDE PRALIDOXIME MESILATE PYRIMIDOXIME R-665 SAD-128 TRIMEDOXIME BROMIDE CHOREA BERGERON-DISEASE BRISSAUD-SYNDROME DUBINI-DISEASE CHORIOCARCINOMA JEG3-CELL CHROMATOGRAPHY ELECTROCHROMATOGRAPHY GEL-FILTRATION GEL-PERMEATION GLC HPLC TLC CHROMOSOME CHROMATID CHYMOTRYPSIN-INHIBITORS BOWMAN-BIRK-INHIBITOR CHYMOSTATIN OSCILLAMIDE-Y POLYACRYLATE CIRRHOSIS chron.congestive-= splenomegaly CLIMATE SEASON WEATHER CLIN.TRIAL BLIND-TEST PHASE-I PHASE-II PHASE-III PHASE-IV CLOTTING-FACTOR-VIII VON-WILLEBRAND-FACTOR CLOTTING-FACTOR-XAINHIBITORS BX-807834 DPC-423 FXV-673 RPR-128515 RPR-208707 SK-549 SN-292 SN-602 COCAINE-ANTAGONISTS 1-RV-96-A COCCIDIOSTATICS ABIERIXIN AKLOMIDE AMPROLIUM AMQUINATE ARPRINOCID BAYG-7183 BCR-4 BECLOTIAMINE BITIPAZONE BOROMYCIN BUQUINOLATE CIPROQUINATE CLAZURIL CLIRAMIN CLOPIDOL COCCICOL CP-25415 CP-30542 CP-53607 CP-82009 CP-84657 DACIGAL DECOQUINATE DIAVERIDINE DICLAZURIL DIMETHIALIUM DINSED DIOLMYCIN-A1 DUOKVIN EFLORNITHINE FARMCOCCSID FRENOLICIN-B GLYCARBYLAMIDE GRISEOCHELIN HALOFUGINONE IRAMINE ISOLASALOCID-A KISIMICIN KLIRAMIN-20 L-628914 LASALOCID LASALOCID-A LASALOCID-B LASALOCID-C LASALOCID-D LASALOCID-E LY-303366 MADURAMICIN MADURAMICIN-ALPHA MESULFAMIDE METHYLDINITROBENZAMIDE MIKS-10 MIKS-9 MONENSIN MOYUKAMYCIN NARASIN NEQUINATE NICARBAZIN NITROMIDE NITROPHENIDE ORMETOPRIM PORTMICIN POSACONAZOLE PROQUINOLATE ROBENIDINE SALINOMYCIN SEMDURAMICIN SULAZURIL SULFACLOZINE SULFAMETROLE SULFAQUINOXALINE TIAZURIL TOLTRAZURIL TOSULUR VORICONAZOLE WS-5995A WS-5995B WS-5995C X-14868A X-14868B X-14868C X-14868D X-14885A XANTHOQUINODIN-A1 XANTHOQUINODIN-A2 XANTHOQUINODIN-A3 XANTHOQUINODIN-B1 XANTHOQUINODIN-B2 ZINCOPHORIN COENZYME ACETYL-COA COA COLLAGENASE-INHIBITORS ACETYLCYSTEINE CIPEMASTAT DOXYCYCLINE FUTOENONE GM-6001 GW-4459 HYDROXYACECLOFENAC-4 MINOCYCLINE PRINOMASTAT RHEIN RIFAMPICIN RIFAMYCIN RIFAMYCIN-B TENIDAP TIAPROFENATE TRANSFORMING-GROWTH-= FACTOR-BETA-1 VANADATE COLLAGENOSIS DERMATOMYOSITIS

Derwent Drug File 1121 Thesaurus ELASTOSIS localized-scleroderma LUPUS-ERYTH. morphea POLYARTERITIS-NODOSA SCLEREDEMA SCLERODERMA SCLEROMYXEDEMA SHARP-SYNDROME SICCA-SYNDROME SJOEGREN-SYNDROME sle systemic-lupus-eryth. THIBIERGE-WEISSENBACH-= SYNDROME COLLOID HYDROCOLLOID COLON CC531 CT26 HCT116 COMB. CYTOSTATIC-COMB. COMPATIBILITY INCOMPATIBILITY COMPLEMENT ALTERNATIVE-PATHWAY ANAPHYLATOXIN C1-ESTERASE C1-ESTERASE-INHIBITOR = (endogenous) COMPLEMENT-C1Q COMPLEMENT-C1R COMPLEMENT-C1S COMPLEMENT-C2 COMPLEMENT-C3 COMPLEMENT-C3A COMPLEMENT-C3B COMPLEMENT-C3B-= INACTIVATOR COMPLEMENT-C3C COMPLEMENT-C3D COMPLEMENT-C4 COMPLEMENT-C4B COMPLEMENT-C4D COMPLEMENT-C5 COMPLEMENT-C5A COMPLEMENT-C5A-DE-ARG COMPLEMENT-C6 COMPLEMENT-C7 COMPLEMENT-C9 FACTOR-B COMPLEX ALUMINUM-COMPLEX ANTIMONY-COMPLEX BARIUM-COMPLEX BERYLLIUM-COMPLEX BISMUTH-COMPLEX BORON-COMPLEX CADMIUM-COMPLEX CALCIUM-COMPLEX CESIUM-COMPLEX CHROMIUM-COMPLEX CLATHRATE COBALT-COMPLEX COPPER-COMPLEX DYSPROSIUM-COMPLEX EUROPIUM-COMPLEX GADOLINIUM-COMPLEX GALLIUM-COMPLEX GOLD-COMPLEX HAFNIUM-COMPLEX HOLMIUM-COMPLEX INDIUM-COMPLEX IODINE-COMPLEX IRIDIUM-COMPLEX IRIDIUM-COMPLEX IRON-COMPLEX LANTHANUM-COMPLEX LEAD-COMPLEX LITHIUM-COMPLEX MAGNESIUM-COMPLEX MANGANESE-COMPLEX MERCURY-COMPLEX MOLYBDENUM-COMPLEX NEODYMIUM-COMPLEX NICKEL-COMPLEX OSMIUM-COMPLEX PALLADIUM-COMPLEX PLATINUM-COMPLEX POTASSIUM-COMPLEX PRASEODYMIUM-COMPLEX RHENIUM-COMPLEX RHODIUM-COMPLEX RUBIDIUM-COMPLEX RUTHENIUM-COMPLEX SCANDIUM-COMPLEX SILVER-COMPLEX SODIUM-COMPLEX STRONTIUM-COMPLEX TECHNETIUM-COMPLEX TELLURIUM-COMPLEX TERBIUM-COMPLEX THORIUM-COMPLEX THULIUM-COMPLEX TIN-COMPLEX TITANIUM-COMPLEX TUNGSTEN-COMPLEX URANIUM-COMPLEX VANADIUM-COMPLEX YTTERBIUM-COMPLEX YTTRIUM-COMPLEX ZINC-COMPLEX ZIRCONIUM-COMPLEX CONDITIONED-REFLEX CONDITIONED-AVOIDANCE CONGENITAL-DISEASE ACHONDROPLASIA ACROCEPHALOSYNDACTYLY ADACTYLIA ADRENOGENITAL-SYNDROME ADRENOLEUKODYSTROPHY AKABANE-DISEASE ALBINISM ALKAPTONURIA ANGIOHEMOPHILIA ANGIOSTEOHYPER= TROPHIC-SYNDROME ANORCHIDISM AORTIC-ARCH-ANOMALY ARTHROGRYPOSIS ATAXIA-TELANGIECTASIA ATRESIA BARTENWERFER-SYNDROME BECKWITH-SYNDROME BLOCH-SULZBERGER-= SYNDROME BLOOM-SYNDROME BONNEVIE-ULLRICH-= SYNDROME BRACHYDACTYLIA BRACHYGNATHIA buerger-grutz-syndrome caffey-silverman-syndrome CAPDEPONT-SYNDROME CARDIOAUDITORY-= SYNDROME CEPHALOSYNDACTYLIA cerebral-gigantism charcot-marie-tooth-= syndrome CHEDIAK-HIGASHI-= SYNDROME CHILAIDITI-SYNDROME christ-siemens-touraine-= syndrome chron.hereditary-= lymphedema COCKAYNE-SYNDROME COLOBOMA congenital-adrenal-= hyperplasia congenital-aplastic-anemia congenital-arthromyo= dysplasia congenital-chorea congenital-dyskeratosis congenital-hypoplastic-= anemia congenital-hypotrichosis congenital-megacolon congenital-musc.dystrophy CONRADI-HUNERMAN-= SYNDROME COPROPORPHYRIA CRANIOSCHISIS CRETINISM crigler-najjar-disease CROSBY-SYNDROME CROUZON-SYNDROME CURSCHMANN-BATTEN-= STEINERT-SYNDROME CYSTIC-FIBROSIS CYSTINURIA DACRYOCYSTOCELE DANDY-WALKER-SYNDROME DE-LANGE-SYNDROME DE-SANCTIS-CACCHIONE-= SYNDROME DE-VRIES-SYNDROME debler-syndrome diamond-blackfan-anemia DIGEORGE-SYNDROME disseminated-= lipogranulomatosis DOLLINGER-= BIELSCHOWSKY-= SYNDROME DUBOVITZ-SYNDROME DURAND-ZUNIN-SYNDROME DYSAUTONOMIA DYSCHONDROSTEOSIS DYSRAPHIA DZIERZYNSKY-SYNDROME EBSTEIN-ANOMALY ECKLIN-SYNDROME ECTODERMAL-DYSPLASIA EHLERS-DANLOS-SYNDROME EISENMENGER-SYNDROME ELLIS-VAN-CREVELD-= SYNDROME EPIDERMOLYSIS-BULLOSA ERYTHROKERATODERMIA-= VARIABILIS EXENCEPHALY FABRY-SYNDROME familial-benign-pemphigus familial-dysautonomia familial-hemolytic-anemia familial-hyperlipoproteinemia familial-nonhemolytic-icterus familial-periodic-paralysis familial-spastic-paraplegia FANCONI-ALBERTINI-= ZELLWEGER-SYNDROME fanconi-disease FANCONI-PETRASSI-= SYNDROME

1122 APPENDIX D FANCONI-SCHLESINGER-= SYNDROME FANCONI-SYNDROME farber-syndrome FISCHER-SYNDROME FOESTER-SYNDROME FOX-DISEASE FRANCOIS-SYNDROME FRIEDREICH-ATAXIA FRUCTOSE-INTOLERANCE FUCOSIDOSIS GALACTOSEMIA GARDNER-SYNDROME GILBERT-DREYFUS-= SYNDROME GILBERT-SYNDROME glanzmann-disease GLOBOID-CELL-= LEUKODYSTROPHY GLUTARIC-ACIDURIA GORDAN-OVERSTREET-= SYNDROME GOTTRON-SYNDROME GREIG-SYNDROME guerin-stern-syndrome GUNN-SYNDROME hailey-hailey-disease HALLERVORDEN-SPATZ-= SYNDROME HARELIP HARTNUP-DISEASE HELLER-NELSON-SYNDROME HEMIMELIA HEMOGLOBINOPATHY HEMOLYTIC-DISEASE-OF-= NEONATE HEMOPHILIA HEMOPHILIA-B hepatorenal-glycogenosis hereditary-ectodermal-= dysplasia hereditary-hem.telangiectasia hereditary-thrombasthenia hereditary-thrombopathy HERMANSKY-PUDLACK-= SYNDROME HERTWIG-WEYERSSYNDROME hirschprung-disease HISTIDINEMIA HOLT-ORAM-SYNDROME HORSESHOE-KIDNEY HUNTER-SYNDROME huntington-chorea HURLER-SYNDROME HYPERARGININEMIA HYPERPHOSPHATASIA idiopathic-osteopsathyrosis infantile-cortical-hyperostosis JOSEPH-DISEASE KALLMANN-SYNDROME KLEIN-WAARDENBURG-= SYNDROME KLINEFELTER-SYNDROME KLIPPEL-FEIL-SYNDROME KUFS-DISEASE KUGEL-STOLOF-SYNDROME LAURENCE-MOON-BIEDL-= SYNDROME LEBER-DISEASE LEPRECHAUNISM LESCH-NYHAN-SYNDROME LITTLE-DISEASE lobstein-syndrome MAL-DE-MELEDA MANNOSIDOSIS MAPLE-SYRUP-DISEASE MARCHESANI-SYNDROME MARFAN-SYNDROME maroteaux-lamy-syndrome MARTIN-BELL-SYNDROME MELKERSSON-ROSENTHAL-= SYNDROME MENKES-SYNDROME METACHROMATIC-= LEUKODYSTROPHY METHYLMALONICACIDEMIA METHYLMALONICACIDURIA MICROCEPHALY MICROGNATHIA MICROMELIA MICROPHTHALMUS MICROSTOMIA MONGOLISM MONILETHRIX MONOSOMY-7 MORQUIO-DISEASE MOSAICISM MULT.NEUROFIBROMA MYOTONIC-DYSTROPHY NAEGELI-SYNDROME NEUROFIBROMATOSIS neuropathic-musc.atrophy NEZELOF-SYNDROME NIEMANN-PICK-DISEASE NIEVERGELT-SYNDROME nonne-milroy-meige-= syndrome NOONAN-SYNDROME OCULOCEREBRORENAL-= SYNDROME OCULOMANDIBULOFACIAL-= SYNDROME OESTERREICHER-TURNER-= SYNDROME OLIGODACTYLIA OPHTHALMORRHEXIS OROTIC-ACIDURIA osler-syndrome OSTEOPETROSIS OSTEOPSATHYROSIS PAPILLON-LEFEVRE-= SYNDROME PARAHEMOPHILIA PATAU-SYNDROME PATENT-DUCTUS-= ARTERIOSUS PATENT-FORAMEN-OVALE PELGER-HUEET-ANOMALY PENDRED-SYNDROME PEUTZ-JEGHER-SYNDROME PHENYLKETONURIA PHOCOMELIA PIERRE-ROBIN-SYNDROME POLYDACTYLISM polydystrophic-dwarfism POLYSOMIA PORENCEPHALY POROKERATOSIS POTTER-DISEASE PRADER-WILLI-SYNDROME PREMATURE-SENILITY-= SYNDROME prim.familial-xanthomatosis progressive-familial-= myoclonic-epilepsy PSEUDOHYPOALDO= STERONISM PSEUDOHYPOPARA= THYROIDISM PSEUDOPSEUDOHYPO= PARATHYROIDISM pure-red-cell-aplasia RECURRENT-POLYSEROSITIS red-cell-aplasia,pure REFSUM-DISEASE REIFENSTEIN-SYNDROME RETICULAR-DYSGENESIS RICHNER-HANHART-= SYNDROME riley-day-syndrome ROTHMUND-SYNDROME ROUSSY-LEVI-SYNDROME RUBINSTEIN-TAYBI-= SYNDROME RUNDLES-FALLS-SYNDROME RUSSELL-SILVER-SYNDROME RUVACALBA-MYHRE-= SMITH-SYNDROME SANDHOFFS-DISEASE SANFILIPPO-SYNDROME schaefer-syndrome SCHEIE-SYNDROME sickle-cell-anemia SITUS-INVERSUS SJOEGREN-LARSSON-= SYNDROME soto-syndrome SPANLANG-TAPPEINER-= SYNDROME SPIELMEYER-SJOEGREN-= DISEASE SPINA-BIFIDA SPLENIC-AGENESIS-= SYNDROME SPONGE-KIDNEY struempell-lorrain-disease STURGE-WEBER-SYNDROME TANGIER-DISEASE TAUSSIG-BING-SYNDROME TAY-SACHS-DISEASE TETRALOGY-OF-FALLOT thomsen-disease THYMIC-ALYMPHOPLASIA TREACHER-COLLINS-= SYNDROME TREMBLING-DISEASE TRISOMY-16-18 trisomy-21 TRISOMY-4 TRISOMY-8 TUBEROUS-SCLEROSIS TURNER-SYNDROME ULLRICH-SYNDROME unna-syndrome unverricht-disease vogt-syndrome von-gierke-syndrome von-willebrand-disease WERNER-SYNDROME westphal-syndrome WEYER-SYNDROME willebrand-juergen-disease WILLIAMS-BEUREN-= SYNDROME WILSON-DISEASE WISKOTT-ALDRICH-= SYNDROME wolman-disease zinsser-engman-cole-= syndrome CONJUGATE ICI-D-0490 CONN.TISSUE ELASTIC-FIBERS ENDOMYSIUM EPIMYSIUM FASCIA MESENCHYMA PERINEURIUM CONTAINER AMPULE BOTTLE BOX

Derwent Drug File 1123 Thesaurus CLOSURE VIAL CONTRACEPTIVE SPERMATOCIDE CONTRACEPTIVES 70026 ACACIASIDE-A ACACIASIDE-B ACETOMEPREGENOL AF-1312-TS ALGESTONE-ACETOPHENIDE ALKYLOXYNOL-741 ANORDIOL ANORDRIN ANTIDE AZASTEN BDH-2700 CDRI-84-35 CDRI-85-287 CDRI-86-333 CDRI-88-495 CELLULOSE-SULFATE CENTCHROMANE CHLOROHYDRIN-ALPHA CHLOROLACTALDEHYDE-3 CI-680 DIENOGEST DL-111-IT DL-204-IT EPOSTANE ETHYLNORGESTRIENONE F-6103 FERTILYSIN FRAXINELLONE GESTRINONE GOSSYPOL GOSSYPOL-ACETATE GOSSYPOLONE H-1067 H-1075 H-1076 H-774 HIPPADINE J-96 LEVONORGESTREL-ACETATE LEVONORGESTREL-= BUTYRATE LEVONORGESTREL-= CAPROATE LEVONORGESTREL-= CYCLOBUTANOATE LEVONORGESTREL-= CYCLOHEXANOATE LEVONORGESTREL-= CYCLOPENTANOATE LEVONORGESTREL-= CYCLOPROPANOATE LEVONORGESTREL-= PENTANOATE LEVONORGESTREL-= PROPIONATE LILOPRISTONE LONIDAMINE LOTRIFEN LY-317236 MENFEGOL METALLIBURE MIFEPRISTONE NAFOXIDINE NANDROLONE-HEXYLOXY= PHENYLPROPIONATE NIM-76 NISTERIME NISTERIME-ACETATE NITROMIFENE NONOXINOL NONOXINOL-10 NONOXINOL-11 NONOXINOL-15 NONOXINOL-20 NONOXINOL-30 NONOXINOL-4 NONOXINOL-40 NONOXINOL-5 NONOXINOL-6 NONOXINOL-9 NORELGESTROMIN NORETHISTERONE-= ACETATE-OXIME NORETHISTERONE-BENZOATE NORETHISTERONE-= ENANTHATE NORETHISTERONE-OXIME-3 NORETHISTERONE-= PHENYLACETATE OCTOXINOL-9 ONAPRISTONE ORF-13811 ORF-13904 PENTARANE-B PSEUDOLARATE-A PSEUDOLARATE-B QUADROSILAN RMI-12936 RS-37367 SCH-10015 SP-562 SP-563 SP-564 SPERMATOCIDES ST-1435 STYRENE-MALEIC-= ANHYDRIDE-POLYMER SU-13320 TETRADECYLSULFATE = SODIUM TOLNIDAMINE U-11634 U-15646 VICOLIDE-B VICOLIDE-D WHI-07 WIN-18446 XINIDAMINE YUEHCHUKENE ZOAPATANOL CONVULSANTS ALLYLGLYCINE AMINOPHOSPHONO= CAPROATE BRUCINE BUTYLBICYCLOPHOSPHORO= THIONATE-TERT CHEB CORIAMYRTIN DENDROBINE FG-7106 FG-7142 FLUROTYL FUMITREMORGIN-A H-13-04 LON-954 MERCAPTOPROPIONATE OXOTREMORINE PENTETRAZOL PN-309 RO-5-3663 RU-5135 SECURININE STRYCHNINE TETRAMETHYLSUCCINIMIDE TREMORINE TUTIN VIROSECURININE ZK-90798 CORONARY-DISEASE ANGINA-PECTORIS DRESSLER-SYNDROME MYOCARD.INFARCT. VASOSPASM CORONAVIRUS CAT-ENTERIC-CORONAVIRUS EVD-VIRUS HEMAGGLUTINATING-= ENCEPHALOMYELITIS-= VIRUS INFECTIOUS-BRONCHITIS-= VIRUS INFECTIOUS-PERITONITIS-= VIRUS MOUSE-HEPATITIS-VIRUS SIALODACRYOADENITIS-= VIRUS TGE-VIRUS TRANSMISSIBLE-ENTERITIS-= VIRUS CORTICOLIBERIN-AGONISTS CORTICOLIBERIN CORTICOLIBERIN-CATTLE CORTICOLIBERIN-HUMAN CORTICOLIBERIN-SHEEP UROCORTIN CORTICOLIBERINANTAGONISTS ANTALARMIN ANTISAUVAGINE-30 ASTRESSIN CORTICOLIBERIN-12-41,D-PHE CORTICOLIBERIN-9-41 CP-154526 CRA-1000 CRA-1001 SC-241 SD-357 SP-904 CORTICOSTEROIDANTAGONISTS AMINOCHOLESTEROL-22-= ALPHA AMINOCHOLESTEROL-22-= BETA AMINOGLUTETHIMIDE CYANOKETONE DDE DDT DDT-ORTHO-PARA DECYLROXIBOLONE KETOCONAZOLE METYRAPONE MIFEPRISTONE MITOTANE ONAPRISTONE ROXIBOLONE RU-25055 RU-25593 SKF-12185 SKF-12185-D SOLIDAGENONE SU-8000 TRILOSTANE U-30870 CORTICOSTEROIDS ACETOXYPREGNENOLONE-= 21 ACROCINONIDE ALCLOMETASONE ALCLOMETASONE-= DIPROPIONATE ALGESTONE

1124 APPENDIX D ALGESTONE-ACETONIDE AMCINAFAL AMCINAFIDE AMCINONIDE AZACORT BECLOMETASONE BECLOMETASONE-= DIPROPIONATE BECLOMETASONE-= PROPIONATE-17 BECLOMETASONE-= PROPIONATE-21 BETAMETHASONE BETAMETHASONE-ACETATE BETAMETHASONE-ACIBUTATE BETAMETHASONEADAMANTOATE BETAMETHASONE-BENZOATE BETAMETHASONE-= BUTYRATE-17 BETAMETHASONE-= BUTYRATE-21 BETAMETHASONE-= DIPROPIONATE BETAMETHASONE-= DIVALERATE-17,21 BETAMETHASONE-= ISOBUTYRATE-17 BETAMETHASONE-= PHOSPHATE SODIUM BETAMETHASONE-= PROPIONATE-21 BETAMETHASONE-VALERATE BETAMETHASONE-= VALERATE-21 BUDESONIDE CCD-3693 CHLOROPREDNISONE CHLOROPREDNISONE-= ACETATE CICLESONIDE CICORTONIDE CIPROCINONIDE CLOBETASOL CLOBETASOL-DIPROPIONATE CLOBETASOL-PROPIONATE CLOBETASONE CLOBETASONE-BUTYRATE CLOBETASONE-PROPIONATE CLOCORTOLONE CLOCORTOLONE-CAPROATE CLOCORTOLONE-PIVALATE CLOPREDNOL CORMETASONE CORMETASONE-ACETATE CORTEXONE-ENANTHATE CORTICOSTERONE CORTICOSTERONE-ACETATE CORTICOSTERONE-= HEMISUCCINATE CORTISONE CORTISONE-ACETATE CORTISONE-ACETATE-17 CORTISONE-BUTYRATE CORTISONE-CAPROATE CORTISONE-HEMISUCCINATE CORTISONE-OCTANOATE CORTISONE-PALMITATE CORTISUZOL CORTIVAZOL CORTODOXONE CORTODOXONE-ACETATE-21 CORTOL-ALPHA DEACETYLDEFLAZACORT DEFLAZACORT DEHYDROCORTICOSTERONE DEOXYHYDROCORTISONE-21 DEPRODONE DEPRODONE-PROPIONATE DESCINOLONE DESONIDE DESOXIMETASONE DEXAMETHASONE DEXAMETHASONE-ACETATE DEXAMETHASONE-= DIPROPIONATE DEXAMETHASONE-= GLUCOSIDE DEXAMETHASONE-= ISONICOTINATE DEXAMETHASONE-= MESILATE-21 DEXAMETHASONE-= PALMITATE DEXAMETHASONE-= PHENYLPROPIONATE DEXAMETHASONE-= PHOSPHATE DEXAMETHASONE-SULFATE DEXAMETHASONE-= SULFOBENZOATE-META DEXAMETHASONE-TEBUTATE DEXAMETHASONE-= TRIMETHYLACETATE DEXAMETHASONE-= TRIOXAUNDECANOATE DEXAMETHASONE-= TRIOXAUNDECANOATE-21 DEXAMETHASONE-VALERATE DICHLORISONE DIFLORASONE DIFLORASONE-DIACETATE DIFLUCORTOLONE DIFLUCORTOLONE-VALERATE DIFLUPREDNATE DIHYDROCORTISOL DIHYDROCORTISOL-20-= ALPHA DIMESONE DOMOPREDNATE DOXIBETASOL DOXIBETASOL-PROPIONATE DROCINONIDE ENDRISONE EPICORTISOL-11 FLUAZACORT FLUCLOROLONE-ACETONIDE FLUDOXYCORTIDE-ACETATE FLUDROCORTISONE FLUDROCORTISONE-ACETATE FLUDROXYCORTIDE FLUMETASONE FLUMETASONE-PIVALATE FLUMOXONIDE FLUNISOLIDE FLUNISOLIDE-ACETATE FLUOCINOLONE FLUOCINOLONE-ACETONIDE FLUOCINONIDE FLUOCORTIN FLUOCORTIN-BUTYL FLUOCORTOLONE FLUOCORTOLONE-CAPROATE FLUOCORTOLONE-PIVALATE FLUOROCORTISONE-9-ALPHA FLUOROMETHOLONE FLUPAMESONE FLUPEROLONE FLUPEROLONE-ACETATE FLUPREDNIDENE FLUPREDNIDENE-ACETATE FLUPREDNISOLONE FLUTICASONE FLUTICASONE-PROPIONATE FORMOCORTAL GT-256729-X HALCINONIDE HALOCORTOLONE HALOMETASONE HALOPREDONE HALOPREDONE-ACETATE HYDRALLOSTANE HYDROCORTAMATE HYDROCORTISONE HYDROCORTISONE-= ACEPONATE HYDROCORTISONE-ACETATE HYDROCORTISONE-= ACETATE-17 HYDROCORTISONE-= BUTEPRATE HYDROCORTISONE-= BUTYRATE HYDROCORTISONE-= BUTYRATE-21 HYDROCORTISONE-= CAPROATE HYDROCORTISONE-= CIPIONATE HYDROCORTISONE-= ENANTHATE HYDROCORTISONE-= HEMISUCCINATE HYDROCORTISONE-= LYSINATE-21 HYDROCORTISONE-= MESILATE-21 HYDROCORTISONE-= OCTANOATE HYDROCORTISONE-= PHOSPHATE SODIUM HYDROCORTISONE-= PROPIONATE HYDROCORTISONEPROPIONATE-17 HYDROCORTISONE-VALERATE HYDROXY= CORTICOSTERONE-18 HYDROXYCORTISOL-18 HYDROXYCORTISOL-6-BETA HYDROXYPREDNISOLONE-= 16-ALPHA HYDROXYPREDNISOLONE-= 6-BETA HYDROXYPREGNENOLONE-= 17 ISOFLUPREDONE ISOFLUPREDONE-ACETATE ISOPREDNIDENE JO-1605 JO-1717 LNF-209 LOTEPREDNOL-ETABONATE MAZIPREDONE MECLORISONE MECLORISONE-DIBUTYRATE MEDRYSONE MEPREDNISONE METHYL-DIHYDRO= PREDNISOLONATE-20-= ALPHA METHYL-DIHYDRO= PREDNISOLONATE-20-BETA METHYLPREDNISOLONE METHYLPREDNISOLONE-= ACEPONATE METHYLPREDNISOLONE-= ACETATE METHYLPREDNISOLONE-= PHOSPHATE METHYLPREDNISOLONE-= PROPIONATE-17 METHYLPREDNISOLONE-= SUCCINATE METHYLPREDNISOLONE-= SULEPTANATE METHYLPREDNISONE-6-= ALPHA

Derwent Drug File 1125 Thesaurus MOMETASONE-FUROATE NAFLOCORT NCX-1015 NCX-1020 NICOCORTONIDE NIVACORTOL OXISOPRED OXOHYDROCORTISONE-18 PARAMETHASONE PARAMETHASONE-ACETATE PJ-91 PREDNAZATE PREDNAZOLE PREDNAZOLINE PREDNISOLAMATE PREDNISOLONATE-METHYL-= ESTER PREDNISOLONE PREDNISOLONE-ACETATE PREDNISOLONE-CAPROATE PREDNISOLONE-ETHYL= CARBONATE-17 PREDNISOLONE-ETHYL= CARBONATE-21 PREDNISOLONE-= FARNESYLATE-21 PREDNISOLONE-META-= SULFOBENZOATE PREDNISOLONE-PALMITATE PREDNISOLONE-PHOSPHATE PREDNISOLONE-PHTHALATE PREDNISOLONE-STEAGLATE PREDNISOLONE-SUCCINATE PREDNISOLONE-TEBUTATE PREDNISOLONE-TETRA= HYDROPHTHALATE PREDNISOLONE-TRIMETHYL= ACETATE PREDNISOLONE-VALERATE-= ACETATE PREDNISONE PREDNISONE-ACETATE PREDNISONE-ACETATE-17 PREDNISONE-= HEMISSUCCINATE PREDNISONE-PHOSPHATE PREDNISONE-VALERATE-17 PREDNYLIDENE PREGNENOLONE PREGNENOLONE-16-= ALPHA-CARBONITRILE PREGNENOLONE-ACETATE PREGNENOLONE-SULFATE PROCINONIDE PROMESTRIENE RIMEXOLONE RPR-106541 RU-26988 RU-28362 SH-713 SQ-15361 SQ-28300 SQ-31853 SQ-31854 SQ-31855 TETRAHYDROCORTI= COSTERONE TETRAHYDROCORTISOL TETRAHYDROCORTISONE TIMOBESONE-ACETATE TIPREDANE TIXOCORTOL TIXOCORTOL-BUTYRATE-= 17-PROPIONATE-21 TIXOCORTOL-PIVALATE TRALONIDE TRIAMCINOLONE TRIAMCINOLONE-ACETONIDE TRIAMCINOLONE-= ACETONIDE-PALMITATE-21 TRIAMCINOLONE-= ACETONIDE-PHOSPHATE TRIAMCINOLONE-= BENETONIDE TRIAMCINOLONE-DIACETATE TRIAMCINOLONE-= FURETONIDE TRIAMCINOLONE-= HEXACETONIDE TRICLONIDE U-42129 ULOBETASOL ULOBETASOL-PROPIONATE WIN-44577 CRAMP GRAPHOSPASM CRYSTALLOGRAPHY X-RAY-DIFFRACTION CURARE-ANTAGONISTS EDROPHONIUM CHLORIDE RX-72601 CYCLIN-DEPENDENT-KINASEINHIBITORS BOHEMINE GW-420371-X NSC-521164 NSC-680434 OXINDOLE-I PGJ2-DEOXY-15-DELTA-12,14 CYCLOOXYGENASE-1INHIBITORS ASPIRIN AURANOFIN EPIAFZELECHIN IBUPROFEN INDOMETACIN MOFEZOLAC NEPAFENAC NORARTOCARPANONE OSTHENOL SC-560 SC-58560 SOPHORAFLAVONE-G CYCLOOXYGENASE-2INHIBITORS A-79175 AGNUSIDE AURANOFIN AVICIN-G BRL-10720 CELECOXIB E-6087 ETORICOXIB FLOSULIDE FR-140423 INDOMETACIN KETOPROFEN L-745337 LICOFELONE LUMIRACOXIB M-5011 MELOXICAM MF-TRICYCLIC MK-966 NABUMETONE NCX-701 NIMESULIDE NITROACETYLSALICYLATE NS-398 PARADOL-8 PARECOXIB PD-164387 ROFECOXIB SC-299 SC-57666 SC-58125 SC-58236 SP-600125 TP-151 TRICHODION UR-8880 VALDECOXIB CYCLOOXYGENASE-INHIBITOR CYCLOOXYGENASE-1-= INHIBITOR CYCLOOXYGENASE-2-= INHIBITOR CYCLOOXYGENASEINHIBITORS A-79175 ACECLOFENAC AGNUSIDE AMENTOFLAVONE ASPIRIN AURANOFIN AVICIN-G BRL-10720 BUDDLEDIN-A CELECOXIB CYCLOOXYGENASE-1-= INHIBITORS CYCLOOXYGENASE-2-= INHIBITORS E-6087 EPIAFZELECHIN ETORICOXIB FLOSULIDE FLURBIPROFEN FR-123826 FR-140423 HCT-3012 IBUPROFEN INDOMETACIN KETOPROFEN L-745337 LAGASCATRIOL LICOFELONE LUMIRACOXIB M-5011 MECLOFENAMATE MELOXICAM MF-TRICYCLIC MK-966 MOFEZOLAC NABUMETONE NCX-701 NEPAFENAC NIMESULIDE NITROACETYLSALICYLATE NORARTOCARPANONE NS-398 OSTHENOL PARADOL-8 PARECOXIB PD-164387 PIROXICAM ROFECOXIB RUTECARPINE SC-299 SC-560 SC-57666 SC-58125 SC-58236 SC-58560 SOPHORAFLAVONE-G SP-600125 TEPOXALIN TP-151 TRICHODION

1126 APPENDIX D UR-8880 VALDECOXIB CYTOCHROME P-450 P-452 P-488 CYTOLOGY CELL-CYCLE MEIOSIS METAPHASE MITOSIS PROPHASE TELOPHASE CYTOSTATICS 101-M 1031-U-89 1396-U-88 1400-W 1843U89 1944-U-88 2-12362 253-152 254-S 261-96 272-131 428-U-89 502-U-83 502U83 506-U 543-U-76 593-A 773-U-82 A-007 A-137 A-145 A-151011 A-191 A-192 A-195 A-204197 A-3-P-166 A-4-P-73 A-62176 A-748 A-74932 A-80198 A-85226 A-91 A-924 AB-163 ABARELIX ABIRATERONE ABMFPP ABRIN ABRIN-A-CHAIN ABT-510 ABT-526 AC-3579 AC-394 AC-7700 AC-7739 ACADESINE ACALYCIXENIOLIDE-A ACALYCIXENIOLIDE-B ACEGLATONE ACETALDOPHOSPHAMIDE ACETAMIDOBENZAMIDE-3 ACETOMYCIN ACETOXYCYCLOHEXIMIDE ACETYLDAUNORUBICIN-N ACETYLDISCODERMOLIDE-7 ACETYLDOPA-N ACETYLDOPAMINE-N ACETYLDOXORUBICIN-N ACETYLGONIOTRIOL-8 ACETYLMELODORINOL ACETYLMELPHALAN-N ACETYLPANAXYDOL ACETYLPHOMALACTONE ACETYLSHIKONIN ACICULATIN ACITRETIN ACIVICIN ACLACINOMYCIN ACLACINOMYCIN-B ACLACINOMYCIN-S ACLACINOMYCIN-T ACLARUBICIN ACODAZOLE ACRONINE ACTINOMYCIN-C2 ACTINOMYCIN-C3 ACTINOMYCIN-D ACTINOMYCIN-K2T ACTINOMYCIN-V ACTINOMYCIN-Z5 ACTINOPLANONE-A ACTINOPYRONE-A ACTIVIN-A ACUTISSIMIN-A ACYCLORETINOATE AD-143 AD-194 AD-198 AD-199 AD-20 AD-202 AD-280 AD-284 AD-285 AD-288 AD-312 AD-32 ADA-202-718 ADAPHOSTIN ADENOPTERIN ADENOSINE-DIALDEHYDE ADOZELESIN AE-941 AEROPLYSININ-1 AG-1112 AG-14031 AG-1517 AG-2 AG-2034 AG-2037 AG-331 AG-3340 AG-337 AG-377 AG-394 AG-494 AG-514 AG-538 AG-556 AG-568 AG-775 AG-85 AG-879 AG-879 AG-952 AG-957 AGELASIMINE-A AGELASIMINE-B AGELASPHIN-11 AGELASPHIN-13 AGELASPHIN-7A AGELASPHIN-9A AGELASPHIN-9B AGELASTATIN-A AGL-1872 AGL-517 AGLAFOLINE AGOSTEROL-A AGROSTISTACHIN AICA AICA-RIBOTIDE AILANTHINONE AIMFPP AJULEMATE AKLAVIN AKROBOMYCIN ALALON ALANINE-MUSTARD ALANOSINE ALAZOPEPTIN ALBOMITOMYCIN-A ALBONOURSIN ALCINDOROMYCIN ALDOIFOSFAMIDE ALDOPHOSPHAMIDE ALISAMYCIN ALLAMANDIN ALLAMCIN ALLDIMYCIN-A ALLIACOLIDE ALLOCOLCHICINE ALLYL-MERCAPTAN ALLYL-METHYL-DISULFIDE ALLYL-METHYL-TRISULFIDE ALRT-1550 ALSTERPAULLONE ALTEMICIDIN ALTHOLACTONE ALTOHYRTIN-B ALTOHYRTIN-C ALTRETAMINE ALTROMYCIN-A ALTROMYCIN-D ALTROMYCIN-H ALTROMYCIN-I AM-132 AM-555-S AMAMISTATIN-A AMAMISTATIN-B AMBROSIN AMETANTRONE AMETOHEPASONE AMIDOX AMINO-ANFOL AMINOALANFOL AMINOCAMPTOTHECIN-9 AMINOCHLORAMBUCIL AMINOELLIPTICINE-9 AMINOGELDANAMYCIN-17 AMINOGLUTETHIMIDE AMINOPTERIN AMINOPTERIN SODIUM AMONAFIDE AMONAFIDE-ACETYL-N AMORPHISPIRONONE AMPHETHINILE AMPHIDINOLIDE-A AMPHIDINOLIDE-B AMPHIDINOLIDE-C AMPHIDINOLIDE-D AMPHIDINOLIDE-J AMPHIDINOLIDE-K AMPHIMEDINE AMPHIREGULIN AMRUBICIN AMSACRINE AMSALOG AMYGDALIN AN-152 AN-201I AN-201II AN-207 AN-215 AN-238

Derwent Drug File 1127 Thesaurus AN-9 ANASTROZOLE ANAXIRONE ANCITABINE ANFOL-R ANGELMICIN-B ANGINEX ANGIOSTATIN ANGIOZYME ANGOLENSATE-METHYL ANGUIDIN ANHYDROVINBLASTINE ANILINE-MUSTARD ANISOMELATE ANKINOMYCIN ANNAMYCIN ANNOMONTACIN ANNONACIN ANNONACINONE ANNORETICUINONE-9 ANOLIGNAN-A ANSAMITOCIN-P3 ANTAGONIST-G ANTINEOPLASTON-A10 ANTINEOPLASTON-A2 ANTINEOPLASTON-A3 ANTINEOPLASTON-A5 ANTINEOPLASTON-AS2-1 ANTINEOPLASTON-AS2-5 AP-5280 APHE-1 APHE-2 APHIDICOLINE-GLYCINATE APHOLATE APICULAREN-A APLAMINONE APLIDIASPHINGOSINE APLYRONINE-A APLYRONINE-B APLYRONINE-C APLYSIANIN-E APLYSIAPYRANOID-A APLYSIAPYRANOID-D APLYSIATERPENOID-A APLYSISTATIN APLYSISTATIN APOGOSSYPOL APOLIZUMAB APOPICROPODOPHYLLIN-= BETA APOPTOLIDIN AQ4 AQ4N AQUAYAMYCIN ARABINOGALACTAN ARABINOSYLAZACYTOSINE-= TRIPHOSPHATE ARABINOSYLGUANINE ARABINOSYLGUANINE-= TRIPHOSPHATE ARABINOSYLTIOGUANINE ARAGUSTEROL-A ARAGUSTEROL-B ARAGUSTEROL-C ARANCIAMYCIN ARANOROSIN ARANOZA ARBUSCULIN-A ARCTIIN ARDISENONE ARENASTATIN-A ARGENTININE ARGIMESNA ARGINASE ARGININE-DEIMINASE ARGYRIN-B ARIMIDEX ARISTOLACTAM-AII ARISTOLOCHATE-I ARISTOLOCHATE-IA ARISTOLOCHATE-II ARJUNOLATE AROTENOID ARPHAMENINE-A ARPHAMENINE-B ARTEMISITENE ARUGOMYCIN ARVANIL ARZOXIFENE AS-101 ASALEI ASALIN ASAPHAN ASCIDIACYCLAMIDE ASCIDIDEMIN ASCOCHITAL ASCORBATE-DOCOSA= HEXAENOATE-6 ASEBOGENIN ASIMICIN ASITRILOBIN-A ASPARAGAMINE-A ASPARAGINASE ASPARTATE-= HYDROXAMATE-BETA ASPCNU ASPERDIOL ASPERLIN ASTA-5607 ASTA-5783 ASTA-7037 ASTA-Z-7654 ASTERIN ASTERRIQUINONE ASTIN-A ASTIN-B ASTROGORGIADIOL ASTROGORGIN AT-2433-A1 AT-2433-B1 AT-486 AT-760 ATF-H-18 ATHEROSPERMIDINE ATRASENTAN AURISTATIN-PE AUROMOMYCIN AUTUMNOLIDE AVAROL AVARONE AVELLANEOL AVI-4126 AVICIN-D AVICIN-G AW-464 AWAMYCIN AXILLARIN AXISONITRILE-3 AZAADENINE-8 AZAADENOSINE-2 AZAADENOSINE-8 AZACYTIDINE AZACYTIDINE-6 AZAGUANINE AZAHYPOXANTHINE-2 AZAPICYL AZASERINE AZATEPA AZATHIOPRINE AZATOXIN AZAURACIL AZAURIDINE AZB-017 AZEPINOMYCIN AZETOMYCIN-I AZETOMYCIN-II AZIDOCYTIDINE-2+ AZIDOPYRIMETHAMINE-= META AZINOMYCIN-A AZINOMYCIN-B AZIPAC AZOMYCIN AZOPROCARBAZINE AZOTOMYCIN AZOXYPROCARBAZINE B-1086 B-15 B-1600 B-201 B-2844 B-3-243 B-327 B-3839 B-3958 B-3970 B-3995 B-3996 B-4152 B-429 B-581 B-623 (benzothiophene) B-850040 B-956 BA-32248B BACCHARIN BACCHARIN-B4 BACCHARIN-B5 BACCHOTRICUNEATIN-A BACTERIOHOPANOL-32 BACTOBOLIN BAKKENOLIDE-A BAL-9611 BARMINOMYCIN-I BARMINOMYCIN-II BASIDALIN BASTADIN-4 BASTADIN-8 BASTADIN-9 BATIMASTAT BAUMYCIN-B2 BAUMYCIN-C1 BAY-11-7085 BAY-11-7821 BAY-12-9566 BAY-38-3441 BAY-43-9006 BAY-50-4798 BAYER-A139 BB-3103 BBR-2207 BBR-2209 BBR-2378 BBR-2577 BBR-2778 BBR-2828 BBR-2867 BBR-2868 BBR-2894 BBR-3005 BBR-3171 BBR-3390 BBR-3464 BCH-2051 BCH-4556 BCN-326862 BE-10988 BE-12406A BE-12406B BE-14348-B BE-18591 BE-23372-M

1128 APPENDIX D BE-23372M BE-3333 BE-373 BE-4444 BENAXIBINE BENDAMUSTINE BENFLURON BENGAMIDE-A BENGAMIDE-B BENGAMIDE-C BENZAMIDE-RIBOSIDE BENZANTHRIN-A BENZANTHRIN-B BENZODEPA BENZOQUINONE-MUSTARD BENZOTEF BENZYLDAUNORUBICIN-N BENZYLIDENE-ASCORBATE-= 5,6 BENZYLIDENE-D-GLUCOSE-= 4,6 BENZYLSPARSOMYCIN BETACLAMYCIN-A BETATHINE BETULETOL BEVACIZUMAB BFNU BHCNU BIBF-1000 BIBW-022 BILOBOL BIM-26189 BIM-26226 BIM-46174 BIMOLANE BIPINNATIN-A BIPINNATIN-B BIPINNATIN-C BIPINNATIN-C BIPINNATIN-D BISANTRENE BISBRUCEANTINYL-= MALONATE BISBRUCEANTINYL-= SUCCINATE BISBRUSATOLYL-MALONATE BISBRUSATOLYL-SUCCINATE BISNAFIDE BISTHEONELLIDE-A BISTRAMIDE-A BISTRAMIDE-D BISTRATENE-A BISTRATENE-B BISUCABERIN BIZELESIN BIZELESIN BL-269 BL-473 BL-554 BL-562 BL-6783 BLEOMYCIN BLEOMYCIN-A1 BLEOMYCIN-A2 BLEOMYCIN-A5 BLEOMYCIN-B2 BLEOMYCIN-B4 BLEOMYCINATE BM-920700 BMS-180820 BMS-181167 BMS-181681 BMS-182178 BMS-184476 BMS-184481 BMS-185411 BMS-185660 BMS-188797 BMS-191352 BMS-214662 BMS-239091 BMS-247550 BMS-250749 BMS-250904 BMS-275291 BMS-310705 BMY-25067 BMY-25282 BMY-25551 BMY-26107 BMY-26605 BN-52205 BN-52207 BN-52211 BN-80927 BNP-1100 BNP-1350 BNP-7787 BNPI-1100 BOFUMUSTINE BOHEMINE BOLESATINE BONE-MORPHOGENETIC-= PROTEIN-2 BONE-MORPHOGENETIC-= PROTEIN-6 BONELLIN BORNYL-COUMARATE BORNYL-FERULATE BORONOPHENYLALANINE-= PARA BOSWELLATE-ALPHA BOTRYODIPLODIN BOUVARDIN BP-179 BR-1376 BRASILIQUINONE-A BRASSILEXIN BRASSININ BRC-16-HT BREFLATE BREMFOL BREQUINAR SODIUM BROMACRYLIDE BROMEBRATE BROMOACETYLCHOLINE BROMODAUNORUBICIN BROMODEOXYCYTIDINE BROMOFOSFAMIDE BROMOTOPSENTIN BROMOVINYLDEOXY= CYTIDINE BROMOVULONE-I BROPIRIMINE BROSTALLICIN BROXURIDINE BROXURIDINE-= MONOPHOSPHATE BROXURIDINE-TRIPHOSPHATE BRUCEANTIN BRUCEANTINOSIDE-C BRUCEOLIDE BRUCEOSIDE-A BRUCEOSIDE-D BRUSATOL BRYOPHYLLIN-A BRYOSTATIN-1 BRYOSTATIN-10 BRYOSTATIN-11 BRYOSTATIN-12 BRYOSTATIN-13 BRYOSTATIN-2 BRYOSTATIN-3 BRYOSTATIN-4 BRYOSTATIN-5 BRYOSTATIN-6 BRYOSTATIN-7 BRYOSTATIN-8 BRYOSTATIN-9 BS-1 BSU-1051 BT-99-25 BU-3129T BUDOTITANE BULLATACIN BULLATACINONE BULLATALICIN BURSERAN BUSRAMUSTINE BUSULFAN BUTHIOPURINE BUTOCIN BUTYLATED-= HYDROXYTOLUENE BUTYLGUANINE-O-6 BUTYLTHIOPHENE-2 BUTYRYLMALLOTOCHROMENE BW-1069-C-85 BW-1843U89 BW-A-1169U BW-A-1261U BW-A-1454U BW-A-353U BW-A-354U BW-A-424U BW-A-453U BW-A-457U BW-A-502U BW-A-503U BW-A-773U BW-A-822U BW-A-90U BW-A-91U BW-A7U BZA-2-B C-1005 C-1006 C-1020 C-1027 C-1263 C-1310 C-1311 C-1371 C-175 C-176 C-205 C-232 C-257 C-264 C-265 C-308 C-309 C-337 C-338 C-410 C-516 C-609 C-73 C-75 C-829 C-835 C-846 C-849 C-857 C-867 C-878 C-881 C-887 C-921 CACOSPONGIONOLIDE CACTINOMYCIN CADEGUOMYCIN

Derwent Drug File 1129 Thesaurus CAFFEATE-PHENETHYL-ESTER CALCIUM-GLUCARATE CALICHEAMICIN CALICHEAMICIN-ALPHA-2-I CALICHEAMICIN-ALPHA-3-I CALICHEAMICIN-BETA-1-BR CALICHEAMICIN-BETA-1-I CALICHEAMICIN-DELTA-1-I CALICHEAMICIN-GAMMA-1-I CALICHEAMICIN-THETA-I-1 CALLIPELTIN-A CALLYSTATIN-A CALONECTRIN CALOTHRIXIN-A CALPHOSTIN-A CALPHOSTIN-B CALPHOSTIN-C CALPHOSTIN-D CALPHOSTIN-I CALUSTERONE CALYCULIN-A CALYCULIN-B CALYCULIN-C CALYCULIN-D CALYCULINAMIDE-A CALYCULINAMIDE-B CALYXIN-J CALYXIN-K CAM-1481 CAMELLIIN-A CAMELLIIN-B CAMPTOTHECIN CANAVALMINE CANTALASAPONIN-1 CANVENTOL CAP-1 CAP-2 CAPARRATRIENE CAPOAMYCIN CAPSICASTRINE CAPSIMINE CARACEMIDE CARBAZYLQUINONE CARBETIMER CARBOPLATIN CARBOQUONE CARBORANYLDEOXY= URIDINE-2+ CARBOXYPEPTIDASE-G2 CARBOXYPHOSPHAMIDE CARMETHIZOLE CARMINAZONE CARMUSTINE CARNIVORA CARUBICIN CARZELESIN CARZINOPHILIN CASEARIN-A CASEARIN-B CASEARIN-C CASEARIN-D CASEARIN-E CASEARIN-F CASEARIN-G CASEARIN-H CASEARIN-I CASEARIN-J CASEARIN-K CASEARIN-L CASEARIN-M CASEARIN-N CASEARIN-O CASEARIN-P CASEARIN-Q CASEARIN-R CATHARININE CB-10-200 CB-10-252 CB-10-277 CB-10-286 CB-1093 CB-1267 CB-1414 CB-1837 CB-1850 CB-1954 CB-300638 CB-300907 CB-300919 CB-30865 CB-30900 CB-3705 CB-3717 CB-3804 CB-3988 CB-7103 CB-7547 CB-7639 CB-7669 CB-7675 CB-7741 CB-966 CBM-11 CC-1065 CC-313 CC-5013 CCI-779 CCRG-82019 CD-388 CD-86022 CD40-LIGAND CDC-501 CDRI-86-333 CEALYSIN CECROPIN-B CECROPIN-B-1 CECROPIN-P-1 CELLADAM CEP-2563 CEP-5214 CEP-701 CEP-751 CEPHALOCHROMIN CEPHALOSTATIN-1 CEPHALOSTATIN-10 CEPHALOSTATIN-12 CEPHALOSTATIN-2 CEPHALOSTATIN-3 CETUXIMAB CG-8840 CGP-19984 CGP-33829 CGP-35753 CGP-36958 CGP-39937-A CGP-41251 CGP-42700 CGP-4303 CGP-48664 CGP-48664-A CGP-520 CGP-53716 CGP-59326 CGP-60261 CGP-60474 CGP-62706 CGP-645 CGP-6809 CGP-69846-A CGS-18320B CGS-20267 CGX-571 CH-23 CHAETOCHROMIN-A CHAETOGLOBOSIN-K CHAPARRINONE CHARTREUSIN CHETRACIN-A CHICAMYCIN-A CHINESIN-II CHITOHEXAOSE CHLAMYDOCIN CHLORAMBUCIL CHLORAMBUCIL-N-OXIDE CHLORAMBUCIL-T-BUTYL-= ESTER CHLORETHYLAMINOURACIL CHLORIMIDAZINE CHLORIN-E6-IRON CHLORMETHINE CHLORNAPHAZINE CHLOROADENOSINE-2 CHLORODEOXYADENOSINETRIPHOSPHATE CHLORODEOXYCYTIDINE-5 CHLORODEOXYURIDINE-5 CHLOROLISSOCLIMIDE CHLOROMALOSIDE-A CHLOROPHENYLACETATE-= PARA CHLOROQUINOXALINE-= SULFONAMIDE CHLOROTAMOXIFEN-4 CHLOROVULONE-I CHLOROVULONE-II CHLOROVULONE-III CHLOROZOTOCIN CHLORPHENACIL CHLORSULFAQUINOXALINE CHONDRAMIDE-A CHONDRAMIDE-B CHONDRAMIDE-C CHONDRAMIDE-D CHONDRILLIN CHROMIC-PHOSPHATE CHROMODOROLIDE-A CHROMOMYCIN-A3 CHROMOXYMYCIN CHRYMUTASIN-A CHRYMUTASIN-B CHRYMUTASIN-C CHRYSENAMINE CHRYSOMYCIN-A CHRYSOMYCIN-B CHRYSOTRICINE CHS-828 CI-1010 CI-937 CI-958 CI-980 CIBA-21381-BA CICLAMYCIN-0 CICLOSPORIN CICUTOXIN CINERUBIN-A CINERUBIN-B CINNAMODIAL CINNAMTANNIN-B2 CISPLATIN CITROPEPTIN CITRUSININE-II CJM-05 CJM-126 CJS-11 CKD-602 CL-232468 CL-246738 CL-387785 CLADRIBINE CLADRIBINE-= MONOPHOSPHATE CLAENONE

1130 APPENDIX D CLANFENUR CLAVEPICTINE-A CLAVEPICTINE-B CLAVULARIN-A CLAVULARIN-B CLAVULONE CLAVULONE-I CLAVULONE-II CLAVULONE-III CLAVULONE-IV CLAZAMYCIN CLAZAMYCIN-A CLAZAMYCIN-B CLEISTANTHIN-A CLEOMISCOSIN-A CLEROCIDIN CLITOCINE CLOFARABINE CLOFARABINE-TRIPHOSPHATE CLOMESONE CLOTURIN CLUSIPARALICOLINE-A CM-101 CMT-3 CMT-6 CMT-7 CNUA COBRA-1 COCHLEAMYCIN-A COCHLEAMYCIN-A2 COCHLEAMYCIN-B COCHLEAMYCIN-B2 COFORMYCIN COFORMYCINMONOPHOSPHATE COFPLATON COLABOMYCIN-A COLCHICIDE COLCHICINE COLCHICOSIDE COLLINEMYCIN COLLISMYCIN-A COLLISMYCIN-B COLOSOLATE COMBRESTATIN-A4-= PHOSPHATE COMBRETASTATIN COMBRETASTATIN-A-1 COMBRETASTATIN-A-4 COMBRETASTATIN-A2 COMBRETASTATIN-A3 COMBRETASTATIN-B-1 COMBRETASTATIN-B2 COMBRETASTATIN-B3 COMBRETASTATIN-B4 COMBRETASTATIN-D-1 COMBRETASTATIN-D-2 CONOPHYLLINE CONVOLUTAMINE-A COPOVITHANE CORALYNE CORDIACHROMENE-A CORDIAQUINONE-B CORDYCEPIN-N-OXIDE-1 CORIARIIN-A CORIOLIN CORNIGERINE CORNUSIIN-A CORONARIN-A CORONARIN-B CORONARIN-C CORONARIN-D CORONARIN-E COROSSOLIN COROSSOLONE CORTIFEN COSMOCARCIN-A COSMOMYCIN-A COSMOMYCIN-B COSMOMYCIN-C COSMOMYCIN-D COUMAROYLTYRAMINE-N COUMATE CP-115953 CP-115955 CP-127374 CP-248 CP-358774 CP-461 CP-46665-1 CP-547632 CP-67804 CPI-0004 CRAMBESCIDIN-800 CRAMBESCIDIN-816 CRANOMYCIN CRASSIN CRC-680578 CRIBROSTATIN-2 CRISNATOL CRL-8275 CRL-8276 CRL-8277 CRL-8299 CROTEPOXIDE CROTONIN CROTOXIN CRX-103 CRYPTOPHYCIN CRYPTOPHYCIN-52 CRYPTOPHYCIN-55 CRYPTOPHYCIN-8 CRYPTOPHYCIN-A CRYPTOPHYCIN-B CRYPTOPHYCIN-C CRYPTOPHYCIN-D CRYPTOPLEURINE CRYPTOPORATE-A CS-682 CT-052923 CT-17 CT-1746 CT-2103 CT-2106 CT-2251 CT-2583 CT-2584 CT-3501 CTNU-3+ CUBEBIN CUCURBITACIN-B CUCURBITACIN-D CUCURBITACIN-F CUCURBITACIN-Q CUMINGIANOSIDE-A CURACIN-A CURACIN-B CURACIN-C CURCUMENE-ALPHA CURCUPHENOL CURDLAN-CM CURROMYCIN-A CURROMYCIN-B CURVULARIN CV-787 CVT-313 CYANOCINNAMATE-ALPHA CYANOCYCLINE-A CYANOMORPHOLINO= DAUNORUBICIN CYANOPUUPEHENOL-15 CYCLIC-AMP-AMINO-8 CYCLIDISONE CYCLOBRASSININ CYCLOCOMMUNOL CYCLODERCITIN CYCLOHEXANO-15-= CROWN-5 CYCLOLEUCINE CYCLOMULBERRIN CYCLOPHOSPHAMIDE CYCLOPLATAM CYCLOSPORIN-B CYCLOSPORIN-C CYCLOSPORIN-D CYCLOSPORIN-H CYCLOSPORIN-K CYCLOSPORIN-M CYCLOSPORIN-O CYCLOSPORIN-Q CYCLOSPORIN-U CYCLOSPORIN-V CYCLOSPORIN-Z CYCLOXAZOLINE CYLINDROCYCLOPHANE-A CYLINDROCYCLOPHANE-D CYLINDROCYCLOPHANE-F CYNAROPICRIN CYSTAPHOS CYSTAPHOS CYSTEAMINYLPHENOL-4-S CYSTEINYLCATECHOL-3-S CYSTEINYLCATECHOL-4-S CYSTEINYLDOPA-5-S CYSTEINYLPHENOL-4-S CYSTEINYLRESORCINOL-2-S CYSTEMUSTINE CYSTODAMINE CYSTODYTIN-A CYSTODYTIN-B CYSTODYTIN-C CYSTODYTIN-J CYTARABINE CYTARABINE-DIPHOSPHATE CYTARABINE-= DIPHOSPHOCHOLINE CYTARABINE-= MONOPHOSPHATE CYTARABINE-PHOSPHATE-5+ CYTARABINE-= STEARYLPHOSPHATE-5+ CYTARAZID CYTOCHALASINE-B CYTOCHALASINE-F CYTOCHALASINE-J CYTOCHALASINE-N CYTOCHALASINE-O CYTOGENIN CYTORHODIN-A CYTORHODIN-D CYTOROS CYTOSINE-DEAMINASE CYTOSTATIN CZ-112 CZ-48 D-150 D-17872 D-18621 D-18954 D-19575 D-20133 D-21266 D-21805 D-24851 D-435 D-609 D-788-1 DA-125 DACARBAZINE DACLIXIMAB DANIQUIDONE DAPHNETICIN

Derwent Drug File 1131 Thesaurus DAPHNODORIN-B DAPHNORETIN DATELLIPTIUM-CHLORIDE DAUNOFORM DAUNORUBICIN DAUNORUBICIN-CYCLO= HEXYLIDINEHYDRAZONE DAUNORUBICINOL DB-174 DB-67 DC-101 DC-81 DC-92-B DC-92-D DC-TA-46 DDE-131 DEACETOXYOLEPUPUANE-7 DEACETOXYTAXOL-10 DEACETYLGEDUNIN DEACETYLRAVIDOMYCIN DEACETYLTAXOL-10 DEACETYLVINBLASTINE DEACETYLVINCRISTINE DEACYLCYNAROPICRIN DEAMIDOBLEOMYCIN-A2 DEAMIDOBLEOMYCIN-B2 DEAZAADENOSINE-1 DEAZAADENOSINE-9 DEAZAAMINOPTERIN-5 DEAZAAMINOPTERIN-8 DEAZAARISTEROMYCIN-3 DEAZAGUANOSINE-3 DEAZAGUANOSINE-7 DEAZAMETHOTREXATE-5 DEAZAMETHOTREXATE-8 DEAZANEPLANOCIN-3 DEAZATETRAHYDRO= FOLATE-5 DEAZAURIDINE-3 DEBROMOAPLYSIATOXIN DECILORUBICIN DECITABINE DECLOPRAMIDE DEDP DEFOSFAMIDE DEGUELIN DEHYDROALTENUSIN DEHYDROCARBODINE DEHYDROCURVULARIN DEHYDRODIDEMNIN-B DEHYDROISOPATULIN DEHYDROMATRICARIA-ESTER DEHYDROTELOBINE-1,2 DEHYDROXYSPARSOMYCIN DELAMINOMYCIN-A DELAMINOMYCIN-B DELAMINOMYCIN-C DEMECOLCINE DEMETHOXY= FUMITREMORGIN-C DEMETHYLBLEOMYCIN-A2 DEMETHYLCHARTREUSIN-= 3++ DEMETHYL= CHROMOMYCIN-A2 DEMETHYL= CHROMOMYCIN-A3 DEMETHYLDACARBAZINE DEMETHYLDEOXYPODO= PHYLLOTOXIN-4+ DEMETHYLOLIVOMYCIN-A DEMETHYLTHIO= COLCHICINE-3 DEMETHYLTUBULOSINE-9 DENDROAMIDE-A DENOPTERIN DENSICOMACIN DENTICULATOLIDE DEOXOFAVELINE DEOXYAKLAVINONE-7 DEOXYBOUVARDIN DEOXYCARUBICIN-13 DEOXYCARUBICIN-6 DEOXYDAUNORUBICIN-11 DEOXYDAUNORUBICINONE-= 11 DEOXYDOXORUBICIN-13 DEOXYDOXORUBICIN-9 DEOXYEPOTHILONE-A DEOXYEPOTHILONE-B DEOXYEPOTHILONE-F DEOXYFORMYCIN-2+ DEOXYLIMONIN DEOXYNOGAROL-7 DEOXYOXANOSINE-2+ DEOXYPODORHIZON DEOXYSPERGUALIN DEOXYTAXOL-7 DEOXYTAXOTERE-10 DEOXYTHIOGUANOSINE DEOXYTOPSENTIN DEOXYURIDINE-3+ DEOXYVERNOLEPIN DEPHOSPHONOCALYCULIN-A DEPROPYLORYZALIN-N DEPUDECIN DERCITIN DERETICULATIN-TRIACETATE DESMAL DESTRUXIN-B DESTRUXIN-E DETALLIPTINIUM DETORUBICIN DEXTRAN-CM-BENZYLAMIDE DEXTRIN-2-SULFATE DEXVERAPAMIL DEZAGUANINE DF-129 DF-203 DF-209 DF-229 DIACETYLDIANHYDRO= GALACTITOL DIACETYLDISCO= DERMOLIDE-3,7 DIACETYLPUTRESCINE DIAM-3 DIAMINOMITOSENE-2,7 DIAMINOPURINE-2,6 DIANHYDROGALACTITOL DIAZAN DIAZAQUINOMYCIN-A DIAZAQUINOMYCIN-B DIAZIQUONE DIBENZYL-DISELENIDE DIBENZYLDAUNORUBICIN-N,N DIBUTYLTIN DICHLOROBENZOPRIM DICHLOROINDOPHENOL-2,6 DICHLOROLISSOCLIMIDE DICHLOROMETHOTREXATE DICHOTOMIN-A DICHOTOMIN-H DICHOTOMIN-I DICLOFENAC-GLUCURONIDE DICTYOTALIDE-B DIDEAZAADENOSINE-1,3 DIDEAZAISOFOLATE-5,8 DIDEAZATETRAHYDRO= FOLATE-5,10 DIDEMETHYLROCAGLAMIDE DIDEMNENONE-C DIDEMNENONE-D DIDEMNIN-A DIDEMNIN-B DIDEMNIN-C DIDEMNIN-D DIDEOXYCYTIDINENE-2+,3+ DIDOX DIETHYLSPERMINE-1,12 DIFFERANISOLE-A DIFLOMOTECAN DIFLUORODEOXY-CTP DIFLUORODEOXYGUANOSINE DIHETEROPEPTIN DIHYDROAMBAZONE DIHYDROAZACYTIDINE-5 DIHYDROBENFLURON-7 DIHYDROCICLOSPORIN DIHYDROCOUMARIN DIHYDROCUCURBITACIN-D-= 23,24 DIHYDROCYCLOSPORIN-C DIHYDROFLUOROURACIL DIHYDROHALICHONDRAMIDE DIHYDROILLUDIN-M DIHYDROISOCYCLOARTOMUNIN DIHYDRONARCICLASINE-= TRANS DIHYDROORACINE-11 DIHYDROOXONATE DIHYDROPANAXACOL DIHYDROSPHINGOSINE-= THREO DIHYDROXYBUTYR= ALDEHYDE DIHYDROXYCHALCONE-= 2+,4+ DIMETHYL-PAMIDRONATE DIMETHYLBUSULFAN DIMETHYLDAUNORUBICIN-= N,N DIMETHYLMITOZOLOMIDE-= N,N DINALINE DIOPTERIN DIOSPYRIN DIOSPYRIN-DIMETHYL-ETHER DIOXADET DIPHYLLIN DIPIN DIPLAMINE DIPROSPIDIUM BROMIDE DIRCIN DIRHODIUM-TETRAACETATE DISCODERMOLIDE DISCORHABDIN-A DISCORHABDIN-C DISCORHABDIN-D DISTAMYCIN-2 DISTAMYCIN-5 DISTAMYCIN-A DISTEL DITERCALINIUM CHLORIDE DITHIZON DITHYMOQUINONE DITIOMUSTINE DITIOMUSTINE-SULFONE DITIOMUSTINE-SULFOXIDE DITRISARUBICIN-A DITRISARUBICIN-B DIVICINE DM-75 DM-96 DMP-315 DNACIN-A1 DNACIN-B1 DOB-41 DODECYLPHOSPHOCHOLINE DOLABELLANIN-A DOLASTATIN-10 DOLASTATIN-11 DOLASTATIN-12 DOLASTATIN-13

1132 APPENDIX D DOLASTATIN-14 DOLASTATIN-15 DOLASTIN-3 DON DOPA-METHYL-ESTER DORRIGOCIN-A DORRIGOCIN-B DOXIFLURIDINE DOXOFORM DOXORUBICIN DRAGMACIDIN-D DRF-1042 DRIMENINE DRUMMONDIN-A DRUMMONDIN-B DRUMMONDIN-C DRUMMONDIN-F DS-4152 DSB-120 DT-5461 DT-5461-A DU-14 DU-86 DUAZOMYCIN DUOCARMYCIN-A DUOCARMYCIN-B1 DUOCARMYCIN-B2 DUOCARMYCIN-C1 DUOCARMYCIN-C2 DUOCARMYCIN-SA DURYNE DWA-2114R DWA-2114S DX-52-1 DX-8951 DX-8951-F DYNEMICIN-A DYNEMICIN-H DYNEMICIN-N DYSIDAZIRINE DYSIDIOLIDE DYSOXYSULFONE E-126 E-7010 E-94 EB-1213 EB-1231 EBIFURAMIN ECOMUSTINE ECTEINASCIDIN-729 ECTEINASCIDIN-743 ECTEINASCIDIN-745 ECTEINASCIDIN-759A ECTEINASCIDIN-759B ECTEINASCIDIN-770 ED-110 ED-749 EDATREXATE EDIKRON EDRECOLOMAB EFLORNITHINE EKB-569 ELACTOCIN ELAEOCARPUSIN ELAEODENDROSIDE-A ELAEODENDROSIDE-E ELAEODENDROSIDE-J ELEMENE-BETA ELENATE ELENOSIDE ELEPHANTIN ELEPHANTOPIN ELEUTHERIN ELEUTHEROBIN ELLIPTICINE ELLIPTINIUM ELLIPTINIUM-OLEATE ELLIPTINIUM-PALMITATE ELLIPTINIUM-STEARATE ELMUSTINE ELSAMICIN ELSAMICIN-A ELSAMICIN-B EM-652 EM-800 EMD-121974 EMD-55900 EMD-66203 EMITEFUR EMOXYL ENDOSTATIN ENDOSTATIN-HUMAN ENDOSTATIN-MOUSE ENLOPLATIN ENMEIN ENOCITABINE ENPROMATE EO-15 EO-5A EO-68 EO-72 EO-9 EPI-OLEANOLATE EPICALYXIN-F EPICALYXIN-I EPICALYXIN-K EPILIMONOL EPIPODOPHYLLOTOXIN EPIPOLYGODIAL EPIPROPIDINE EPIRUBICIN EPIRUBICINOL EPITAXOL-7 EPITIOSTANOL EPONEMYCIN EPOTHILONE-A EPOTHILONE-B EPOTHILONE-D EPOXOMICIN EPOXYLUPINIFOLIN EPOXYQUINOMICIN-A EPOXYQUINOMICIN-B EPRATUZUMAB ER-076349 ER-086526 ER-35744 ER-68203-00 ER-69029 ERBSTATIN ERGOLIDE ERGOSTEROL-PEROXIDE ERIOLANIN ERUCYLPHOSPHOCHOLINE ES-921 ES-922 ESORUBICIN ESPERAMICIN ESPERAMICIN-A1 ESPERAMICIN-A1B ESPERAMICIN-A2 ESPERAMICIN-C ESPERAMICIN-D ESPERAMICIN-E ESPERAMICIN-X ESPERAMICIN-Z ESTRAMUSTINE ESTRAMUSTINE-PHOSPHATE ESTROMUSTINE ET-16S-OET ET-18-OCH3 ETANERCEPT ETAROTENE ETHOXIDINE ETHOXYESTRADIOL-2 ETHYLDEHYDROXY= SPARSOMYCIN ETHYLESTRONE-3-O-= SULFAMATE-2 ETHYLMERCAPTOPURINE-6 ETHYLNITROSOUREA ETHYMIDINE ETHYNYLCYTIDINE-3+ ETHYNYLURIDINE-3+ ETIOLINE ETOGLUCID ETOPOFOS ETOPOSIDE ETOPOSIDE-QUINONE-O ETOPRINE ETRETINATE EUCANNABINOLIDE EUGENIIN EUGLOBAL-G5 EUGLOBAL-IA1 EUGLOBAL-IA2 EUGLOBAL-IIB EUGLOBAL-IVA EUGLOBAL-IVB EUGLOBAL-VII EUONYMOSIDE-A EUPAROTIN EUPATOLIDE EUPATORIOPICRIN EUROPINE EURYCOMALACTONE EURYCOMANONE EVEROLIMUS EVOLITRINE EXCOECARIA-TOXIN EXEMESTANE EXISULIND F-11782 F-4168 F-4236 F-4614 F-910826 FAD-001 FADROZOLE FAGARONINE FASCAPLYSIN FASTIGILIN-C FAVELANONE FAVELINE FAZARABINE FCE-23762 FCE-24561 FCE-25217 FCE-25450-A FCE-26366 FCE-26367 FCE-26541 FCE-26605 FCE-26644 FCE-26806 FCE-27164 FCE-28068 FCE-28164 FCE-28729 FCE-28987 FCE-29006 FCE-29272 FCNU FD-1 FD-594 FD-891 FEAC FEBRIFUGINE FELLUTAMIDE-A FENRETINIDE FERROCENE-A FETINDOMIDE FEUDOMYCIN-B

Derwent Drug File 1133 Thesaurus FEUDOMYCIN-D FIBROBLAST-GROWTH-= FACTOR-BASIC-SAPORIN FIDUXOSIN FINROZOLE FLAVIPUCINE FLAVOPIRIDOL FLOXURIDINE FLOXURIDINE-DICAPRYLATE-= 3+,5+ FLOXURIDINE-DIPALMITATE-= 3+,5+ FLOXURIDINE-PHOSPHATE FLOXURIDINE-TRIPHOSPHATE FLU-401 FLU-402 FLUASTERONE FLUDARABINE FLUDARABINE-PHOSPHATE FLUOROCYTIDINE FLUOROCYTOSINE-= ARABINOSIDE FLUORODAUNORUBICIN-2+ FLUORODEOXYCYTIDINE-= PHOSPHATE FLUORODOPAN FLUOROFORMYCIN-2 FLUOROIDARUBICIN-2 FLUOROIDARUBICIN-3 FLUOROIDARUBICIN-8R FLUOROIDARUBICIN-8S FLUOROMETHOTREXATE-= GAMMA FLUOROOROTATE FLUOROPYRIMIDINONE FLUOROURACIL FLUOROURACIL-ARABINOSIDE FLUOROURACIL-PHTHALIDYL FLUOROURIDINE FLUOROURIDINE-PHOSPHATE FLUOROURIDINE-= TRIPHOSPHATE FLUROCITABINE FMAU FORFENIMEX FORMAMICIN FORMESTANE FORMOSANIN-C FORMYCIN FORMYCIN-B FORPHENICINOL FOSFESTROL FOSQUIDONE FOSTRIECIN FOTEMUSTINE FR-182877 FR-66973 FR-66979 FR-66980 FR-900405 FR-900482 FR-900840 FR-901228 FR-901463 FR-901464 FR-901465 FR-901537 FREDERICAMYCIN-A FRENTIZOLE FTI-2148 FTI-2153 FTI-276 FTI-277 FUMAGILLOL FUMITREMORGIN-C FURAQUINOCIN-A FURAQUINOCIN-B FURAQUINOCIN-C FURAQUINOCIN-D FURAQUINOCIN-E FURAQUINOCIN-F FURAQUINOCIN-G FUROSIN FUSARICIDE FYTATE G-3139 G-4073 GACAVIT GALACTOSE-MUSTARD-C6 GALANOLACTONE GALLIUM-CHLORIDE GALOCITABINE GALOCITABINE GALTAMYCIN GANODERATE-E GANODERATE-T GANODERATE-Y GANU GAUDICHAUDIONE-A GAUDICHAUDIONE-B GBC-590 GE-132 GE-3 GECLOSPORIN GEIPARVARIN GEM-231 GEMCITABINE GEMIN-A GEMTUZUMAB OZOGAMICIN GENKWADAPHNIN GEODIAMOLIDE-A GEODIAMOLIDE-B GERANYLGERANIOL GG-211 GGTI-286 GGTI-287 GGTI-297 GGTI-298 GI-147211 GI-147211-C GI-147211C GI-149893 GIGANTECIN GIGANTETROCIN-A GIGANTETROCIN-B GIGANTETRONENIN GILVOCARCIN-M GILVOCARCIN-V GINSENOSIDE-RG5 GINSENOSIDE-RH2 GIRACODAZOLE GIRINIMBINE GL-331 GLACIASTEROL-A GLAUCARUBINONE GLIDOBACTIN-A GLIDOBACTIN-B GLIDOBACTIN-C GLUCAN-CM GLUCAN-HA GLUCOSE-MUSTARD-C6 GLUTAMATE-GAMMA-= MONOHYDROXAMATE GLUTAMATE-MONO= HYDROXAMATE GLUTAMIN-(ASPARAGIN-)ASE GLYCIPHON GM-1474 GMD-4-C GNIDIDIONE GNIDILATIDIN GNIDILATIN GNIDIMACRIN GOE-4902 GOE-5549 GONIODIOL GONIODIOL-DIACETATE GONIODIOL-= MONOACETATE-7 GONIODIOL-= MONOACETATE-8 GONIOFUFURONE GONIOPYPYRONE GONIOTHALAMICIN GONIOTRIOL GP-27 GP-48989 GP-7 GPA-1734 GR-54374 GR-54374X GRAPE-SEED-EXTRACT GREVILLOL GRIFOLAN GRIFOLAN-LE GRIFOLAN-NMF-5N GROSHEIMIN GROSSULARINE-1 GROSSULARINE-2 GS-1500 GUANAZOLE GUANIDINOPROPIONATE-3 GUANOSINE-N-OXIDE-7 GUATTEGAUMERINE GW-154 GW-158 GW-187 GW-2016 GW-347845-X GW-420371-X GW-7845 GW-8510 GW-974 GYKI-13324 H-200-68 H-76-8159 HA-14-1 HADACIDIN HAEMANTHAMINE HALICHONDRIN-B HALICLAMINE-A HALIMEDATRIAL HALISTATIN-1 HALISTATIN-2 HALLERIDONE HALOMON HARRINGTONINE HATOMARUBIGIN-B HC-TOXIN HEDAMYCIN HEDERACOLCHISID-A1 HELENALIN HELICHRYSETIN HELIOPORIN-D HELIQUINOMYCIN HELIXOR HEMIASTERLIN HENU HEPATOCYTE-GROWTH-= FACTOR-NK4 HEPSULFAM HEPTELIDATE HEPTYLCHAPARRINONE-15-= BETA HERACLENIN HERBIMYCIN-A HERBIMYCIN-B HERBIMYCIN-C HERBINDOLE-A HERBINDOLE-B HERBINDOLE-C HERBOXIDIENE HEREGULIN-HUMAN

1134 APPENDIX D HERICENONE-A HERNOVINE HERSTATIN HEXANOYLSPHINGOSINE-N HEXAPHOSPHAMIDE HIBARIMICIN-A HIBARIMICIN-C HIBARIMICIN-D HIBURIPYRANONE HIMASTATIN HINOKININ HIPPOCRATEINE-I HIRTELLIN-A HIRTELLIN-B HISPHEN HITACHIMYCIN HIYODORILACTONE-E HMN-176 HO-221 HODGKINSINE HOLACANTHONE HOMOHALICHONDRIN-B HOMOHARRINGTONINE HOMOLYCORINE HORMOTHAMNIONE HORSERADISH-PEROXIDASE HR-2074 HR-2153 HR-2257 HRK-055512 HRK-429 HYB-190 HYDNOCARPIN HYDRAZINE-SULFATE HYDROPEROXYCYCLO= PHOSPHAMIDE HYDROPEROXYIFOSFAMIDE HYDROXYACIVICIN-4 HYDROXYACLARUBICIN-2 HYDROXYACLARUBICIN-II HYDROXYBULLATACINONE-30 HYDROXYBULLATACINONE-31 HYDROXYBULLATACINONE-32 HYDROXYBULLATACINONE-32 HYDROXYCAMPTOTHECIN-= 10 HYDROXYCYCLO= PHOSPHAMIDE-4 HYDROXYDOXORUBICIN-3+ HYDROXYEURYCOMA= LACTONE-6-ALPHA HYDROXYGLUTAMATE-4 HYDROXYIFOSFAMIDE-4 HYDROXYLOMUSTINE-2-= TRANS HYDROXYLOMUSTINE-4-CIS HYDROXYMETHOTREXATE-7 HYDROXYMETHYLELLIPTICINE HYDROXYMETHYLPENTA= METHYLMELAMINE HYDROXYNONENAL-4 HYDROXYNONYLADENINE HYDROXYRUBICIN-D HYDROXYUREA HYDROXYVITAMIN-D5,1-= ALPHA HYMENISTATIN-1 HYMENOXIN IBANDRONATE IBRITUMOMAB-TIUXETAN ICI-198583 ICI-47776 ICI-D-0490 ICIG-1105 ICIG-1163 ICIG-1164 ICP-1 ICR-170 ICR-191 ICRF-154 ICRF-158 ICRF-193 ICRF-197 ICRF-202 ICRF-500 ICRF-505 ICRF-510 ICRF-602 IDARUBICIN IDARUBICINOL IDEC-152 IDN-5109 IDN-5390 IDOXURIDINE IDOXURIDINE-= MONOPHOSPHATE IEJIMALIDE-B IFOSFAMIDE IH-636 IKD-8344 IKIMINE-A ILIMAQUINONE ILLUDIN ILLUDIN-M ILLUDIN-S ILLUDOFULVENE ILMOFOSINE ILX-23-7553 IM-862 IMATINIB IMBRICATINE IMET-28-67 IMET-2951 IMET-3164 IMET-3293 IMET-3379 IMIDACRINE IMINODAUNORUBICIN-5 IMINODOXORUBICIN-5 IMIPHOS IMMUCILLIN-H IMPROSULFAN IMUVERT INCADRONATE INCRUSTASTEROL-A INCRUSTASTEROL-B INDANOCINE INDICINE-N-OXIDE INOLIDE-A INOSTAMYCIN INOTODIOL INOXINE INPROQUONE INSULARINE INTERFERON INTERFERON-ALPHA INTERFERON-ALPHA,BETA INTERFERON-ALPHA,BETA-= MOUSE INTERFERON-ALPHA,BETA-= RAT INTERFERON-ALPHA-1 INTERFERON-ALPHA-1-= ALPHA-8-HUMAN INTERFERON-ALPHA-1-= CATTLE INTERFERON-ALPHA-1-= HUMAN INTERFERON-ALPHA-1MOUSE INTERFERON-ALPHA-2 INTERFERON-ALPHA-2-1-= HUMAN INTERFERON-ALPHA-2-ARG INTERFERON-ALPHA-2-= HUMAN INTERFERON-ALPHA-2-LYS-= HUMAN INTERFERON-ALPHA-2MOUSE INTERFERON-ALPHA-2A INTERFERON-ALPHA-2A-= HUMAN INTERFERON-ALPHA-2B INTERFERON-ALPHA-2B-= HUMAN INTERFERON-ALPHA-2C INTERFERON-ALPHA-2C-= HUMAN INTERFERON-ALPHA-4-= HUMAN INTERFERON-ALPHA-4-= MOUSE INTERFERON-ALPHA-4A INTERFERON-ALPHA-54 INTERFERON-ALPHA-6 INTERFERON-ALPHA-7-= HUMAN INTERFERON-ALPHA-8 INTERFERON-ALPHA-A-D INTERFERON-ALPHA-A-D= (BGL-II) INTERFERON-ALPHA-B INTERFERON-ALPHA-B-D INTERFERON-ALPHA-B-D-= HUMAN INTERFERON-ALPHA-B-= HUMAN INTERFERON-ALPHA-BDBB INTERFERON-ALPHA-C INTERFERON-ALPHA-C-= CATTLE INTERFERON-ALPHA-C-= HUMAN INTERFERON-ALPHA-CATTLE INTERFERON-ALPHA-CON-1 INTERFERON-ALPHA-CON1-= HUMAN INTERFERON-ALPHA-F-D INTERFERON-ALPHA-F-= HUMAN INTERFERON-ALPHA-GAMMA INTERFERON-ALPHA-HUMAN INTERFERON-ALPHA-I INTERFERON-ALPHA-I-HUMAN INTERFERON-ALPHA-I1 INTERFERON-ALPHA-I1-= CATTLE INTERFERON-ALPHA-II-1 INTERFERON-ALPHA-J INTERFERON-ALPHA-J-C INTERFERON-ALPHA-J1-= SER116 INTERFERON-ALPHA-K INTERFERON-ALPHA-MOUSE INTERFERON-ALPHA-N INTERFERON-ALPHA-N1 INTERFERON-ALPHA-N1-= HUMAN INTERFERON-ALPHA-N3-= HUMAN INTERFERON-ALPHA-PIG INTERFERON-BETA INTERFERON-BETA-1 INTERFERON-BETA-1-HORSE INTERFERON-BETA-1-HUMAN INTERFERON-BETA-1A INTERFERON-BETA-1A-= HUMAN INTERFERON-BETA-1B INTERFERON-BETA-2 INTERFERON-BETA-2-HUMAN INTERFERON-BETA-CAT INTERFERON-BETA-CATTLE INTERFERON-BETA-HUMAN INTERFERON-BETA-MOUSE

Derwent Drug File 1135 Thesaurus INTERFERON-BETA-SER INTERFERON-BETA-SER-= HUMAN INTERFERON-CAT INTERFERON-CATTLE INTERFERON-CONCENSUS INTERFERON-DELTA-4-= ALPHA-2-ALPHA-1 INTERFERON-GAMMA INTERFERON-GAMMA-1B INTERFERON-GAMMA-4A INTERFERON-GAMMA-= CATTLE INTERFERON-GAMMA-= HUMAN INTERFERON-GAMMA-= INDUCING-FACTOR-MOUSE INTERFERON-GAMMA-= MOUSE INTERFERON-GAMMA-PIG INTERFERON-GAMMA-RABBIT INTERFERON-GAMMA-RAT INTERFERON-HUMAN INTERFERON-INDUCIBLE-= PROTEIN-10-HUMAN INTERFERON-MOUSE INTERFERON-PI INTERFERON-RAT INTERFERON-TAU INTERFERON-TAU-HUMAN INTERFERON-TAU-SHEEP INTERLEUKIN-13,LYS-13 INTERLEUKIN-13,LYS-13-= ASP-112 INTERLEUKIN-18 INTOPLICINE INUVISCOLIDE INX-3280 IODODEOXYDOXO= RUBICINOL-4+ IODOMYCIN IODOTAMOXIFEN IODOVULONE-I IPOMEANOL IPROPLATIN IRCINAL-A IRINOTECAN IROFULVEN ISCADOR ISIS-11061 ISIS-12449 ISIS-12959 ISIS-13650 ISIS-2503 ISIS-3521 ISO-DC-81 ISOACTEOSIDE ISOANNONACIN ISOANNONACINONE ISOBATZELLINE-A ISOBATZELLINE-C ISOBLEOMYCIN-A2 ISOBUTYRYLMALLOTO= CHROMENE ISOCRYPTOMERIN ISOCUCURBITACIN-B ISODEOXYPODOPHYLLOTOXIN ISODONAL ISODONOATE ISODOXORUBICIN ISOHOMOHALICHONDRIN-B ISOISOVELLERAL ISOKIDAMYCIN ISOMELODIENONE ISOMITOMYCIN-A ISOMITRAPHYLLINE ISOPENTENYLADENOSINE ISOPHOSPHORAMIDE-= MUSTARD ISOPLUMERICIN ISOPSYCHOTRIDINE-C ISOSTEGANE ISOSWINHOLIDE-A IST-622 IT-62-B IVALIN J-109404 JACEOSIDIN JARANOL JATROPHONE JK-1624-2 JK-1624-3 JM-1 JM-10 JM-11 JM-118 JM-120 JM-122 JM-125 JM-132 JM-149 JM-185 JM-2 JM-20 JM-216 JM-221 JM-222 JM-223 JM-225 JM-229 JM-231 JM-236 JM-244 JM-251 JM-256 JM-260 JM-262 JM-2644 JM-269 JM-271 JM-273 JM-274 JM-291 JM-3 JM-334 JM-335 JM-40 JM-407 JM-473 JM-480 JM-5 JM-6 JM-64 JM-68 JM-82 JM-93 JUNCUSOL JUSTICIDIN-B JV-1-36 JWH-133 K-11002 K-11017 K-11777 KAHALALIDE-F KALOPANAXSAPONIN-B KALOPANAXSAPONIN-H KALOPANAXSAPONIN-I KANSHONE-A KAPURIMYCIN-A1 KAPURIMYCIN-A2 KAPURIMYCIN-A3 KAR-2 KAZUSAMYCIN KAZUSAMYCIN-B KB-R-8498 KEDARCIDIN KELLETININ-I KENGSHENGMYCIN KERAMAPHIDIN-B KERICEMBRENOLIDE-D KERICEMBRENOLIDE-E KERRIAMYCIN-A KERRIAMYCIN-B KERRIAMYCIN-C KETOIFOSFAMIDE-4 KETOTREXATE KF-25706 KF-58333 KH-1059 KH-1139 KH-1230 KHPC-002 KI-8110 KIJANIMICIN KM-966 KN-827 KO-132 KO-134 KO-143 KOKUSAGININE KOLAVENOL KP-1019 KP-418 KP-735 KRAUSSIANIN KRESTIN KRN-5500 KRN-7000 KRN-8602 KT-6006 KT-6124 KT-6149 KT-6528 KT-7692 KW-2170 KW-2189 KYN-54 L-39 L-651582 L-731734 L-731735 L-739749 L-744832 L-778123 L-86-8275 L-METHIONINE-GAMMA-= LYASE LACTOQUINOMYCIN LACTOQUINOMYCIN-A LAETRILE LAF-389 LAHERRADURIN LAMELLARIN-D LAMELLARIN-I LAMELLARIN-K LAMELLARIN-M LAMIVUDINE-TRIPHOSPHATE LAMOROLIDE LANNEAQUINOL LANTHIOPEPTIN LAPACHOL LAPACHONE-BETA LARGOMYCIN LARGOMYCIN-F-II LARICIRESINOL LARREANTIN LASIOCARPINE-N-OXIDE LASIODIPLODIN LASOFOXIFENE LASONOLIDE-A LAVANDUCYANIN LAVENDAMYCIN

1136 APPENDIX D LAVENDAMYCIN-METHYL-= ESTER LAVENDUSTIN-A LAXIFLORIN-C LB-42908 LBIF LEAKADIN LEINAMYCIN LENTINAN LEPTOFURANIN-A LEPTOFURANIN-B LEPTOFURANIN-C LEPTOFURANIN-D LEPTOLSTATIN LEPTOMYCIN-A LEPTOMYCIN-B LERIDISTIM LEUCASCANDROLIDE-A LEUCINOSTATIN-D LEUKEMIA-INHIBITORY-= FACTOR-HUMAN LEUKOREGULIN LEURUBICIN LEUSTRODUCSIN-B LEVAN LFM-A-13 LG-100268 LG-101305 LGD-1069 LIAROZOLE LIBLOMYCIN LIMONIN LIQUIRITIN LIRIODENDRIN LISSOCLINAMIDE-4 LISSOCLINAMIDE-5 LISSOCLINAMIDE-7 LISSOCLINOTOXIN-A LITHOSPERMATE-B LK-11 LL-14-I-352-ALPHA LL-C10037-ALPHA LL-D-49194-ALPHA-1 LL-D49194-ALPHA-1 LM-609 LM-975 LM-985 LMB-2 LOBAPLATIN LOBOHEDLEOLIDE LOFENAL LOMETREXOL LOMUSTINE LONGIKAURIN-A LONGIKAURIN-B LONGIKAURIN-D LONGILACTONE LONGILENE-PEROXIDE LONGIMICIN-B LONIDAMINE LOSAXANTRONE LOSOXANTRONE LOUISIANIN-A LS-2715 LS-2724 LU-103793 LU-224332 LU-55446 LU-79553 LUCIDENATE-A LUFFARIELLOLIDE LUMICOLCHICINE LUNASIN LUOTONIN-A LUZOPEPTIN LUZOPEPTIN-A LUZOPEPTIN-B LUZOPEPTIN-C LUZOPEPTIN-D LY-119932 LY-121887 LY-181984 LY-181985 LY-186391 LY-195448 LY-195779 LY-203725 LY-207702 LY-219703 LY-231514 LY-243246 LY-254155 LY-256787 LY-266070 LY-295501 LY-298207 LY-309887 LY-316373 LY-317236 LY-317615 LY-326315 LY-335563 LY-335979 LY-487355 LY-509207 LYCORENINE LYCORICIDINE LYSINE-ALPHA-OXIDASE M-40403 M-83 MA-144-N1 MACBECIN-I MACBECIN-II MACLURAXANTHONE MACROCLINISIDE-A MACROCLINISIDE-C MACROLACTIN-A MACROLACTIN-B MACROLACTIN-E MACROLACTIN-F MACROLACTINATE MACROMOMYCIN MACROSPHELIDE-A MADINDOLINE-A MADINDOLINE-B MADUROPEPTIN MAESAQUINONE MAFOSFAMIDE MAFOSFAMIDE LYSINE MAGNOLIALIDE MAHARISHI-4 MAITANSINE MAKALUVAMINE-A MAKALUVAMINE-B MAKALUVAMINE-C MAKALUVAMINE-D MAKALUVAMINE-E MAKALUVAMINE-F MALLOTOCHROMENE MALLOTOLERIN MALLOTOPHENONE MAMANUTHAQUINONE MAMMASTATIN MANNOMUSTINE MANNOSULFAN MANOOL MANSONIN MANUMYCIN MANUMYCIN-B MANUMYCIN-C MANWUWEIZATE MANZAMINE-A MANZAMINE-B MANZAMINE-C MANZAMINE-D MANZAMINE-Y MARCELLOMYCIN MARCHANTIN-A MARCHANTIN-C MARIMASTAT MASPIN MATLYSTATIN-A MATLYSTATIN-B MAYTANBUTINE MBI-28 MC-1301 MC-62 MC-77 MDL-101731 MDL-103323 MDL-27048 MDL-72175 MDX-H-210 ME-2303 ME-3229 MECHLORETHAMINE-OXIDE MEDITERRANEOL-A MEDORUBICIN MEDPHALAN MEGAPHONE MEISOINDIGO MELANOCIDIN-A MELANOCIDIN-B MELANOTAN-I MELANOTAN-II MELIANONE MELINONINE-F MELODIENONE MELODORINOL MELPHALAN MELPHALAN-METHYL-ESTER MEN-10397 MEN-10400 MEN-10567 MEN-10706 MEN-10710 MEN-10755 MENOGARIL MEQUINOL MERANZIN MERBARONE MERCAPTOPOLY= CYTIDYLATE-5 MERCAPTOPURINE MERCAPTOPURINE-RIBOSIDE MERCAPTOPURINE-RIBOTIDE MERIDINE MERODANTOIN MEROPHAN MERULIDIAL MESO-DIHYDRO= GUAIARETATE METACHROMIN-A METACHROMIN-C METAMELFALAN METAZATHIOPRINE METHANOCARBA= THYMIDINE-N METHASQUIN METHOPTERIN METHOTREXATE METHOTREXATE-ALPHA-= ALANINE METHOTREXATE-ALPHA-= ARGININE METHOTREXATE-ALPHA-= ASPARTATE METHOTREXATE-DIBUTYL-= ESTER METHOTREXATE-= DIMETHYL-ESTER METHOTREXATE-GAMMA-= ASPARTATE

Derwent Drug File 1137 Thesaurus METHOTREXATE-= MONOBUTYL-GAMMA-= ESTER METHOXYBENZENE= SELENOL-PARA METHOXYELLIPTICINE-9 METHOXYPHASEOLLIDIN-1 METHOXYPODOPHYLLO= TOXIN-5 METHOXYSTROBILURIN-K-9 METHYL-DOXORUBICIN-O-4+ METHYL-MESILATE METHYL-TRAMETENOLATE METHYLANGUSTOLINE-19-O METHYLBETACLAMYCIN-= T,4-O METHYLCYCLO= PHOSPHAMIDE-4 METHYLDACARBAZINE-1 METHYLDEOXYCYTIDINE-5 METHYLELLIPTICINIUM-2 METHYLENE-DIMESILATE METHYLENOLACTOCIN METHYLEPOXYSHIKOCCIN-O METHYLFORMAMIDE METHYLFORMYCIN-4 METHYLGLYOXAL METHYLMERCAPTOPURINE METHYLMERCAPTO= PURINE-RIBOSIDE METHYLMITOZOLOMIDE-N METHYLQUADRANGU= LARATE-D METHYLSELENINATE METHYLSELENOCYSTEINE-SE METHYLSELENOL METHYLSHIKOCCIN-O METHYLTHIOFORMYCIN METHYLURIDINE-5 METOPRINE METROGIL METUREDEPA MF-13 MG-115 MG-341 MG-98 MI-1544 MICROLENIN MICROSTEGIOL MIGRASTATIN MIKANIAHUMULENE-I MIKANIAHUMULENE-II MILDIOMYCIN MILTEFOSINE MILTIPOLONE MIMIMYCIN MIMOSINE MIPROXIFENE MIRABIMIDE-E MISTLETOE-LECTIN MITINDOMIDE MITOBRONITOL MITOCLOMINE MITOGUAZONE MITOLACTOL MITOMYCIN MITOMYCIN-A MITOMYCIN-B MITOMYCIN-D MITOMYCIN-F MITOMYCIN-G MITOMYCIN-H MITOMYCIN-K MITONAFIDE MITOPODOZIDE MITOQUIDONE MITOSPER MITOTENAMINE MITOXANTRONE MITOZOLOMIDE MKT-077 MMI-166 MNNG MOBILETREX MOFAROTENE MOLVIZARIN MOLYBDATE MOLYBDENOCENE-= DICHLORIDE MONASTROL MONOAZIRIDINYL= PUTRESCINE MONOLINOLEIN-ALPHA MONORDEN MONTIPORATE-A MONTIPORATE-B MORONATE MORPHOLINODAUNORUBICIN MOTRETINIDE MOTUPORAMINE-C MOTUPORIN MPV-2213-AD MR-566-A MR-566-B MRS-1067 MRS-1191 MRS-1220 MS-247 MS-27-275 MSI-238 MST-16 MUCONIN MULLERIAN-INHIBITING-= SUBSTANCE-HUMAN MUP-98156 MURICATACIN MURICATETROCIN-A MURICATETROCIN-B MURISOLIN MURISOLINONE-CIS MURISOLINONE-TRANS MURRAPANINE MURRAYANINE MUSETTAMYCIN MVE-5 MX MX-2 MX-3350-1 MY-5 MYCALAMIDE-B MYCALISINE-A MYCALOLIDE-B MYCALOLIDE-C MYCAPEROXIDE-A MYCAPEROXIDE-B MYCOPHENOLATE MYCORRHIZIN-B1 MYCORRHIZIN-B2 MYCOTRIENIN-I MYCOTRIENIN-II MYROCIN-C MZ-5-156 N-30 N-5228 NA-22598-A-1 NAKIJIQUINONE-A NAKIJIQUINONE-B NAPAVIN NAPHTHGERANINE-A NAPHTHOPYRANOMYCIN NAPHTHYRIDINOMYCIN NAPYRADIOMYCIN-A1 NAPYRADIOMYCIN-B1 NAPYRADIOMYCIN-C1 NARCICLASINE NARDOSINONE NB-1011 NB-506 NBQ-38 NBQ-48 NBQ-59 NC-190 NCS-686760 NDDP NDH-3080 NE-10244 NE-58051 NECTANDRIN-B NEIHUMICIN NELARABINE NEOAMBROSIN NEOAPLAMINONE NEOCARZILIN-A NEOMANOALIDE NEOOXAZOLOMYCIN NEOSENKIRKINE NEOTHRAMYCIN NEOTHRAMYCIN-A NEOTHRAMYCIN-B NEPLANOCIN-A NEPRILYSIN NEPTAMUSTINE NEUROLENIN-B NEYTUMORIN NF-023 NF-031 NF-032 NF-103 NF-110 NF-201 NF-503 NF-504 NF-506 NIFURON NIGRANOATE NIMBOLIDE NIMUSTINE NIOBOCENE-DICHLORIDE NIPHATESINE-A NIPHATESINE-B NIPHATESINE-C NIPHATESINE-D NITIDINE NITRACRINE NITROCAMPTOTHECIN-9 NITROCHOLESTEROL-6 NITROIBUPROFEN NITRULLINE NK-121 NK-611 NLCQ-1 NOBOTANIN-G NOBOTANIN-H NOBOTANIN-I NOBOTANIN-K NOCARDICYCLIN-A NOCODAZOLE NOGARENE NOMILIN NONYLOXYCARBONYL-= MITOMYCIN NOR-ISOGUAIACIN NORCANTHARIDIN NORCHLORMETHINE NORDERCITIN NORDIDEMNIN-B NORPACLITAXEL-C NORSANGUINARINE NORSPERMIDINE NORTOPSENTIN-A NORTRACHELOGENIN NOSTOCYCLOPHANE-D NOVOBIOCIN

1138 APPENDIX D NOVOEMBICHIN NPF-86-IA NPF-86-IB NPF-86-IIA NPF-86-IIB NPF-86IA NPF-86IB NPF-86IIA NPF-86IIB NS-1C NS-1D NSC-100880 NSC-101327 NSC-107392 NSC-110333 NSC-113423 NSC-114460 NSC-117614 NSC-126771 NSC-140117 NSC-140701 NSC-145813 NSC-146067 NSC-146068 NSC-158197 NSC-170895 NSC-170898 NSC-170899 NSC-176319 NSC-181928 NSC-191295 NSC-194814 NSC-215914 NSC-224070 NSC-224964 NSC-23909 NSC-239717 NSC-239851 NSC-246112 NSC-250427 NSC-251635 NSC-255110 NSC-259946 NSC-262666 NSC-267213 NSC-269130 NSC-269416 NSC-271674 NSC-278214 NSC-278467 NSC-278999 NSC-281246 NSC-289517 NSC-290205 NSC-296964 NSC-303861 NSC-30705 NSC-311469 NSC-314622 NSC-321567 NSC-321584 NSC-324368 NSC-328002 NSC-330507 NSC-330770 NSC-335154 NSC-337238 NSC-338600 NSC-338698 NSC-339675 NSC-340307 NSC-341082 NSC-341936 NSC-341964 NSC-343513 NSC-343529 NSC-344270 NSC-344280 NSC-347515 NSC-350102 NSC-350386 NSC-350602 NSC-352683 NSC-352692 NSC-352875 NSC-352876 NSC-353649 NSC-354646 NSC-355277 NSC-357704 NSC-361456 NSC-364720 NSC-365171 NSC-366140 NSC-370147 NSC-370277 NSC-373232 NSC-38280 NSC-402538 NSC-47547 NSC-49272 NSC-521164 NSC-56336 NSC-57153 NSC-57155 NSC-60339 NSC-606174 NSC-606698 NSC-607732 NSC-609974 NSC-612567 NSC-613060 NSC-613862 NSC-613863 NSC-615830 NSC-615831 NSC-619444 NSC-619446 NSC-619531 NSC-627505 NSC-629243 NSC-630176D NSC-639366 NSC-639829 NSC-640488 NSC-645306 NSC-647884 NSC-649488 NSC-654261 NSC-655649 NSC-662304 NSC-662306 NSC-663284 NSC-665517 NSC-667005 NSC-66761 NSC-668380 NSC-680434 NSC-680718 NSC-686288 NSC-693567 NSC-71261 NSC-714187 NSC-76509 NSC-82196 NSC-83265 NSC-84954 NSC-84963 NSC-86047 NSC-87974 NSC-88104 NSC-95397 NSC-95580 NSC-D-699127 NU-2058 NU-6027 NU-UB-199 NU-UB-31 NUCLEOTICIDIN NY-3170 NY-3460 NY-4137 NY-4138 OC-144093 OCTADECYLMETHYLGLYCEROL OCTALACTIN-A OENOTHEIN-A OENOTHEIN-B OF-4949-I OGT-719 OHIOENSIN-A OKICENONE OKILACTOMYCIN OLEANONATE OLEOYLETHANOLAMINE-N OLIVACINE OLIVOMYCIN OLOMOUCINE ONCHITRIOL-I ONCHITRIOL-II ONCOSTATIN-M ONO-3403 ONOPORDOPICRIN ONYX-015 OPHIDIACEREBROSIDE-E ORG-31710 ORI-1202 ORI-1313 ORI-1327 ORIDONIN ORMAPLATIN OSI-774 OSSAMYCIN OSTEOCLASTOGENESIS-= INHIBITORY-FACTOR OSTOPANATE OSW-1 OVALICIN OVATODIOLIDE OXALIPLATIN OXALYSINE OXANOSINE OXAUNOMYCIN OXAZOLOMYCIN OXETANOCIN-A OXI-4503 OXINDOLE-I OXISURAN OXOPLATIN OXOPROPALINE-D OXOSTAUROSPORINE-7 OXOTINGENOL-6 P-1015 P-30 P-4018 PAB-13 PAB-13 PAB-23 PAB-23 PACHYMAN PACOVATININ-A PACTAMYCIN PAFENCYL PALAUOLOL PALMATINE PALOMINOL PALUSTRAN PALVANIL PANAXACHLOR PANAXACOL PANAXYDOL PANAXYTRIOL

Derwent Drug File 1139 Thesaurus PANCRATISTATIN PANICEIN-B3 PANICEIN-C PAPYRACON-A PARADOL-6 PAREIRUBRINE-A PARTHENIN PARVIFLORIN PATELLAMIDE-A PATELLAMIDE-B PATELLAMIDE-C PATELLAMIDE-D PATELLAZOLE-B PATRIN-2 PAZELLIPTINE PC-766B PCNU PD-0183085 PD-083176 PD-098059 PD-110095 PD-110334 PD-110911 PD-111391 PD-112940 PD-113270 PD-113271 PD-113377 PD-113876 PD-114027 PD-114057 PD-114245 PD-114254 PD-114541 PD-114595 PD-114631 PD-115934 PD-116152 PD-116250 PD-116740 PD-117802 PD-118309 PD-119556 PD-130883 PD-141955-2 PD-153717 PD-157655 PD-158780 PD-161176 PD-161570 PD-161956 PD-165557 PD-166285 PD-166793 PD-167462 PD-168368 PD-168393 PD-169451 PD-169540 PD-171026 PD-180970 PD-183805 PD-184352 PD-83176 PD-98059 PE-1001 PECTINIOSIDE-C PECTINIOSIDE-D PECTINOLIDE PEGVISOMANT PELIOMYCIN PELORUSIDE-A PELTATIN-ALPHA PELTATIN-BETA PENASTEROL PENBEROL PENCLOMEDINE PENDOLMYCIN PENTABROMOPSEUDILINE PENTAMETHYLMELAMINE PENTOSTATIN PENTYLSPARSOMYCIN PEPLOMYCIN PEPTICHEMIO PERENIPORIN-A PERENIPORIN-B PEREZONE PERFRAGILIN-B PERIDININ PEROXISOMICINE-A1 PEROXISOMYCIN PETROFORMYNE-1 PETROFORMYNE-2 PETROFORMYNE-3 PETROFORMYNE-4 PETROSYNOL PEX PGA1-DELTA-7-METHYL-= ESTER PGJ2-DEOXY-15-DELTA-12,14 PHAKELLISTATIN-11 PHAKELLISTATIN-8 PHASEOLLIDIN PHENAZINOMYCIN PHENESTER PHENESTERIN PHENETHYL-= ISOTHIOCYANATE PHENOMYCIN PHENYL-ISOTHIOCYANATE PHENYLACETATE-MUSTARD PHENYLAHISTIN PHENYLAZOXYCYANIDE PHENYLKETOCYCLO= PHOSPHAMIDE PHENYLPROPYLISO= THIOCYANATE PHORBOXAZOLE-A PHORBOXAZOLE-B PHORTRESS PHOSMIDOSINE PHOSMIDOSINE-B PHOSPHOLINE (antibiotic = cytostatic) PHOSPHORAMIDE-MUSTARD PHTHALIDE PHYLLANTHOCIN PHYLLANTHOSIDE PHYLLANTHOSTATIN-1 PHYLLANTHOSTATIN-2 PHYLLANTHOSTATIN-3 PHYLLOSTACHYSIN-A PHYLLYRAEOIDIN-A PI-88 PIBENZIMOL PICLAVINE-A1 PICLAVINE-A2 PICLAVINE-A3 PICLAVINE-A4 PICROPODOPHYLLOTOXIN PIFITHRIN-ALPHA PILATIN PIMECAR PIMELEA-FACTOR-P2 PINAFIDE PIPENDOXIFENE PIPERADUNCIN-B PIPERLONGUMINE PIPOBROMAN PIPOSULFAN PIRARUBICIN PIRARUBICIN PIRITREXIM PIRONETIN PIROXANTRONE PKI-166 PLAKINIDINE-A PLAKINIDINE-B PLAKORIN PLAKORTONE-D PLENOLIN PLEUROTIN PLICAMYCIN PLURAMYCIN-A PMEG PMEHX PMS-1 PNU-101383 PNU-145156-E PNU-157820 PNU-157924 PNU-159682 PNU-99533 PODOFILOX PODOPHYLLATE POLY-I-C-12-U POLY-OXYPEPTIN POLYACTIN-A POLYCARPINE POLYDATIN POLYERGA POLYGODIAL POLYPORATE POLYPRENOATE POMOLATE PORFIROMYCIN PORICOATE-A POROTHRAMYCIN-B POTASSIUMTETRACHLOROPLATINATE PR-1501 PREDNIMUSTINE PRETAZETTINE PREUSSOMERIN-D PREUSSOMERIN-E PREUSSOMERIN-F PREUSSOMERIN-G PREUSSOMERIN-H PREUSSOMERIN-I PRIANOSIN-C PRIANOSIN-D PRIEURIANIN PRINOMASTAT PROCARBAZINE PROCODAZOLE PROCYANIDIN-B2-DIGALLATE PRODIGIOZAN PROLACTIN-HUMAN-G129R PROSPIDIUM CHLORIDE PROSTRATIN PROTHRACARCIN PROTOANEMONIN PROXIFEINE PSAMMAPLIN-A PSEUDODISTOMIN-A PSEUDODISTOMIN-B PSEUDODISTOMIN-C PSEUDOISOCYTIDINE PSEUDOLARATE-B PSEUDOPTEROLIDE PSEUDOSTELLARIN-D PSEUDOUREA PSICOFURANINE PSOROSPERMIN PSYCHOTRIDINE PT-441 PT-523 PT-619 PT-633 PTEROPODINE PTEROSTILBENE

1140 APPENDIX D PTILOMYCALIN-A PTMC PTT-119 PUMITEPA PUNAGLANDIN-3 PUNAGLANDIN-4 PUROMYCIN PUROMYCIN-= AMINONUCLEOSIDE PURPURAMINE-H PUUPEHENONE PX-12 PXD-101 PY-490 PYRAONCOZINE PYRAZOMYCIN PYRIDINDOLOL-K2 PYRIDOXATIN PYROXAMIDE PYRROLOSPORIN-A PYRROMYCIN Q-85 QUADRIGEMINE-A QUADRIGEMINE-B QUADRONE QUELAMYCIN QUINOCARCIN QUINOCARCINOL QUINOCARMYCIN QUINOLACTACIN-A QUINOLACTACIN-B QUINOLIDOMICIN-A1 R-101933 R-76713 R-83842 RA-700 RA-X RABDOCOETSIN-B RABDOCOETSIN-C RACEMELFALAN RALTITREXED RANIMUSTINE RANTES RAVIDOMYCIN RAZOXANE RB-6145 RB-7040 RB-90740 RB-91724 RB-92816 RB-93918 RB-94571 RB-95629 RC-3940-II RC-3950-II REBECCAMYCIN REBLASTATIN RESIQUIMOD RESORTHIOMYCIN RESPINOMYCIN-A1 RESPINOMYCIN-A2 RESPINOMYCIN-B RESPINOMYCIN-C RESPINOMYCIN-D RESTRICTOCIN RETELLIPTINE RETICULATACIN RETINOATE-9-CIS RETINOL-GLUCURONIDE RETINOYL-BETA-= GLUCURONIDE RETINOYL-PHENYLALANINE RETINYL-METHYL-ETHER RETINYLIDENE-DIMEDONE REUMYCIN REVEROMYCIN-A REVEROMYCIN-B REVEROMYCIN-C REVEROMYCIN-D RG-13022 RG-14620 RG-50858 RHIZOXIN RHIZOXIN-D RHODAMINE-110 RHODAMINE-123 RHODOMYCIN-A RHODOMYCIN-B RHODOMYCIN-I-BETA RHOPALOATE-A RIBOPRINE RICCARDIN-A RICCARDIN-B RICCARDIN-C RICIN RICIN-A-CHAIN RICIN-A-CHAIN-= DEGLYCOSYLATED RICIN-B-CHAIN RICIN-BLOCKED RITROSULFAN RITTERAZINE-A RITTERAZINE-B RITTERAZINE-C RITTERAZINE-K RK-286C RK-397 RK-682 RM-175 RO-09-3431 RO-09-4889 RO-10-1770 RO-12-9933 RO-13-2389 RO-14-3899 RO-14-9572 RO-24-2090 RO-24-2287 RO-24-2637 RO-24-5531 RO-25-2032 RO-25-3036 RO-25-4020 RO-25-5318 RO-25-6603 RO-25-6760 RO-25-7553 RO-25-9022 RO-25-9887 RO-28-2653 RO-31-1215 RO-31-1740 RO-31-1741 RO-31-1749 RO-31-1966 RO-31-2035 RO-31-3294 RO-31-7453 RO-4-6824 RO-4020 RO-41-4439 RO-46-7864 RO-47-3359 RO-47-5944 RO-8-4969 RO-8-7699 RO-8-9372 ROCAGLAMIDE RODORUBICIN ROGLETIMIDE ROLLINACIN ROLLINIASTATIN-2 ROLLINICIN ROLLINONE ROLLITACIN RON ROQUINIMEX ROSCOVITINE ROSEOPHILIN ROYLEANONE RP-20132 RP-60475 RPR-113829 RPR-114334 RPR-121056 RR-150 RS-0481 RS-1541 RS-83277 RS-83287 RSR-13 RSU-1069 RSU-1131 RSU-1150 RSU-1164 RSU-1165 RSU-1170 RSU-1172 RTI-3021-020 RU-58668 RUBAMPICIN RUBEOMYCIN-A RUBEOMYCIN-A1 RUBEOMYCIN-B RUBICYCLAMIN RUBOXYL RUDMOLLIN RUDOLPHOMYCIN RUFOCROMOMYCIN S-10036 S-12362 S-137 S-16020-2 S-182 S-23906-1 S-247 S-27609 S-28463 S-55 S-785026 S-830544 SAE9 SAFRACIN-A SAFRACIN-B SAFRAMYCIN-A SAFRAMYCIN-AD-1 SAFRAMYCIN-B SAFRAMYCIN-C SAFRAMYCIN-D SAFRAMYCIN-F SAFRAMYCIN-G SAFRAMYCIN-H SAFRAMYCIN-MX-1 SAFRAMYCIN-R SAFRAMYCIN-S SAFRAMYCIN-Y2B SAFRAMYCIN-Y2B-D SAFRAMYCIN-Y3 SAFRAMYCIN-YD-1 SAFRAMYCIN-YD-2 SAINTOPIN SALICYLIHALAMIDE-A SALVICINE SALVIOLONE SALYNE SAMPANGINE SANDARACOPIMARATE SANDRAMYCIN SANGGENON-B SANGIVAMYCIN SANGUIIN-H11 SANGUIIN-H2

Derwent Drug File 1141 Thesaurus SANGUIIN-H6 SANTALOL-ALPHA SANTAMARIN SAPHENAMYCIN SAPONACEOLIDE-A SAPONACEOLIDE-B SAPORIN SAPORIN-6 SAPTOMYCIN-A SAPTOMYCIN-B SAPTOMYCIN-C1 SAPTOMYCIN-C2 SAPTOMYCIN-D SAPTOMYCIN-E SAPTOMYCIN-F SAPTOMYCIN-G SAPTOMYCIN-H SAPURIMYCIN SARASINOSIDE-A1 SARASINOSIDE-B1 SARCIN-ALPHA SARCNU SARCODICTYIN-A SARCODICTYIN-B SARCOPHYTOL-A SARCOPHYTOL-B SARKOMYCIN SARKOMYCIN-A SATIVAN SB-203347 SB-220025 SB-238039 SB-T-1213 SB-T-12843 SC-33428 SC-41661A SCH-207758 SCH-226374 SCH-44342 SCH-50673 SCH-56582 SCH-59228 SCH-60677 SCH-61129 SCH-66336 SCHA-764 SCOPADULCATE-A SCOPADULCATE-B SCYTOPHYCIN-B SCYTOPHYCIN-C SCYTOPHYCIN-D SCYTOPHYCIN-E SDK-103 SDK-110 SDK-12B-13 SDK-12B-5 SDZ-212-122 SDZ-266336 SDZ-266337 SDZ-280-446 SDZ-35-682 SECALONATE-D SECOMANOALIDE SEF-19 SELENAZOFURINE SEMAXANIB SEMPERVIRINE SEMUSTINE SENDANIN SENEGALENE SENKIRKINE SEOCALCITOL SESBANIMIDE SESBANIMIDE-A SESBANIMIDE-B SF-2575 SHERMILAMINE-B SIBIROMYCIN SIMALIKALACTONE-D SIMPLEXIN SIMTRAZENE SINOCOCULINE SINUGIBBEROL SIPLIZUMAB SIWENMYCIN SIZOFIRAN SJG-136 SK-31662 SK-31694 SKF-101772 SKF-102912 SKF-104524 SKF-45905 SKF-98625 SKI-2053-R SKULLCAPFLAVONE-II SM-108 SM-11355 SMA-41 SMA-52 SMENOQUINONE SMENORTHOQUINONE SMENOSPONDIOL SMENOSPONGIARINE SMENOSPONGIDINE SMENOSPONGINE SN-13553 SN-14771 SN-16507 SN-16713 SN-18071 SN-20779 SN-22 SN-22-NA SN-22981 SN-23862 SN-24771 SN-25084 SN-25261 SN-25341 SN-25507 SN-38 SN-4094 SN-6053 SN-6113 SN-6132 SN-6324 SN-6570 SN-6999 SO-75R1 SOAZ SODIUM-ARSENATE SOLAMARGINE SOLAMIN SOLIDAGENONE SOMATOMEDIN-C-BINDING-= PROTEIN-3 SOPHORAFLAVONE-G SP-500263 SP-600125 SP-904 SP-G SPARFOSATE SPARSOMYCIN SPATHULENOL SPATOL SPC-100270 SPERGUALIN SPHINGOSINE-PHOSPHATE-1 SPHINXOLIDE SPHINXOLIDE-B SPHINXOLIDE-C SPHINXOLIDE-D SPICAMYCIN SPIKET-P1 SPINAMYCIN SPIRANTHOL-A SPIRASINEOL-A SPIRAZIDIN SPIROBRAMINE SPIROGERMANIUM SPIROMUSTINE SPIROPLATIN SPIROTRYPROSTATIN-B SPONGISTATIN-1 SPONGISTATIN-3 SQUAMOCIN SQUAMONE SQUAMOSTATIN-A SR-11220 SR-11238 SR-11246 SR-11302 SR-11364 SR-144528 SR-16234 SR-4330 SR-4452 SR-4482 SRI-2712-24 SRI-62-834 SSG SSM ST-1481 ST-1646 STAUROSPORINE STEARYLPHOSPHOCHOLINE STEFFIMYCIN-D STEGANACIN STEGANOLIDE-A STEGANONE STELLETTIN-C STELLETTIN-D STELLETTIN-E STELLETTIN-F STIPIAMIDE STOLONIDIOL STOLONIDIOL-= MONOACETATE-17 STREBLOSIDE STREPTOCOCCAL-= ANTITUMOR-= GLYCOPROTEIN STREPTOVITACIN-A STRICTININ STROBILURIN-E STROBILURIN-F STROBILURIN-G STROBILURIN-H STRYCHNOPENTAMINE SU-4984 SU-5402 SU-5416 SU-6668 SU-9516 SUBEROYLANILIDE-= HYDROXAMATE SUCCINYLACETONE SUFOSFAMIDE SULFENOSINE SULFINOSINE SULFONOSINE SULFORAPHANE SULFUR-MUSTARD SULINDAC-SULFONELACTONE SULOFENUR SUN-4599 SUVANINE SWINHOLIDE-A SWINHOLIDE-H SY-801

1142 APPENDIX D SYMPLOSTATIN-1 SYZYGIOL T-0128 T-121-B T-138067 T-23 T-900607 T-98 TA-077 TACHPYRIDINE TAGITININ-C TAGITININ-F TALISOMYCIN TALISOMYCIN-B TALISOMYCIN-S10B TALLIMUSTINE TAMARIXININ-A TAMOXIFEN METHIODIDE TAN-1518-A TANTAZOLE-A TANTAZOLE-B TAPP-BR TAPP-H TAS-103 TAURINE-MUSTARD TAUROMUSTINE TAUTOMYCIN TAXODIONE TAXOL-C TAXOTERE TAXUSPINE-D TBI-361 TECTORIDIN TEGAFUR TEI-9826 TELEKIN TELOMESTATIN TELOXANTRONE TEMAROTENE TEMOZOLOMIDE TENIPOSIDE TENIPOSIDE-QUINONE-O TENUAZONATE TEPA TER-286 TERFLURANOL TEROXIRONE TERPENTECIN TESMILIFENE TESTIPHENONE TESTOLACTONE TETRADECYLPHOSPHOCHOLINE TETRAHYDRODAIDZEIN-CIS TETRAMETHYLSCUTELLAREIN TETRAMETHYLUREA TETRAMIN TETRAZOMINE TETROCARCIN-A TEURILENE THALICARPINE THALICOSIDE-A THALIFABERINE THALRUGOSINE THEONELLADIN-A THEONELLADIN-B THEONELLADIN-C THEONELLADIN-D THEONELLAPEPTOLIDE-ID THEONEZOLIDE-A THERMINE THEVETOSIDE THIAZINOTRIENOMYCIN-B THIOASTIN-B THIOCOLCHICINE THIOCORALINE THIOCYANATONEOPUPU= KEANANE-2 THIODIGLYCOL THIODIPIN THIOGUANOSINE THIOGUANOSINE-= MONOPHOSPHATE THIOPHENFURINE THIOPLATIN THIOTEPA THIOURIDINE-4 THIOXANTHINE-6 THIOXANTHINE-RIBOTIDE THORECTANDROL-A THORECTANDROL-B THUJAPLICIN-BETA THYRSIFEROL THYRSIFERYL-ACETATE-23 TIAMIPRINE TIAZOFURINE TIAZOFURINE-ADENINE-= DINUCLEOTIDE TIAZOFURINE-PHOSPHATE TILIVALLINE TIOGUANINE TIPIFARNIB TIPIFARNIB TIRAPAZAMINE TITANOCENE-DIBROMIDE TITANOCENE-DICHLORIDE TK-5477 TMC-151-A TMC-151-B TMC-151-C TMC-151-D TMC-151-F TMC-69 TN-16 TNF-RELATED-APOPTOSIS-= INDUCING-LIGAND TNO-38 TNP-351 TOK-4528 TOLYPORPHIN-A TOLYTOXIN TOMAYMYCIN TOMIZINE TOP-53 TOPOTECAN TOPSENTIN TORILIN TOSITUMOMAB TOYOCAMYCIN TP-151 TP-40 TP-69 TP-72 TRAMETENOLATE TRANSFORMING-GROWTH-= FACTOR-ALPHA-PE40 TRANSFORMING-GROWTH-= FACTOR-B1-CATTLE TRANSFORMING-GROWTH-= FACTOR-B2-CATTLE TRANSFORMING-GROWTH-= FACTOR-BETA TRANSFORMING-GROWTH-= FACTOR-BETA-1 TRAPOXIN-A TREOSULFAN TRESTOLONE TRESTOLONE-ACETATE TRETAMINE TREWIASINE TRIACETYLDYNEMICIN-A TRIACETYLSCIRPENETRIOL TRIAPINE TRIAZINATE TRIAZIQUONE TRIBETAMIDE TRICHLORMETHINE TRICHODERMIN TRICHOKIRIN TRICHORABDAL-A TRICHORABDAL-B TRICHORABDAL-C TRICHORABDAL-D TRICHORABDAL-F-ACETATE TRICHORABDAL-G-ACETATE TRICHOSTATATE TRICHOSTATIN-A TRICIN TRICIRIBINE TRICIRIBINE-PHOSPHATE TRICOLORIN-A TRIENOMYCIN-A TRIENOMYCIN-B TRIENOMYCIN-C TRIFLUOROMETHYLDEOXY= CYTIDINE TRIFLUOROMETHYLHOMO= CYSTEINE TRIFLURIDINE TRIFLURIDINE-PHOSPHATE TRILOBACIN TRILOBOLIDE TRIMELAMOL TRIMETHYLCOLCHICINATE TRIMETREXATE TRIMIDOX TRIPDIOLIDE TRIPHENYLSELENONIUM= CHLORIDE TRIPTOLIDE TRK-710 TROFOSFAMIDE TRYPROSTATIN-A TRYPROSTATIN-B TRYPTOPHAN-2,3-= DIOXYGENASE TST-220 TST-334 TT-232 TUBEIMOSIDE-I TUBEIMOSIDE-III TUBERCIDIN TUBERCIDIN-= MONOPHOSPHATE TUBULOZOLE TULIPALIN-A TUMOR-INVASION-= INHIBITING-FACTOR-2 TUMOR-NECROSIS-FACTOR TUMOR-NECROSIS-FACTOR-= ALPHA TUMOR-NECROSIS-FACTOR-= ALPHA-BETA TUMOR-NECROSIS-FACTOR-= ALPHA-CATTLE TUMOR-NECROSIS-FACTOR-= ALPHA-HUMAN TUMOR-NECROSIS-FACTOR-= ALPHA-MOUSE TUMOR-NECROSIS-FACTOR-= BETA TUMOR-NECROSIS-FACTOR-= BETA-HUMAN TUMOR-NECROSIS-FACTOR-= HUMAN TUMOR-NECROSIS-FACTOR-= MOUSE TUMOR-NECROSIS-FACTOR-= S-AM2-HUMAN TUMOR-NECROSIS-FACTOR-= SAM2 TUMSTATIN TURMERONE-AR TW-13 TW-19 TW-22

Derwent Drug File 1143 Thesaurus TW-25 TW-26 TW-32 TW-39 TW-50 TX-1123 TX-1856 TX-522 TX-527 TYLOCREBRINE TYLOPHORINE TYLOPHORINIDINE TYLOPILAN TYRPHOSTIN-A-23 TYRPHOSTIN-A-47 TZ-93 TZT-1027 U-108333-E U-62736 U-63360 U-66226 U-66664 U-66694 U-66866 U-67786 U-68415 U-68819 U-71184 U-72799 U-75559 U-76074 U-76579 U-76915 UCE-1022 UCE-6 UCF-1-C UCH-9 UCN-01 UCN-02 UCT-4B UK-1 (Cytostatic) UK-2-A UK-21 UK-25 ULITHIACYCLAMIDE UNCARINE-C UNCARINE-E UNGEREMINE URAMUSTINE URDAMYCINONE-B UREDEPA URETHANE URICYTIN UROGUANYLIN UROTERPENOL USTILOXIN-D UVARETIN VALANIMYCIN VANADOCENE-DICHLORIDE VANOXONIN VARACIN VARAMINE-A VARAMINE-B VARIABILIN VARIAMYCIN VARIOLIN-B VATALANIB VATDIOSPYROIDOL VELLERAL VELUTIN VERACTAMYCIN-A VERACTAMYCIN-B VERMIXOCIN-A VERMIXOCIN-B VERNOLEPIN VERNOMENIN VEROTOXIN-1 VEROTOXIN-2 VERRUCARIN-A VERRUCARIN-J VERUCOPEPTIN VF-122 VF-147 VICENISTATIN VIDARABINE VIDARABINE-ACETATE VIDARABINE-DIACETATE2+,3+ VIDARABINE-OCTANOATE VIDARABINE-PHOSPHATE VIDARABINE-TRIPHOSPHATE VIDARABINE-VALERATE VINBLASTINE VINBLASTINE-ISOLEUCINATE VINCRISTINE VINDESINE VINEOMYCIN-A1 VINEPIDINE VINESTRAMIDE VINFLUNINE VINFORMIDE VINFOSILTINE VINGLYCINATE VINLEUCINOL VINLEUROSINE VINORELBINE VINROSIDINE VINTRIPTOL VINZOLIDINE VIOLAMYCIN VIROSECURININE VIRULIZIN VITAXIN VN-85-1 VN-87-1 VNP-20009 VOROZOLE VRCTC-310-ONCO VX-497 W-68 WAKAYIN WAY-140424 WB-4291 WB-608 WF-3161 WHI-P-131 WHI-P-154 WHI-P-353 WHI-P-97 WHK-BF-1 WIKSTROMOL WIN-32950 WIN-33123 WIN-33156 WIN-33377 WIN-58161 WIN-63320 WIN-64593 WITHANGULATIN-A WITHANOLIDE-D WITHASOMNINE WMC-26 WOODFORDIN-A WOODFORDIN-C WOODFORDIN-D WP-401 WP-546 WP-549 WP-608 WP-631 WP-652 WU-345 WV-15 WX-360 WX-UK-1 WY-13876 XANTHENONE-ACETATE-4 XANTHOCHYMOL XANTHORRHIZOL XB-596 XK-469 XR-11576 XR-5944 XR-5967 XR-9576 XYLOTUBERCIDIN Y-18598 Y-27632 YADANZIOSIDE-A YADANZIOSIDE-B YADANZIOSIDE-C YADANZIOSIDE-D YADANZIOSIDE-E YADANZIOSIDE-F YADANZIOSIDE-G YADANZIOSIDE-H YADANZIOSIDE-I YADANZIOSIDE-J YADANZIOSIDE-L YADANZIOSIDE-P YAKUCHINONE-B YELLAMYCIN-A YELLAMYCIN-B YELLAMYCIN-C YH-439 YLL-224 YM-30059 YM-47522 YM-534 YNKO-1 YOMOGIARTEMIN YOMOGIN YOSHIXOL YUANHUACINE Z-100 ZAHAVIN-A ZD-1839 ZD-2767 ZD-2767-D ZD-2767-P ZD-4190 ZD-6126 ZD-9331 ZEBULARINE ZENIPLATIN ZERUMBONE ZILASCORB (2H) ZINOSTATIN ZINOSTATIN-POLY-STYRENE-= MALEATE ZIRCONOCENE-DICHLORIDE ZK-156718 ZK-191703 ZL-III-43-A ZM-249148 ZM-252868 ZM-258754 ZOLEDRONATE ZORUBICIN DELUSIONAL-DISORDER EROTOMANIA PARANOIA paranoid-schizophrenia PARAPHRENIA DEMENTIA ALZHEIMER-DISEASE ALZHEIMER-DISEASE KLUVER-BUCY-SYNDROME DEMYELINATING-DISEASE BALO-DISEASE

1144 APPENDIX D GLOBOID-CELL-= LEUKODYSTROPHY HALLERVORDEN-SPATZ-= SYNDROME METACHROMATIC-= LEUKODYSTROPHY MULT.SCLEROSIS OPTIC-NEUROMYELOPATHY SCHILDER-DISEASE DEODORANTS LIMONENE DERMATOLOGY ACANTHOLYSIS ACANTHOSIS ACNE ACRODERMATITIS ACROKERATOSIS ACROPUSTULOSIS acute-parapsoriasis ALVELD ANETODERMA ANGIODERMATITIS athletes foot atopic-dermatitis atopic-eczema BACTERID bedsore BLISTER bowen-disease BULLA CAMELPOX CARBUNCLE CHROMOBLASTOMYCOSIS CHROMOMYCOSIS CHRYSIASIS COLLOID-MILIUM COMEDO CONDYLOMA condyloma-acuminatum congenital-dyskeratosis contact-dermatitis COWPOX decubitus-ulcer degos-delort-tricot-syndrome DERMATITIS dermatitis-herpetiformis DERMATOLYSIS DERMATOMYOSITIS DERMATOPHILOSIS DERMATOPHYTOSIS DERMATOPOLYNEURITIS DERMATOSIS DYSKERATOSIS ECTHYMA ECZEMA EPIDERMODYSPLASIA EPIDERMOLYSIS EPIDERMOLYSIS-BULLOSA EPITHELIOLYSIS ERYSIPELAS ERYTHEMA ERYTHEMA-CHOLINERGIC ERYTHEMA-ELEVATUM-= DIUTINUM ERYTHRASMA ERYTHRODERMA ERYTHRODYSESTHESIA-= SYNDROME ERYTHROKERATODERMIA ERYTHROKERATODERMIA-= VARIABILIS EXUD.DIATHESIS EXUD.EPIDERMITIS familial-benign-pemphigus FIXED-ERUPTION FOLLICULITIS FOX-DISEASE FOX-FORDYCE-DISEASE FROSTBITE FURUNCLE FURUNCULOSIS GOUGEROT-BLUM-= SYNDROME hailey-hailey-disease hallopeau-syndrome hand-foot-syndrome HELOMA herpes-gestationis HIDRADENOMA HORSEPOX HYDROA HYPERKERATOSIS ICHTHYOSIS IMPETIGO INTERTRIGO KELOID KERATOACANTHOMA KERATODERMA KERATOMA KERATOSIS LEWANDOWSKY-LUTZ-= SYNDROME LICHEN (disease) LOEFGREN-SYNDROME LUMPY-SKIN-DISEASE LUPOID-ULCER LUPUS-VULGARIS MAJOCCHI-DISEASE MAL-DE-MELEDA malignant-atrophic-papulosis malignant-erythema-= multiforme MELANODERMA melanoma, skin MELASMA MELEDA-DISEASE mesnier-prurigo MILIARIA MILIUM MOLLUSCUM-= CONTAGIOSUM mucha-habermann-syndrome MUCINOSIS MYCOSIS-FUNGOIDES NECROBIOSIS-LIPOIDICA NETHERTON-DISEASE nettlerash neumann-disease neurodermatitis NEVUS NODULAR-ELASTOIDOSIS ORF PAPULE PAPULOSIS PARAKERATOSIS PARAPSORIASIS PEMPHIGOID PEMPHIGUS pemphigus-erythematosus pemphigus-vegetans PHOTODERMATITIS PHOTODERMATOSIS PHRYNODERMA PIGEONPOX PIGPOX PILONIDAL-SINUS PINTA PITYRIASIS PODODERMATITIS POIKILODERMA POMPHOLYX POROKERATOSIS POROMA PORPHYRIA-CUTANEA-TARDA precancerous-dermatosis PRURIGO PSEUDO-COWPOX PSEUDOPORPHYRIA PSEUDOXANTHOMA-= ELASTICUM PSORIASIS pustular-dermatitis PUSTULOSIS PYODERMA RADIODERMATITIS RASH RICHNER-HANHART-= SYNDROME ROSACEA SAPHO-SYNDROME SCABIES schaefer-syndrome SEBORRHEA seborrheic-eczema senear-usher-syndrome SEZARY-SYNDROME SIEMENS-SYNDROME skin-melanoma sneddon-wilkinson-syndrome SPANLANG-TAPPEINER-= SYNDROME STEATOMATOSIS stevens-johnson-syndrome STRIAE-ATROPHICAE subcorneal-pustular-= dermatosis SULZBERGER-GARBE-= SYNDROME SUNBURN SWEET-SYNDROME SYCOSIS-VULGARIS SYRINGOCYSTADENOMA THIBIERGE-WEISSENBACH-= SYNDROME TINEA TOX.EPIDERMAL-NECROLYSIS TRICHOEPITHELIOMA unna-disease UNNA-THOST-SYNDROME URTICARIA URTICARIA-CHOLINERGIC UVEOMENINGEAL-= SYNDROME VESICULAR-EXANTHEMA WART WELLS-SYNDROME WINTER-ULCER XERODERMA zinsser-engman-cole-= syndrome DESENSITIZERS ALLERGOVIT ALLERKIN ALLPYRAL ALPARE ALUTARD ANJUVAC BRL-42245 CONJUVAC HEPP IPOINAL PHARMALGEN POLINEX POLLINEX PURETHAL SPECTRALGEN TYROSIN-ALLERGOID DIABETES DAWN-PHENOMENON diabetic-retinopathy

Derwent Drug File 1145 Thesaurus DIAGNOSIS ANGIOCARDIOGRAPHY ANGIOGRAPHY AORTOGRAPHY APEXCARDIOGRAPHY ARTERIOGRAPHY ARTHROGRAPHY ARTHROSCOPY BALLISTOCARDIOGRAPHY BRONCHOSCOPY CAPILLAROSCOPY CAPNOGRAPHY CARDIOGRAPHY CARDIOTOCOGRAPHY CAVERNOSOGRAPHY CHOLANGIOCHOLE= CYSTOGRAPHY CHOLANGIOCYSTOGRAPHY CHOLANGIOGRAPHY CHOLANGIOPANCREATO= GRAPHY CHOLECYSTOGRAPHY CINEANGIOGRAPHY CISTERNOGRAPHY COLONOSCOPY COLPOSCOPY CRANIOCORPOGRAPHY CYSTOSCOPY CYSTOURETHROGRAPHY CYTODIAGNOSIS CYTOSCOPY ECHOCARDIOGRAPHY ECHOSCOPY ELECTROCORTICOGRAPHY ELECTROGASTROGRAPHY ELECTRORETINOGRAPHY ELECTROSPINOGRAPHY ENCEPHALOGRAPHY ENDOSCOPY EPIDUROGRAPHY FIBEROSCOPY GASTROSCOPY HOESCH-TEST HYSTEROSALPINGOGRAPHY HYSTEROSCOPY LAPAROSCOPY LARYNGOSCOPY LYMPHANGIOGRAPHY LYMPHOGRAPHY MISDIAGNOSIS MYELOGRAPHY MYOGRAPHY OPHTHALMOSCOPY PANCREATOGRAPHY PATCH-TEST PHALLOGRAPHY PHLEBOGRAPHY PLETHYSMOGRAPHY PLEUROGRAPHY PNEUMOENCEPHALOGRAPHY PNEUMOVENTRICULOGRAPHY PORTOGRAPHY PYELOGRAPHY RHEOGRAPHY RORSCHACH-TEST SCHILLING-TEST SCINTILLOGRAPHY SIALOGRAPHY SIGMOIDOSCOPY SONOGRAPHY SPLENOPORTOGRAPHY THERMOGRAPHY THORN-TEST THROMBOELASTOGRAPHY THROMBOGRAPHY TOMODENSITOMETRY TOMOGRAPHY TUSSOMETRY TZANCK-TEST ULTRASONOGRAPHY UROGRAPHY VECTORCARDIOGRAPHY VENOGRAPHY VENTRICULOGRAPHY DIAGNOSTICS ACETAMIDOHIPPURATE-PARA ACHOLEST ACU-TEST AMERLEX AMINOHIPPURATE ANAZOLENE SODIUM ANSWER ARCLOFENIN BASOKIT BENPENOLISIN BENTIROMIDE BETA-NEOCEPT BETAZOLE BIOPHAN-C BROMSULFALEIN BUTILFENIN CHEMSTRIP-BG CLINISTIX CLINITEST COMBOSTAT-2 CONGO-RED CYTUR-TEST DAISY-2 DEXTROSTIX DIABUR-5000 DIASTIX DIBROMSULFALEIN DISOFENIN DUALCOUNT E.P.T. ECHOCON ECUR-4-TEST ENZYGNOST-RUBELLA ETIFENIN FE-CULT FECATEST FECATWIN FECATWIN-SENSITIVE FLUORESCEIN FLUORESCEIN-DILAURATE FLUORODEOXYGLUCOSE-2 GLUCOHEPTONATE GYNAEGNOST HAEMOGLUKOTEST HEMAFECIA HEMOCCULT HEMOQUANT IMMOPHASE INDOCYANINE-GREEN IODOESTRADIOL-16-ALPHA IOMETIN KETODIASTIX KETOSTIX LIDOFENIN MEBROFENIN MERCKOGNOST MONOTEST N-LABSTIX N-MULTISTIX NEOCUPROINE NEPHUR-TEST PAH PENTETATE PHADEBAS PHADEBAS-AMYLASE-TEST PHENOLSULFONPHTHALEIN PREDICTOR PREGNASTICK QUANTAPHASE RAPIGNOST-AMYLASE RAPIGNOST-BASIS-SCREEN REFLOCHECK REFLOLUX ROTAZYME SIMULTRAC STAT-TEK SUCCIMER TES-TAPE TEST-TAPE THROMBOFAX TRILUTE VISIDEX DIET HYPERALIMENTATION THERAPEUTIC-FASTING DIGESTANTS ACID-PHOSPHATASE AGALSIDASE-ALPHA AMAFERM CELLULASE CHOLENZYME ENDO-1,3(4)-BETA-D-= GLUCANASE ENZYNORM GLUCANASE-BETA KEMZYME NORTASE PANCREATIN PANCRELIPASE VITA-FERM XYLANASE DISPERSION MIST DIURETICS A-49816 A-56234 A-68828 ABBOTT-56234 ABT-702 ACEFYLLINE ACEFYLLINE-PIPERAZINE ACETAZOLAMIDE ALIPAMIDE ALTIZIDE AMANOZINE AMBUPHYLLINE AMBUSIDE AMILORIDE AMINOMETRADINE AMINOPHYLLINE AMISOMETRADINE AMMONIUM-ACETATE AMPHENONE AMPYRIMINE ANARITIDE AP-539 AP-811 APIOL ARBUTIN ATRIAL-NATRIURETIC-FACTOR ATRIAL-NATRIURETIC-= FACTOR-1-24-RAT ATRIAL-NATRIURETIC-= FACTOR-104-126-RAT ATRIAL-NATRIURETIC-= FACTOR-105-126-HUMAN ATRIAL-NATRIURETIC-= FACTOR-105-126-RAT ATRIAL-NATRIURETIC-= FACTOR-54-126 ATRIAL-NATRIURETIC-= FACTOR-8-33 ATRIAL-NATRIURETIC-= FACTOR-8-33-HUMAN

1146 APPENDIX D ATRIAL-NATRIURETIC-= FACTOR-A-HUMAN-1-11 ATRIAL-NATRIURETIC-= FACTOR-A-HUMAN-18-28 ATRIAL-NATRIURETIC-= FACTOR-A-HUMAN-5-28 ATRIAL-NATRIURETIC-= FACTOR-A-HUMAN-7-28 ATRIAL-NATRIURETIC-= FACTOR-ALPHA ATRIAL-NATRIURETIC-= FACTOR-ALPHA-RAT ATRIAL-NATRIURETIC-= FACTOR-BETA-+-HUMAN ATRIAL-NATRIURETIC-= FACTOR-BETA-HUMAN ATRIAL-NATRIURETIC-= FACTOR-C-HUMAN ATRIAL-NATRIURETIC-= FACTOR-C-RAT ATRIAL-NATRIURETIC-= FACTOR-GAMMA-HUMAN ATRIAL-NATRIURETIC-= FACTOR-HUMAN ATRIAL-NATRIURETIC-= FACTOR-I-RAT ATRIAL-NATRIURETIC-= FACTOR-II ATRIAL-NATRIURETIC-= FACTOR-III-RAT ATRIAL-NATRIURETIC-= FACTOR-IV-RAT ATRIAL-NATRIURETIC-= FACTOR-RAT ATRIAL-NATRIURETIC-= FACTOR-RAT-13-28 ATRIAL-NATRIURETIC-= PEPTIDE-79-98 ATRIOPEPTIN ATRIOPEPTIN-I ATRIOPEPTIN-II ATRIOPEPTIN-II-AMIDE ATRIOPEPTIN-III AURICULIN-A AZOLIMINE AZOSEMIDE BAROKATON BAX-439 BAY-N-1468 BEMETIZIDE BEMITRADINE BENDROFLUMETHIAZIDE BENZMETANIDE BENZOLAMIDE BENZTHIAZIDE BENZYLHYDROCHLORO= THIAZIDE BESULPAMIDE BESUNIDE BM-106 BM-15 BM-17 BM-20 BM-24 BN-50157 BRAIN-NATRIURETIC-= PEPTIDE-32-HUMAN BRAIN-NATRIURETIC-= PEPTIDE-32-RAT BRAIN-NATRIURETIC-= PEPTIDE-45-RAT BRAIN-NATRIURETIC-= PEPTIDE-PIG BRAIN-NATRIURETIC-= PEPTIDE-PIG-32 BROCRINAT BUMETANIDE BUTAZOLAMIDE BUTIZIDE C-3534 C-3535 C-TYPE-NATRIURETIC-= PEPTIDE C3-76 CAFFEINE CAFFEINE-SODIUM-= BENZOATE CAFFEINE-SODIUM-= SALICYLATE CANDOXATRILAT CANRENOATE CANRENOATE POTASSIUM CANRENONE CANTHARIDIN CARMETIZIDE CARPERITIDE CARZENIDE CHLORAZANIL CHLORMERODRIN CHLOROTHIAZIDE CHLORTALIDONE CHOLINE-THEOPHYLLINATE CICLETANINE CL-13580 CL-5343 CLAZOLIMINE CLOFENAMIDE CLOPAMIDE CLOREXOLONE CVT-124 CYCLOHEXYLSUBERO= GORGAMIDE-N CYCLOPENTHIAZIDE CYCLOTHIAZIDE DEHYDROCHOLATE DENDROASPIS-= NATRIURETIC-PEPTIDE DEXTRONATRIN DICIRENONE DICLOFENAMIDE DIMETHAZAN DIPHENYLMETHANE= SULFONAMIDE DISULFAMIDE DR-3438 DS-210 DS-511 EPITIZIDE EPLERENONE ER-32935 ETACRYNATE ETAMIPHYLLIN ETHIAZIDE ETHOXYZOLAMIDE ETOZOLIN FENOLDOPAM FENQUIZONE FK-838 FLUMETHIAZIDE FORMONONETIN FR-161282 FURACRINATE FUROSEMIDE FURTERENE GALOSEMIDE GLYCERYLNONIVAMIDE GOE-5584-A GOE-6070 H-5350 HEXAMETHYLENE-= AMILORIDE-5 HYDRACARBAZINE HYDROBENTIZIDE HYDROCHLOROTHIAZIDE HYDROFLUMETHIAZIDE HYDROXINDASATE HYDROXYTRIAMTERENE-= PARA IBOPAMINE ICI-206970 ICI-207828 INDACRINONE INDAPAMIDE IODOAMILORIDE-6 IRL-1620 ISOSORBIDE JTV-605 KF-15372 KW-3902 L-589420 L-593511 L-632481 L-643799 L-645151 LEIOCARPOSIDE LEMIDOSUL LESPENEPHRYL M-12285 M-17055 MANNITOL MDL-100173 MDL-100240 MEBUTIZIDE MEDULLIPIN-I MEFRUSIDE MERALLURIDE MERBIURELIDIN MERCAPTOMERIN MERCUDERAMIDE MERCUMATILIN SODIUM MERCUROPHYLLINE MERSALYL METHALTHIAZIDE METHAZOLAMIDE METHYCLOTHIAZIDE METICRANE METIPAMIDE METOLAZONE METYRAPOL METYRAPONE MEXRENOATE POTASSIUM MJ-8592-1 MK-447 MK-473 MK-597 MUZOLIMINE NATRIURETIC-HORMONE NIRAVOLINE NNC-70-0270 NOC-7 OPC-31260 OXPRENOATE POTASSIUM OZOLINONE P-275 PAMABROM PARAFLUTIZIDE PENFLUTIZIDE PENTIFYLLINE PIRETANIDE POLYTHIAZIDE POLYURENE POMISARTAN PRAMIPEXOLE PROPAZOLAMIDE PRORENOATE POTASSIUM PROTHEOBROMINE PYTAMINE QUINCARBATE QUINETHAZONE RB-105 RO-14-9012 RO-64-6198 RPH-2823 S-8666 SA-7090

Derwent Drug File 1147 Thesaurus SC-16100 SC-16102 SKF-100273 SKF-100398 SKF-100501 SKF-100885 SKF-101071 SKF-101485 SKF-101496 SKF-101497 SKF-101498 SKF-101926 SKF-17467 SKF-R-87516 SORBITOL SPIRONOLACTONE SPIROXASONE SQ-27786 SQ-46542 SR-121463-B SR-144528 SU-15049 SULCLAMIDE SULICRINAT SULOCARBILATE SUMETIZIDE TECLOTHIAZIDE THEOBROMINE THEOBROMINE-= SALICYLATE-SODIUM THEOBROMINE-SODIUM-= ACETATE THEOPHYLLINE THEOPHYLLINE-LYSINE THEOPHYLLINE-SODIUM-= ANISATE THEOPHYLLINE-SODIUM-= GLYCINATE TIAMIZIDE TIENILATE TIENOXOLOL TIZOLEMIDE TORASEMIDE TRAXANOX TRIAMTERENE TRICHLORMETHIAZIDE TRIFLOCIN TRIFLUORMETHAZOLAMIDE TRIPAMIDE TROMETAMOL U-1003 U-18177-A U-2113 U-38658-A UK-69578 URODILATIN VASONATRIN-PEPTIDE VP-343 WAY-VPA-985 WY-5256 XIPAMIDE YM-430 YM-435 ZP-120-C DNA-INTERCALATORS ACTINOMYCIN AMSACRINE BISNAFIDE BROSTALLICIN CI-958 DAUNORUBICIN DOXORUBICIN ECHINOMYCIN ESPERAMICIN HOMIDIUM BROMIDE IDARUBICIN JM-473 KW-2170 LU-79553 MITOXANTRONE NOGALAMYCIN NSC-655649 PD-115934 DOPA-DECARBOXYLASEINHIBITORS BENSERAZIDE CARBIDOPA MDL-71801 NSD-1015 NSD-1024 NSD-1034 RO-4-5127 DOPAMINE-ANTAGONISTS 1192-U-90 A-37850 A-69024 ACEPERONE ACEPROMAZINE ACETOPHENAZINE AD-5423 AD-8112 AHR-1709 AJ-76 ALIMEMAZINE ALPIROPRIDE AMISULPRIDE AZAPERONE AZAPRIDE BALAPERIDONE BENPERIDOL BENZQUINAMIDE BRL-20596 BRL-25594 BRL-34778 BROMOLISURIDE-2 BROMOSPIPERONE-PARA BROMPERIDOL BROMPERIDOL-DECANOATE BUTACLAMOL BUTAPERAZINE BW-737-C CARFENAZINE CHLOROETHYLNORAPO= MORPHINE CHLOROSCOULERINE-12 CHLORPROMAZINE CHLORPROMAZINE-= METHIODIDE CHLORPROTHIXENE CICLOFENAZINE CITATEPINE CLOFLUPEROL CLOMACRAN CLOPENTHIXOL CLOPENTHIXOL-DECANOATE CLOPIMOZIDE CLOPITHEPIN CLOROTEPINE CLOTIAPINE CLOTIXAMIDE CLOZAPINE CP-293019 CP-88059 DEMETHYLLEVOME= PROMAZINE-O DEMETHYLNEMONAPRIDE-N DIHYDROBENPERIDOL DIHYDROTETRABENAZINE DIHYDROWISANINE DIMETPRAMIDE DO-710 DOMPERIDONE DROPERIDOL DS-121 DU-29894 EGYT-2474 EGYT-2509 ERIZEPINE ETHOMOXANE ETICLOPRIDE F-1603 F-1806 F-1808 FENTANYL-ISOTHIOCYANATE FLA-659 FLA-797 FLA-873 FLA-908 FLA-961 FLA-988 FLB-457 FLB-463 FLB-472 FLB-524 FLUANISONE FLUMEZAPINE FLUPENTIXOL FLUPENTIXOL-DECANOATE FLUPHENAZINE FLUPHENAZINE-DECANOATE FLUPHENAZINE-ENANTHATE FLUSPIPERONE FLUSPIRILENE GABA-LINOLEAMIDE GBR-12783 GR-103691 H-44-68 HALOPERIDOL HALOPERIDOL-DECANOATE HOMOFENAZINE HP-236 HP-370 HPP HSR-803 HYDROXYCHLOR= PROMAZINE-3 HYDROXYLEVOME= PROMAZINE-3 HYDROXYLEVOME= PROMAZINE-7 ILOPERIDONE IMICLOPAZINE IODOAZAPRIDE IODOCLEBOPRIDE IODOSULPRIDE ISOBUTACLAMOL L-646462 L-741626 L-741742 L-745870 L-750667 LE-300 LEK-8829 LENPERONE LEVOMEPROMAZINE LEVOSULPIRIDE LOXAPINE LU-13-117 LU-14-068 LU-17-123 LU-17-151 LU-17-152 LU-18-006 LUR-2366 LUZINDOLE MAFOPRAZINE MAROXEPIN MEMANTINE MESORIDAZINE METHOPROMAZINE

1148 APPENDIX D METHYLSPIPERONE METOCLOPRAMIDE METOFENAZATE METOPIMAZINE MEZILAMINE MILENPERONE MILIPERTINE MJ-13980-1 MOLINDONE MOPERONE MOSAPRAMINE MS-377 NAFADOTRIDE NCQ-115 NCQ-318 NCQ-344 NCQ-436 NCQ-616 NEFLUMOZIDE NEMONAPRIDE NGD-94-1 NNC-01-0687 NNC-0112 NNC-22-0010 NNC-22-0031 NNC-22-0215 NO-01-0756 NORCHLORPROMAZINE NORTHIORIDAZINE NRA-0045 NRA-0160 NRA-0161 NRA-0215 NRA-0562 OCAPERIDONE OLANZAPINE OPC-14597 OPC-4392 OSU-6162 OXIPEROMIDE OXYPERTINE P-9236 PD-152255 PD-158771 PD-172760 PENFLURIDOL PENTIAPINE PERICIAZINE PERLAPINE PERPHENAZINE PERPHENAZINE-DECANOATE PERPHENAZINE-ENANTHATE PIFLUTIXOL PIMOZIDE PINOXEPIN PIPAMAZINE PIPAMPERONE PIPERACETAZINE PIQUINDONE PROCHLORPERAZINE PROMAZINE PROPIOMAZINE PROPYPERONE PSD-958 QF-0307-B QF-0313-B QM-7184 QUETIAPINE R-2572 R-48455 RACLOPRIDE RED.HALOPERIDOL REMOXIPRIDE RESERPINE RISPERIDONE RMI-11974 RO-22-6600 ROMERGOLINE RTI-55 RU-41656 RWJ-37796 S-14297 S-18327 SARIZOTAN SAVOXEPIN SB-277011 SCH-12679 SCH-15199 SCH-23388 SCH-23390 SCH-38840 SCH-39165 SCH-39166 SCH-40853 SCH-66712 SDZ-212-327 SEROQUEL SETOPERONE SH-3-24 SKF-103108A SKF-7172A SKF-83566 SKF-83692 SKF-83742 SM-13496 SND-919 SOLYPERTINE SPIPERONE SPIRAMIDE SPIRILENE ST-1460 SULPIRIDE TAK-218 TEFLUTIXOL TEPIRINDOLE TETRABENAZINE THIETHYLPERAZINE THIOPROPERAZINE THIORIDAZINE THIORIDAZINE-= DISULFOXIDE-2,5 THIORIDAZINE-OXIDE-5 TIOPERIDONE TIOSPIRONE TIOTIXENE TRIFLUOPERAZINE TRIFLUPERIDOL TRIFLUPROMAZINE TROPAPRIDE U-101387 U-101958 U-99194-A U-99363-E UH-232 UH-242 VERALIPRIDE Y-20024 YM-0850 YM-43611 ZETIDOLINE ZUCLOPENTHIXOL ZUCLOPENTHIXOL-ACETATE ZUCLOPENTHIXOL-= DECANOATE DOPAMINERGICS 201-403 201-678 205-501 A-68930 A-77636 A-85380 A-86929 AB-118 AB-85 ABT-431 ADTN AGROCLAVINE ALENTEMOL ALNESPIRONE APOMORPHINE AR-C-68397-AA AS-8 BAM-1110 BAM-1303 BAZINAPRINE BRL-16657 BROMERGURIDE BROMOCRIPTINE BROMOERGOSINE BY-101 CABERGOLINE CARMOXIROLE CGP-3466-B CGS-15855A CGS-15873A CHF-1035 CI-1007 CI-201-678 CILADOPA CQA-206-291 CS-263 CS-265 CY-208-243 DCN-203-922 DELERGOTRILE DICLOFENSINE DIETHYLDOPAMINE-N,N DIHYDREXIDINE DIHYDROERGOCORNINE DIHYDROERGOCRISTINE DIHYDROERGOCRYPTINE DIHYDROERGOCRYPTINE-= ALPHA DIHYDROERGOCRYPTINE-= BETA DIHYDROERGOSINE DIHYDROERGOSININE DIHYDROERGOTOXINE DIMETHYLDOPAMINE-N,N DIPROPYLDOPAMINE-N,N DISULERGINE DK-118 DO-897 DOCARPAMINE DOPAMINE DOPEXAMINE DU-127090 ELYMOCLAVINE EMD-23448 EMD-38362 ERGOCORNINE ERGOCRISTINE ERGOCRYPTINE ERGOCRYPTINE-ALPHA ERGOCRYPTINE-BETA ERGOMETRINE ERGOSINE ERGOSININE ERGOTOXINE ERGOVALINE ETISULERGINE FCE-22716 FCE-27395 FENOLDOPAM FLUORODOPAMINE-6 FPL-63012AR GBR-11513 GBR-12909 GBR-12922 GBR-12935 GBR-13069

Derwent Drug File 1149 Thesaurus GBR-13098 GBR-13119 GK-13 GLIAL-CELL-DERIVED-= NEUROTROPHIC-FAC.HUM GLIAL-CELL-DERIVED-= NEUROTROPHIC-FAC.RAT GLIAL-CELL-DERIVED-= NEUROTROPHIC-FACTOR GLUDOPA GMC-1-169 GYKI-32887 GYKI-35064 HA-117 HA-118 HA-97 HW-165 HYDROXYDIPROPYLAMINO= TETRALIN-7 HYDROXYMETHYL= PHENIDATE-PARA IBOPAMINE ISOAPOMORPHINE JGC-174 JMB-249 JOD-173 JPC-266 KSU-1415 LERGOTRILE LEVODOPA LEVODOPA-METHYL-ESTER LISURIDE LU-24-040 LY-062 LY-137157 LY-141865 LY-149179 LY-156525 LY-158A LY-175877 LY-202475 LY-202991 LY-202992 LY-206243 LY-254490 MASTODYNON MERGOCRIPTINE MESULERGINE MPTP N-0425 N-0434 N-0435 N-0436 N-0437 N-0438 N-0498 N-0499 N-0918 N-0923 NAXAGOLIDE NB-355 NO-434 NO-437 NOMIFENSINE NORAPOMORPHINE NS-2359 OPC-14597 PD-118717 PD-119819 PD-128907 PD-143188 PD-158771 PERGOLIDE PIRIBEDIL PR-000001 PR-000608 PRAMIPEXOLE PRECLAMOL PROPYLBUTYLDOPAMINE PROTERGURIDE QUINAGOLIDE QUINELORANE QUINPIROLE RD-219 RDS-127 RO-41-9067 ROMERGOLINE ROPINIROLE ROXINDOLE RS-25560-197 RU-24213 RU-24926 RU-29717 RU-41656 S-3608 SANDOZ-27403 SDZ-212-327 SIB-1765-F SKF-28393 SKF-38393 SKF-38393-A SKF-75670 SKF-77434 SKF-80723 SKF-81297 SKF-82957 SKF-82958 SKF-83189 SKF-83565 SKF-83959 SKF-85174 SKF-85738 SKF-88827 SKF-89124 SKF-89615 SKF-89626 SKF-R-105058 SKF-R-106114 SKF-R-87516 ST-1943 SUNEPITRON TERGURIDE TIENOCARBINE TL-102 TL-137 TL-140-III TL-232 TL-259 TL-302 TL-304 TL-308 TL-312 TL-333 TL-334 TL-350 TL-68 TL-99 TOLNAPERSINE U-66444B U-68552B U-86170-F U-91356 U-91356-A UH-148 VANOXERINE WF-23 WF-31 WIN-28929 YM-435 Z-1046 Z-10997-A ZK-112566 DOSAGE ALTERNATE-DAY B.I.D. ONCE-DAILY Q.I.D. SELF-ADMINISTRATION T.I.D. DRESSING ABSORBABLE-SUTURE BANDAGE COLLODION PLASTER STOMAHESIVE SUTURE DRUG-DELIVERY SYNCHRON TARGETING DRUG-DESIGN COMBINATORIAL-LIBRARY DWARFISM RUSSELL-SILVER-SYNDROME DYE ACID-YELLOW-9 AMARANTH CARMINATE CARMOISINE CHRYSOINE-S COCHINEAL LIGHT-GREEN-SF-YELLOWISH NEW-COCCINE PATENT-BLUE-V QUINOLINE-YELLOW SCARLET-GN SUDAN-II SUDAN-IV SULFAN-BLUE DYSAUTONOMIA KEY-GASKELL-SYNDROME EAR AUDITORY-MEATUS COCHLEA ENDOCOCHLEAR ORGAN-OF-CORTI PINNA ROUND-WINDOW TYMPANIC-MEMBRANE EATING-DISORDER ANOREXIA-NERVOSA BULIMIA-NERVOSA EDEMA PAPILLEDEMA SPONGIOSIS EGG OOCYTE YOLK ELECTROCHEM. AMPEROMETRY COULOMETRY ELECTROLYSIS POLAROGRAPHY POTENTIOMETRY VOLTAMMETRY VOLTAMPEROMETRY ELECTROLYTE-METAB. ALKALI-RESERVE ELECTROLYTEMETAB.DISORDER ACIDOSIS ALKALOSIS CALCINOSIS CHONDROCALCINOSIS

1150 APPENDIX D DOWNER-COW-SYNDROME HYPERCALCEMIA HYPERCALCIURIA HYPERCHLOREMIA HYPERKALEMIA HYPERMAGNESEMIA HYPERNATREMIA HYPERPHOSPHATEMIA HYPERZINCEMIA HYPOCALCEMIA HYPOCHLOREMIA HYPOCUPREMIA HYPOKALEMIA HYPOMAGNESEMIA HYPONATREMIA HYPOPHOSPHATASIA HYPOPHOSPHATEMIA HYPOSTHENURIA HYPOZINCEMIA LACTIC-ACIDOSIS LIGHTWOOD-ALBRIGHT-= SYNDROME MILK-ALKALI-SYNDROME MILK-FEVER NEPHROCALCINOSIS PHOSPHATURIA WILSON-DISEASE ELECTROPHORESIS CHROMATOFOCUSING ELECTROCHROMATOGRAPHY ISOTACHOPHORESIS ELECTROPHYSIOL. ACTION-POTENTIAL AFTERDEPOLARIZATION AFTERPOLARIZATION DEPOLARIZATION DROMOTROPIC HYPERPOLARIZATION MEMBRANE-POTENTIAL MIGRATING-MYOELECTRIC-= COMPLEX POTENTIAL-DIFFERENCE QT-INTERVAL REFRACTORY-PERIOD RHEOBASE EMBOLISM AIR-EMBOLISM FAT-EMBOLISM EMBRYO AMNION BLASTOCYST BLASTULA FETUS GASTRULA MESENCHYMA MESODERM MORULA MYOBLAST YOLK-SAC EMULSIFIER THICKENER ENCEPHALITIS HERPES-ENCEPHALITIS ENCEPHALOPATHY 9L-GLIOSARCOMA acute-cerebellar-ataxia acute-prim.hem.encephalitis ADRENOLEUKODYSTROPHY AKABANE-DISEASE ALZHEIMER-DISEASE ALZHEIMER-DISEASE AMNESIA ANGULAR-GYRUS-= SYNDROME APHASIA APRAXIA ATAXIA ATAXIA-TELANGIECTASIA ATHETOSIS aujeszkys-disease aujeszkys-disease AVELLIS-SYNDROME BABINSKI-NAGEOTTE-= SYNDROME BALO-DISEASE BARANY-SYNDROME bayle-disease BENEDIKT-SYNDROME BERGERON-DISEASE BINSWANGER-DEMENTIA BONNIER-SYNDROME BORDER-DISEASE BORNA-DISEASE BRISSAUD-SYNDROME caprine-arthritis-encephalitis CEREBELLAR-SYNDROME CEREBELLITIS cerebral-edema cerebral-gigantism CEREBRAL-PALSY cerebral-poliomyelitis CEREBRAL-VASOMOTOR-= SYNDROME CESTAN-CHENAIS-= SYNDROME CHOREA CHOREOATHETOSIS CHORIOMENINGITIS CLAUDE-SYNDROME COMA CONCUSSION congenital-chorea DANDY-WALKER-SYNDROME DIPLEGIA DUBINI-DISEASE DYSARTHRIA DYSAUTONOMIA DYSKINESIA ENCEPHALITIS ENCEPHALOCELE ENCEPHALOMALACIA encephalomeningitis ENCEPHALOMYELITIS ENCEPHALOMYELOPATHY ENCEPHALOMYOCARDITIS EPILEPSY EXTRAPYRAMIDAL-DISORDER FAHR-DISEASE familial-dysautonomia FOVILLE-SYNDROME FRIEDREICH-ATAXIA FUCOSIDOSIS gerlier-disease GLIOBLASTOMA GLIOMA GLIOSARCOMA GLIOSIS GOLDSTEIN-SYNDROME GRAND-MAL HALLERVORDEN-SPATZ-= SYNDROME HEAD-HOLMES-SYNDROME HEIDENHAIN-SYNDROME HEMIBALLISMUS HEMIPLEGIA hepatic-coma hepatic-encephalopathy HERPES-ENCEPHALITIS huntington-chorea HYDROCEPHALUS HYPERBARIC-NERVOUS-= SYNDROME JAKOB-CREUTZFELDT= SYNDROME japanese-b-encephalitis JOSEPH-DISEASE KERNICTERUS KORSAKOFF-SYNDROME KOZHEVNIKOV-SYNDROME LESCH-NYHAN-SYNDROME LEUKOENCEPHALITIS LEUKOENCEPHALOPATHY LITTLE-DISEASE LOUPING-ILL lymphocytic-choriomeningitis MANN-SYNDROME MENINGISM MENINGITIS MENINGOCELE MENINGOENCEPHALITIS MENINGOENCEPHALOCELE MENINGOENCEPHALOMYELITIS MENINGORADICULITIS MENKES-SYNDROME MICROCEPHALY MILLARD-GUBLER-= SYNDROME MULT.SCLEROSIS MULTI-INFARCT-DEMENTIA MYELOENCEPHALITIS MYOCLONUS NEUROSYPHILIS OLIVOPONTOCEREBELLAR-= ATROPHY ORGANIC-BRAIN-SYNDROME orthostatic-dysautonomic-= hypotension PACHYMENINGITIS PALINACOUSIS PANENCEPHALITIS paralytic-dementia paralytic-vertigo PARKINSONISM PETIT-MAL POLIOENCEPHALITIS POLIOENCEPHALOMALACIA PORENCEPHALY progressive-familial-= myoclonic-epilepsy progressive-supranuclear-= paralysis PSEUDORABIES PSEUDOSCLEROSIS PYKNOLEPSY RABIES RADICULOMYELO= ENCEPHALITIS RAYMOND-CESTAN-= SYNDROME REYE-SYNDROME riley-day-syndrome SCHILDER-DISEASE SCHILDER-FOIX-DISEASE shy-drager-syndrome spastic-paresis SPIELMEYER-SJOEGREN-= DISEASE steele-richardson-olszewski-= syndrome struempell-disease struempell-lichtenstern-= encephalitis TARDIVE-DYSKINESIA TESCHEN-DISEASE THALAMIC-SYNDROME THOMAS-SYNDROME TREMBLING-DISEASE TUBEROUS-SCLEROSIS unverricht-disease

Derwent Drug File 1151 Thesaurus UVEOMENINGEAL-= SYNDROME UVEOMENINGOENCEPHALITIS VENTRICULITIS VISNA vogt-syndrome WEST-SYNDROME WILSON-DISEASE zappert-syndrome ENDOCARDITIS THROMBOENDOCARDITIS ENDOMYCETALES SACCHAROMYCESCEREVISIAE ENDOTHELIN-ANTAGONISTS A-127722 A-158112 A-182086 A-192621 ATRASENTAN ATZ-1993 BE-18257B BMS-182874 BMS-193884 BOSENTAN BQ-123 BQ-485 BQ-610 BQ-788 BQ-928 CGS-31447 CGS-34043 CGS-35066 DARUSENTAN FR-139317 IRL-1620 IRL-2500 J-104132 L-749329 LABEDIPINEDILOL-A LU-127043 LU-135252 LU-224332 LU-302146 LU-302872 LU-420627 PD-142893 PD-145065 PD-155080 PD-156252 PD-156707 PD-159433 PD-163070 RES-1149-1 RES-701-1 RO-46-2005 RO-46-8443 S-0139 SB-209670 SB-217242 SB-234551 SB-247083 SCH-54470 T-0115 T-0201 TAK-044 TBC-11241 TBC-11251 TEZOSENTAN TTA-386 YM-62899 ENDOTHELIN-CONVERTINGENZYME-INHIBITORS CGS-25015 CGS-26303 CGS-26582 CGS-26670 CGS-31447 CGS-34043 CGS-35066 PHOSPHORAMIDON SCH-42354 THIORPHAN WS-75624-A WS-75624-B ENZYME-IMMUNODET. ELISA EMIT ENZYMES ACETYLCHOLINESTERASE ACETYLTHROMBIN ACID-PHOSPHATASE ACYLSTREPTASE ADENOSINE-DEAMINASE AGALSIDASE-ALPHA ALKALINE-PHOSPHATASE ALPHA-AMYLASE ALPHA-D-GALACTOSIDASE ALPHA-D-GLUCOSIDASE ALPHA-D-MANNOSIDASE AMAFERM AMP-DEAMINASE AMYLASE ANCROD ANCROD ANISTREPLASE ANTILEUKOPROTEASE APYRASE ARGINASE ARGININE-DEIMINASE ASPARAGINASE ASPERASE ATROXASE AVIZYME-TX AVIZYME-TX BATROXOBIN BETA-D-GALACTOSIDASE BETA-GLUCURONIDASE BILIRUBIN-OXIDASE BRINASE BRL-26920 BRL-33575 BROMELAIN BUTYRYLCHOLINESTERASE CALPAIN CARBONATE-DEHYDRATASE CARBOXYPEPTIDASE-A CARBOXYPEPTIDASE-B CARBOXYPEPTIDASE-G2 CATALASE CELLULASE CERASTASE-F4 CHOLENZYME CHOLINESTERASE CHONDROITINSULPHATASE CHYMOPAPAIN CHYMOTRYPSIN CLOSTRIDIOPEPTIDASE-A CLOTTING-FACTOR-XA COLLAGENASE CYTOSINE-DEAMINASE DEOXYRIBONUCLEASE-I DESTABILASE DEXTRANASE DIAMINE-OXIDASE DIGESTAL DIPEPTIDYL-PEPTIDASE-IV ECARIN ELASTASE ENDO-1,3(4)-BETA-D-= GLUCANASE ENDODEOXYRIBONUCLEASE ENKEPHALINASE ENZYNORM EXO-1,4-BETA-D-= GLUCOSIDASE FIBROLASE G-11035 GALACTOSE-OXIDASE GLUCANASE-BETA GLUCOSE-OXIDASE GLUCOSYLCERAMIDASE GLUTAMIN-(ASPARAGIN-)ASE GLUTAMINASE HEMENTIN HEMICELLULASE HEPARIN-LYASE HORSERADISH-PEROXIDASE HYALURONIDASE IDURONIDASE IMMOZYME INULASE KALLIKREIN KEMZYME KIDNEY-BRUSH-BORDER-= NEUTRAL-PROTEINASE KRILL-PROTEASES L-AMINO-ACID-OXIDASE L-METHIONINE-GAMMA-= LYASE LACTATE-DEHYDROGENASE LACTOPEROXIDASE LEUCINE-AMINOPEPTIDASE LIPASE LONGOLYTIN LYSINE-ALPHA-OXIDASE LYSOSTAPHIN LYSOSUBTILIN-G10X LYSOZYME MALTASE MONTEPLASE MUCOPOLYSACCHARIDASE MUTANOLYSIN MYELOPEROXIDASE NATTOKINASE NEPRILYSIN NEURAMIDE NEURAMINIDASE NIGADASE NORTASE ORGANOPHOSPHATE-= ANHYDRASE ORGOTEIN ORNITHINE-CARBAMOYL= TRANSFERASE PAF-ACETYLHYDROLASE PANCREATIN PANCRELIPASE PANCURMEN PAPAIN PENICILLINASE PENTOSANASE PEPSIN PEROXIDASE PHENYLALANINE-= AMMONIA-LYASE PHOSPHOLIPASE-A2 PHOSPHOLIPASE-C PHOSPHOLIPASE-D PHOSPHOTRIESTERASE PHYTASE PLASMIN POLYGALACTURONASE PROLINE-DIPEPTIDASE PRONASE PROTEASE-C PSEUDOCATALASE PURINE-NUCLEOSIDE-= PHOSPHORYLASE

1152 APPENDIX D RENIN RETEPLASE RIBONUCLEASE RIBONUCLEASE-A SEAPROSE SERRAPEPTASE SERRATIOPEPTIDASE SFERICASE SPHINGOMYELINASE STAPHYLOKINASE STREPTODORNASE STREPTOKINASE SUBTILISIN SUCROSE-ALPHA-D-= GLUCOHYDROLASE SUTILAINS TENECTEPLASE TERRILYTINE THROMBIN THROMBIN-ALPHA-HUMAN THYMIDINE-PHOSPHORYLASE TRIACYLGLYCEROL-LIPASE TRYPSIN TRYPTOPHAN-2,3-= DIOXYGENASE TYROSINASE URATE-OXIDASE UREASE UROKINASE VITA-FERM XANTHINE-OXIDASE XYLANASE YM-866 EOSINOPHILIA EOSINOPHILIA-MYALGIA-= SYNDROME HYPEREOSINOPHILIC-= SYNDROME EPILEPSY GRAND-MAL KOZHEVNIKOV-SYNDROME MYOCLONUS PETIT-MAL PYKNOLEPSY ERYTHEMA ERYTHEMA-ELEVATUM-= DIUTINUM ERYTHROCYTE ELLIPTOCYTE ERYTHROBLAST HEINZ-BODY HEMATOCRIT MACROCYTE MEGALOBLAST MEGALOCYTE MICROCYTE NORMOCYTE POIKILOCYTE RETICULOCYTE SICKLE-CELL SPHEROCYTE SPHEROSTOMATOCYTOSIS ERYTHROLEUKEMIA FSD1-F4-CELL K562-CELL ESOPHAGUS CROP ESOPHAGUS-DISEASE ACHALASIA BARRETT-SYNDROME BOERHAAVE-SYNDROME DYSPHAGIA esophageal-varices ESOPHAGITIS MALLORY-WEISS-SYNDROME MEGAESOPHAGUS NUTCRACKER-ESOPHAGUS ODYNOPHAGIA PLUMMER-VINSON-= SYNDROME PRESBYESOPHAGUS PYROSIS reflux-esophagitis ESS.OIL ANISE-OIL ARTEMISIA-OIL BALM-LEAF-OIL BAY-OIL BERGAMOT-OIL CAJEPUT-OIL CALAMUS-OIL CAMELLIA-OIL CARDAMOM-OIL CHENOPODIUM-OIL CINNAMON-OIL CITRONELLA-OIL COPAIBA-OIL CORIANDER-OIL CUMIN-OIL EUCALYPTUS-OIL GERANIUM-OIL JOJOBA-OIL JUNIPER-OIL KANUKA-OIL LAUREL-OIL LAVENDER-OIL LEMON-GRASS-OIL LEMON-OIL MACE-OIL MANUKA-OIL MINT-OIL MONARDA-OIL NIAOULI-OIL NUTMEG-OIL ORANGE-OIL ORIGANUM-OIL PINE-OIL ROSEMARY-OIL SAGE-OIL SANDALWOOD-OIL SASSAFRAS-OIL THYME-OIL YLANG-YLANG-OIL ESTROGEN-ANTAGONIST AROMATASE-INHIBITOR ESTROGEN-ANTAGONISTS 9599 A-007 ANASTROZOLE AROMATASE-INHIBITORS ATAMESTANE BISPHENOL BUSRAMUSTINE CB-7675 CCRL-1002 CCRL-1008 CCRL-1009 CDRI-85-287 CDRI-86-333 CDRI-88-495 CENTCHROMANE CGP-44645 CGP-47645 CGS-18320B CGS-20267 CHLOROPHENYLACETATE-= PARA CHLOROTAMOXIFEN-4 CI-628M CLOMETERONE CLOMIFENE CLOMIFENOXIDE COUMATE CP-336156 D-15413 D-15414 D-18954 DELMADINONE DELMADINONE-ACETATE DEMETHYLDROLOXIFENE-N DEMETHYLTAMOXIFEN DEMETHYLTOREMIFENE-N DIDEMETHYLTAMOXIFEN DIHYDROXYTAMOXIFEN-3,4 DIMEPREGNEN DIPHENYLENEDENE DROLOXIFENE EM-139 EM-170 EM-652 EM-776 EM-800 EMD-16795 ENCLOMIFENE EPITIOSTANOL ETHAMOXYTRIPHETOL EXEMESTANE FADROZOLE FINROZOLE FORMESTANE FULVESTRANT GW-5638 H-1285 HB-66 HEXESTROL-META HYDROXYANDROSTENE= DIONE-19 HYDROXYCHALCONE-4+ HYDROXYCLOMIFENE-4 HYDROXYESTRADIOL HYDROXYTAMOXIFEN HYDROXYTAMOXIFEN-4+ HYDROXYTOREMIFENE-4 ICI-133312 ICI-140447 ICI-141389 ICI-142269 ICI-145458 ICI-145663 ICI-145680 ICI-164384 ICI-47699 ICI-55548 ICI-79792 ICI-85966 ICI-90069 IDOXIFENE IODOTAMOXIFEN LASOFOXIFENE LEVORMELOXIFENE LILLY-88571 LN-1643 LN-2833 LN-2839 LY-117018 LY-317236 LY-326315 LY-335563 LY-357489 LY-56110 MDL-103323 MDL-18962 MEPITIOSTANE MINAMESTANE MIPROXIFENE MPV-2213-AD

Derwent Drug File 1153 Thesaurus MR-20492 NAFOXIDINE NITROMIFENE OSW-1 PANOMIFENE PIPENDOXIFENE R-1128-A R-1128-B R-1128-C R-1128-D R-151885 R-76713 R-83839 R-83842 RALOXIFENE RU-16117 RU-39411 RU-45144 RU-58668 SC-12222 SP-500263 SR-16234 TAMOXIFEN TAMOXIFEN METHIODIDE TAMOXIFEN-N-OXIDE TAT-59 TOREMIFENE TRIOXIFENE U-23469 VICOLIDE-B VOROZOLE WAY-140424 WSP-1 WSP-3 ZINDOXIFENE ZK-114043 ZK-119010 ZK-135695 ZK-191703 ZUCLOMIFENE ESTROGENS ALMESTRONE ANORDIOL ANORDRIN BE-14348-B BENZESTROL BIFLURANOL BIOCHANIN-A BROMOESTRADIOL-4 BROMOVINYLESTRADIOL-= 17-ALPHA BROPARESTROL BUAME BUTOLAME CHLOROTRIANISENE CL-868 CLOXESTRADIOL CLOXESTRADIOL-ACETATE COUMESTROL CP-336156 CYCLOFENIL DEHYDROESTRONE-8,9 DIBROMOESTRADIOL-2,4 DIENESTROL DIENESTROL-ALPHA DIENESTROL-BETA DIENESTROL-DIACETATE DIETHYLSTILBESTROL DIETHYLSTILBESTROL-3,4-= OXIDE DIETHYLSTILBESTROL-= DIPALMITATE DIETHYLSTILBESTROL-= DIPROPIONATE DIETHYLSTILBESTROL-= EPOXIDE DIETHYLSTILBESTROL-= GLUCURONIDE-SULFATE DIETHYLSTILBESTROL-= MONOGLUCURONIDE DIETHYLSTILBESTROL-= MONOPHOSPHATE DIETHYLSTILBESTROL-= MONOSULFATE DIETHYLSTILBESTROL-= QUINONE DIHYDROEQUILENIN-17-= ALPHA DIHYDROEQUILENIN-17-BETA DIHYDROEQUILIN DIHYDROEQUILIN-17-ALPHA DIHYDROEQUILIN-SULFATE DIMESTROL DIMETHYLSTILBESTROL DOISYNESTROL DOISYNOLATE EIPW-111 EM-652 EMD-20262 EPIESTRIOL EPIMESTROL EQUILENIN EQUILENIN-SULFATE EQUILIN EQUILIN-SULFATE ESTETROL ESTRADIOL ESTRADIOL-17-ALPHA ESTRADIOL-ACETATE ESTRADIOL-BENZOATE ESTRADIOL-CYCLOOCTYL= ACETATE-17 ESTRADIOL-CYPIONATE ESTRADIOL-DIACETATE ESTRADIOL-DIENANTHATE ESTRADIOL-DIPROPIONATE ESTRADIOL-DISULFATE ESTRADIOL-ENANTHATE ESTRADIOL-HEMISUCCINATE ESTRADIOL-METHYL-= ETHER-3 ESTRADIOL-METHYL= DIHYDRONICOTINATE ESTRADIOL-OCTANOATE ESTRADIOL-PALMITATE ESTRADIOL-PHENYL= PROPIONATE ESTRADIOL-PHOSPHATE ESTRADIOL-PROPIONATE ESTRADIOL-STEARATE-17 ESTRADIOL-SULFATE-17 ESTRADIOL-SULFATE-3 ESTRADIOL-UNDECYLATE ESTRADIOL-VALERATE ESTRAPRONICATE ESTRAZINOL ESTRIOL ESTRIOL-GLUCURONIDE-16 ESTRIOL-GLUCURONIDE-17 ESTRIOL-GLUCURONIDE-3 ESTRIOL-SUCCINATE ESTRIOL-SULFATE-17 ESTRIOL-SULFATE-3 ESTROFURATE ESTROGEN-CONJUGATED ESTRONE ESTRONE-ACETATE ESTRONE-METHYL-ETHER ESTRONE-SULFATE ESTROPIPATE ESTRYNAMINE ETHINYLESTRADIOL ETHINYLESTRADIOL-= SULFONATE ETHINYLESTRIOL ETHYLESTRONE-3-O-= SULFAMATE-2 ETOLAME F-6060 FENESTREL FI-6173 FLUOROESTRADIOL-16-= ALPHA FLUOROESTRADIOL-16-BETA FLUOROESTRADIOL-2 FLUOROESTRADIOL-4 FLUORONORHEXESTROL FLUOROTAMOXIFEN-4 FORMONONETIN FOSFESTROL FUKINOLATE FUROSTILBESTROL GW-154 GYNOESTRYL-FORT HEXESTROL HEXESTROL-DICAPRYLATE HEXESTROL-ORTHO HYDROXYESTRADIOL HYDROXYESTRADIOL-4 HYDROXYESTRADIOL-6-= ALPHA HYDROXYESTRIOL-2 ICI-3188 ICI-77949 INDANESTROL INDENESTROL-A INDENESTROL-B IODOESTRADIOL-16-ALPHA ISODIENESTROL J-303 J-628 J-811 J-824 J-96 J-995 KCA-098 LASOFOXIFENE LY-139478 MESO-HEXESTROL MESTILBOL MESTRANOL METHALLENESTRIL METHESTROL METHESTROL-DIPROPIONATE METHOXYESTRADIOL-2 METHOXYESTRADIOL-4 METHYLENEESTRADIOL-16 METHYLESTRADIOL MOXESTROL MRL-37 NALOXONE-ESTRONE-AZINE NILESTRIOL NISTRANOL NORETHISTERONE-OXIME-3 NYASOL ORESTRATE ORF-5330 ORF-5331 P-5780 PENTAFLURANOL PENTOLAME POLYESTRADIOL-PHOSPHATE PRENYLNARINGENIN-8 PROACAME PROLAME PROMESTRIENE QUINESTRADOL QUINESTROL RVC-588 SC-9022 SEGETALIN-A SIGETIN

1154 APPENDIX D STS-153 STS-456 STS-593 STS-64 U-10293 WAY-140424 WS-7528 WY-5090 ZEARALANONE ZEARALENONE ZERANOL ESTRUS DIESTRUS METESTRUS PROESTRUS EUNUCHOIDISM FERTILE-EUNUCH-SYNDROME EXPECTORANTS AMBROXOL AMBROXOL = THEOPHYLLINATE AMMONIUM-ACETATE ANETHOLE APOMORPHINE BR-227 BROMELAIN BROMHEXINE CEPHAELINE CISTINEXINE DEMBREXINE EMETINE EUCALYPTOL GLYCYRAM GLYCYRRHIZATE GUACETISAL GUAIETOLIN GUAIFENESIN HELENIN IDB-1031 IODINATED-GLYCEROL IRFI-005 IRFI-016 LIMONENE LYCORINE PLATYCODIN-D PRENISTEINE SULFOGAIACOL TEREBINTH-OIL TERPIN-HYDRATE TIPEPIDINE EXTRAPYRAMIDAL-DISORDER JOSEPH-DISEASE PARKINSONISM EXTREMITY ARM FINGER FOOT HAND LEG LIMB PAW THIGH TOE WING EYE AQUEOUS-HUMOR CHOROID CILIARY-PROCESS CONJUNCTIVA CORNEA DARK-ADAPTATION EALE-DISEASE intraocular-pressure IRIS LENS MIOSIS MYDRIASIS PUPIL RETINA SCLERA VITREOUS-BODY VITREOUS-HUMOR EYE-DISEASE ADIE-SYNDROME ALACRIMA AMBLYOPIA ANISOCORIA ANKYLOBLEPHARON ANOPHTHALMUS APHAKIA BEHR-DISEASE BLEPHARITIS BLEPHAROCONJUNCTIVITIS BLINDNESS BLURRED-VISION BRIGHT-BLINDNESS BROWN-SYNDROME CATARACT CHALAZION charlin-syndrome CHEMOSIS CHORIORETINITIS CHOROIDITIS ciliary-neuralgia cogan-syndrome COLOBOMA CONJUNCTIVITIS CORNEAL-DYSTROPHY CYCLOKERATITIS DACRYOADENITIS DACRYOCYSTITIS DACRYOCYSTOCELE DACRYORRHEA DELLEN diabetic-retinopathy DIPLOPIA DISTICHIA EALE-DISEASE ENDOPHTHALMITIS EPISCLERITIS EXOPHTHALMOS GLAUCOMA graefe-syndrome granular-corneal-dystrophy HEMERALOPIA HEMIANOPIA HERPES-CORNEAE herpes-keratitis HORDEOLUM HYALITIS HYDROPHTHALMOS HYPHEMA HYPOPYON infantile-glaucoma infectious-keratoconjunctivitis IRIDOCORNEAL-= ENDOTHELIAL-SYNDROME IRIDOCYCLITIS IRIDOSCHISIS IRITIS KERATITIS KERATOCELE KERATOCONJUNCTIVITIS KERATOCONUS KERATOMALACIA KERATOPATHY KERECTASIS LAGOPHTHALMOS LEBER-DISEASE macular-corneal-dystrophy MICROPHTHALMUS MONOCHROMATISM MYDRIASIS MYOPIA NEURORETINITIS nonsyphilitic-interstitial-= keratitis NYCTALOPIA NYSTAGMUS OCULO-RESPIRATORY-= SYNDROME OCULOGYRIC-CRISIS OPHTHALMIA OPHTHALMITIS OPHTHALMOPLEGIA OPHTHALMORRHEXIS OPSOCLONUS ORBITAL-PSEUDOTUMOR painful-ophthalmoplegia PANNUS PANOPHTHALMITIS PAPILLEDEMA PARATRACHOMA PARINAUD-SYNDROME PHOTOPHOBIA progressive-ophthalmoplegia PTOSIS REITER-SYNDROME RETINITIS RETINOCHOROIDITIS RETINOPATHY RUBEOSIS-IRIDIS SCLERITIS SCLEROMALACIA SCOTOMA SPANLANG-TAPPEINER-= SYNDROME STAPHYLOMA STRABISMUS SYNECHIAE TERRY-SYNDROME tolosa-hunt-syndrome TRACHOMA TUBULAR-VISION UVEITIS UVEOMENINGEAL-= SYNDROME VOGT-DISEASE XEROPHTHALMIA FACTITIOUS-DISORDER acute-hallucinatory-mania ganser-syndrome MUENCHAUSEN-SYNDROME MUENCHAUSEN-= SYNDROME-BY-PROXY polle-syndrome PSEUDODEMENTIA FARNESYL-PROTEINTRANSFERASE-INHIBITORS ACTINOPLANONE-A BMS-214662 BZA-2-B CB-7741 FTI-2148 FTI-2153 HYDROXYCINNAM= ALDEHYDE-2+ L-744832 L-778123 LB-42908 MANUMYCIN PD-83176 PREUSSOMERIN-D PREUSSOMERIN-G RPR-114334 SCH-207758 SCH-226374

Derwent Drug File 1155 Thesaurus SCH-44342 SCH-56582 SCH-66336 TIPIFARNIB TIPIFARNIB UCF-1-C FEEDSTUFF RAPESEED-MEAL FERTILITY FECUNDITY FERTILIZATION IN-VITRO-FERTILIZATION FIBRINOGEN-ANTAGONIST GP-IIB-IIIA-ANTAGONIST FIBRINOGEN-ANTAGONISTS ARC-69931-MX CRL-42796 ELAROFIBAN EPTIFIBATIDE GP-IIB-IIIA-ANTAGONISTS HMR-1794 L-736622 LOTRAFIBAN ME-3229 ORBOFIBAN PS-028 ROXIFIBAN SC-57101-A SR-121566 T-250 TIROFIBAN UR-12947 XEMILOFIBAN XU-063 XV-454 YM-57029 FIBROBLAST 3T3-CELL 3T6-CELL A31-CELL AD6-CELL AP9-CELL B82-CELL CCD18-CELL CCF-CELL CCL84-CELL CH23-CELL DON-CELL EHB-CELL GM258-CELL L-CELL L929-CELL LM-CELL MC5-5-CELL RNF22-CELL RTG2-CELL ST-BALB-CELL ST-CELL V79-CELL W138-CELL FIBROSARCOMA HT1080-CELL MC7-CELL MCB6-1-CELL METH-A METH-A-CELL SA5-CELL FILTRATION DIALYSIS HEMODIALYSIS HEMOFILTRATION MICRODIALYSIS ULTRAFILTRATION FISH CARP CATFISH LAMPREY ORYZIAS PIKE POECILIA SALMON TORPEDO TROUT FLAVOR FISH-TAINT GARLIC TASTE-REPELLENT THAUMATIN FLUORESCENCE FLUORIMETRY FLUORIMETRY fpia FOLATE-ANTAGONISTS ADITOPRIM AG-2034 AG-2037 AG-377 AG-394 AG-85 AM-92008 AZIDOPYRIMETHAMINE-= META CB-30865 CB-3717 CB-3804 CB-3988 DEAZATETRAHYDRO= FOLATE-5 DICHLOROBENZOPRIM DICHLOROMETHOTREXATE DIDEAZATETRAHYDRO= FOLATE-5,10 FLUORONITROPYRIMETH= AMINE ICI-198583 K-107 K-120 K-122 K-137 K-138 K-150 K-96 LOMETREXOL LY-231514 LY-243246 LY-309887 METHOBENZAPRIM MOBILETREX MX-68 NSC-118203 NSC-125358 NSC-128189 NSC-211327 NSC-232965 NSC-235777 NSC-3077 NSC-330465 PIRITREXIM PT-441 PT-523 PT-619 PT-633 PYRIMETHAMINE RALTITREXED RO-11-8958 TNP-351 TRIMETHOPRIM TRIMETREXATE FOLLIBERIN-AGONISTS ACTIVIN FOLLIBERIN FRAGMENT DIGIBIND FRUIT APPLE BERRY COCONUT OLIVE ORANGE PEAR FUNGICIDES A-32390-A ACETYLHETEROPHYLLISINE-8 ACRISORCIN ACULEACIN-A AFK-108 AGELASIDINE-A AKUAMMIDINE ALBIDIN ALICONAZOLE ALISAMYCIN ALLIXIN ALLOSAMIDIN ALOE-EMODIN ALPHA-D-MANNOSIDASE AMBRUTICIN AMIJITRIENOL AMOROLFINE AMPHOGLUCAMINE AMPHOTERICIN-A AMPHOTERICIN-B AMPHOTERICIN-B-= METHYLESTER ANDROCTONIN ANILAZINE ANTOFINE ARANOROSIN AROMADENDRIN ARVENSOSIDE-D ASCOMYCIN ASCOSFEROL ASPIROCHLORINE ATHEROSPERMININE ATHEROSPERMININE-N-OXIDE ATPENIN-A4 ATPENIN-A4 ATPENIN-A5 ATPENIN-B AUREOBASIDIN-B AUREOBASIDIN-C AUREOBASIDIN-D AUREOBASIDIN-E AUREOBASIDIN-F AUREOBASIDIN-G AUREOBASIDIN-H AUREOBASIDIN-I AUREOBASIDIN-J AUREOBASIDIN-K AUREOBASIDIN-L AUREOBASIDIN-M AUREOBASIDIN-N AUREOBASIDIN-O AUREOBASIDIN-P AUREOBASIDIN-Q AUREOBASIDIN-R AUREOFUNGIN AURISTATIN-PHE AVAROL AVARONE AVENACIOLIDE AZACONAZOLE AZALOMYCIN-F4

1156 APPENDIX D AZASERINE AZOXYBACILIN BAFILOMYCIN-D BASIFUNGIN BASIL-OIL BAY-L-9139 BAY-R-3783 BAY-U-3625 BE-18591 BELAMCANIDIN BENANOMICIN-A BENANOMICIN-B BENASTATIN-A BENASTATIN-B BENOMYL BENQUINOX BENSULDAZATE BETA-DEFENSIN-3-HUMAN BIFONAZOLE BITERTANOL BIVITTOSIDE-A BIVITTOSIDE-B BIVITTOSIDE-C BIVITTOSIDE-D BLASTICIDIN-S BMS-181184 BMY-28864 BRASINOLIDE-A BUCLOSAMIDE BUDDLEDIN-A BUTENAFINE BUTOCONAZOLE CAERULOMYCIN-A CALBISTRIN-A CALBISTRIN-B CALCOFLUOR-WHITE CALLIPELTIN-A CALOPOROSIDE CAN-296 CANADENSOLIDE CAP-18-HUMAN CAPTAN CARBAZOMYCIN-B CARBAZOMYCIN-G CARBAZOMYCINAL CARBENDAZIME CARBOXIN CASPOFUNGIN CEPACIDINE-A1 CEPACIDINE-A2 CERCOSPORAMIDE CHAETIACANDIN CHAKSINE CHLORACETOPHOS CHLORANIL CHLORHEXIDINE-= PHOSPHANILATE CHLORMIDAZOLE CHLOROMALOSIDE-A CHLORONEB CHLOROPHETANOL CHLOROTETAIN CHLOROTHALONIL CHLORPHENESIN CHLORPHENOCTIUM = AMSONATE CHLORQUINALDOL CHOKOL-A CHONDRAMIDE-A CHONDRAMIDE-B CHONDRAMIDE-C CHONDRAMIDE-D CHRYSCANDIN CICLOPIROX CILOFUNGIN CISPENTACIN CLATHRAMIDE-A CLAUSSEQUINONE CLAVARIOPSIN-A CLAVARIOPSIN-B CLIMBAZOLE CLODANTOIN CLOFENOXYDE CLOPROTHIAZOLE CLOTIOXONE CLOTRIMAZOLE CLOXIQUINE COLLISMYCIN-A COLLISMYCIN-B COPIAMYCIN COPPER-OXYCHLORIDE CORDIAQUINONE-B CRIBROSTATIN-2 CROCONAZOLE CROTMADINE CURCUPHENOL CYANOPUUPEHENOL-15 CYCLO-TRP-PRO CYCLO-TRP-TRP CYCLOHEXIMIDE D-0870 DAPHNODORIN-B DAZOMET DEACETOXYOLEPUPUANE-7 DEDITONIUM BROMIDE DEHYDROACETATE DEHYDROALTENUSIN DEHYDROCURVULARIN DEMETHOXYVIRIDIN DEMETHYLALLOSAMIDIN DEMETHYLOLIVOMYCIN-B DEMETHYLRAPAMYCIN-O-27 DEMOCONAZOLE DENMERT DEQUALINIUM CHLORIDE DERMACID DERMASEPTIN DERMASEPTIN-S3-1-16 DERMOCEPT DICHLONE DICHLORBENZALKONIUM DICHLOROPHEN DICLOBUTRAZOL DIDEMNENONE-A DIDEMNENONE-B DIETIFEN DIHYDROGENISTEIN DIHYDROHALICHONDRAMIDE DIHYDROTANSHINONE-I DIMAZOLE DIMETHIRIMOL DINICONAZOLE DINOCAP DIPYRITHIONE DITHIANONE DOCONAZOLE DODEMORPH DODINE DORRIGOCIN-A DORRIGOCIN-B DRAGMACIDIN-D DRAZOXOLON DUNAIMYCIN-A1 DUNAIMYCIN-C2 DUNAIMYCIN-D2 DUNAIMYCIN-D2S DUNAIMYCIN-D3 DUNAIMYCIN-D4S DUP-860 DYSIDAZIRINE ECHINOCANDIN-B ECHINOCANDIN-C ECHINOCANDIN-D ECHINOCYSTATE ECHINOSIDE-B ECONAZOLE ELACTOCIN EMESTRIN EMODIN ENACTIN-IA ENACTIN-IB1 ENACTIN-IB2 ENACTIN-VA ENCELIN ENILCONAZOLE EPIPOLYGODIAL ER-30346 ETHIRIMOL ETHISOLIDE ETHYLMERCURIC-CHLORIDE ETISAZOLE ETONAM EUPOLAURIDINE EUPOLAURIDINE-N-OXIDE EUROPINE EXALAMIDE FAERIEFUNGIN-A FAERIEFUNGIN-A FAERIEFUNGIN-B FALCARINOL FATTIVIRACIN-FV-8 FENARIMOL FENPROPIMORPH FENTICLOR FENTICONAZOLE FENTIN HYDROXIDE FERBAM FEZATIONE FILIPIN FLAVIPUCINE FLUCONAZOLE FLUCYTOSINE FLUSILAZOLE FLUTRIAFOL FLUTRIMAZOLE FLUVIRUCIN-A1 FLUVIRUCIN-A2 FLUVIRUCIN-B1 FLUVIRUCIN-B2 FLUVIRUCIN-B3 FOLPET FORMAMICIN FR-131535 FR-900848 FR-901469 FUNICULOSIN FURACRYLIN FURAZONAL FURFURAL FUSACANDIN-A FUSACANDIN-B FUSARICIDE GALANOLACTONE GALBONOLIDE-A GALBONOLIDE-B GAMBIERATE-A GAMBIERATE-B GAMBIERATE-C GC-1993 GEODIAMOLIDE-A GEODIAMOLIDE-B GLOMOSPORIN GLYCYCOUMARIN GM-160575 GM-193663 GM-237354 GRANULYSIN GRISEOFULVIN GUANIDYLFUNGIN-A HALICHONDRAMIDE HALISULFATE-1 HALOPENIUM CHLORIDE

Derwent Drug File 1157 Thesaurus HALOPROGIN HAPALINDOLE-E HAPALINDOLE-G HAPALINDOLE-H HAPALINDOLE-J HAPALINDOLE-M HAPALINDOLE-O HAPALINDOLE-U HAZIMYCIN-5 HAZIMYCIN-6 HEDAQUINIUM CHLORIDE HEDERACOLCHISID-A1 HEDERACOLCHISIDE-A HEXACHLOROBENZENE HEXACONAZOLE HEXAMIDE HISPANOLONE HISTATIN-5 HISTIDINOMYCIN HOLOTHURIN-B HOLOTOXIN-A1 HUMULONE HYDRANGENOL HYDRARGAPHEN HYDROXYETHYLCLAVAM HYDROXYITRACONAZOLE HYDROXYMARASMATE-9-= BETA HYDROXYSTILBAMIDINE ICI-153066 ICI-195739 ILLUDIN-C3 INCRUSTOPORIN INDISOCIN INDOLICIDIN IRUMAMYCIN ISOAVENACIOLIDE ISOBATZELLINE-A ISOBATZELLINE-C ISOCONAZOLE ISOISOVELLERAL ISOPULEGOL ISOVELLERAL ISOWIGHTEONE ITRACONAZOLE ITURIN-AL JACAREUBIN JASPAMIDE JASPLAKINOLIDE JULIFLORINE KABIRAMIDE-C KAHALALIDE-F KALIHINOL-A KALIHINOL-F KALIHINOL-X KALIHINOL-Y KALIHINOL-Z KANCHANAMYCIN-A KANCHANAMYCIN-D KANUKA-OIL KAZUSAMYCIN KAZUSAMYCIN-B KETOCONAZOLE KHAFREFUNGIN KP-103 KY-62 L-660631 L-687781 L-688786 L-693989 L-705589 L-731373 L-733560 L-743872 L-793422 LACHNELLULONE LACHNUMON-B1 LACHNUMON-B2 LACTOFERRICIN-B LAGOSIN LANOCONAZOLE LANOMYCIN LASIOCARPINE-N-OXIDE LAXAPHYCIN-A LAXAPHYCIN-B LAXAPHYCIN-D LAXAPHYCIN-E LEPTOMYCIN-A LEPTOMYCIN-B LEUCASCANDROLIDE-A LEUCINOSTATIN-A LEUCINOSTATIN-B LEUCINOSTATIN-C LEUCINOSTATIN-D LEUCINOSTATIN-F LEUCINOSTATIN-H LEUCINOSTATIN-K LEUSTRODUCSIN-A LEUSTRODUCSIN-B LEUSTRODUCSIN-C LICOCOUMARONE LIDIMYCIN LIGSTROSIDE LIME-SULFUR LINEARMYCIN-A LIRIODENINE LISSOCLINOTOXIN-A LUCKNOMYCIN LUPULONE LY-303366 LY-307853 LY-317584 LY-448212 LY-448731 LYSOVET MAACKIAIN MAGAININ-1 MAGAININ-2 MAGAININ-B MALABARICONE-C MANEB MANIWAMYCIN-A MANIWAMYCIN-B MANUKA-OIL MANUMYCIN MARASMATE MARCHANTIN-C ME-1401 MEDICAGENATE MEDICAGENATE-= GLUCOSIDE-3 MEGLUMINE-DITHIO= CARBAMATE MER-WF-3010 MERCAPTOBENZOTHIAZOLE MERIDINE MERULIDIAL METHAM SODIUM METHOXYCARBAZO= MYCINAL-6 METHOXYCINNAM= ALDEHYDE-ORTHO METHOXYPHASEOLLIDIN-1 METHOXYSTROBILURIN-K-9 METHYL-ORSELLINATE-= ORTHO METHYLENOLACTOCIN METHYLMERCURY-CHLORIDE METIPIROX METRIFONATE-ACETATE MICACOCIDIN MICAFUNGIN MICONAZOLE MILDIOMYCIN MONOPROP MONORDEN MS-8209 MSI-1436 MULUNDOCANDIN MUSIZIN MYCO-CURB MYCOHEPTIN MYCOPENTEN MYCORRHIZIN-B1 MYCORRHIZIN-B2 MYCOTRIENIN-I MYCOTRIENIN-II MYCOVERSILIN MYOMYCIN MYRIOCIN MYRISTOYLCHOLINE = BROMIDE MYROCIN-C MYXALAMIDE-A MYXALAMIDE-B MYXALAMIDE-C MYXALAMIDE-D NABAM NAFTIFINE NAFTOXATE NAKIJIQUINONE-A NAKIJIQUINONE-B NANNOCHELIN-A NATAMYCIN NEIHUMICIN NEO-ENACTIN-A NEO-ENACTIN-B1 NEO-ENACTIN-B2 NEO-ENACTIN-M2 NEO-ENACTIN-NL1 NEO-ENACTIN-NL2 NEOCNIDILIDE NEOPYRROLOMYCIN NETZAHUALCOYONE NIAOULI-OIL NIBROXANE NIFURALIDE NIFURMERONE NIKKOMYCIN-J NIKKOMYCIN-PSEUDO-J NIKKOMYCIN-PSEUDO-Z NITRALAMINE NITROFEN NITROFUNGIN NITROSOFUNGIN NITROXOLINE NOBILETIN NORTOPSENTIN-A NSC-615985 NYSTATIN NYSTATIN-A1 NYSTATIN-A2 OCEANAPISIDE OIDIODENDROLIDE-A OIDIOLACTONE-A OLIGOMYCIN OLIGOMYCIN-A OLIGOMYCIN-B OLIGOMYCIN-C OMOCONAZOLE ONTIANIL ONYCHINE OPHIOBOLIN-A ORCONAZOLE OSTHENOL OUDEMANSIN OUDEMANSIN-A OUDEMANSIN-B OUDEMANSIN-X OXANTHROMICIN OXETIN OXICONAZOLE OXIFUNGIN

1158 APPENDIX D OXYCARBOXIN PACLOBUTRAZOL PAMAMYCIN-607 PANICUTINE PAPUAMINE PAPYRACON-A PARACONAZOLE PARADOL-6 PARCONAZOLE PATULOLIDE-A PATULOLIDE-B PATULOLIDE-C PC-766B PECILOCIN PENCYCURON PENOCTONIUM BROMIDE PENTACHLORONITROBENZENE PENTACHLOROPHENOL PENTALAMIDE PERVICOSIDE-A PERVICOSIDE-B PERVICOSIDE-C PETROSYNOL PF-1163-A PGE-4175997 PHENOXYACETATE PHENYLHEPTATRIYNE PHENYLMERCURIC-BORATE PHENYLPHENOL-2 PHOMALACTONE PHOMENOATE PHORBOXAZOLE-A PHORBOXAZOLE-B PICLAVINE-A2 PILATIN PIPERAZINOMYCIN PIRITETRATE PLAKINATE-A PLAKINATE-B PLAKORTATE PLD-118 PNEUMOCANDIN-A0 PNEUMOCANDIN-A1 PNEUMOCANDIN-A2 PNEUMOCANDIN-A3 PNEUMOCANDIN-A4 PNEUMOCANDIN-B0 PNEUMOCANDIN-B2 PNEUMOCANDIN-C0 PODOSPORIN-A POLYNOXYLIN POSACONAZOLE POTASSIUM-IODIDE PR-967-234 PR-967-248 PR-969-566 PRADIMICIN-A PRADIMICIN-B PRADIMICIN-S PRADIMICIN-T1 PRADIMICIN-T2 PRAMANICIN PRENYLNARINGENIN-8 PREUSSIN PREUSSOMERIN-D PREUSSOMERIN-G PROCHLORAZ PROCLONOL PROPHAM PROPICONAZOLE PROPIONATE SODIUM PROTIOFATE PRUNIN PSEUDOLARATE-B PSEUDOMYCIN-C+ PTILOMYCALIN-A PUNCTATIN-A PUNCTATIN-D PYRIDINITRILE PYRROLNITRIN PYRROXAMYCIN QUADRIGEMINE-C QUINOLACTACIN-A QUINOLACTACIN-B QUINTOZENE R-39519 R-63373 RANALEXIN RAVUCONAZOLE RESTRICTICIN REVEROMYCIN-A REVEROMYCIN-B REVEROMYCIN-C REVEROMYCIN-D RHEIN RHIZOXIN RHIZOXIN-D RI-331 RIMOCIDIN RIMOPROGIN RK-397 ROFLAMYCOIN ROSELIPIN-1A ROSELIPIN-1B ROSELIPIN-2A ROSELIPIN-2B ROSEOFUNGIN ROXATICIN RS-22-A RS-22-B RS-22-C RUTAMYCIN RUTAMYCIN-B SALICYLANILIDE SALICYLATE SALICYLATE TROLAMINE SALVICYKLIN SAMPANGINE SAPERCONAZOLE SAPINDOSIDE-A SAPINDOSIDE-B SAPINDOSIDE-C SAPINDOSIDE-D SAPONOSIDE-S2 SAPTOMYCIN-D SC-58272 SC-59840 SC-61213 SCH-28191 SCH-37137 SCH-38518 SCH-39304 SCH-40873 SCH-42427 SCH-50002 SCH-51048 SCH-53174 SCH-54445 SCOULERINE SCYTOPHYCIN-B SCYTOPHYCIN-C SCYTOPHYCIN-D SCYTOPHYCIN-E SDZ-87-469 SDZ-89485 SDZ-SBA-586 SELENIUM-SULFIDE SERTACONAZOLE SF-2370 SF-85-190 SKF-3301-A SKF-7997-A3 SM-8668 SM-9164 SMAP-28 SOLACONGESTIDINE SORANGICIN-A SORANGICIN-B SORBATE SPA-S-753 SPA-S-843 SPHINGOFUNGIN-A SPHINGOFUNGIN-B SPHINGOFUNGIN-C SPHINGOFUNGIN-D SPICAMYCIN SPINAMYCIN SQUALESTATIN-1 SS-717 SS-750 STAUROSPORINE STEMPHOL STICHOPOSIDE-A STIGMATELLIN STIGMATELLIN-A STILBAMIDINE ISETIONATE STREPTIMIDONE STREPTOTHRICIN-B STROBILURIN-A STROBILURIN-B STROBILURIN-E STROBILURIN-F STROBILURIN-G STROBILURIN-H SULBENTINE SULCONAZOLE SULFONIDAZOLE SURINAMENSIN SWINHOLIDE-A SYN-2836 SYN-2869 SYN-2903 SYN-2921 SYRINGOMYCIN-E SYRINGOSTATIN-A TAK-456 TAN-1518-A TAN-950-A TAURULTAM TAUTOMYCIN TECNAZENE TENONITROZOLE TENUIFOLIN TERBINAFINE TERCONAZOLE TETRACHLORSALICYLANILIDE TETRACONAZOLE TETRAHYDROECHINO= CANDIN-B TETRAHYDROSECAMINE THIARUBRINE-A THIOLUTIN THIOPHANATE THIOPHANATE-METHYL THIOPYRONINE THIRAM THYMOL TIABENDAZOLE TICLATONE TIGERININ-1 TIOCONAZOLE TIOXOLONE TJIPANAZOLE-A1 TOLCICLATE TOLINDATE TOLNAFTATE TOLYTOXIN TOMATINE TRACHEAL-ANTIMICROBIAL-= PEPTIDE TRIACETIN TRIADIMEFON

Derwent Drug File 1159 Thesaurus TRIADIMENOL TRIAFUNGIN TRICHLOROPHENOL TRICHLOROPHENOL-2,4,5 TRICHOCARPIN TRICHODERMIN TRICHOMYCIN-A TRICHOMYCIN-B TRICHOSETIN TRICHOSTATIN-A TRICHOSTATIN-C TRIDEMORPH TRIMORPHAMIDE TRITRPTICIN UK-2-A UK-3-A UK-47265 UNCINATONE UR-9825 VALCLAVAM VALCONAZOLE VALDEZIN-D VALIDAMYCIN-A VALIDAMYCIN-B VALIDAMYCIN-G VALIDOXYLAMINE-G VANILLATE-ETHYL VARACIN VELLERAL VIBUNAZOLE VILMORRIANONE VIOLACEIN VIRGAUREASAPONIN-1 VIRGAUREASAPONIN-2 VIRIDOFULVIN VIRIDOFULVIN-A VIRIDOFULVIN-B VORICONAZOLE VUF-8501 VUF-8842 WARBURGANAL WS-9659A WS-9659B WYERONE X-14873A X-14889A X-14889C X-14889D XENYSALATE YM-47522 YM-75518 YOSHIXOL YS-822A ZARAGOZATE-A ZARAGOZATE-B ZARAGOZATE-C ZG-1494-ALPHA ZINC-UNDECENOATE ZINEB ZINOCONAZOLE ZIRAM ZOFICONAZOLE FUNGUS ABSIDIA ACHLYA ACREMONIUM ACROPHIALOPHORA ACTINOSPORANGIUM ACTINOSYNNEMA ALLESCHERIA ALTERNARIA AMAUROASCUS APHANOMYCES ARTHROBOTRYS ASCOCHYTA ASCOSPHAERA ASP. AUREOBASIDIUM BACTERIONEMA BASIDIOBOLUS BEAUVERIA BLAKESLEA BLASTOMYCES BOTRYODIPLODIA BOTRYOTINIA BOTRYTIS CALDARIOMYCES CANDIDA CEPHALOSPORIUM CERATOCYSTIS CHAETOMIUM CHROMOSPORIUM CHRYSOSPORIUM CLADOSPORIUM CLAVICEPS COCCIDIOIDES COCHLIOBOLUS COLEOSPORIUM COLLETOTRICHUM CONDIOBOLUS CONIOPHORA COPRINUS CORTICIUM CRYPTOCOCCUS CUNNINGHAMELLA CURVULARIA DEUTEROPHOMA DICHOTOMYCES DICTYOSTELIUM DIPODASCUS ELSINOE ENANTIOTHAMNUS ENTOMOPHTHORA EPICOCCUM EPIDERMOPHYTON EREMOTHECIUM ERYSIPHE EUPENICILLIUM EXOPHIALA FONSECAEA FUSARIUM FUSIDIUM GEOTRICHUM GLIOCLADIUM GLOEOSPORIUM GLOMERELLA GONGRONELLA GRAPHIUM HANSENULA HELICOSTYLUM HELMINTHOSPORIUM HENDERSONIA HENDERSONULA HISTOPLASMA HORMODENDRUM HUMICOLA HYPHOMYCES KERATINOMYCES KIBDELOSPORANGIUM KLOECKERA LEPTOSPHERIA LOBOA LYCOGALA MACROPHOMINA MADURELLA MALASSEZIA METARHIZIUM MICROBOTRYUM MICROSPORUM MONASCUS MONOCILLIUM MONOSPORIUM MORTIERELLA MUCOR MYCELIA MYRIODONTIUM MYROTHECIUM NADSONIA NEMATOSPORA NEUROSPORA OIDIODENDRON OOSPORA PAECILOMYCES PARACOCCIDIOIDES PELLICULARIA PEN. PETRIELLA PETRIELLIDIUM PETRIELLIDUM PHAEOTRICHOCONIS PHANEROCHAETE PHIALOPHORA PHYSALOSPORA PHYSARUM PICHIA PIRICULARIA PITHOMYCES PITYROSPORON PLASMOPARA PLEOSPORA PSEUDALLESCHERIA PSEUDOPERONOSPORA PUCCINIA PYRICULARIA PYTHIUM RAMICHLORIDIUM RHINOSPORIDIUM RHIZOBIUM RHIZOCTONIA RHIZOPODA RHIZOPUS RHODOSPORIDIUM RHODOTORULA ROTHIA SACCH. SACCHAROMYCOPSIS SACCHAROPOLYSPORA SAKSENAEA SAPROLEGNIA SCHIZONELLA SCHIZOSACCH. SCHWANNIOMYCES SCLEROTINIA SCOPULARIOPSIS SEBEKIA SEPEDONIUM SPOROBOLOMYCES SPOROTHRIX STACHYBOTRYS STEMPHYLIUM SYNCEPHALASTRUM TORULA TORULOPSIS TRICHODERMA TRICHOPHYTON TRICHOSPORON TRICHOTHECIUM UROCLADIUM USTILAGO VALSA VENTURIA WANGIELLA WINGEA YEAST ZYGOSACCH. G.U.TRACT BLADDER neurogenic-bladder URACHUS URETER

1160 APPENDIX D URETHRA GABA-ANTAGONISTS ALLOKAINATE-ALPHA AMINOBUTYL= PHOSPHONATE-4 AMINOPROPYL= PHOSPHONATE-3 BICUCULLINE BICUCULLINE-METHIODIDE BICUCULLINEMETHOBROMIDE BICUCULLINE-= METHOCHLORIDE BUTYLBICYCLOPHOSPHORO= THIONATE-TERT CGP-35348 CGP-36742 CGP-44533 CGP-46381 CGP-51176 CGP-52432 CGP-54062 CGP-55845 CGP-55845A CGP-56433 CGP-56433A CGP-56999 CGP-56999-A CGP-61334 CGP-62349 CM-42641 D-20443 FAMIRAPRINIUM CHLORIDE FGIN-1-27 GABAZINE HYDROXYSACLOFEN KAINATE NORBICUCULLINE PHACLOFEN PITRAZEPIN R-5135 RU-5135 SACLOFEN SCH-50911 SN-606078 SR-42641 THIOSEMICARBAZIDE (Drug) U-93631 VIROSECURININE GABAMINERGICS ACAMPROSATE ACETYLTAURINE AHR-14042 AMINOBENZOATE-META AMINOBUTYRATE-BETA AMINOPROPYL= PHOSPHINATE-3 AMINOVALERATE-DELTA AR-A-008055 AWD-131-138 CALCIUM-BIS-ACETYL-= HOMOTAURINE CEGABA CGP-29030-A CGP-44532 CGP-44533 CO-5-2791 CYCLOSERINE,LDIAMINOBUTYRATE-2,4 DIHYDROMUSCIMOL EMODEPSIDE FENGABINE GABA GABA-CETYL-ESTER GABA-ISOBUTYL GABA-MEVALONATE GABA-PALMITAMIDE GABA-STEATAMIDE GABOXADOL GANAXOLONE GLUTAPYRONE GUVACINE HOPANTENATE CALCIUM HYDROXYNIPECOTATE-4 IMIDAZOLEACETATE-4 ISOBUTYL-GABA ISOGUVACINE ISONICOTINOYL-GABA ISONIPECOTATE L-655708 LY-81067 MDL-26479 MDL-27192 MUSCIMOL NCC-05-0711 NICOTINOYL-GABA NIPECOTAMIDE NNC-711 NO-329 ORG-20380 ORG-20599 ORG-21465 PD-144550 PHTHALYL-GABA-N PIPERIDINESULFONATE-4 PROGABIDE PROGABIDE-ACID RETIGABINE ROD-185 RP-59037 RP-60503 SALUTARIDINE SKF-100330A SKF-100561 SKF-100591A SKF-100844A SKF-89976 SKF-89976A SKF-97541 SL-79-182 THIOMUSCIMOL THPO TIAGABINE U-89843-A UROCANATE GALLBLADDER CYSTIC-DUCT GANGLION-STIMULANTS AHR-602 DMPP MCN-A-343 NICOTINE NICOTINE-POLACRILEX OG-21 OG-30 OG-57 OG-90 OH-87 TETRAMETHYLAMMONIUM TETRAPROPYLAMMONIUM GANGLIONOPLEGICS AF-64A AZAMETHONIUM BROMIDE BENZOQUINONIUM CHLORISONDAMINE CHLORIDE CINNAMAMIDE DICOLINIUM IODIDE DIMECAMINE DIMECOLONIUM IODIDE DROPEMPINE EMEPRONIUM BROMIDE FUBROGONIUM IODIDE GALLAMINE-TRIETHIODIDE GANGLEFENE GUANADREL H-635 HEPTAMETHONIUM BROMIDE HEXAMETHONIUM HEXAMETHONIUM BROMIDE HEXAMETHONIUM CHLORIDE IMEQUINE LEPTODACTYLINE MECAMYLAMINE NANOFIN NEOTETRAZOLIUM OCTAMETHONIUM BROMIDE OXAPROPANIUM IODIDE P-286 PACHYCARPINE PANCURONIUM BROMIDE PEMPIDINE PENTACYNIUM CHLORIDE PENTAMETHONIUM BROMIDE PENTOLONIUM TARTRATE PHENACTROPINIUM = CHLORIDE QUATERON STILONIUM IODIDE TEMECHIN TETRAMETHONIUM BROMIDE TETRYLAMMONIUM = BROMIDE TETRYLAMMONIUM = CHLORIDE TIAMETONIUM IODIDE TREPIRIUM IODIDE TRIMETAPHAN CAMSILATE TRIMETAPHAN = NITROPRUSSIDE TRIMETHIDINIUM-= METHOSULFATE VINCANINE-= METHYLCHLORIDE GANGRENE IMMERSION-FOOT GARFT-INHIBITORS AG-2034 AG-2037 LOMETREXOL LY-298207 LY-309887 LY-316373 GASTRIC-SECRETIONINHIBITORS ACEROXATIDINE AD-2646 AG-041-R AG-1812 AG-2000 AH-22216 AHR-9294 ALE-36 AMINOINDAZOLE-6 ANTIGASTRIN AU-1421 AWD-26-06 AWD-26-39 AY-28200 AY-29315 AY-9928 B-813-19 B-831-56 BAXITOZINE BENTIPIMINE BEPERIDIUM IODIDE BL-6341A BMY-25271

Derwent Drug File 1161 Thesaurus BMY-25368 BMY-25405 BTM-1041 BTM-1042 BTM-1086 BURIMAMIDE BY-841 CAM-1028 CHLORBENZOXAMINE CI-588 CI-624 CIMETIDINE CL-115574 CL-1700 CLIDINIUM BROMIDE D-51-9927 DA-4643 DBM-819 DECITROPINE DEMETHYLNIZATIDINE-N2 DEPTROPINE-= METHOBROMIDE DICLOGUAMINE DICYCLOVERINE DONETIDINE DQ-2511 DS-4574 EBROTIDINE ELUCAINE EPIPACHYSAMINE-A ESAPRAZOLE ETINTIDINE FAMOTIDINE FENOCTIMINE FM-100 FPL-52694 FR-145715 FRG-8813 GUALENATE SODIUM GV-150013 H-200-62 H-200-66 H-200-68 H-224-25 H-335-25 HEXAPRAZOL HEXOCYCLIUM = METILSULFATE HF-2035 IBI-P-05006 ICI-162846 IGN-2098 IK-82029 ISOTHIOBARBAMINE IT-066 IY-81149 KU-1257 KW-5805 L-643411 L-643441 L-740093 LAMTIDINE LANSOPRAZOLE LEMINOPRAZOLE LOXTIDINE MAZ-525 MCN-A-1293 ME-3407 MECIADANOL METHANTHELINIUM = BROMIDE METHYLBENACTYZIUM = BROMIDE METIAMIDE METOQUIZINE MIFENTIDINE NC-1300 NC-1300-B NC-1300-SULFIDE NIK-228 NIZATIDINE NO-794 NOLINIUM BROMIDE NORBURIMAMIDE NUVENZEPINE OMEPRAZOLE ORF-17910 OXOPROSTOL P-371-A-1 PANTOPRAZOLE PARIPRAZOLE SODIUM PHENTHIMENTONIUM PICARTAMIDE PICOPRAZOLE PIFARNINE PIRENZEPINE POLDINE-METILSULFATE PROGLUMIDE PROPANTHELINE PROPANTHELINE BROMIDE QUIDITENE QUISULTAZINE RABEPRAZOLE RAMIXOTIDINE RANITIDINE RANITIDINE-BISMUTH-= CITRATE RGH-5981 RO-18-5362 RO-18-5364 ROXATIDINE RS-2039 S-0509 S-1924 S-4216 SAVIPRAZOLE SCH-28080 SCH-32651 SKF-93479 SKF-95601 SKF-96067 SOFALCONE ST-341 SU-740 SUFOTIDINE T-330 T-593 TELENZEPINE TIOTIDINE TIQUINAMIDE TOQUIZINE TRITIOZINE TRM-115 TRY-200 TU-199 TUVATIDINE TY-11345 UH-AH-37 WHR-1370A WHR-2568 WY-26769 WY-45086 WY-45662 WY-45727 YJA-20379-1 YJA-20379-8 YM-022 YM-14471 YM-220 Z-300 Z-360 ZALTIDINE ZINC-ACEXAMATE GASTRIN-ANTAGONISTS AG-041-R BENZOTRIPT CAM-1028 CAM-1481 CR-2017 CR-2093 D-51-9927 DEXLOXIGLUMIDE JB-93182 L-365260 L-368935 L-740093 P-371-A-1 PD-134308 PD-136450 PD-140548 PROGLUMIDE RC-3095 RC-3105 RC-3125 RC-3420 RC-3940-II RP-69758 RS-2039 S-0509 SPIROGLUMIDE YM-022 YM-220 GASTROENTEROPATHY ABOMASITIS ABOMASUM-DISPLACEMENT ACHALASIA ACHLORHYDRIA ACHYLIA ANAL-SACCULITIS ANUSITIS APERISTALSIS APPENDICITIS BEZOAR BLIND-LOOP-SYNDROME BLUECOMB BORBORYGMUS BRADYGASTRIA BRAXY BROWN-BOWEL-SYNDROME CARCINOID CC531 CHILAIDITI-SYNDROME CHOLERA COLECTASIA COLIC COLITIS congenital-megacolon CONSTIPATION CROHN-DISEASE CRONKHITE-CANADA-= SYNDROME CT26 DIARRHEA DIVERTICULITIS DUMPING-SYNDROME DUODENITIS DYSENTERY DYSPEPSIA EGG-YOLK-PERITONITIS EMESIS ENTERITIS ENTEROCOLITIS ENTEROHEPATITIS ENTEROLITHIASIS ENTERORRHAGIA EPIGASTRALGIA EPIPLOCELE FLATULENCE GARDNER-SYNDROME GASTRALGIA

1162 APPENDIX D GASTRITIS GASTRODUODENITIS GASTROENTERITIS GASTROPARESIS GASTROSPASM GRAIN-OVERLOAD GRASS-SICKNESS HCT116 HEM.BOWEL-SYNDROME HEM.ENTERITIS HERNIA hirschprung-disease HYPERCHLORHYDRIA HYPERCHYLIA HYPEREMESIS HYPERGASTRINEMIA HYPOCHLORHYDRIA ILEITIS ILEOCECITIS ILEUS INDIGESTION INTEST.ADENOMATOSIS INTEST.ATONY INTEST.TORSION INTUSSUSCEPTION IRRITABLE-COLON JEJUNITIS MALLORY-WEISS-SYNDROME MEGACOLON MELENA MESENTERITIS METEORISM MUCOSAL-DISEASE PARATYPHOID PERITONITIS PNEUMATOSIS-CYSTOIDES PROCTITIS PROCTOSIGMOIDITIS PROLAPSE PROTEIN-LOSING-= ENTEROPATHY PULLORUM-DISEASE PYLORIC-STENOSIS PYROSIS RECTOCELE RECTOSIGMOIDITIS RETICULITIS RINDERPEST RUMENITIS SAINT-TRIAD SALPINGOPERITONITIS SIGMOIDITIS SPRUE TACHYGASTRIA TRICHOBEZOAR TYPHLITIS ULCER VOLVULUS VOMITING-AND-WASTING-= DISEASE WHIPPLE-DISEASE GASTROINTEST.HORMONE PANCREOZYMIN-AGONIST GASTROINTEST.HORMONES A-71378 A-71623 A-72962 ACETYL-TETRAGASTRIN BC-197 BC-264 CAPROYL-TETRAGASTRIN CCK-12 CCK-5 CCK-6 CCK-7 CCK-JMV-180 DEAMIDOSINCALIDE DP-432 ENTEROGASTRONE ENTEROGLUCAGON GALANIN GALANIN-HUMAN GALANIN-PIG GASTRIC-INHIBITORY-PEPTIDE GASTRIC-INHIBITORY-= PEPTIDE-CATTLE GASTRIC-INHIBITORY-= PEPTIDE-HUMAN GASTRIC-INHIBITORY-= PEPTIDE-PIG GASTRIN GASTRIN-I GASTRIN-I-HUMAN GASTRIN-I-HUMAN-1-13 GASTRIN-I-PIG GASTRIN-II GASTRIN-II-HUMAN GASTRIN-II-PIG GASTRIN-RELEASING-PEPTIDE GASTRIN-RELEASING-= PEPTIDE-DOG GASTRIN-RELEASING-= PEPTIDE-DOG-21-27 GASTRIN-RELEASING-= PEPTIDE-HUMAN GASTRIN-RELEASING-= PEPTIDE-PIG GASTRIN-RELEASING-= PEPTIDE-PIG-1-16 GASTRIN-RELEASING-= PEPTIDE-PIG-14-27 GASTRIN-RELEASING-= PEPTIDE-PIG-18-27 GLUCAGON-37 JMV-170 JMV-180 JMV-236 JMV-310 JMV-320 JMV-328 JMV-332 KW-5139 LAUROYL-TETRAGASTRIN MEN-10208 MOTILIN MOTILIN-DOG MOTILIN-NLE-13 P-BC-264 PANCREOZYMIN PANCREOZYMIN-39 PANCREOZYMIN-AGONISTS PANCREOZYMIN-DOG-58 PANCREOZYMIN-HUMAN PANCREOZYMIN-NON-= SULFATED PANCREOZYMIN-PIG-58 PENTAGASTRIN PHI (Drug) PHI-CATTLE PHI-HUMAN PHI-PIG PHV-42-HUMAN PROGLUCAGON-78-107-PIG SECRETIN SECRETIN-5-27 SINCALIDE SNF-8702 SNF-9007 SQ-19265 SQ-19297 SQ-19300 SQ-19301 SQ-20204 SQ-20294 SUT-8701 TETRAGASTRIN UROGASTRONE VALOSIN VASOACT.INTEST.PEPTIDE VASOACT.INTEST.PEPTIDE-= 10-28 VASOACT.INTEST.PEPTIDE-= 7-11 VASOACT.INTEST.PEPTIDE-= FOWL GELATINASE-A-INHIBITORS ACETYLCYSTEINE BAY-12-9566 DOXYCYCLINE L-805645 MMI-166 PD-166793 RO-28-2653 YLL-224 GELATINASE-B-INHIBITORS ACETYLCYSTEINE BAY-12-9566 DOXYCYCLINE GW-4459 L-805645 MMI-166 PD-166793 RO-28-2653 YLL-224 GELATINASE-INHIBITORS SC-44463 GEN.ANESTHETICS ALFADOLONE ALFADOLONE-ACETATE ALFAXALONE ALIFLURANE ANAVENOL BENZYL-ALCOHOL BUTANETHIOL BUTHALITAL SODIUM CHLOROFORM CRYOFLUORANE CYCLOHEXAMINE CYCLOPENTANE CYCLOPROPANE (Drug) DESFLURANE DICHLOROETHANOL DICHLOROMETHANE DIETHYL-ETHER DIMETHYLPHENOL-2,6 DIVINYL-ETHER ELTANOLONE ENFLURANE ESTIL ETICYCLIDINE ETOXADROL FLUROXENE GYKI-21114 HALOPROPANE HALOTHANE HEPTANE HYDROXYDIONE-= SUCCINATE SODIUM I-537 ISOFLURANE KETAMINE METHITURAL METHOHEXITAL METHOXYFLURANE MIDAZOLAM MINAXOLONE NITROUS-OXIDE NORFLURANE NORKETAMINE ORG-20380 ORG-20549

Derwent Drug File 1163 Thesaurus ORG-20599 ORG-21465 PENTANE PHENCYCLIDINE PROPANIDID PROPOFOL RENANOLONE RO-21-6347 ROFLURANE SEVOFLURANE TEFLURANE THIALBARBITAL THIAMYLAL THIOBUTABARBITAL SODIUM THIOHEXITAL THIOMETHOXYFLURANE THIOPENTAL THIOPENTAL SODIUM THIOTETRABARBITAL TILETAMINE TRIBROMOETHANOL TRICHLOROETHANOL TRICHLOROETHYLENE TRIFLUOROETHANOL U-0949 URETHANE XYLAZINE GENE ONCOGENE GENE-THERAPY ANTIGENE-THERAPY GDEPT RNA-INTERFERENCE SUICIDE-GENE-THERAPY GENE-TRANSFER GENE-GUN VIRAL-VECTOR GENETICS ALLELE ANEUPLOIDY CLONE CYTOGENETICS DIPLOIDY GENE GENOTYPE HAPLOIDY HAPLOTYPE HEREDITY HETEROZYGOTE HOMOZYGOTE INHERITANCE KARYOTYPE MUTATION ONCOGENE OPERON PHENOTYPE PLEIOTROPY PLOIDY POLYPLOIDY R-FACTOR TETRAPLOIDY TRIPLOIDY GERANYLGERANYL-PROTEINTRANSFERASE-INHIBITORS BAL-9611 BZA-2-B CB-7741 GGTI-2154 GGTI-287 GGTI-297 GINKGO LI-1370 GLIOBLASTOMA CBT-CELL GLIOMA ASTROCYTOMA C6-GLIAL-CELL CG-GLIOMA EPENDYMOMA NG108-15-CELL OLIGODENDROGLIOMA SF126-CELL SF375-CELL SF407-CELL GLIOSARCOMA 9L-CELL 9L-GLIOSARCOMA GLOBULIN ADALIMUMAB ALS ALS-ANTITHYMOCYTE ALS-ANTITHYMOCYTE-= GLOBULIN ALS-ANTITHYMOCYTE-= GLOBULIN-HORSE ALS-ANTITHYMOCYTE-= GLOBULIN-RABBIT ALS-GLOBULIN ALS-HORSE ALS-RABBIT ANGIOTENSINOGEN = (Endogenous) APOLIZUMAB AUNATIV BASILIXIMAB BERIGLOBIN BEVACIZUMAB BM-01014 BT-563 BW-494 C1-ESTERASE-INHIBITOR CAMPATH-1 CAMPATH-1G CAMPATH-1H CAMPATH-1M CAMPATH-6 CENTOXIN CETUXIMAB CMV-IMMUNOGLOBULIN COLECALCIFEROL-BINDING-= GLOBULIN COLOSTRX CRP CRP-HUMAN CRYOGLOBULIN CYTOGAM CYTOTECT DACLIXIMAB DC-101 DIGIBIND DIGIDOT ECULIZUMAB EDRECOLOMAB EMD-55900 EMD-72000 ENDOBULIN EPRATUZUMAB EUGLOBULIN FLEBOGAMMA GAMIMUNE GAMIMUNE-N GAMMA-16 GAMMA-VENIN GAMMAGARD GAMMAPROTECT GAMMAR-IV GAMMASTAN GAMMIMUNE-N GAMMONATIVE GEMTUZUMAB OZOGAMICIN GLOBULIN-N GLOBUMAN HEP-B-GAMMAGEE HEPATECT HEPATITIS-B-= IMMUNOGLOBULIN HYPER-HEP IBRITUMOMAB-TIUXETAN IDEC-131 IDEC-152 IMC-1C11 INTRAGAM INTRAGLOBIN INTRAGLOBIN-F KELIXIMAB LACTOBIN MACROGLOBULIN MDX-33 MDX-H-210 MICROGLOBULIN MUROMONAB-CD3 NATALIZUMAB OCTAGAM OMALIZUMAB PALIVIZUMAB PENTAGLOBIN PENTIGETIDE POLYGAM POLYGLOBIN PSOMAGLOBIN PURIMMUN R3-36-16 RHEUMATOID-FACTOR SANDOGLOBULIN SB-249417 SEX-HORMONE-BINDING-= GLOBULIN SIPLIZUMAB SM-4300 THROMBOGLOBULIN-BETA THYROXINE-BINDING-= GLOBULIN TOSITUMOMAB VARITECT VEINOGLOBULIN VENILON VENIMMUN VENOGLOBULIN-I VENOGLOBULIN-S WINRHO GLUCAGON-AGONISTS ALX-0600 ENTEROGLUCAGON EXENDIN-4 GLICENTIN GLUCAGON GLUCAGON-1-21 GLUCAGON-37 GLUCAGON-LIKE-PEPTIDE-1 GLUCAGON-LIKE-PEPTIDE-= 1,7-36-AMIDE GLUCAGON-LIKE-PEPTIDE-= 1,7-37 GLUCAGON-LIKE-PEPTIDE-2 GLUCAGON-LIKE-PEPTIDE-= 2-HUMAN LY-307161 NN-2211 GLUCAGON-ANTAGONISTS EXENDIN-9-39-AMIDE NNC-25-2504 GLUCOSIDASE-INHIBITORS ACARBOSE AO-128 BAY-M-1099

1164 APPENDIX D CASTANOSPERMINE DEOXYNOJIRIMYCIN-1 DEOXYNOJIRIMYCIN-1-= METHYL-N EMIGLITATE MIGLITOL NONYL-DEOXYNOJIRI= MYCIN-N QUERCETIN GLUTAMATE-ANTAGONIST AMPA-ANTAGONIST KAINATE-ANTAGONIST METHYLASPARTATE-N-= ANTAGONIST GLUTAMATE-ANTAGONISTS ACEA-0593 ACEA-0762 ACEA-1021 ACEA-1031 ACEA-1328 AMPA-ANTAGONISTS B-3-277 E-2050 EGIS-8332 FG-9041 FG-9202 GAVESTINEL GYKI-52466 IEM-1460 KAINATE-ANTAGONISTS KAITOCEPHALIN LY-215490 LY-293558 LY-302679 METHYLASPARTATE-N-= ANTAGONISTS NPS-846 PD-152247 PHENIDONE RILUZOLE S-17625 SIB-1893 TOPIRAMATE YM-900 GLUTAMATEDECARBOXYLASEINHIBITORS PHENELZINE PIRACETAM SANGUINARINE TIAGABINE VIGABATRIN GLUTAMATE-RECEPTOR AMPA-RECEPTOR GLYCINE-RECEPTOR KAINATE-RECEPTOR METHYLASPARTATE-N-= RECEPTOR GLYCERIDE CASTOR-OIL (endogenous) CHAULMOOGRA-OIL EMULSION-E300 FAT INTRALIPID LIPOFUNDIN REALMENTYL TRIGLYCERIDE GLYCINE-ANTAGONISTS ACEA-0762 GLYCOGENOSIS ANDERSEN-DISEASE MCARDLE-DISEASE GLYCOLIPID GANGLIOSIDE GLOBOSIDE GLYCOPROTEIN ALPHA-1-ACID-= GLYCOPROTEIN ALPHA-2-GLYCOPROTEIN FETUIN SP-1 GLYCOSIDASE-INHIBITORS AO-128 BAY-M-1099 CASTANOSPERMINE CYCLOPHELLITOL DEOXYNOJIRIMYCIN-1 DEOXYNOJIRIMYCIN-1-= METHYL-N EMIGLITATE MANNOSTATIN-A MIGLITOL QUERCETIN GNOTOBIOTICS AXENIC HOLOXENIC MONOXENIC SPF GONADOLIBERIN-AGONISTS GONADOLIBERIN GONADOLIBERIN-SALMON GONAVET OVURELIN SUPERGESTRAN GONADOLIBERINANTAGONISTS ABARELIX ACYLINE AG-045572 AZALINE AZALINE-B CDB-2085A MI-1544 RWJ-47428-021 GONADOTROPINANTAGONISTS DANAZOL FENABUTENE INHIBIN INHIBIN-ALPHA-92 INHIBIN-ALPHA-PIG INHIBIN-BETA-HUMAN INHIBIN-CATTLE INHIBIN-PIG INHIBIN-SHEEP PENTARANE-B TALERANOL TX-380 VICOLIDE-B WY-45760 GONADOTROPINS CHORIONIC-= GONADOTROPHIN FSH FSH-ALPHA FSH-BETA FSH-CATTLE FSH-HORSE FSH-HUMAN FSH-PIG FSH-RAT FSH-SHEEP GONADOTROPIN-CARP HCG HCG-ALPHA HCG-ASIALO-= DEGLYCOSYLATED HCG-BETA HHG HMG ICSH ICSH-BETA ICSH-CATTLE ICSH-HORSE ICSH-HUMAN ICSH-PIG ICSH-SHEEP PMSG GONORRHEA fitz-hugh-syndrome gonococcal-perihepatitis GPIIB-IIIA-ANTAGONISTS ARC-69931-MX CRL-42796 ELAROFIBAN EPTIFIBATIDE F-4168 HMR-1794 L-736622 LOTRAFIBAN ME-3229 ORBOFIBAN PS-028 ROXIFIBAN SC-57101-A SR-121566 T-250 TIROFIBAN XEMILOFIBAN XJ-754 XU-063 XV-454 YM-337 YM-57029 GRAM-NEG. ACETOBACTER ACHOLEPLASMA ACHROMOBACTER ACIDAMINOCOCCUS ACINETOBACTER ACTINOBAC. AEROBACTER AEROMONAS AGROBACT. ALCALIGENES ALTEROMONAS ANAEROVIBRIO AZOTOBACTER BACTEROIDES BARTONELLA BORDETELLA BRANHAMELLA BRUC. BURKHOLDERIA BUTYRIVIBRIO CALYMMATOBACT. CAMPYLOBACTER CAPNOCYTOPHAGA CARDIOBACT. CAULOBACTER CEDECEA CHROMOBACT. CITROBACTER COMAMONAS CYTOPHAGA DICHELOBACTER E.COLI EDWARDSIELLA EMPEDOBACTER ENTEROBACTER ERWINIA ESCHERICHIA

Derwent Drug File 1165 Thesaurus FLAVOBACT. FLEXIBACTER FRANCISELLA FUSOBACT. GARDNERELLA GLUCONOBACTER HAEMOPHILUS HAFNIA HALOBACT. HELICOBACTER HISTOPHILUS KINGELLA KLEBS. LEGIONELLA LEPTOTRICHIA LYSOBACTER MEGASPHAERA meningococcus MOBILUNCUS MORAXELLA MORGANELLA MYCOPLASMA MYXOCOCCUS NEISSERIA neisseria-meningitidis PAENIBAC. PAENIBACT. PARACOCCUS PASTEURELLA PLESIOMONAS PROTEUS PROVIDENCIA PS. RHODOPS. RHODOSPIRILLUM RUMINOBACTER SALM. SAPROSPIRA SELENOMONAS SERRATIA SHIGELLA SPHAEROTILUS SPIROPLASMA STREPTOBAC. SUCCINIVIBRIO SULFOLOBUS TAYLORELLA THIOBAC. THIOBACT. UREAPLASMA VEILLONELLA VIBRIO WOLINELLA XANTHOMONAS YERSINIA ZOOGLOEA GRAM-POS. ACTINOMADURA ACTINOMYCES ACTINOPLANES AEROCOCCUS AMPULLARIELLA ARACHNIA ARTHROBACTER BAC. BIFIDOBACT. BREVIBACT. CLOSTR. CORYNEBACT. DERMATOPHILUS ENTEROCOCCUS ERYSIPELOTHRIX EUBACT. GAFFKYA GEMELLA LACTOBAC. LEUC. LISTERIA MICROCOCCUS MICROMONOSPORA MYCOBACT. NOCARDIA PEPTOCOCCUS PEPTOSTREPT. PHOTOBACT. PROPIONIBACT. RAMIBACT. RENIBACT. RHODOCOCCUS RUMINOCOCCUS SARCINA STAPH. STREPT. STREPTOMYCES STREPTOSPORANGIUM STREPTOVERTICILLIUM THERMOACTINOMYCES THERMOMONOSPORA GRANULE MICROGRANULE GRANULOMA MYOSPHERULOSIS GRANULOMATOUS-DISEASE ALLERGIC-GRANULOMATOSIS GRANULOMATOSIS idiopathic-retroperitoneal-= fibrosis JOB-SYNDROME LETHAL-MIDLINE-= GRANULOMA nodular-nonsuppurative-= panniculitis ormond-syndrome PANNICULITIS RETROPERITONEAL-FIBROSIS RHINOSCLEROMA SARCOIDOSIS weber-christian-disease WEGENER-= GRANULOMATOSIS GROWTH DIAPAUSE HEADACHE GUANYLATE-CYCLASEINHIBITORS LINSIDOMINE METHYLTHIONINIUM = CHLORIDE YC-1 GYNECOLOGY ADNEXITIS AMENORRHEA ANOVULATION BREAKTHROUGH-BLEEDING BREISKY-DISEASE CERVICITIS CYSTIC-OVARY DECIDUOSIS DYSMENORRHEA ENDOMETRIOSIS ENDOMETRITIS ENDOMYOMETRITIS FRITSCH-ASHERMAN-= SYNDROME HYPERMENORRHEA HYPOMENORRHEA MENOMETRORRHAGIA MENORRHAGIA MENSTRUAL-IRREGULARITY METRITIS METRORRHAGIA OLIGOMENORRHEA pelvic-inflammatory-disease pelvic-peritonitis PERIMETRITIS POLYMENORRHEA PYOMETRA PYOSALPINX SALPINGITIS SALPINGOPERITONITIS VULVITIS H-K-ATPASE-INHIBITORS DBM-819 MAZ-525 RABEPRAZOLE SPI-447 TY-11345 YJA-20379-1 YJA-20379-8 HEMICRANIA MIGRAINE HEART A.V.NODE ATRIUM ENDOCARDIUM EPICARDIUM HIS-BUNDLE MYOCARDIUM PAPILLARY-MUSCLE PARANODAL-FIBERS PERICARDIUM PURKINJE-FIBERS QT-INTERVAL SINOATRIAL-NODE SINUS-NODE SUBENDOCARDIUM SUBEPICARDIUM VENTRICLE HEM.DIATHESIS AFIBRINOGENEMIA ANGIOHEMOPHILIA AUTOERYTHROCYTE-= SENSITIZATION COAGULOPATHY DE-VRIES-SYNDROME DEFIBRINATION DISSEMINATED-= INTRAVASCULAR-= COAGULATION DYSFIBRINOGENEMIA EUROPEAN-BROWN-HARE-= SYNDROME glanzmann-disease HEMOPHILIA HEMOPHILIA-B HENOCH-SCHOENLEIN henoch-schoenlein-purpura hereditary-thrombasthenia hereditary-thrombopathy HYPOFIBRINOGENEMIA HYPOPROTHROMBINEMIA idiopathic-thrombocyto= penic-purpura JUERGEN-SYNDROME HAIR ALOPECIA congenital-hypotrichosis PIEDRA PILOERECTION TRICHORRHEXIS unna-syndrome HARDNESS BREAKING-STRENGTH

1166 APPENDIX D KASABACH-MERRITT-= SYNDROME MOSCHOWITZ-SYNDROME PARAHEMOPHILIA PELIOSIS-HEPATIS PLATELET-STORAGE-POOL-= DISEASE PURPURA SEIDLMAYER-SYNDROME THROMBASTHENIA THROMBOCYTOPATHY thrombocytopenic-purpura THROMBOPATHY von-willebrand-disease willebrand-juergen-disease HEMODYNAMICS AFTERLOAD BLOOD-FLOW BLOOD-PRESSURE CARDIAC-INDEX CARDIAC-OUTPUT CAROTID-BODY-REFLEX CAROTID-SINUS-REFLEX CHRONOTROPIC DIASTOLE ejection-fraction HEART-RATE HEART-RHYTHM INOTROPIC PRELOAD pulmonary-capillary-wedge-= pressure PULSE STROKE-INDEX STROKE-VOLUME STROKE-VOLUME-INDEX SYSTOLE VASCULAR-COMPLIANCE VASCULAR-RESISTANCE HEMOGLOBIN HEMOGLOBIN-F HEMOGLOBIN-S HEMORRHAGE EALE-DISEASE ECCHYMOSIS ENTERORRHAGIA EPISTAXIS HEM.TELANGIECTASIA HEMARTHROSIS HEMATEMESIS HEMATOCELE HEMATOMA HEMATURIA HEMOPERICARDIUM HEMOPERITONEUM HEMOPTYSIS HEMOTHORAX hereditary-hem.telangiectasia MELENA osler-syndrome HEMOSTATICS ADRENALONE ADRENOCHROME AETHIOPINONE AGL-1872 AMINAFTONE AMINOCAPROATE-EPSILON BATROXOBIN BENZARONE BISMUTH-TRIBROMPHENATE CALCIUM-ALGINATE CARBAZOCHROME CARBAZOCHROME-= SALICYLATE CARBAZOCHROME-= SULFONATE SODIUM CLOTTING-FACTOR-IX CLOTTING-FACTOR-IX CLOTTING-FACTOR-IXAI CLOTTING-FACTOR-VII CLOTTING-FACTOR-VIIA CLOTTING-FACTOR-VIII CLOTTING-FACTOR-VIII-= DELTA-II CLOTTING-FACTOR-VIII-= HUMAN CLOTTING-FACTOR-VIII-SQ-= HUMAN CLOTTING-FACTOR-X CLOTTING-FACTOR-XI CLOTTING-FACTOR-XII clotting-factor-xiii CONGO-RED COTARNINE DEMETHYLWEDELOLACTONE DOBESILATE CALCIUM ECARIN ELLAGATE ERGOTAMINE ESCULAMINE ESTRIOL-SUCCINATE ETAMSYLATE ETIPIRIUM IODIDE FERACRYL FIBRACCEL FIBRIN-STABILIZING-FACTOR GLUTAMYL-PLASMINOGEN GLYCYRAM GLYCYRRHIZATE HEPARIN-LYASE HISTIDINE-RICH-= GLYCOPROTEIN HYDRASTININE KABI-2161 KONYNE LERIDISTIM LEUCOCIANIDOL LEUSTRODUCSIN-H LYSYL-PLASMINOGEN MENATETRENONE METESCUFYLLINE MOBECARB NAFTAZONE NARINGIN OXAMARIN PAMBA PHTHIOCOL PHYLLOQUINONE-BETA PHYTOMENADIONE PHYTOMENADIONE-OXIDE PHYTONADIOL-= DIPHOSPHATE SODIUM PIBECARB PLATELET-FACTOR-4 PLATELET-FACTOR-4-HUMAN POLYCRESOLSULFONATE PROTEIN-C (Pharmaceutical) PROTHROMBIN SULMARIN SODIUM THROMBOPLASTIN TOLONIUM CHLORIDE TRANEXAMATE TRIMETHYLELLAGATE-3,3+,4 TRK-219 VUEFFE WEDELOLACTONE ZOOXANTHELLATOXIN-A HEPARINOIDS ACETYLHEPARIN-N APROSULATE SODIUM ARDEPARIN SODIUM ARMATAN BEMIPARIN SODIUM BM-21-23 CERTOPARIN CHONDROITINSULFATE CHONDROITINSULFATE-A CHONDROITINSULFATE-C CHONDROITINSULFATE-E CY-222 DALTEPARIN SODIUM DANAPAROID SODIUM ENOXAPARIN SODIUM FR-860 G-31150 GALACTAN-POLYSULFATE GL-522 GLUCURONYLGALACTOS= AMINO-GLYCAN-SULFATE GLUCURONYLGLUCOS= AMINO-GLYCAN-SULFATE GLYCOSAMINOGLYCAN-= POLYSULFATE GM-1077 HEPARAN-SULFATE HEPARIN HEPARIN CALCIUM HEPARIN LITHIUM HEPARIN MAGNESIUM HEPARIN SODIUM HEPARIN-BETA HEPARIN-DESULFATED HEPARIN-PENTASACCHARIDE HEPARITIN HIRUDOID IC-83-1423 INTIMATAN ITF-1300 ITF-300 LW-10078 LW-10079 LW-10086 MEPESULFATE MESOGLYCAN NADROPARIN CALCIUM OH-10172 OP-2123 OP-386 OP-622 ORG-10172 ORG-31540 ORG-31550 ORG-34006 PARNAPARIN PENTOSAN-POLYSULFATE PI-88 REVIPARINE RO-1-8307 RO-2-7509 SANORG-32701 SR-90107 SULEPAROIDE SULODEXIDE TEDELPARIN THROMBOCID TINZAPARIN SODIUM HEPATITIS SERUM-HEPATITIS VIRUS-HEPATITIS HEPATITIS-VIRUS HEPATITIS-A-VIRUS HEPATITIS-B-VIRUS HEPATITIS-C-VIRUS WOODCHUCK-HEPATITIS-= VIRUS HEPATOBLASTOMA HEP-G2-CELL

Derwent Drug File 1167 Thesaurus HEPATOMA AH130-CELL AH66-CELL H35-CELL H4-CELL HEPA1-CELL HTC-CELL KIRKMAN-ROBBINS-= HEPATOMA MH134-CELL MORRIS-HEPATOMA MORRIS-HEPATOMA-CELL NOVIKOFF-HEPATOMA NOVIKOFF-HEPATOMA-CELL SK-HEP1-CELL HEPATOPATHY ACHOLIA alcoholic-cirrhosis ANDERSEN-DISEASE angara-disease banti-syndrome bronze-diabetes budd-chiari-syndrome cholangiolitic-hepatitis cholestatic-hepatitis cholestatic-icterus chron.aggressive-hepatitis chron.congestive-= splenomegaly CIRRHOSIS CRUVEILHEIR-= BAUMGARTEN-SYNDROME DERZSY-DISEASE ENTEROHEPATITIS fat-cow-syndrome FATTY-LIVER fitz-hugh-syndrome GILBERT-SYNDROME gonococcal-perihepatitis HEMOCHROMATOSIS HEMOSIDEROSIS hepatic-coma hepatic-encephalopathy hepatic-vein-thrombosis HEPATITIS HEPATOBLASTOMA HEPATOCHOLANGITIS HEPATOLITHIASIS HEPATOMA HEPATOMEGALY HEPATORENAL-SYNDROME HEPATOSIS HEPATOSIS-DIETETICA HEPATOSPLENOMEGALY HERS-DISEASE hydropericardium-syndrome HYPERBILIRUBINEMIA ICTERUS INCLUSION-BODY-HEPATITIS KIRKMAN-ROBBINS-= HEPATOMA laennec-cirrhosis leptospiral-icterus MORRIS-HEPATOMA MOSSE-SYNDROME NOVIKOFF-HEPATOMA PELIOSIS-HEPATIS PERIHEPATITIS REYE-SYNDROME SERUM-HEPATITIS STEATOSIS TRIADITIS TYPHLOHEPATITIS VIRUS-HEPATITIS weil-disease WHITE-LIVER-DISEASE WILSON-DISEASE xanthomatous-biliary-cirrhosis ZIEVE-SYNDROME HEPATOTROPICS ACUMINATIN AGATHISFLAVONE ANDROGRAPHOLIDE ARJUNOLATE BETULONATE BPC-157 CAFFEOYLHISTAMINE CAPSICASTRINE CAPSIMINE CARPESTEROL CARSIL CELOSIAN CIANIDANOL CICLOXILATE CINNAMOYLHISTAMINE CITIOLONE CLAUSENAMIDE CLEOMISCOSIN-A COUMAROYLHISTAMINE-= PARA CPS-161 CUMAMBRIN-A CURCUMENONE DDB DEHYDROCLAUSENAMIDE DEMETHYLRICININE-N DEMETHYLWEDELOLACTONE DEOXYGOMISIN-A DEOXYPODOPHYLLOTOXIN DEOXYSHIZANDRIN DIBENZOTHIOLINE DILUDINE DIMERCAPTOPROPANE= SULFONATE-2,3 DV-7021 E-3330 EPLIR EPOMEDIOL ETIOLINE FERULOYLHISTAMINE FLAMIN GENIPOSIDE GLUTATHIONE-= MONOETHYL-ESTER GLYCYRRHETINATE-ALPHA-= 18 GOMISIN-A GOMISIN-C GOMISIN-N HEPAPOIETIN HEPATIC-STIMULATOR-= SUBSTANCE HEPATOCYTE-GROWTH-= FACTOR-DELETED HEPATOCYTE-GROWTH-= FACTOR-HUMAN HQ-275 INFLORAN ISOCHLOROGENATE-B ISOPROPOXYGERMATRANE KAIKASAPONIN-I KAIKASAPONIN-III KF-14363 KHASIANINE KOPSININE KUTKOSIDE KZ-1026 LAENNEC LECITHIN-POLYENE LEUKOMISIN LIPEXAL LIV-52 LIVOL MENBUTONE MESO-DIHYDRO= GUAIARETATE MESOPORPHYRIN-COBALT MESOPORPHYRIN-TIN MESOPORPHYRIN-ZINC METOCHALCONE MYRICADIOL MYRICANOL NCX-1000 NH-40 NICOGAMOL NKK-100 ORAZAMIDE ORNITHINE-ASPARTATE ORNITHINE-CARBAMOYL= TRANSFERASE OXOTHIAZOLIDINE-2-= CARBOXYLATE-4 PHYCOCYANIN-C PICROLIV PICROSIDE-1 PICROSIDE-2 POLYDATIN PREPARATION-E PROTEIN-C-INHIBITOR PROTOPORPHYRIN PROTOPORPHYRIN-ZINC QUADRANOSIDE-I QUADRANOSIDE-II QUADRANOSIDE-V REGOPAR REPIN RESVERATROL RHATANNIN RHODODENDRIN RICININE S-15176 SA-3443 SAIKOSAPONIN-A SAIKOSAPONIN-D SAUCHINONE SCHISANTHERIN-D SENECIONINE SHOSAIKO-TO SILANDRIN SILIBININ SILIBININ-DIHEMISUCCINATE SILICRISTIN SILIDIANIN SILIPIDE SILYHERMIN SINAPOYLHISTAMINE SOPHORADIOL-= GLUCURONIDE SY-640 TARAXEROL TARAXERONE TAUROMURICHOLATE-BETA TEFROLI TEI-2306 TENYLIDONE TETRAHYDRONEOPTERIN-= 5,6,7,8 TETRAHYDROSWERTIANOLIN THIOCTATE TIDIACIC TIMONACIC TIOPRONIN TIOTRIAZOLIN TJ-135 TOMERZOLE TR-1722 TROFOPAR TUBULOSIDE-B URAZAMIDE UVAOL WEDELOLACTONE WUWEIZISU-C Y-8845

1168 APPENDIX D YH-438 YH-439 ZY-15039 HERBICIDES 2,4,5-T 2,4-D 2,4-DB AMETRYNE AMINOZIDE AMIPROFOS-METHYL AMITROLE AMO-1618 ATRAZINE BARBAN BENFLURALIN BENSULIDE BUTURON CACODYLATE CHLORMEQUAT CHLOROACETATE CHLORPHONIUM CHLORPROPHAM CHLORSULFURON CHLORTOLURON DALAPON DAZOMET DCU DEF DI-ALLATE DICAMBA DINOSAM DINOSEB DIPHENAMID DIQUAT DIURON DNOC ETHOXYQUIN FENOPROP FLUOMETURON GLUFOSINATE GLYPHOSATE LINURON MCPA MECOPROP METFLURAZONE METHABENZTHIAZURON METHANEARSONATE METHOPROTRYNE METHYL-SULFOMETURON MOLINATE MONOLINURON MONURON MORFAMQUAT NITROFEN PARAQUAT PHOSALACINE PHOSPHINOTHRICIN PICLORAM PROMETON PROMETRYNE PROPACHLOR PROPANIL PROPHAM PROXIMPHAM SIMAZINE SWEP TERBACIL TERBUTRYNE TRI-ALLATE TRIFLURALIN VERNOLATE HERNIA ENCEPHALOCELE EPIPLOCELE MENINGOCELE MENINGOENCEPHALOCELE MENINGOMYELOCELE RECTOCELE HERPES-SIMPLEX HERPES-CORNEAE HERPES-ENCEPHALITIS HERPES-SIMPLEX-VIRUS HERPES-SIMPLEX-VIRUS-1 HERPES-SIMPLEX-VIRUS-2 HERPESVIRUS CHANNEL-CATFISH-VIRUS COITAL-EXANTHEMA-VIRUS CYTOMEGALO-VIRUS EPSTEIN-BARR-VIRUS HERPES-SIMPLEX-VIRUS HERPES-SIMPLEX-VIRUS-1 HERPES-SIMPLEX-VIRUS-2 IBR-IPV-VIRUS INCLUSION-BODY-RHINITIS-= VIRUS INFECTIOUS-= LARYNGOTRACHEITIS-= VIRUS MALIGNANT-CATARRHAL-= FEVER-VIRUS MAMILLITIS-VIRUS MAMMILITIS-VIRUS MOUSE-THYMIC-VIRUS ONCORHYNCHUS-MASOU-= VIRUS PACHECO-DISEASE-VIRUS PIGEON-HERPESVIRUS PSEUDORABIES-VIRUS PULMONARY-= ADENOMATOSIS-VIRUS RHINOPNEUMONITIS-VIRUS RHINOTRACHEITIS-VIRUS SIMIAN-VARICELLA-VIRUS VARICELLA-ZOSTER-VIRUS HIPPOCAMPUS PYRAMIDAL-CELL HISTAMINERGICS 1935-L 48-80 AMTHAMINE ANTRAMINE ARPROMIDINE BETAHISTINE BP-2-94 BU-E-75 BU-E-76 DIMAPRIT DIMETHYLHISTAMINE-N,N DIMETHYLHISTAPRODIFEN-= N,N FR-A-19 FUB-373 FUB-407 HE-30346 HE-90481 HISTAMINE HISTAPRODIFEN HOMODIMAPRIT IMETIT IMMEPIP IMPROMIDINE METHYLDIMAPRIT-N METHYLHISTAMINE-2 METHYLHISTAMINE-5 METHYLHISTAMINE-ALPHA METHYLHISTAMINE-N METHYLHISTAMINE-P METHYLHISTAMINE-T METHYLHISTAPRODIFEN-N NORDIMAPRIT PLOCAMADIENE-A SCH-49648 SCH-50971 SKF-71432-A2 SKF-71481-A2 SKF-91606 SOPROMIDINE ST-363 ST-464 ST-608 ST-93 THAPSIGARGICIN THAPSIGARGIN THAPSIGARGIN TRILOBOLIDE VUF-5297 VUF-8401 VUF-8405 VUF-8407 VUF-8411 VUF-8413 VUF-8532 VZ-20 Z-12000 Z-12001 Z-12007 HISTIDINE-DECARBOXYLASEINHIBITORS AIS-48 BROCRESINE CAFFEOYLHISTAMINE CINNAMOYLHISTAMINE COUMAROYLHISTAMINE-= PARA FERULOYLHISTAMINE HYDRAZINOHISTIDINE MCN-A-1293 MECIADANOL MONOFLUOROMETHYL= HISTIDINE SINAPOYLHISTAMINE HISTIOCYTOSIS-X eosinophilic-granuloma HAND-SCHULLER-= CHRISTIAN-DISEASE LETTERER-SIWE-DISEASE HISTOCOMPATIBILITY HLA HISTOLOGY HISTOCHEM. HISTONE NUCLEOHISTONE HISTONE-DEACETYLASEINHIBITORS BUTYRATE MS-27-275 SUBEROYLANILIDE-= HYDROXAMATE HIV-INTEGRASE-INHIBITORS AG-556 AVAROL AVARONE DICAFFEOYLTARTRATE GAP-31 HYDROXOCOBALAMIN ISOCHLOROGENATE-A ISOCHLOROGENATE-B ISOCHLOROGENATE-C L-708906 L-731988 LITHOSPERMATE-B MAP-30 NSC-115290 NSC-158393

Derwent Drug File 1169 Thesaurus ROSMARINATE T-30177 HIV-PROTEASE-INHIBITORS A-98881 AG-1402 AMARIIN AMPRENAVIR CGP-73547 DIDANOSINE DMP-450 GW-433908 H-19 INDINAVIR JE-2147 KYNOSTATIN-272 L-689502 LOPINAVIR LY-289612 NELFINAVIR NSC-158393 PD-178390 PD-178392 PNU-109112 QUERCETIN RITONAVIR SAQUINAVIR SB-203238 SC-52151 SD-146 STAVUDINE TIPRANAVIR U-103017 U-96988 UIC-94003 XR-457 XV-638 ZALCITABINE ZIDOVUDINE HIV-VIRUS HIV-1-VIRUS HIV-2-VIRUS HMG-COA-REDUCTASEINHIBITORS CERIVASTATIN CRILVASTATIN D-003 DALVASTATIN DIALLYL-DISULFIDE DIHYDROMEVINOLIN DMP-565 FLUVASTATIN GARLIC-EXTRACT LOVASTATIN MDL-28815 MEVASTATIN NK-104 PERFLUOROOCTANE-= SULFONATE PERFLUOROROOCTANOATE PRAVASTATIN ROSUVASTATIN S-1321 S-1322 SIMVASTATIN SIMVASTATIN SKF-99085 SR-9223-I SR-9223I U-20685 U-51862 U-76190 U-9888 HPLC ELECTROCHROMATOGRAPHY HYBRID INTERFERON-DELTA-4-= ALPHA-2-ALPHA-1 HYGIENE PUBLIC-HEALTH QUARANTINE HYPERBILIRUBINEMIA GILBERT-SYNDROME HYPERPIGMENTATION CHRYSIASIS MELANODERMA HYPERTENSIVES AMEZINIUM METILSULFATE CICLAFRINE CP-0597 DIMETOFRINE ETIFELMINE ETILEFRINE ETILEFRINE-PIVALATE GEPEFRINE IMINOETHYL-ORNITHINE-N K-6341 K-6343 L-163491 LACRIMIN-A M-40403 MEPHENTERMINE METARAMINOL METHOXAMINE METHYLARGININE-N-G MIDODRINE NORFENEFRINE OCTOPAMINE OENETHYL PHENYLEPHRINE SYNEPHRINE U-37883A HYPERVITAMINOSIS HYPERCAROTENEMIA HYPOCHONDRIA BODY-DYSMORPHIC-= DISORDER cardiac-neurosis da-costa-syndrome dysmorphophobia roemheld-syndrome HYPOGONADISM KALLMANN-SYNDROME HYPOLIPOPROTEINEMIA TANGIER-DISEASE HYPOTENSIVES 1045-U-85 1229-U-91 606-A 8363-S 97-139 A-025 A-127722 A-131701 A-147627 A-182086 A-192621 A-72517 A-74273 A-81988 AB-47 ABBOTT-81282 ACEPERONE ACETRYPTINE ACETYLJERVINE-O ACETYLPEPSTATIN-N ACETYLSELENONIUM-= CHOLINE ACOXATRINE ACRIP ADIMOLOL ADRENOMEDULLIN ADRENOMEDULLIN-HUMAN ADRENOMEDULLIN-RAT AE-0047 AGN-191976 AGN-193080 AHR-16303B AHR-5360 AHR-5360C AJ-2615 AJMALICINE AL-0671 ALACEPRIL ALATRIOPRIL ALFUZOSIN ALINIDINE ALIPAMIDE ALPRENOXIME ALTIOPRIL CALCIUM ALTIZIDE AMINOBENZOATE-META AMIQUINSIN AMLODIPINE AMOSULALOL ANARITIDE ANCOVENIN ANTALARMIN APORPHINE APRACLONIDINE APSTATIN AR-12463 ARANIDIPINE ARNOLOL ATENOLOL ATIPROSIN ATRASENTAN ATRIAL-NATRIURETIC-= PEPTIDE-79-98 AY-28925 AZAMETHONIUM BROMIDE AZEPEXOLE B-120 BAM-2101 BARBATUSOL BARNIDIPINE BAY-10-6734 BAY-41-2272 BAYA-6781 BENALFOCIN BENAZEPRIL BENAZEPRILAT BENCLONIDINE BENDAZOL BENDROFLUMETHIAZIDE BENIDIPINE BENOXATHIAN BENSERAZIDE BENZOYLCAPTOPRIL BENZTHIAZIDE BENZYLHYDROCHLORO= THIAZIDE BESULPAMIDE BETANIDINE BEVANTOLOL BHT-958 BIBP-3226 BIBS-222 BIBS-39 BIETASERPINE BILA-2157-BS BIMAKALIM BMS-180560 BMS-182657

1170 APPENDIX D BMS-182874 BMS-183920 BMS-184698 BMS-193884 BN-063 BN-50157 BOSENTAN BQ-123 BREFONALOL BRETYLIUM TOSILATE BRIMONIDINE TARTRATE BRL-36378 BS-1-81 BUCINDOLOL BUDRALAZINE BUFENIODE BUMEPIDIL BUPICOMIDE BUTIZIDE BUTYLPHTHALIDE-3 BUTYNAMINE BW-A575C CADRALAZINE CAFFEOYLHISTAMINE CANBISOL CANDESARTAN CANDESARTAN-CILEXETIL CANDOXATRIL CANDOXATRILAT CAPTOPRIL CAPTOPRIL-CYSTEINE CAPTOPRIL-DISULFIDE CAPTOPRIL-GLUTATHIONE CARACASANDIAMIDE CARBAMOYLTRYPTAMINE-5 CARMETIZIDE CARVEDILOL CASTALAGIN CD-349 CELIPROLOL CENTAQUINE CENTHAQUIN CENTPYRAQUIN CEREBROCRAST CERONAPRIL CETAMOLOL CGP-18137A CGP-22979A CGP-29287 CGP-38560 CGS-10078B CGS-13928C CGS-19281-A CGS-22492 CGS-22989 CGS-25155 CGS-25462 CGS-26303 CGS-26393 CGS-28106 CGS-30440 CGS-34043 CGS-35066 CHLOROBETANIDINE CHLOROTHIAZIDE CHLORTALIDONE CHOLATE CI-925 CI-926 CI-927 CI-996 CIANERGOLINE CICLETANINE CICLOSIDOMINE CIHEPTOLANE CILAZAPRIL CILAZAPRILAT CILNIDIPINE CINNAMOYLHISTAMINE CITRUSIN-C CK-53 CL-242817 CL-329167 CLADIELLOLIDE CLENTIAZEM CLOFENAMIDE CLONIDINE CODONOPSINE COUMAROYLHISTAMINE-= PARA CP-23445 CP-2907 CP-71362 CP-80794 CPU-23 CPU-57 CRISTEPIN CROMAKALIM CS-905 CV-11194 CV-5975 CYCLAZOSIN CYCLOPENTHIAZIDE CYCLOTHIAZIDE D-573 DARODIPINE DARUSENTAN DEACETYLALACEPRIL DEBRISOQUINE DEHYDROEVODIAMINE DELAPRIL DELAPRIL-DIACID DEMETHYLNAFTOPIDIL DENDROASPIS-= NATRIURETIC-PEPTIDE DENITRONIPRADILOL DEXNIGULDIPINE DEXTRONATRIN DIACETOLOL DIAZOXIDE DIBOZANE DICLOFURIME DICRANENONE-A DIHYDRALAZINE DIHYDROERGOSINE DILEVALOL DIMETHOLIZINE DIMETHYLHISTAPRODIFEN-= N,N DIPERDIPINE DIPIVALYL-TERBUTALONE DITEKIREN DMP-581 DMP-811 DORIDOSINE DOXAZOSIN DR-3438 DRAMEDILOL DROPEMPINE DU-1227 DU-1777 DU-717 DUP-532 DY-9708 E-4177 E-4701 EFONIDIPINE EG-1088 ELEDOISIN ELENOLIDE ELGODIPINE EM-311 EM-336 EM-65 EMD-52-297 EMD-56133 ENALAPRIL ENALAPRILAT ENALKIREN ENDRALAZINE EPANOLOL EPICAPTOPRIL EPITIZIDE EPROSARTAN ER-32935 ERGOSININE ES-295 ES-300 ES-305 ES-313 ES-316 ES-317 ES-6864 ES-8891 ESPROQUINE ETHINYLPROGESTERONE-18 EU-4867 EU-5476 EUPHOL EXP-063 EXP-3174 EXP-3312 EXP-3892 EXP-597 EXP-6155 EXP-6159 EXP-6803 EXP-7711 EXP-9270 FARGLITAZAR FCE-22716 FD-008 FELODIPINE FENOLDOPAM FENPERATE FERULOYLHISTAMINE FK-409 FK-739 FK-906 FLAVODILOL FLESINOXAN FLORDIPINE FLUPRANONE FLUTONIDINE FOROXYMITHINE FORSYTHIASIDE FOSINOPRIL FOSINOPRILAT FR-144420 FR-35447 FR-900359 FURIDARONE FUSARATE GALANTHINE GALLOCATECHIN-GALLATE GEA-3175 GEMOPATRILAT GHRELIN-HUMAN GINGEROL-6 GOE-5584-A GOE-6070 GOUTENIN-4 GOUTENIN-5 GR-117289-C GR-138950 GRAYANOTOXIN-1 GUABENXAN GUANABENZ GUANACLINE GUANADREL GUANAZODINE GUANCIDINE

Derwent Drug File 1171 Thesaurus GUANCLOFINE GUANETHIDINE GUANFACINE GUANISOQUINE GUANOCLOR GUANOCTINE GUANOXABENZ GUANOXAN GUANOXYFEN GW-1929 GYKI-11679 GYKI-12743 GYKI-32887 H-113 H-142 H-261 H-76 H-77 HAEMANTHAMINE HAPLOPINE HEXAMETHONIUM HEXAMETHONIUM BROMIDE HEXAMETHONIUM CHLORIDE HF-2035 HIMBACINE HIMBADINE HISTAPRODIFEN HN-65021 HOE-065 HOE-288 HOMOLYCORINE HR-720 HYDRACARBAZINE HYDRALAZINE HYDROCHLOROTHIAZIDE HYDROFLUMETHIAZIDE HYDROXYACTEOSIDE-BETA HYDROXYINDORAMIN-6 ICI-101187 ICI-106270 ICI-206970 ICI-207828 ICI-D-6888 ICI-D-8731 IDRALFIDINE IDRAPRIL IF-C-45 IGANIDIPINE IMIDAPRIL IMIDAPRILAT INDAPAMIDE INDOLAPRIL INDOLAPRILAT INDORAMIN INDORENATE IODOAMILORIDE-6 IP-66 IRBESARTAN ISF-2405 ISOBARIN ISOMANNIDE-MONONITRATE ISOTEOLINE J-104132 JERVINONE JTP-2724 K-3827 K-4011 K-4300 KC-515 KF-4307 KF-4942 KI-3005 KMD-3213 KOPSINGINE KP-403 KR-30450 KR-30988 KRI-1177 KRI-1230 KRI-1314 KRN-2391 KRN-4884 KT-3-671 KT-3-671 KUM-32 KUWANON-G KW-3433 KW-3902 L-158809 L-159689 L-159913 L-16052 L-161177 L-162223 L-162441 L-163017 L-632481 L-681176 L-749329 L-765314 L-8040 L-8142 LABEDIPINEDILOL-A LABETALOL LACIDIPINE LAMININE LEMIDOSUL LENIQUINSIN LERCANIDIPINE LEUALACIN LEVCROMAKALIM LF-20254 LIBENZAPRIL LIGUSTRAZINE LISINOPRIL LITHOSPERMATE-B LL-1418 LL-21945 LOFEXIDINE LOSULAZINE LR-693 LR-99853 LR-B-057 LR-B-081 LU-420627 LU-49938 LY-127210 LY-134046 LY-222675 LY-301875 LYCORENINE M-12285 MA-540 MCC-134 MCN-5691 MDL-100173 MDL-100240 MDL-27088 MDL-27210 MDL-43925 MECAMYLAMINE MECARBINATE MECINARONE MEDROXALOL MEDULLIPIN-I MEFENIDIL MEFESERPINE METAZOSIN METHALTHIAZIDE METHOSERPIDINE METHYLDOPA METHYLDOPATE METHYLHISTAPRODIFEN-N METHYLOXAMETHONIUM = IODIDE METHYLURAPIDIL-5 METIAPRIL METIOPRIL METIPAMIDE METIROSINE METIROSINE-METHYLESTER METOLAZONE MIBEFRADIL MIMAX MINDODILOL MINOXIDIL MJ-451 MK-286 MK-761 MK-996 MOEXIPRIL MOEXIPRILAT MOLSIDOMINE MONATEPIL MOPIDRALAZINE MOTAPIZONE MOXISYLYTE MOXONIDINE MPC-2101 MPV-207 MPV-295 MPV-304 MPV-305 MPV-390 MUZOLIMINE MYSTIXIN-11 MYSTIXIN-7 N-1518 NA-0344 NA-0345 NA-0346 NAFTOPIDIL NCX-1000 ND-186 NEBIDRAZINE NEBIVOLOL NEFERINE NEOTETRAZOLIUM NESAPIDIL NEXOPAMIL NGP-1-01 NICOPHOLINE NIGULDIPINE NIP-121 NIPRADILOL NIRAVOLINE NITRAMARINE NITRENDIPINE NITRICHOLINIUM = PERCHLORATE NITROPRUSSIDE SODIUM NITROSOCAPTOPRIL-S NOC-7 NORSALSOLINOL NPK-1867 NPK-1868 NPK-1886 OFORNINE OLEUROPEIN OLEUROPEOSIDE OLMESARTAN-MEDOXOMIL OLMIDINE OMAPATRILAT ONO-1301 ONO-AP-227 OPB-9195 OPC-28326 ORH-3088 OT-24 OUDENONE OXAMETHONIUM IODIDE OXDRALAZINE

1172 APPENDIX D OXONAZINE OXYDILIN OXYLIDINE P-1075 P-11 P-1188 P-23 PACRINOLOL PALONIDIPINE PAMATOLOL PARGYLINE PAZOXIDE PD-123177 PD-132002 PD-155080 PD-156252 PD-156707 PD-163070 PELANSERIN PEMPIDINE PENFLUTIZIDE PENPROSTENE PENTACYNIUM CHLORIDE PENTAMETHONIUM BROMIDE PENTOPRIL PENTOPRILAT PERADOXIME PERAQUINSIN PERATIZOLE PERINDOPRIL PERINDOPRILAT PH-881-7 PHENACEIN PHENACTROPINIUM = CHLORIDE PHENITRONE PHENOXYBENZAMINE PHYSALEMIN PILDRALAZINE PINACIDIL PINACIDIL-N-OXIDE PIPOCTANONE PITENODIL PIVOPRIL PM-1000 PO-285 PODILFEN POLYTHIAZIDE POMISARTAN PRACTOLOL PRAMIPEXOLE PRANIDIPINE PRAZOSIN PRIMAPERONE PRIMIDOLOL PRIZIDILOL PROPRANOLOL PROTEASOME-INHIBITOR-1 PROTOSTEPHANINE PROTOVERATRINE PROTOVERATRINE-A PROTOVERATRINE-B PST-2238 PYRROXANE QF-303 QF-307 QF-311 QF-313 QF-603 QUINAPRIL QUINAPRILAT QUINAZOSIN QUINETHAZONE QUINPIROLE QUINUCLIUM R-28935 R-29814 R-67138 R-67145 RACEMETIROSINE RAMIPRIL RAMIPRILAT RB-105 REC-0-0232 REC-15-2739 RESCIMETOL RESCINNAMINE RESERPILINE RESERPINE REV-6207 RILMAKALIM RILMENIDINE RIODIPINE RK-30 RMI-71963 RNH-6270 RO-12-4713 RO-3-7410 RO-31-6930 RO-31-8472 RO-47-8634 ROPINIROLE RP-49356 RP-61419 RPR-111844 RS-100975 RS-25560-197 RS-4045 RS-51324 RS-93522 RU-13 RUPATADINE RWJ-46458 S-0139 S-11568 S-12967 S-12968 S-23515 S-2864 S-312 S-8307 S-8350 S-8666 SA-2572 SA-7090 SALSOLINE SALSOLINOL SARALASIN SARMESIN SARPAGINE SATERINONE SAUVAGINE SB-203220 SB-209670 SB-217242 SB-239063 SC-30552 SC-46944 SC-52458 SC-52608 SCA-40 SCH-37398 SCH-39370 SCH-42495 SCH-54470 SCH-59498 SCRIP SDZ-PCO-400 SDZ-WAG-994 SEMOTIADIL SGB-1534 SGB-483 SHOGAOL-6 SINAPOYLHISTAMINE SIRATIAZEM SKF-101368 SKF-102048 SKF-102698 SKF-104856 SKF-24260 SKF-29661 SKF-64139 SKF-7698 SKF-85738 SKF-88827 SKF-89124 SKF-95018 SL-890591 SM-6586 SPHAEROPHYSINE SPIRAPRIL SPIRAPRILAT SPIRGETINE SPM-4744 SPM-5185 SPONGIATRIOL SQ-27786 SQ-32547 SQ-33351 SR-120819-A SR-121463-B SR-42128 SR-42128A SR-43845 SR-44866 SR-47063 SR-49059 ST-1913 ST-1943 ST-363 ST-464 ST-475 ST-476 ST-606 ST-608 ST-666 ST-732 ST-91 ST-93 ST-95 STAUROSPORINE STEPHARININE STH-2100 STH-2224 SULFINALOL SUN-9221 SUSPENSASIDE SY-9215 SYROSINGOPINE T-0115 T-0201 T-1032 TA-606 TAK-044 TAK-536 TAK-636 TALIPEXOLE TALUDIPINE TCV-295 TELMISARTAN TEMOCAPRIL TEMOCAPRILAT TEPROTIDE TERAZOSIN TEZOSENTAN TH-142177 THEANINE TIAMENIDINE TIAMIZIDE TIBALOSIN TIGLOIDINE TIODAZOSIN

Derwent Drug File 1173 Thesaurus TIPENTOSIN TJN-220 TOCOPHEROL-ALPHA-= FUSARATE TOCOPHERYL-QUINONE TODRALAZINE TOLMESOXIDE TOLONIDINE TRANDOLAPRIL TRANDOLAPRILAT TREQUINSIN TRETHINIUM TOSILATE TRIACSIN-C TRIACSIN-D TRICHLORMETHIAZIDE TRIMAZOSIN TRIMETAMIDE TRIMETAPHAN CAMSILATE TRIMETAPHAN = NITROPRUSSIDE TRIMETHIDINIUM-= METHOSULFATE TRIMOXAMINE TRIPAMIDE TROXONIUM TOSILATE TROXYPYRROLIUM TOSILATE TTA-386 TZC-1370 TZC-5665 U-1003 U-20057 U-2113 U-62168-E U-62168E U-71909E U-72407-E U-72407E U-72408-E U-72408E U-72409-E U-72409E U-73777-E U-77451-E U-77451E U-77455-E U-77646-E U-77646E U-77647E U-80215-E U-80215E UK-52831 UK-69578 UP-269-6 UR-12592 UR-7280 UR-8225 URAPIDIL UROCANATE UTIBAPRIL VALSARTAN VANINOLOL VERATRAMINE VICO-81 VINCAMINE VINCAMINE ADENYLATE VINIGROL VINYLPROGESTERONE-18 WAY-120491 WAY-126227 WK-1492 WS-009A WS-75624-B WY-44221 XIPAMIDE XR-510 XYLOCHOLINE Y-19638 Y-26763 Y-27152 Y-27632 YM-099 YM-11133 YM-21095 YM-358 YM-430 YM-435 YM-62899 YM-934 YP-279 Z-1046 Z-10997-A Z-13752-A ZD-1611 ZD-7155 ZK-112566 ZK-33839 ZOFENOPRIL ZOFENOPRILAT ZOFENOPRILAT-ARGININE-= SALT ZOLERTINE HYPOTHALAMUS MEDIAN-EMINENCE PARAVENTRICULAR-NUCLEUS PREMAMILLARY-NUCLEUS PREOPTIC-NUCLEUS SUPRACHIASMATIC-NUCLEUS SUPRAOPTIC-NUCLEUS VENTROMEDIAL-NUCLEUS HYPOTHALAMUS-DISEASE ADIPOSOGENITAL-= DYSTROPHY HYPOVITAMINOSIS BERIBERI BLACK-TONGUE EXUD.DIATHESIS HEPATOSIS-DIETETICA KERATOMALACIA osteodystrophia-fibrosa PELLAGRA PHRYNODERMA POLIOENCEPHALOMALACIA RACHITIS renal-osteodystrophy renal-rachitis renal-rickets SCURVY STRACHAN-SCOTT-= SYNDROME WHITE-LIVER-DISEASE ZUELZER-OGDEN-= SYNDROME ICAM-ANTAGONISTS A-286982 A-292949 ADXANTHROMYCIN ADXANTHROMYCIN-B CICLOSPORIN PD-117302 TOCOPHEROL-ALPHA ICTERUS ARIAS-SYNDROME GILBERT-SYNDROME HYPERBILIRUBINEMIA KERNICTERUS ILEUS INTEST.ATONY IMAGING-AGENTS AF-0150 AMI-121 AMI-227 AMINOINDAZOLE-6 BMS-181321 BROMOHIPPURATE BY-963 CGP-12388 CYT-356 DIISOPROPYLIMINODIACETATE DYSPROSIUM-PENTETATE DYSPROSIUM-PENTETATE-= BISMETHYLAMIDE ECHOGEN EDTA-CHROMIUM ETIOTRAST FC-3280 FERRIC-OXIDE FERRITE FLUOROCARAZOLOL FLUOROMISONIDAZOLE FS-069 GADOBENATE-DIMEGLUMINE GADOBUTROL GADODIAMIDE GADOFLUORINE-M GADOLINIUM TEXAPHYRIN GADOLINIUM-BOPTA GADOLINIUM-DO3A GADOLINIUM-DOTA GADOLINIUM-DOTA-= POLYLYSINE GADOLINIUM-= ETHOXYBENZYL-DTPA GADOLINIUM-OXALATE GADOLINIUM-TEXAPHYRIN GADOPENAMIDE GADOPENTETATE GADOPENTETATE-= BISMETHYLAMIDE GADOPENTETATE-= DIMEGLUMINE GADOPENTETATE-= DIMEGLUMINE-POLYLYSINE GADOPENTETATE-= POLYLYSINE GADOTERIDOL GADOVERSETAMIDE HL-91 IODODEXETIMIDE-4 ISOPROPYL-= IODOAMPHETAMINE L-366012 LBT-44 LU-29024 MESOPORPHYRIN-= GADOLINIUM MESOPORPHYRIN-= MANGANESE METHYLQUIPAZINE-N MRX-115 MRX-408 MS-325 NC-100100 NM-324 NM-404 NSC-678515 P-280 P-792 PALMITATE-METHYL-ESTER PENTETREOTIDE PERFLEXANE PERFLUBRON PERFLUOROPENTANE PERFLUTREN PESDA Q-12 QW-3600 RP-30 RP-30A SBK-II

1174 APPENDIX D SCH-38548 SHL-643-A SHU-454 SHU-508 SHU-508A SHU-555-A SHU-563-A SP-4 SQ-32014 SR-144385 SR-4554 TEBOROXIME TECHNEPINE TETROFOSMIN WIN-39996 IMMUNE-COMPLEX ARTHUS-REACTION IMMUNITY ANTIBODY-RESPONSE ANTIBODY-TITER IMMUNE-RESPONSE IMMUNODEFICIENCY-DISEASE AGAMMAGLOBULINEMIA AIDS AIDS-RELATED-COMPLEX ANERGY DIGEORGE-SYNDROME HYPOCOMPLEMENTEMIA HYPOGAMMAGLOBULINEMIA NEZELOF-SYNDROME RETICULAR-DYSGENESIS THYMIC-ALYMPHOPLASIA WISKOTT-ALDRICH-= SYNDROME IMMUNODET. ELISA EMIT ENZYME-IMMUNODET. GONOZYME PETINIA RADIOENZYME-IMMUNODET. RADIOIMMUNODET. IMMUNOGENICITY HACA-RESPONSE HAMA-RESPONSE IMMUNOGLOBULIN ADALIMUMAB ALS ALS-ANTITHYMOCYTE ALS-ANTITHYMOCYTE-= GLOBULIN ALS-ANTITHYMOCYTE-= GLOBULIN-HORSE ALS-ANTITHYMOCYTE-= GLOBULIN-RABBIT ALS-GLOBULIN ALS-HORSE ALS-RABBIT AMEVIVE APOLIZUMAB AUNATIV BASILIXIMAB BERIGLOBIN BEVACIZUMAB BM-01044 CAMPATH-1G CAMPATH-1H CAMPATH-1M CAMPATH-6 CENTOXIN CETUXIMAB CMV-IMMUNOGLOBULIN CYTOGAM CYTOTECT DACLIXIMAB DC-101 DIGIBIND DIGIDOT ECULIZUMAB EDRECOLOMAB EMD-55900 EMD-72000 ENDOBULIN EPRATUZUMAB FLEBOGAMMA GAMIMUNE GAMIMUNE-N GAMMA-16 GAMMA-VENIN GAMMAGARD GAMMAPROTECT GAMMAR-IV GAMMASTAN GAMMIMUNE-N GAMMONATIVE GEMTUZUMAB OZOGAMICIN GLOBULIN-N GLOBUMAN HEP-B-GAMMAGEE HEPATECT HEPATITIS-B-= IMMUNOGLOBULIN HYPER-HEP IBRITUMOMAB-TIUXETAN IDEC-131 IDEC-152 IGA IGD IGE IGG IGG1 IGG2 IGG2A IGG2B IGG3 IGG4 IGM IMC-1C11 INTRAGAM INTRAGLOBIN INTRAGLOBIN-F KELIXIMAB LACTOBIN MDX-H-210 MUROMONAB-CD3 NATALIZUMAB OCTAGAM OMALIZUMAB PALIVIZUMAB PENTAGLOBULIN POLYGAM POLYGLOBIN PSOMAGLOBIN PURIMMUN PYROGLOBULIN R3-36-16 SANDOGLOBULIN SB-249417 SIPLIZUMAB SM-4300 TOSITUMOMAB VARITECT VEINOGLOBULIN VENILON VENIMMUN VENOGLOBULIN-I VENOGLOBULIN-S WINRHO IMMUNOSTIMULANTS 104 34-M 506 86-448 A-171 A-172 ABMFPP ACEMANNAN ADA-202-718 ADAMANTANEDIOL-1,4 ADAMANTYLAMIDE-= DIPEPTIDE ADROXAZINE AGL-517 AIMFPP AL-721 ALDESLEUKIN ALOCTIN-A AM-3 AMIPRILOSE APURINIC-ACID ARABINOGALACTAN ARBIDOL ARPHAMENINE-A ARPHAMENINE-B AS-101 ASCOGEN ASCOSFEROL ASTRAGALOSIDE-I AVS-1018 AZIMEXON BAY-50-4798 BB-10010 BCG BCH-069 BCH-1393 BETATHINE BIOMUNIL BIOSTIM BLASTOLYSIN BORDETELLA PERTUSSIS BROMANTANE BROMOPHENAZONE-4 BRONCHO-VAXOM BROPIRIMINE BRU-PEL BSK BUCILLAMINE CD40-LIGAND CELLADAM CHACONINE-ALPHA CHITOHEXAOSE CIANIDANOL CID-85 CINNAMAN-AX CL-246738 CL-259763 COLIBIOGEN CONAGENIN CORD-FACTOR CORYNEBACT. PARVUM CORYNEBACT. UBERIS CORYNEBACT.CUTIS CP-46665-1 CP-64131 CRL-1005 CYANOETHYLUREA CYCLIZIDINE CYTOBLASTIN CYTOGENIN DEAZAGUANOSINE-7 DECORIN DENGUE-VACCINE DEODAN-AB DETOX DIETHYLDITHIOCARBAMATE DIHYDROHEPTAPRENOL DIUCIPHON DJ-7041

Derwent Drug File 1175 Thesaurus DODECONIUM DT-5461 DT-5461-A EPIMEDIN-C ESCULENTOSIDE-H EXODUS FACTOR-AF2 FANETIZOLE FCE-20696 FCE-24578 FK-156 FK-23 FK-565 FORFENIMEX FORMOSANIN-C FORPHENICINOL FR-46091 FR-46758 FR-47920 FR-48217 FR-900483 FR-900490 GALLIUM-NITRILOTRIACETATE GBC-590 GLA-27 GLA-40 GLA-57 GLA-58 GLA-59 GLA-60 GLA-63 GLA-65 GLA-66 GLA-70 GLUCAN-M GLYCYRRHIZAN-GA GLYCYRRHIZAN-UA GLYCYRRHIZAN-UB GM-53 GPI-0100 HEMALIN HEPTAMINOL-AMP-AMIDATE HYDROXYISOVALERATE-BETA IMEXON IMIQUIMOD IMMTHER IMREG-1 IMUVERT INTERFERON INTERFERON-ALPHA INTERFERON-ALPHA,BETA INTERFERON-ALPHA,BETAMOUSE INTERFERON-ALPHA,BETA-= RAT INTERFERON-ALPHA-1 INTERFERON-ALPHA-1-= ALPHA-8-HUMAN INTERFERON-ALPHA-1-= CATTLE INTERFERON-ALPHA-1-= HUMAN INTERFERON-ALPHA-1-= MOUSE INTERFERON-ALPHA-2 INTERFERON-ALPHA-2-1-= HUMAN INTERFERON-ALPHA-2-ARG INTERFERON-ALPHA-2-= HUMAN INTERFERON-ALPHA-2-LYS-= HUMAN INTERFERON-ALPHA-2-= MOUSE INTERFERON-ALPHA-2A INTERFERON-ALPHA-2A-= HUMAN INTERFERON-ALPHA-2B INTERFERON-ALPHA-2B-= HUMAN INTERFERON-ALPHA-2C INTERFERON-ALPHA-2C-= HUMAN INTERFERON-ALPHA-4-= HUMAN INTERFERON-ALPHA-4-= MOUSE INTERFERON-ALPHA-4A INTERFERON-ALPHA-54 INTERFERON-ALPHA-6 INTERFERON-ALPHA-7-= HUMAN INTERFERON-ALPHA-8 INTERFERON-ALPHA-A-D INTERFERON-ALPHA-A-= D(BGL-II) INTERFERON-ALPHA-B INTERFERON-ALPHA-B-D INTERFERON-ALPHA-B-D-= HUMAN INTERFERON-ALPHA-B-= HUMAN INTERFERON-ALPHA-BDBB INTERFERON-ALPHA-C INTERFERON-ALPHA-C-= CATTLE INTERFERON-ALPHA-C-= HUMAN INTERFERON-ALPHA-CATTLE INTERFERON-ALPHA-CON-1 INTERFERON-ALPHA-CON1-= HUMAN INTERFERON-ALPHA-F-D INTERFERON-ALPHA-F-= HUMAN INTERFERON-ALPHA-GAMMA INTERFERON-ALPHA-HUMAN INTERFERON-ALPHA-I INTERFERON-ALPHA-I-= HUMAN INTERFERON-ALPHA-I1 INTERFERON-ALPHA-I1-= CATTLE INTERFERON-ALPHA-II-1 INTERFERON-ALPHA-J INTERFERON-ALPHA-J-C INTERFERON-ALPHA-J1-= SER116 INTERFERON-ALPHA-K INTERFERON-ALPHA-MOUSE INTERFERON-ALPHA-N INTERFERON-ALPHA-N1 INTERFERON-ALPHA-N1-= HUMAN INTERFERON-ALPHA-N3-= HUMAN INTERFERON-ALPHA-PIG INTERFERON-BETA INTERFERON-BETA-1 INTERFERON-BETA-1-HORSE INTERFERON-BETA-1-HUMAN INTERFERON-BETA-1A INTERFERON-BETA-1A-= HUMAN INTERFERON-BETA-1B INTERFERON-BETA-2 INTERFERON-BETA-2-HUMAN INTERFERON-BETA-CAT INTERFERON-BETA-CATTLE INTERFERON-BETA-HUMAN INTERFERON-BETA-MOUSE INTERFERON-BETA-PIG INTERFERON-BETA-SER INTERFERON-BETA-SER-= HUMAN INTERFERON-CAT INTERFERON-CATTLE INTERFERON-CON-1 INTERFERON-CONCENSUS INTERFERON-DELTA-4-= ALPHA-2-ALPHA-1 INTERFERON-GAMMA INTERFERON-GAMMA-1B INTERFERON-GAMMA-4A INTERFERON-GAMMA-= CATTLE INTERFERON-GAMMA-= HUMAN INTERFERON-GAMMA-= INDUCING-FACTOR-MOUSE INTERFERON-GAMMA-= MOUSE INTERFERON-GAMMA-PIG INTERFERON-GAMMA-RABBIT INTERFERON-GAMMA-RAT INTERFERON-HUMAN INTERFERON-MOUSE INTERFERON-PI INTERFERON-RAT INTERFERON-TAU INTERFERON-TAU-HUMAN INTERFERON-TAU-SHEEP INTERLEUKIN-1-BETA-163-171 INTERLEUKIN-1-BETA-SHEEP INTERLEUKIN-10-MOUSE INTERLEUKIN-11-HUMAN INTERLEUKIN-12 INTERLEUKIN-12-HUMAN INTERLEUKIN-12-MOUSE INTERLEUKIN-13 INTERLEUKIN-13-HUMAN INTERLEUKIN-13-MOUSE INTERLEUKIN-15 INTERLEUKIN-18-HUMAN INTERLEUKIN-18-MOUSE INTERLEUKIN-2-SER-125 INTERLEUKIN-7-MOUSE IVASTIMUL JENISSEENSOSIDE-C JENISSEENSOSIDE-D JUZENTAIHOTO KEMANTAN KIFUNENSINE KRESTIN KRN-7000 L-644257 LACTOFERRIN-CATTLE LANTHIOPEPTIN LEAKADIN LENOGRASTIM LERIDISTIM LEUCOTROPHIN LEUKOREGULIN LEUSTRODUCSIN-A LEUSTRODUCSIN-B LEUSTRODUCSIN-C LEUSTRODUCSIN-H LEVAMINE-70 LEVAMISOLE LEVAN LF-1695 LIPID-X LK-409 LK-410 LOXORIBINE LW-50020 LZ-8 MACROCYCLON MACROGARD MACROGARD MAESANIN MALTOSE-TETRAPALMITATE MANGIFERIN MARCOL-52 MEDAMINE

1176 APPENDIX D MEDICAGENATE METHACIL MGN-3 MIVAL MSD-53 MURAMETIDE MURAMYL-DIPEPTIDE MURAMYL-DIPEPTIDE-B30 MURAMYL-DIPEPTIDE-= DIPALMITOYL-GLYCEROL MURAMYL-TRIPEPTIDE MVE-4 MVE-5 MY-1 MYCOBACT.BUTYRICUM MYCOBACT.CHELONAE MYCOBACT.PHLEI MYCOBACT.SMEGMATIS MYCOBACT.TUBERCULOSIS MYCOBACT.VACCAE MYELOPID MYTILAN NEURICH NEYTHYMUN NOCARDIA RUBRA NORCANTHARIDIN NOSANTINE NSC-640488 NSC-649488 O-18 OF-4949-I OF-4949-II OM-163 OM-8980 OMNADIN ONO-4007 OXALYSINE OXAMISOLE P40 PALUSTRAN PAP-I PASPAT PCF-39 PICIBANIL PIDOTIMOD PIMELAUTIDE PIND-AVI PIND-ORF POLY-A-U POLY-I-C-12-U POLY-I-C-L-C POLYACTIN-A POLYERGA POLYRIBONATE PPD PR-39 PROPIONIBACT. AVIDUM PROPIONIBACT.GRANULOSUM PYRROLOMYCIN-B QUIL-A QUILLAJA-SAPONIN REGRESSIN REHMANNAN-SA REHMANNAN-SB RESIQUIMOD RESPIVAX RGH-0205 RGH-0206 RIBI-ADJUVANT RIBOMUNYL RIGIN RM-O6 RNA-DOUBLE-STRANDED ROMURTIDE ROQUINIMEX RP-56142 RS-0481 RU-41821 RUBRATIN S-26704 S-27609 S-28463 SA-981 SAF-M SALMOSAN SAPOSHNIKOVAN-A SAPOSHNIKOVAN-C SARGRAMOSTIM SB-225002 SC-55494 SC-68420 SDK-12B-5 SDZ-280-636 SDZ-MRL-953 SITOINDOSIDE-IX SITOINDOSIDE-X SIZOFIRAN SKF-107647 SLO4 SPERGUALIN SPIRULINA-PLATENSIS SSG ST-789 STREPTENOL-A SYMBIOFLOR-I SYNTEX-ADJUVANT-= FORMULATION-1 T150R1 TAK TAN-1030-A TC-13 TEI-3096 THYMOCYTE-GROWTH-= FACTOR THYMOLYMPHOTROPIN THYMOMODULIN THYMOSTIMULIN TILOMISOLE TIPROTIMOD TJ-114 TUFTSIN TUFTSINYLTUFTSIN UKONAN-A UKONAN-B UKONAN-C UKONAN-D UKRAIN URO-VAXOM VEGETAN VILOZEN VIRULIZIN VNP-20009 WHI-P-131 WS-1279 XEROSIN-II Y-25510 Z-100 ZOSTERIN ZY-15039 ZYMOSAN-A IMMUNOSUPPRESSIVES 207-887 4162-W-94 A-771726 A-86281 ACNISTIN-A ACNISTIN-E AG-4263 ALS ALS-ANTITHYMOCYTE ALS-ANTITHYMOCYTE-= GLOBULIN ALS-ANTITHYMOCYTE-= GLOBULIN-HORSE ALS-ANTITHYMOCYTE-= GLOBULIN-RABBIT ALS-GLOBULIN ALS-HORSE ALS-RABBIT ANAKINRA ANGUIDIN ANK-102 ARABINOSYLGUANINE ARGYRIN-B ASARININ ASCOMYCIN AZATHIOPRINE AZODICARBOXAMIDE BAOHUOSIDE-1 BASILIXIMAB BATRIDENE BATZELLADINE-F BCX-34 BIDEMETHYLRAPAMYCIN-O-= 16,27 BMS-188667 BMS-224818 BOFUMUSTINE BRASINOLIDE-A BT-563 BTS-63155 BX-471 CCI-779 CGP-43902B CI-972 CIAMEXON CICLOSPORIN CLADRIBINE CP-123369 CRYPTOMERIN-B CT-2576 CX-659-S CYCLOLINOPEPTIDE-B CYCLOMUNINE CYCLOPHOSPHAMIDE CYCLOSPORIN-B CYCLOSPORIN-C CYCLOSPORIN-D CYCLOSPORIN-K CYCLOSPORIN-M CYCLOSPORIN-O CYCLOSPORIN-Q CYCLOSPORIN-U CYCLOSPORIN-V CYCLOSPORIN-Z CYTOCHALASINE-U CYTOXAZONE DACLIXIMAB DEAZAADENOSINE-3 DEHYDRODIDEMNIN-B DELAMINOMYCIN-A DEMETHYLRAPAMYCIN-O-16 DEMETHYLRAPAMYCIN-O-27 DEMETHYLRAPAMYCIN-O-39 DEOXYMETHYLSPERGUALIN DERCITIN DIHYDROCICLOSPORIN DIHYDROCYCLOSPORIN-C DIHYDROCYCLOSPORIN-D DIHYDROGUAIARETATE DIHYDROXYCHOLESTEROL-= 7,25 DISCODERMOLIDE DUNAIMYCIN-A1 DUNAIMYCIN-C2 DUNAIMYCIN-D2 DUNAIMYCIN-D2S DUNAIMYCIN-D3 DUNAIMYCIN-D4S DY-9973 DYKELLATE

Derwent Drug File 1177 Thesaurus E-5564 ER-69029 ERGOSTEROL-PEROXIDE ETANERCEPT EVEROLIMUS FR-115092 FR-900523 FR-901483 FRENTIZOLE FTY-720 FUMAGILLOL GALECTIN-1 GECLOSPORIN GLAT GLIOTOXIN-E GLIOTOXIN-G HMR-1279 HMR-1715 HP-466 HS-378 HWA-131 IDEC-131 IFOSFAMIDE IMMUCILLIN-H INTERLEUKIN-1-RECEPTOR-= HUMAN ISOCRYPTOMERIN ISOGINKGETIN ISOGUANINE ISP-I-55 J-861 JENISSEENSOSIDE-C JENISSEENSOSIDE-D KB-R-7785 KE-298 KETOIFOSFAMIDE-4 L-682993 L-683590 L-709049 LEFLUNOMIDE LICARIN-B LJP-249 LUTIDINATE LYMPHOSTIN MACHILIN-A MEDAMINE METACYCLOPRODIGIOSINE MICROCOLIN-A MICROCOLIN-B MITOCLOMINE MIZORIBINE MLR-52 MNA-279 MNA-715 MUROMONAB-CD3 MYCESTERICIN-D MYCESTERICIN-E MYCOPHENOLATE-MOFETIL N-30 NAFAMOSTAT OCHNAFLAVONE OM-01 ONO-1714 ORG-4094 OVALICIN OXECLOSPORIN OXISURAN PD-119229 PD-141955 PETUNIASTERONE-A PETUNIASTERONE-C-= ACETATE-22 PHELLODENDRINE PIMECROLIMUS PIRONETIN PNU-156804 PROCODAZOLE RAPAMYCIN RO-25-1553 RO-31-7549 RO-31-8161 RO-31-8220 RO-32-0432 RO-45-2081 RWJ-50271 SANGLIFEHRIN-A SB-210396 SCH-24937 SDZ-212-122 SDZ-214-103 SDZ-281-240 SEPIMOSTAT SIPLIZUMAB SKF-105685 SKF-106615 SM-8849 SP-100030 SPIRAZIDIN SR-31747 STROMAL-CELL-DERIVED-= FACTOR-1 STROMAL-CELL-DERIVED-= FACTOR-1-ALPHA SUFOSFAMIDE SULFAMETHOXAZOLE-= HYDROXYLAMINE SY-640 TACROLIMUS TEI-1338 TEI-6472 TEI-8364 TEL-1338 TERPRENIN TJ-135 TRESPERIMUS TRIPTONIDE TRIPTOPHENOLIDE U-0126 UNDECYLPRODIGIOSIN V-10367 VINAXANTHONE VX-497 XOMA-ZYME-H65 Y-39041 YM-13650 IMMUNOTOXIN ICI-D-0490 INFANT NEONATE INFERTILITY AHUMADA-DEL-CASTILLO-= SYNDROME ANOVULATION ARGONZ-DEL-CASTILLO-= SYNDROME ASTHENOSPERMIA AZOOSPERMIA FRITSCH-ASHERMAN-= SYNDROME HYPERESTRINISM NECROSPERMIA OLIGOSPERMIA REPEAT-BREEDING TERATOSPERMIA TESTICULAR-DYSGENESIS-= SYNDROME INFLUENZA-VIRUS INFLUENZA-A-VIRUS INFLUENZA-B-VIRUS INJECTION BOLUS I.A. I.C. I.M. I.P. I.V. INFUSION MICROINJECTION S.C. INSECT-HORMONES AI3-36206 ECDYSONE ECDYSTERONE JUVENILE-HORMONE PONASTERONE-A PYRIPROXYFEN INSECTICIDES ABAMECTIN ACRODEX ALDICARB ALDICARB-SULFONE ALDICARB-SULFOXIDE ALDRIN ALLETHRIN ALLETHRIN-I ALLETHRIN-II AMINOCARB AMITON ANABASINE APHOLATE ARAMITE ASPERENTIN AZADIRACHTIN AZAMETHIPHOS AZINPHOS-METHYL BAC.THURINGIENSIS BAYER-9017 BENDIOCARB BENOXAFOS BENZYLBENZOATE BETA-BHC BIFENTHRIN BIOALLETHRIN-S BIORESMETHRIN BOLFO BROMOCICLEN BROMOFOS BUTACARB BUTONATE CARBARIL CARBOFURAN CARBOPHENOTHION CGA-19255 CHLORBENSIDE CHLORDANE CHLORDECONE CHLORFENETHOL CHLORFENSON CHLORFENVINPHOS CHLORFLUAZURON CHLORMETHIURON CHLOROBENZILATE CHLOROPROPYLATE CHLORPHENAMIDINE CHLORPYRIFOS CHLORPYRIFOS-METHYL CHLORTHION CLENPIRIN COUMAFOS CROTOXYPHOS CRUFOMATE CYCLOPHOS CYCLOPROTHRIN CYFLUTHRIN CYHALOTHRIN CYHALOTHRIN-LAMBDA CYMIAZOLE CYOLANE

1178 APPENDIX D CYPERMETHRIN CYPERMETHRIN-ALPHA CYROMAZINE CYTHIOATE DDD DDE DDT DDT-ORTHO-PARA DEBROMOLEPTOPHOS DECARAFLURON DELTA-BHC DELTAMETHRIN DEMETON DEMETON-METHYL DENDROBACILLIN DIAZINON DICHLOFENTHION DICHLOROBENZENE-PARA DICHLORVOS DICOFOL DICRESYL DIELDRIN DIFLUBENZURON DIMATIF DIMEFOX DIMETHOATE DIMETILAN DINOCAP DIOXACARB DIOXATION DISULFOTON DIXANTHOGEN DNOC DORAMECTIN DOWCO-214 ENDOSULFAN ENDRIN ENT-51007 ENT-51143 EPN ESFENVALERATE ETAFOS ETHION ETHOATE-METHYL ETOFENPROX FAMPHUR FENAZAFLOR FENCHLORPHOS FENFLUTHRIN FENITROTHION FENOBUCARB FENOXYCARB FENPROPATHRIN FENSON FENSULFOTHION FENTHION FENVALERATE FIPRONIL FLUCYTHRINATE FLUPHENACUR FLUVALINATE FONOFOS FONOFOS-OXON FORMOTHION FOSMETHILAN GAMMA-BHC GH-74 GS-13007 HEMPA HEPTACHLOR HEPTENOPHOS HERCULES-9007 HIMACHALOL HYDROPRENE IBOTENATE IMIDACLOPRID IMIDAN IODOFENPHOS IRIDOMYRMECIN ISO-OMPA ISOFENPHOS ISOLAN ISOPROCARB IVERMECTIN KELEVAN LEPTOPHOS LG-113 LG-114 LG-115 LG-63 LIMONIN LUFENURON MAGNESIUM-= FLUOROSILICATE MALAOXON MALATHION MANUMYCIN MECARBAM MEOBAL MESULFEN METEPA METHAMIDOPHOS METHIDATHION METHIOCARB METHIOCARB-SULFOXIDE METHOCROTOPHOS METHOMYL METHOXYCHLOR METHYLETHYLTHIOPHOS METRIFONATE METRIFONATE-ACETATE MEVINPHOS MEXACARBATE MGK-264 MILBEMYCIN-A MILBEMYCIN-ALPHA-3 MILBEMYCIN-B-41D MILBEMYCIN-BETA-1 MILBEMYCIN-BETA-3 MILBEMYCIN-D MILBEMYCIN-E MILBEMYCIN-G MILBEMYCIN-OXIME MIPAFOX MIREX MITOTANE MOBAM MONOCROTOPHOS MOXIDECTIN NALED NIFLURIDIDE NIMIDANE NONACHLOR-CIS NRDC-156 OMS-15 OXYCHLORDANE OXYDEMETON-METHYL PARATHION PARATHION-METHYL PELLITORINE PERMETHRIN PEROL PHENKAPTON PHENOTHRIN PHENTHOATE PHORATE PHOSALONE PHOSMET PHOSPHAMIDON PHOXIM PINDONE PIPERINE PIPERONYL-BUTOXIDE PIRIMICARB PIRIMIPHOS-METHYL PLIZON POLYBROMINATED-BIPHENYL PROCLONOL PROFENOFOS PROMACYL PROMECARB PROPETAMPHOS PROPOXUR PYRAMAT PYRETHRIN PYRETHRIN-I PYRETHRIN-II PYRETHRUM PYRIMITATE PYRIPROXYFEN PYROCIN PYROLAN QUINALPHOS QUINTIOFOS R-14805 RESMETHRIN ROTENONE RYANODINE SCHRADAN SD-14045 SELAMECTIN SPORANDOL SULFIDOPHOS-20 SULFIRAM SULFOTEPP TEFLUBENZURON TEMEFOS TEPA TEPP TERBUFOS TETRACHLORVINPHOS TETRADIFON TETRALIN TETRAMETHRIN THANITE TOXAPHENE TRALOMETHRIN TRICYCLOHEXYLHYDROXYTIN TRIFLUMURON TRIORTHOCRESYL-= PHOSPHATE VARROXAN-T-1 VERRUCARIN-A VINCOFOS W-328 WL-22864 YT-615 INSULIN-AGONISTS AD-5075 BM-130913 CHIRO-INOSITOL CLX-0901 DIARGINYLINSULIN HOE-71-GT INSULIN INSULIN-A-CHAIN INSULIN-ASPART INSULIN-B-9-23 INSULIN-B-CHAIN INSULIN-CATTLE INSULIN-CATTLE-A-CHAIN INSULIN-CATTLE-B-CHAIN INSULIN-DETEMIR INSULIN-FOWL INSULIN-GLARGINE INSULIN-GUINEA-PIG INSULIN-HORSE INSULIN-HUMAN INSULIN-HUMAN-A-CHAIN INSULIN-HUMAN-B-CHAIN INSULIN-HUMAN-B10-ASP

Derwent Drug File 1179 Thesaurus INSULIN-HUMAN-B10-GLU INSULIN-HUMAN-B28-= LYS,B29-PRO INSULIN-HUMAN-B9-ASP,= B27-GLU INSULIN-PIG INSULIN-RABBIT INSULIN-RAT INSULIN-SAPG INSULIN-SHEEP L-783281 MERCK-L-7 METHYLCYSTEINE-= SULFOXIDE-S NN-304 PROINSULIN PROINSULIN-CATTLE PROINSULIN-HUMAN PROINSULIN-HUMAN-DE-= 64-65 PROINSULIN-MONKEY PROINSULIN-PIG VANADYL DIPICOLINATE INSULIN-ANTAGONISTS BPDZ-44 BPDZ-62 DC-23-99 INTEGRIN-ANTAGONIST VLA-4-ANTAGONIST INTEGRIN-ANTAGONISTS EMD-121974 EMD-270179 EMD-66203 F-4168 LM-609 NEUTROPHIL-INHIBITORY-= FACTOR S-137 S-247 SB-273005 SH-306 SJ-749 SKF-107260 ST-1646 VLA-4-ANTAGONISTS XT-199 INTEGRIN-RECEPTOR alpha4beta1 cd49d-cd29 VLA-4 INTERFERON-INDUCERS 6-MFA AIPP APURINIC-ACID AVRIDINE BAYFERON BL-20803 BRL-10739 BRL-5907 BROPIRIMINE CARBOXYMETHYL= ACRIDANONE-10 ESCULENTOSIDE-H FCE-20696 GLA-27 GLA-40 GLA-57 GLA-58 GLA-59 GLA-60 GLA-66 GLA-70 IMIQUIMOD IMURESP-P INTERLEUKIN-18-MOUSE LAFARINE LARYPHANE MA-56 MOP-35 MOP-79 NSC-46015 NSC-46015-C OXYAMYLOSE POLY-A-U POLY-G-C POLY-I-C POLY-I-C-12-U PXL-6 RIDOSTIN RIFASTINE RMI-10874-DA RMI-11002-DA RMI-11567-DA RMI-11877-DA RMI-9563-DA RMI-9567-DA RNA-DOUBLE-STRANDED S-26704 S-27609 S-28828 SLO4 SSM STATOLON TASH-3 TASH-4 TASH-5 TILORONE TOLPA U-25166 INTERLEUKIN-CONVERTINGENZYME-INHIBITORS EI-1511-3 EI-1625-2 L-709049 MANUMYCIN MANUMYCIN-B MANUMYCIN-G U-56407 WIN-67694 INTERLEUKIN-RECEPTOR INTERLEUKIN-2-RECEPTOR INTERMEDIN-AGONISTS ACTH-1-13-AMIDE HP-466 INTERMEDIN INTERMEDIN,4-NLE-7-D-PHE INTERMEDIN-ALPHA INTERMEDIN-BETA INTERMEDIN-BETA-CATTLE INTERMEDIN-BETA-HORSE INTERMEDIN-BETA-HUMAN INTERMEDIN-BETA-MONKEY INTERMEDIN-BETA-PIG INTERMEDIN-GAMMA INTERMEDIN-GAMMA-3 INTERMEDIN-ANTAGONISTS SHU-9119 INTERSEX GILBERT-DREYFUS-= SYNDROME goldberg-maxwell-morris-= syndrome GORDAN-OVERSTREET-= SYNDROME HELLER-NELSON-SYNDROME HERMAPHRODITISM KLINEFELTER-SYNDROME PSEUDOHERMAPHRODITISM REIFENSTEIN-SYNDROME testicular-feminization TURNER-SYNDROME INTEST.FLORA BIOFLORIN INTESTINE APPENDIX CC531 CECUM COLON CT26 DUODENUM HCT116 ILEUM JEJUNUM MESENTERY PERISTALSIS RECTUM TAENIA-CAECI TAENIA-COLI INTOXICATION ALVELD ARGYRIA BOTULISM BRIGHT-BLINDNESS BROMINISM ERGOTISM FESCUE-FOOT FLUOROSIS LUPINOSIS OSTEOLATHYRISM TOX.OIL-SYNDROME INTRAUTERINE-DEVICE DALKON-SHIELD LIPPES-LOOP MARGULIES-SPIRAL IONEXCHANGERS AMBERLITE AMBERLITE-IRC-50 AMBERLITE-XAD-4 COLESTYRAMINE DOWEX FILICOL MCI-196 POLACRILIN POTASSIUM POLIDEXIDE POLYSTYRENE-SULFONATE = CALCIUM POLYSTYRENE-SULFONATE = SODIUM IONOPHORES A-204A ABIERIXIN ALBORIXIN AS-701 BEAUVERICIN BROMOLASALOCID CALCIMYCIN CARRIOMYCIN CATIONOMYCIN CEZOMYCIN CP-53607 CP-82009 CP-84657 CYCLEX-2E DEOXYSALINOMYCIN DIANEMYCIN EPINIGERICIN ETHEROMYCIN GRAMICIDIN GRAMICIDIN-A GRAMICIDIN-J2 GRAMICIDIN-NF GRAMICIDIN-S GRAMICIDIN-S-2 GRAMICIDIN-S-3

1180 APPENDIX D GRISEOCHELIN GRISORIXIN HEPOXILIN-A3 INDANOMYCIN IONOMYCIN ISOLASALOCID-A KRYPTOFIX-221 LAIDLOMYCIN LAIDLOMYCIN-BUTYRATE LASALOCID LASALOCID-A LASALOCID-B LASALOCID-C LASALOCID-D LASALOCID-E LENOREMYCIN LONOMYCIN LONOMYCIN-A LONOMYCIN-B LONOMYCIN-C LYSOCELLIN MADURAMICIN MADURAMICIN-ALPHA MAMMOSIDE-A MAMMOSIDE-B MAMMOSIDE-H1 MAMMOSIDE-H2 MENENSIN-B MONAZOMYCIN-A MONENSIN MONENSIN-A MONENSIN-B MONENSIN-C MOYUKAMYCIN NARASIN NIGERICIN NOBORITOMYCIN-A NOBORITOMYCIN-B NORBORITOMYCIN-A NORBORITOMYCIN-B OKADAATE OMOMYCIN PAMAMYCIN-607 ROFLAMYCOIN SALINOMYCIN SEMDURAMICIN SEPTAMYCIN T150R1 TETRANACTIN TETRONASIN TETRONOMYCIN VALINOMYCIN X-14667A X-14868A X-14868B X-14868C X-14868D X-14873A X-14885A X-14889C X-206 ZINCOPHORIN IRIDOVIRUS FROG-VIRUS-3 ISOTOPIC-THERAPY NEUTRON-CAPTURE-= THERAPY JOINT ANKLE HIP KNEE LIGAMENT STIFLE WRIST JOINT-DISEASE ALBERT-SYNDROME ARTHRALGIA ARTHRITIS ARTHROSIS BOG-SPAVIN BONE-SPAVIN BURSITIS caplans-syndrome CAPSULITIS CARPITIS CHONDROCALCINOSIS CLUTTON-SYNDROME congenital-= arthromyodysplasia COXARTHROSIS COXITIS DACTYLITIS DISLOCATION FELTY-SYNDROME GONARTHRITIS GONARTHROSIS GONITIS GOUT GRAM-SYNDROME guerin-stern-syndrome HEMARTHROSIS HOFFA-KASTERT-SYNDROME HYDRARTHROSIS hypertrophic-pulmonary-= osteoarthropathy idiopathic-hypertrophic-= osteoarthropathy JOINT-ILL juvenile-rheumatoid-arthritis LYME-ARTHRITIS marie-bamberger-syndrome MARIE-LERI-SYNDROME neuropathic-arthritis OSTEOARTHRITIS OSTEOARTHROPATHY OSTEOARTHROSIS PERIARTHRITIS PNEUMARTHROSIS POLYARTHRITIS POLYMYALGIA-RHEUMATICA POLYSYNOVITIS PONCET-DISEASE PROFICHET-DISEASE PSEUDOGOUT PSEUDOPOLYARTHRITIS putti-syndrome PYOARTHROSIS REITER-SYNDROME RHEUMATIC-FEVER rheumatic-pneumoconiosis rheumatic-sciatica rheumatism rheumatoid-arthritis SACROILIITIS SAPHO-SYNDROME SPRAIN STIEDA-PELLEGRINI-= SYNDROME still-syndrome SWEET-ITCH SYMPHISIS SYNOVITIS TEMPOROMANDIBULAR-= JOINT-SYNDROME touraine-solente-gole-= syndrome uehlinger-syndrome KAINATE-AGONISTS KAINATE KAINATE-ANTAGONISTS FG-9202 GYKI-52466 IEM-1460 PHENIDONE RILUZOLE TOPIRAMATE YM-900 KERATITIS HERPES-CORNEAE herpes-keratitis KERATOLYTICS ALCLOXA ALDIOXA BENZOYLPEROXIDE BMY-30123 IMEDEEN ISOTRETINOIN ISOTRETINOIN-METHYL-= ESTER MOTRETINIDE PICOTRIN PYROGALLOL-TRIACETATE RETINYLIDENE-= METHYLNITRONE RO-12-7554 RO-12-9933 RO-22-6595 SALICYLATE SALICYLATE TROLAMINE SOLCODERM TAZAROTENE TETROQUINONE TRETINOIN TRETINOIN-METHYL-ESTER U-75412E KERATOSIS MAL-DE-MELEDA KIDNEY ANEPHRIC BHK-CELL BHK21-CELL C3H2K-CELL CV1-CELL DIURESIS glomerular-filtration-rate GLOMERULUS GLV3-CELL HAK-CELL HEK-CELL IBRS2-CELL JUXTAGLOMERULAR-CELL kaliuresis LLC-MK2-CELL LLC-PK1-CELL LLC-RK1-CELL LOOP-OF-HENLE MA104-CELL MDBK-CELL MDCK-CELL natriuresis NEPHRON PK15-CELL potassium-diuresis proximal-tubule RK13-CELL sodium-diuresis VERO-CELL KINETOSIS AIR-SICKNESS KININS ADIPOKININ BRADYKININ BRADYKININ,MET-LYS BRADYKININ-8-LEU-DE-ARG-9 BRADYKININ-8-TYR BRADYKININ-DE-ARG-1

Derwent Drug File 1181 Thesaurus BRADYKININ-DE-ARG-9 COLOSTROKININ FR-190997 KALLIDIN KALLIDIN-9-LEU-DE-ARG-10 KALLIDIN-DE-ARG-10 KALLIKREIN T-KININ LAB.ANIMAL ARMADILLO AXOLOTL BABOON BADGER BAT BEAR BUSH-RAT CAPUCHIN CAT CATTLE CHIMPANZEE CHIPMUNK CLAM COTTON-RAT COYPU CRAB CRAYFISH DOG DUCK EEL ewe female-sheep FERRET FOWL FOX FROG GERBIL GOAT GOLDFISH GOOSE GORILLA GROUND-SQUIRREL GUINEA-PIG HAMSTER HARE HORSE JELLYFISH JIRD LEMMING LION LIZARD LOBSTER MACAQUE MARMOSET MINIPIG MINK MONKEY MOUSE MUDPUPPY MULE MUSKRAT OPOSSUM ORANG-UTAN PARTRIDGE PEACOCK PHEASANT PIG PIGEON PRAIRIE-DOG QUAIL QUOKKA RABBIT RAT rhesus-monkey SALAMANDER SHARK SHEEP SHREW SNAIL SPIDER SQUID SQUIRREL-MONKEY SUNCUS TADPOLE TAMARIN TERRAPIN TIGER TOAD TORTOISE TURKEY VOLE WOODCHUCK young-sheep LACTATION GALACTORRHEA HYPOGALACTIA POLYGALACTIA LAXATIVES ABT-229 AGAR AGIOLAX ALOE-EMODIN ALOIN AS-4370 BISACODYL BISOXATIN BOLDINE CASANTHRANOL CASCAROSIDE-A CHOLATE COFISATIN DANTRON DEACETYLBISACODYL DIOCTYLSULFOSUCCINATE CALCIUM DOCUSATE SODIUM GLUCOFRANGULIN GUM-KARAYA ISPAGHULA JALAP KAMALA KF-66854 LACTITOL LACTULOSE MANNITOL MICROLAX NUX-VOMICA OXYPHENISATINE OXYPHENISATINE-ACETATE PARAFFIN-LIQUID PHENOLPHTHALEIN PHENOLPHTHALOL PHORBOL PICOFOSFATE SODIUM PICOSULFATE SODIUM POLOXAMER-188 POLYCARBOPHIL PSYLLIUM RHEINANTHRONE SC-46499 SENNIDIN-A SENNIDIN-B SENNOSIDE SENNOSIDE-A SENNOSIDE-A1 SENNOSIDE-B SENNOSIDE-C SENNOSIDE-D SENNOSIDE-D1 SENNOSIDE-E SENNOSIDE-F SORBITOL SR-57746A SULFOSUCCINATE SULISATIN TANNATE YM-31636 Z-338 LEIOMYOMA MG34-CELL LEUKEMIA AKR-CELL BCL1-CELL CCRF-CEM-CELL FRIEND-LEUKEMIA FRIEND-LEUKEMIA-CELL GROSS-LEUKEMIA GROSS-LEUKEMIA-CELL hairy-cell-leukemia HL60-CELL HUT102B2-CELL J111-CELL JURKAT-CELL KG1-CELL L1210 L1210-CELL L2C-CELL L40 L40-CELL L5222 L5222-CELL LAZ007-CELL leukemic-reticuloendotheliosis MBL2-ASCITES MBL2-CELL ML1-CELL MOLT3-CELL MOLT4-CELL P388 P388-CELL RAW264-CELL RPMI6410-CELL RPMI8402-CELL SKL2-CELL SKL5-CELL U937-CELL LEUKOCYTE BASOPHIL EOSINOPHIL GRANULOCYTE HETEROPHIL LEUKOBLAST LEUKOPOIESIS METAMYELOCYTE MONOBLAST MONOCYTE MYELOBLAST MYELOCYTE NEUTROPHIL POLYMORPHONUCLEAR LEUKOCYTE-DISORDER CHEDIAK-HIGASHI-= SYNDROME EOSINOPHILIA EOSINOPHILIA-MYALGIA-= SYNDROME HYPEREOSINOPHILIC-= SYNDROME KARTAGENER-SYNDROME LEUKOCYTOSIS LEUKOSTASIS MONOCYTOSIS NEUTROPHILIA PELGER-HUEET-ANOMALY PSEUDOLEUKOCYTOSIS LEUKOSIS-COMPLEX ERYTHROLEUKOSIS mareks-disease mareks-disease

1182 APPENDIX D LEUKOTRIENE-ANTAGONISTS 208-199 A-65260 A-69412 A-78773 A-79175 A-93178 AA-1777 AA-863 ABBOTT-63162 ABLUKAST ABT-080 ABT-761 AD-3264 AH-9679 AMLEXANOX ARTOBILOXANTHONE AS-35 ATRACTYLOCHROMENE BAY-U-9773 BAY-X-1005 BAY-X-7195 BAY-Y-1015 BI-L-226XX BI-RM-270 BORNYL-COUMARATE BUDDLEDIN-A BW-755C BW-A137C BW-A4C BW-A797C BW-B218C BW-B70C CANNIPRENE CBS-113A CGP-34064A CGP-35949 CGP-44826 CGP-45715A CGP-47969-A CGP-57698 CGS-23885 CGS-25019-C CGS-25019C CGS-8515 CI-986 CMI-392 CMI-947 CO-1828 CP-105696 CP-195494 CP-195543 CP-199331 CV-6504 DIPHENYL-DISULFIDE DOCEBENONE DOQUALAST DS-4574 DUP-654 E-3040 E-3330 E-6080 EBSELEN EICOSADIENOATE-11,14 EICOSATRIENOATE-11,14,17 EMETHALLICIN-A EMETHALLICIN-B EMETHALLICIN-C EN-105 ENOFELAST EP-045 ETH-615 F-5 FLINDERSINE FLM-5011 FPL-55618 FPL-55712 FPL-57231 FPL-64170-XX FR-71021 FUSCOSIDE-B GLYCERYL-TRIDOCOSA= HEXAENOATE HALICHOLACTONE HQNO ICI-198615 ICI-207968 ICI-211965 ICI-216800 ICI-D-2138 ISOPETASIN KC-404 KZ-111 L-615919 L-648051 L-649923 L-651392 L-651896 L-652343 L-654639 L-655238 L-655240 L-656224 L-657098 L-660711 L-665210 L-669572 L-670592 L-670602 L-670630 L-674573 L-674636 L-686708 L-689037 L-699333 L-699392 L-746530 LEUCETTAMINE-A LEUCETTAMINE-B LINOLENATE-METHYL-ESTER LM-1453 LM-1468 LONAPALENE LY-137617 LY-163443 LY-178002 LY-183001 LY-189585 LY-203647 LY-223980 LY-223982 LY-255283 LY-256548 LY-280810 LY-293111 LY-83583 MCI-826 METHYLFLINDERSINE-N MK-0591 MK-886 MONTELUKAST MY-12-62-C NAFAZATROM NEUTROPHIL-INHIBITORY-= FACTOR NITECAPONE NORDIHYDROGUAIARETATE ONO-LB-457 ONO-RS-347 OSTHENOL OXATOMIDE OXPHALIN OXPHAMAN PF-10042 PF-5901 PGV-20229 PH-163 PHLEBIACHRYSOATE-B PHLEBIACHRYSOATE-D PIRIPROST PZ-25 QA-208-199 QUINOTOLAST R-68151 REV-5901 REV-5901-A RG-12525 RG-12553 RG-14893 RG-6866 RG-7152 RITOLUKAST RO-24-5913 RO-25-3562 RP-64966 RP-69698 RWJ-63556 SANGGENON-B SB-203347 SC-37872 SC-41930 SC-45662 SC-50605 SC-51146 SC-53228 SC-57461 SCH-37224 SCH-40120 SERINE-BORATE SKF-101132 SKF-102081 SKF-102922 SKF-104353 SKF-104353-Z2 SKF-104373 SKF-104493 SKF-105809 SKF-106203 SKF-107310 SKF-86002 SKF-86002-A2 SKF-S-106203 SL-81-0433 SM-11044 SM-15178 SM-9064 SR-2640 SULUKAST T-0757 TEI-1338 TEL-1338 TENIDAP TEPOXALIN TOMELUKAST TX-11027 TZI-41127 U-56467 U-66858 U-75302 U-75305 U-75360 U-75485 U-77692 U-78489 VERLUKAST VZ-65 WAY-120739 WAY-121006 WAY-121520 WEDELOLACTONE WF-11605

Derwent Drug File 1183 Thesaurus WY-44329 WY-45911 WY-47288 WY-48090 WY-49232 WY-50295 WY-50295-C WY-50295-T Y-19432 YM-16638 YM-57158 YPE-01 ZAFIRLUKAST ZARDAVERINE ZILEUTON ZIMET-18-84 ZIMET-19-84 ZIMET-20-84 ZIMET-22-84 ZIMET-25-85 ZIMET-53-84 ZIMET-58-85 ZIMET-61-85 ZIMET-72-85 ZK-158252 LEUKOVIRUS AVIAN-SARCOMA-VIRUS BIV-VIRUS C-TYPE-VIRUS ERYTHROLEUKOSIS-VIRUS FIV-VIRUS FRIEND-VIRUS GROSS-VIRUS HIV-1-VIRUS HIV-2-VIRUS HIV-VIRUS HTLV-I-VIRUS HTLV-II-VIRUS KIRSTEN-VIRUS LEUKOSIS-VIRUS MASON-PFIZER-MONKEY-= VIRUS MOLONEY-VIRUS MOUSE-SARCOMA-VIRUS MYELOBLASTOSIS-VIRUS RAUSCHER-VIRUS RETICULOENDOTHELIOSIS-= VIRUS ROUS-SARCOMA-VIRUS SIMIAN-SARCOMA-VIRUS SIV-VIRUS SQUIRREL-MONKEY-= RETROVIRUS STLV-III-VIRUS LEVO-ISOMER SD-3212 LICHEN CLADONIA DINARIA LECANORA PARMELIA LIFE-CYCLE AMASTIGOTE PROMASTIGOTE LIPID-METAB. BETA-OXIDATION KETOGENESIS LIPID-PEROXIDATION LIPOGENESIS LIPOLYSIS LIPID-METAB.DISORDER ABETALIPOPROTEINEMIA buerger-grutz-syndrome CHYLOMICRONEMIA disseminated-= lipogranulomatosis DOLLINGER-= BIELSCHOWSKY-= SYNDROME FABRY-SYNDROME familial-hyperlipoproteinemia farber-syndrome FAT-NECROSIS GANGLIOSIDOSIS GAUCHER-DISEASE GRAM-SYNDROME hanot-macmahon-= tannhauser-syndrome HYPERCHOLESTEROLEMIA HYPERCHYLOMICRONEMIA HYPERLIPEMIA HYPERLIPOPROTEINEMIA HYPERTRIGLYCERIDEMIA HYPOBETALIPOPROTEINEMIA HYPOCHOLESTEROLEMIA HYPOLIPEMIA HYPOLIPOPROTEINEMIA KETOACIDOSIS KETOSIS KUFS-DISEASE LIPIDOSIS LIPIDURIA LIPODYSTROPHY LIPOGRANULOMATOSIS LIPOMATOSIS metabolic-syndrome METABOLIC-SYNDROME-X NEUROLIPOMATOSIS NIEMANN-PICK-DISEASE PHOSPHOLIPIDOSIS prim.familial-xanthomatosis progressive-lipodystrophy LIPOXYGENASE-INHIBITORS A-78773 A-79175 A-93178 ABBOTT-63162 ABT-761 ATRACTYLOCHROMENE BAY-X-1005 BI-L-226XX BUDDLEDIN-A BW-A4C CENTAUREIDIN CGS-23885 CMI-206 CMI-392 CMI-947 CP-102 CP-25 CP-26 CV-6504 ERIOCEPHALIN F-1067 FPL-64170-XX FUSCOSIDE-B ICI-230487 ICI-D-2138 L-656224 L-670630 L-689065 L-691816 L-699333 L-702539 L-739010 LAGASCATRIOL LAGUNAMYCIN LICOFELONE LY-280810 MK-0591 MK-886 MORNIFLUMATE OSTHENOL SANDHOFFS-DISEASE simons-syndrome SITOSTEROLEMIA SPIELMEYER-SJOEGREN-= DISEASE TANGIER-DISEASE TAY-SACHS-DISEASE wolman-disease XANTHOMA XANTHOMATOSIS xanthomatous-biliary-cirrhosis LIPOSARCOMA SA1-CELL LIPOSOME IMMUNOLIPOSOME P-8977 PD-146176 PRANTSCHIMGIN R-85355 REV-5901 ROOPEROL RWJ-63556 SANDARACOPIMARATE SANGGENON-B SB-202235 SB-210661 SC-41661A SCH-40120 T-0757 TETRAMETHYLLUTEOLIN TETRAMETHYLSCUTELLAREIN TEUCRIN-A TRIMETHYLAPIGENIN TZI-41127 WAY-121520 WY-50295-T YPE-01 ZILEUTON LITHIASIS biliary-calculi CHOLEDOCHOLITHIASIS CHOLELITHIASIS HEPATOLITHIASIS kidney-calculi NEPHROLITHIASIS UROLITHIASIS LITHOLYTICS CHENODEOXYCHOLATE COCONUT-OIL G-871 G-872 ISOPROPYL-ACETATE LIFIBROL METHYLCHENODEOXY= CHOLATE-7-BETA METHYLCHOLATE-7-BETA MONOOCTANOIN MTBE NORURSODEOXYCHOLATE ROSMANOL ROWACHOL SARCOURSODEOXYCHOLATE SF-482 SODIUM-POTASSIUM-= CITRATE URSODEOXYCHOLATE URSULCHOLATE LIVER HEPATOCYTE KUPFFER-CELL

1184 APPENDIX D LIVER-OIL AMEU ANCHOVY-OIL COD-LIVER-OIL FISH-OIL MENHADEN-OIL LOCAL-ANESTHETICS 6211 6603 ACETYLCAINE AGATOXIN-ALPHA-489 ALLOCOCAINE ALLOPSEUDOCOCAINE ALLYLNORCOCAINE AMBUCAINE AMOLANONE AMOXECAINE AMYDRICAINE AMYLOCAINE APTOCAINE ARTICAINE AZACAINE BENAMOCAINE BENCAINE BENZOBUTAMINE BENZOCAINE BENZONATATE BETOXYCAINE BRONCHOCAINE BUCRICAINE BUMECAINE BUPIVACAINE BUPIVACAINE-CARBONATED BUTACAINE BUTAMINE BUTANILICAINE BUTETHAMINE BUTOFORM BW-62-235 CARBISOCAINE CHLOROBUTANOL CHLOROPROCAINE CINCHOCAINE CLIBUCAINE CLODACAINE CLOFEXAMIDE CLORMECAINE COCAINE CYCLOMETHYCAINE CYMENE DEXIVACAINE DIAMOCAINE DICARFEN DIMETHOCAINE DIOCAINE DIPERODON DROXICAINIDE DYCLONINE ECGONINE EDAN EDRONOCAINE ELUCAINE ETHONIUM ETIDOCAINE EUCAINE-BETA EUGENOL EUPROCIN F-1459 FENOXAZOLINE FEXICAINE FOMOCAINE G-491 GEA-968 GUAFECAINOL HEPTACAINE HEXYLCAINE HS-37 HYDROXYCAINE HYDROXYPROCAINE HYDROXYTETRACAINE ICHTHYOCALM IQB-9302 ISOBUTAMBEN ISOBUTYLCAINE K-1905 KETOCAINE KETOCAINOL KP-23 L-30 L-48 L-7810 LEA-103 LEFETAMINE LEUCINOCAINE LIDOCAINE LM-207 LM-246 LOTUCAINE LS-93 MENTHOL MEPIVACAINE MEPRYLCAINE METABUTETHAMINE METACAINE MIDAMALINE MYRTECAINE NAEPAINE NEOPSICAINE NICOTINOYL-PROCAINE NORCOCAINE OCTACAINE OCTYLACAINE ORTHOCAINE OXETACAINE OXYBUPROCAINE PARETHOXYCAINE PARIDOCAINE PHENACAINE PHENODIANISYL PINCAINIDE PINOLCAINE PIPEROCAINE PIPEROCAINE-METHIODIDE PIRIDOCAINE POLIDOCANOL PRAMOCAINE PRIBECAINE PRILOCAINE PROCAINE PROPANOCAINE PROPIPOCAINE PROPOXYCAINE PROXYMETACAINE PSEUDOCOCAINE PYRROCAINE QUATACAINE QUINISOCAINE QX-222 QX-314 QX-572 RAC-109 RAD-150 RAD-154 RAD-179 RAD-240 RAD-241 RAD-242 RAD-243 RAD-244 RAD-393 RAG-505 RHINOCAINE RISOCAINE RODOCAINE ROPIVACAINE SA-130 SA-167 SA-36 SA-61 SA-62 SA-63 SA-67 SAMERIDINE SCH-221 STADACAIN TEECAINE TETRACAINE TOLYCAINE TRAPENCAINE TRIMECAINE TRIMETHISOQUIN W-36017 W-49091 W-6603 W-82139 XENYSALATE ZOLAMINE LOW MOL. WEIGHT ARDEPARIN SODIUM DALTEPARIN SODIUM DANAPAROID SODIUM DEXTRAN-1 ENOXAPARIN SODIUM NADROPARIN CALCIUM OP-2123 OP-386 OP-622 ORG-10172 ORG-31540 ORG-31550 PENTOSAN-POLYSULFATE REVIPARINE SR-90107 TEDELPARIN TINZAPARIN SODIUM LULIBERIN-AGONISTS AN-207 AY-25205 BUSERELIN DEAMIDOLULIBERIN DESLORELIN FERTIRELIN GOSERELIN HISTRELIN LEUPRORELIN LULIBERIN LULIBERIN-3-10 LULIBERIN-4-10 LULIBERIN-D-ALA-6 LULIBERIN-D-LYS-6 LULIBERIN-D-PHE-6 LULIBERIN-D-SER-6 LULIBERIN-FOWL LULIBERIN-I-FOWL LULIBERIN-II-FOWL LUTRELIN MINILULIBERIN NAFARELIN RS-49947 SUPERGESTRAN T-98 TRIPTORELIN LULIBERIN-ANTAGONISTS A-75998 ANTARELIX ANTIDE CDB-2085A CETRORELIX DETIRELIX

Derwent Drug File 1185 Thesaurus DETIRELIXACETATE GANIRELIX NAL-ARG-LULIBERIN NAL-GLU-LULIBERIN ORF-18260 ORF-21243 ORG-30093 ORG-30276 SB-29 SB-30 SB-88 T-121-B TEVERELIX TX-44 TX-51 TX-53 WY-18185 LUNG BRONCHIOLE BRONCHUS FLOW2002-CELL L132-CELL L1321-CELL LEWIS-LUNG-CARCINOMA PLEURA LYMPH-DISEASE BRENNEMANN-SYNDROME BURSAL-DISEASE canale-smith-syndrome chron.hereditary-= lymphedema CHYLOPERICARDITIS CHYLOTHORAX CHYLURIA ELEPHANTIASIS filatov-disease glandular-fever infectious-bursal-disease infectious-mononucleosis LYMPHADENITIS LYMPHADENOPATHY LYMPHANGIECTASIA LYMPHANGIOPHLEBITIS LYMPHANGITIS LYMPHEDEMA LYMPHOCELE LYMPHOGRANULOMATOSIS nonne-milroy-meige-= syndrome pfeiffer-glandular-fever PIRINGER-KUCHINKA-= SYNDROME pseudomalignant-= lymphadenopathy sinus-histiocytosis STRANGLES LYMPHOCYTE B-CELL CD4+-CELL CD8+-CELL HELPER-CELL IM9-CELL LAK-CELL LYMPHOBLAST LYMPHOCYTOSIS LYMPHOPOIESIS NAT.KILLER-CELL PLASMA-CELL PRE-B-CELL RPMI8422-CELL SPLEEN-CELL SUPPRESSOR-CELL TH1-CELL TH2-CELL THYMOCYTE LYMPHOMA ABPL2-CELL B35M-CELL BW5147-CELL DAUDI-CELL DT5-CELL EB-CELL EB-LYMPHOMA EB2-CELL ESB-CELL ESB-LYMPHOMA HODGKIN-DISEASE HRIK-CELL HUT11-CELL L12R4-CELL NEMETH-KELLNER-CELL NEMETH-KELLNER-= LYMPHOMA RAJI-CELL RPMI1346-CELL S49-CELL TLX5 TLX5-CELL LYMPHOPROLIFERATIVEDISEASE BAEFVERSTEDT-SYNDROME burkitt-lymphoma CHLOROMA eosinophilic-granuloma ERYTHROLEUKEMIA follicular-lymphoma hairy-cell-leukemia HAND-SCHULLER-= CHRISTIAN-DISEASE HODGKIN-DISEASE IMMUNOCYTOMA KIMURA-DISEASE LETTERER-SIWE-DISEASE LEUKEMIA leukemia, lymphocytic leukemic-reticuloendotheliosis LYMPHOBLASTOMA lymphocytic-leukemia LYMPHOHISTIOCYTOSIS LYMPHOMA LYMPHOMATOSIS LYMPHOSARCOMA MULT.MYELOMA MYCOSIS-FUNGOIDES MYELOPROLIFERATIVE-= SYNDROME MYELOSIS PLASMACYTOMA RETICULOENDOTHELIOSIS RETICULOSARCOMA RETICULOSIS LYMPHOSARCOMA P1798 MACROPHAGE HISTIOCYTE KUPFFER-CELL MICROGLIA OSTEOCLAST RAW264-CELL MALABSORPTION PROTEIN-LOSING-= ENTEROPATHY SHORT-BOWEL-SYNDROME SPRUE STEATORRHEA WHIPPLE-DISEASE MALARIA BLACK-WATER-FEVER MALNUTRITION HEPATOSIS-DIETETICA KWASHIORKOR MARASMUS MAMMA NIPPLE TEAT MAMMA-DISEASE adenocarcinoma, mamma AGALACTIA COMEDOCARCINOMA CYSTOSARCOMA FIBROADENOSIS GYNECOMASTIA MAMILLITIS mamma-adenocarcinoma mastalgia MASTITIS MASTODYNIA MAO-INHIBITORS AB-15 ACETYLPHENELZINE-N2 AGN-1135 ALMOXATONE AMIFLAMINE BAZINAPRINE BEFLOXATONE BRL-14831 BRL-16644 BROFAROMINE BW-1003-U-88 BW-1024-U-88 BW-1370U87 BW-1552-U-88 BW-183U88 BW-330-U-88 BW-380U88 BW-616U76 BW-A616U CGP-22364A CIMEMOXIN CIMOXATONE CINCHONAMINONE CINCHONICINOL CLORGILINE CVT-P-040 E-2011 ESUPRONE ETRYPTAMINE FA-37 FA-42 FA-43 FA-45 FA-73 FENOXYPROPAZINE FLA-289 FLA-299 FLA-314 FLA-334 FLA-336 FLA-365 FLA-384 FLA-405 FLA-417 FLA-450 FLA-463 FLA-558 FLA-668 FLA-717 FLA-727 FLA-788 FLUOROTRANYLCYPROMINE HARMALINE

1186 APPENDIX D HYDROXYTRANYLCY= PROMINE-PARA IODOCLORGYLINE IPROCLOZIDE IPRONIAZID ISOCARBOXAZID J-512 J-516 LAZABEMIDE LAZABEMIDE LEMUNINOL-A LEMUNINOL-B LEMUNINOL-C LILLY-51641 LK-63 LU-53439 LUTEUSIN-A LY-51641 LY-93716 M-9260 MD-220661 MD-240098 MD-240233 MD-240928 MD-240931 MD-760548 MD-770222 MDL-72145 MDL-72274 MDL-72392 MDL-72394 MDL-72638 MDL-72974 MEBANAZINE METHYLAPLYSINOPSIN METHYLBENZYLAMINE-= ALPHA METHYLSALSOLINOL-N MOCLOBEMIDE N-0425 NBF-003 NBF-008 NBF-021 NIALAMIDE NORSALSOLINOL NORSOLORINATE OCTAMOXIN PARGYLINE PHENELZINE PHENIPRAZINE PIM-35 R-40519 RAN-113 RASAGILINE RO-16-3177 RO-16-6491 RO-18-1675 RO-19-7731 RO-41-1049 RO-43-0463 ROLLINIASTATIN-1 RS-1653 RS-2232 RS-8359 SAFRAZINE SELEGILINE SENNOSIDE-F SERCLOREMINE SU-11739 TRANYLCYPROMINE TUK-9261 TV-3326 TZ-650 U-1424 UP-614-04 VERATRYLHYDRAZINE MAP-KINASE-INHIBITORS BIRB-796 PD-184352 PD-98059 SB-239063 MARROW MEGAKARYOBLAST MEGAKARYOCYTE MYELOPOIESIS PROMYELOCYTE MARROW-DISEASE AGRANULOCYTOSIS AMEGAKARYOCYTOSIS aplastic-anemia congenital-aplastic-anemia congenital-hypoplastic-= anemia diamond-blackfan-anemia EOSINOPENIA ERYTHROBLASTOSIS fanconi-disease HEMOBLASTOSIS LEUKOPENIA LYMPHOPENIA MACROCYTOSIS MARROW-DEPRESSION MOSSE-SYNDROME MYELOFIBROSIS NEUTROPENIA PANCYTOPENIA PANLEUKOPENIA PANMYELOPATHY PLASMACYTOSIS POLYCYTHEMIA POLYCYTHEMIA-VERA PRELEUKEMIA PSEUDOLEUKEMIA pure-red-cell-aplasia red-cell-aplasia,pure STRANSKY-REGALA-= SYNDROME MASTOCYTOMA P815 P815-CELL P815Y P815Y-CELL MATRIX-METALLOPROTEINASEINHIBITOR COLLAGENASE-INHIBITOR GELATINASE-A-INHIBITOR GELATINASE-B-INHIBITOR RO-28-2653 STROMELYSIN-1-INHIBITOR STROMELYSIN-2-INHIBITOR STROMELYSIN-INHIBITOR MATRIX-METALLOPROTEINASEINHIBITORS A-151011 ACETYLCYSTEINE ADALIMUMAB AE-941 ALLICIN BAY-12-9566 BB-3103 BMS-275291 CGS-27023-A CIPEMASTAT CMT-7 COLLAGENASE-INHIBITORS CP-471-474 CT-1746 DOXYCYCLINE EPIGALLOCATECHIN-GALLATE FUTOENONE GELATINASE-A-INHIBITORS GELATINASE-B-INHIBITORS GM-6001 GW-4459 HYDROXYACECLOFENAC-4 L-805645 MARIMASTAT METHYLSELENOL MINOCYCLINE MMI-166 PD-166793 PGE-4410186 PNU-99533 PRINOMASTAT RHEIN RIFAMPICIN RIFAMYCIN RIFAMYCIN-B RO-32-7315 SC-44463 STROMELYSIN-1-INHIBITORS STROMELYSIN-2-INHIBITORS STROMELYSIN-INHIBITORS TENIDAP THEAFLAVIN THEAFLAVIN-DIGALLATE TIAPROFENATE TP-151 TRANSFORMING-GROWTH-= FACTOR-BETA-1 VANADATE YLL-224 MDR-MODULATOR MRP-1-INHIBITOR MDR-MODULATORS AGOSTEROL-A CERAMIDE-C6 DENDROAMIDE-A OC-144093 MELANOLIBERIN-AGONISTS MELANOLIBERIN MELANOMA B16-CELL B16-MELANOMA B16A-CELL B4-CELL CLOUDMAN-CELL CLOUDMAN-MELANOMA CLOUDMAN-S91-CELL G-CELL HAB-CELL HARDING-PASSEY-CELL HARDING-PASSEY-= MELANOMA M21-CELL MM253-CELL RPMI1846-CELL S91-CELL SK-MEL28-CELL SK-MEL37E-CELL TANG-CELL MELANOSTATIN-AGONISTS MELANOSTATIN MELANOSTATIN-I TYROSYL-MELANOSTATIN MELATONIN-AGONISTS LY-156735 TAK-375 MEMBRANE CELL-WALL DESMOSOME LIPOSOME

Derwent Drug File 1187 Thesaurus MENINGITIS lymphocytic-choriomeningitis MENINGORADICULITIS MENSTRUATION AMENORRHEA BREAKTHROUGH-BLEEDING DYSMENORRHEA HYPERMENORRHEA HYPOMENORRHEA MENARCHE MENOMETRORRHAGIA MENORRHAGIA MENSTRUAL-IRREGULARITY METRORRHAGIA OLIGOMENORRHEA POLYMENORRHEA PREMENSTRUAL-SYNDROME premenstrual-tension MENTAL-DISORDER acute-hallucinatory-mania ACUTE-STRESS-DISORDER add adhd ADJUSTMENT-DISORDER ADRENOLEUKODYSTROPHY AGORAPHOBIA ALZHEIMER-DISEASE ALZHEIMER-DISEASE ANOREXIA-NERVOSA ANXIETY ANXIETY-DISORDER ATTENTION-DEFICIT-= DISORDER ATTENTION-DEFICIT-= HYPERACTIVITY-DISORDER autism AUTISTIC-DISORDER AUTOMATISM bayle-disease BINSWANGER-DEMENTIA BIPOLAR-DISORDER BIPOLAR-I-DISORDER BIPOLAR-II-DISORDER BODY-DYSMORPHIC-= DISORDER BRADYKINESIA BRADYPHRENIA BRIEF-PSYCHOTIC-DISORDER BULIMIA-NERVOSA CAPGRAS-SYNDROME cardiac-neurosis catatonic-schizophrenia CLAUSTROPHOBIA CONDUCT-DISORDER CONFUSION CYCLOTHYMIC-DISORDER da-costa-syndrome DELIRIUM DELIRIUM-TREMENS DELUSIONAL-DISORDER DEMENTIA DEPERSONALIZATION DEPRESSION DYSLEXIA dysmorphophobia DYSTHYMIC-DISORDER EATING-DISORDER EROTOMANIA FACTITIOUS-DISORDER ganser-syndrome GENERALIZED-ANXIETY-= DISORDER gilles-de-la-tourette-= syndrome HALLUCINATION hyperactivity-syndrome HYPERBARIC-NERVOUS-= SYNDROME HYPERERGASIA HYPERKINESIA hyperkinesia-syndrome HYPOCHONDRIA HYPOMANIA HYSTERIA KLEINE-LEVIN-SYNDROME KLUVER-BUCY-SYNDROME KORSAKOFF-SYNDROME LOGORRHEA MAJOR-DEPRESSIVE-= DISORDER MANIA manic-depression minimal-brain-dysfunction MOOD-DISORDER MUENCHAUSEN-SYNDROME MUENCHAUSEN-= SYNDROME-BY-PROXY MULTI-INFARCT-DEMENTIA NARCISSISM NEURASTHENIA NEURODYSTONIA NEUROSIS OBSESSIVE-COMPULSIVE-= DISORDER ORGANIC-BRAIN-SYNDROME PAGOPHAGIA PANIC-DISORDER paralytic-dementia PARANOIA paranoid-schizophrenia PARAPHRENIA PEDOPHILIA PERSONALITY-DISORDER PHOBIA PICA polle-syndrome POSTTRAUMATIC-STRESS-= DISORDER PREMENSTRUAL-SYNDROME premenstrual-tension presbyophrenia PSEUDODEMENTIA PSEUDOSEIZURE PSYCHOTIC-DISORDER roemheld-syndrome SADISM SCHIZOAFFECTIVE-DISORDER SCHIZOPHRENIA SCHIZOPHRENIFORM-= DISORDER SEASONAL-AFFECTIVE-= DISORDER SEPARATION-ANXIETY-= DISORDER SOCIAL-PHOBIA TOURETTE-DISORDER TRANSSEXUALISM TRANSVESTISM TRICHOTILLOMANIA wernicke-disease WERNICKE-= ENCEPHALOPATHY wernicke-syndrome METHYLASPARTATE-NANTAGONISTS ACEA-0762 B-3-277 GAVESTINEL GAVESTINEL LY-302679 NPS-846 SDZ-EAB-515 MIGRAINE cluster-headache MILK COLOSTRUM MILK-FOOD BUTTER YOGHURT MINERALOCORTICOIDS ALDOSTERONE ALDOSTERONE-ACETATE CORTEXONE CORTEXONE-ACETATE CORTEXONE-GLUCOSIDE CORTEXONE-= PHENYLPROPIONATE CORTEXONE-PIVALATE DEOXYALDOSTERONE-18 FLUDROCORTISONE FLUDROCORTISONE-ACETATE HYDROXYALDOSTERONE-19 HYDROXYCORTEXONE-18 NORCORTEXONE-19 OXOHYDROCORTISONE-18 MITE lynxacarus-v MOLLUSC APLYSIA BIOMPHALARIA BUSYCON CRASSOSTREA HELIX LOLIGO LYMNAEA ONCOMELANIA OSTREA MOLLUSCICIDES MOLUCID NICLOSAMIDE OLAMINE TRIFENMORPH MONKEY CAPUCHIN MACAQUE SQUIRREL-MONKEY MONOCLONAL APOLIZUMAB BASILIXIMAB BEVACIZUMAB BT-563 CENTOXIN CETUXIMAB DACLIXIMAB EDRECOLOMAB EMD-72000 EPRATUZUMAB GEMTUZUMAB OZOGAMICIN IBRITUMOMAB-TIUXETAN ICI-D-0490 IDEC-131 KELIXIMAB MDX-H-210 MUROMONAB-CD3 NATALIZUMAB OMALIZUMAB PALIVIZUMAB SIPLIZUMAB TOSITUMOMAB MOOD-DISORDER BIPOLAR-DISORDER BIPOLAR-I-DISORDER BIPOLAR-II-DISORDER CYCLOTHYMIC-DISORDER DEPRESSION DYSTHYMIC-DISORDER

1188 APPENDIX D MAJOR-DEPRESSIVE-= DISORDER manic-depression PREMENSTRUAL-SYNDROME premenstrual-tension SEASONAL-AFFECTIVE-= DISORDER MORPHINE-ANTAGONISTS AMIPHENAZOLE BINALTORPHIMINE CASOXIN-6 CHLORNALTREXAMINE CLOCINNAMOX CM-32191 CONORFONE CTAP CTOP CYCLAZOCINE CYCLORPHAN CYPRENORPHINE CYPRODIME DEXTRALLORPHAN DIACETYLNALORPHINE DIALLYLNORMORPHINIUM = BROMIDE DIPRENORPHINE DYNORPHIN-2-17 EN-2260 EN-2265 FUNALTREXAMINE-ALPHA FUNALTREXAMINE-BETA GEMAZOCINE GPA-1843 GPA-1847 GPA-2163 ICI-139462 ICI-154129 ICI-174864 J-113397 KETAZOCINE L-246736 LEVALLORPHAN LEVALLORPHAN-METHIODIDE LY-106737 LY-117413 LY-136595 LY-88329 LY-99335 M-154129 METHYLNALORPHINE-N METHYLNALOXONE-N METHYLNALTREXONE-N METHYLNALTRINDOLE-N MORPHINONE MR-1452 MR-1453 MR-2097-CL MR-2266 MR-2266-BS MR-2267 NALBUPHINE NALBUPHINE-= ACETYLSALICYLATE-3 NALMEFENE NALMEXONE NALORPHINE NALORPHINE-6-= GLUCURONIDE NALORPHINE-6-SULFATE NALORPHINE-EPOXIDE-7,8 NALOXAZONE NALOXOL-ALPHA NALOXONE NALOXONE-BENZOYL= HYDRAZONE NALOXONE-ESTRONE-AZINE NALOXONE-METHOBROMIDE NALTREXONAZINE NALTREXONE NALTREXONE-= METHOBROMIDE NALTRIBEN NALTRINDOLE NALTRINDOLE-= ISOTHIOCYANATE-5 NIH-10236 NORBINALTORPHIMINE OXILORPHAN QUADAZOCINE RX-8008M S-20682 SDZ-210-096 SR-58002-C TENA UM-1037 UM-1046 WIN-42610 WIN-44441-2 XORPHANOL MOSQUITO AEDES ANOPHELES CULEX MUCOLYTICS ACEBROPHYLLINE ACETYLCYSTEINE ADAMEXINE AMBROXOL AMBROXOL = THEOPHYLLINATE AMIFOSTINE AZULAN BENCISTEINE BR-227 BROMHEXINE BRONCOPLUS BROVANEXINE CARBOCISTEINE CARBOCISTEINE-LYSINE-SALT CO-1408 CYSTEINE-ETHYL-ESTER DEMBREXINE DEOXYRIBONUCLEASE-I DOMIODOL EPRAZINONE ERDOSTEINE GELSOLIN GUAIMESAL INS-365 IQB-782 IRFI-005 IRFI-016 LETOSTEIN MESNA MYRTOL NACYSTELYN NELTENEXINE NESOSTEINE OMONASTEINE OXABREXINE PRENISTEINE REGENASOL SEAPROSE SERRATIOPEPTIDASE SFERICASE SS-320A STEPRONIN STEPRONIN-LYSINE-SALT TASULDINE TIMONACIC-METHYL-ESTER TIOPRONIN ZY-15850A MUCOPOLYSACCHARIDOSIS BARTENWERFER-SYNDROME HUNTER-SYNDROME HURLER-SYNDROME maroteaux-lamy-syndrome MORQUIO-DISEASE MUCINOSIS polydystrophic-dwarfism SANFILIPPO-SYNDROME SCHEIE-SYNDROME MULTI-INFARCT-DEMENTIA BINSWANGER-DEMENTIA MUSCLE BICEPS DELTOID DIAPHRAGM G8-CELL GASTROCNEMIUS MYOFIBRIL MYOFIBROBLAST MYOFILAMENT SARCOLEMMA MUSHROOM AGARICUS AMANITA amanita-muscaria ARMILLARIA AURICULARIA FLAMMULINA fly-agaric GRIFOLA INOCYBE OUDESMANIELLA PHOMA POLYPORUS PSILOCYBE SCHIZOPHYLLUM STROPHARIA TRICHOLOMA MYALGIA EOSINOPHILIA-MYALGIA-= SYNDROME MYASTHENIA EATON-LAMBERT-SYNDROME MYDRIATICS APOATROPINE ATROPINE ATROPINE-ETHIODIDE ATROPINE-METHONITRATE CYCLODRINE CYCLOPENTOLATE DIAMIPHENE DIPHEMIN DIPIVEFRINE EUCATROPINE HOMATROPINE HYDROXYAMPHETAMINE LACHESINE PHENYLEPHRINE PHENYLEPHRINE-= OXAZOLIDINE PHOLEDRINE PLATYPHYLLINE SCOPOLAMINE TROPICAMIDE TYRAMINE MYELOMA MPC11-CELL NS1-CELL MYOPATHY ARTHROGRYPOSIS congenital-arthromyo= dysplasia

Derwent Drug File 1189 Thesaurus congenital-musc.dystrophy CURSCHMANN-BATTEN-= STEINERT-SYNDROME DERMATOMYOSITIS DETERMANN-SYNDROME DYSTONIA EOSINOPHILIA-MYALGIA-= SYNDROME familial-periodic-paralysis FIBROMYALGIA FIBROMYOSITIS FIBROSITIS FOESTER-SYNDROME guerin-stern-syndrome MCARDLE-DISEASE muechmeyer-syndrome munchmeyer-syndrome MUSC.ATROPHY MUSC.DYSTROPHY MUSC.SPASM MYALGIA MYASTHENIA MYATONIA MYOGELOSIS MYOSITIS MYOTONIA MYOTONIC-DYSTROPHY NIELSEN-SYNDROME OSTEOMYELOSCLEROSIS POLYMYALGIA-RHEUMATICA POLYMYOSITIS progressive-ossifying-myositis PSEUDOMYOTONIA PYOMYOSITIS RHABDOMYOLYSIS STRINGHALT SWEENEY SYSTREMMA TENDINITIS thomsen-disease TORTICOLLIS ULLRICH-SYNDROME westphal-syndrome ZENKER-DEGENERATION PARAINFLUENZA-VIRUS PARAMYXO-VIRUS PEROMYSCUS-VIRUS PIGEON-PARAMYXO-VIRUS RINDERPEST-VIRUS RS-VIRUS SENDAI-VIRUS SV5-VIRUS NA-CA-ATPASE-INHIBITORS KB-R-7943 NA-H-EXCHANGE-INHIBITORS CARIPORIDE FR-168888 T-162559 NA-K-ATPASE-INHIBITORS ACETYLDIGOXIN ACETYLDIGOXIN-12 ACETYLDIGOXIN-ALPHA ACETYLDIGOXIN-BETA ACETYLGITOXIN AMTIZOLE AU-1421 DEGLUCOHYRCANOSIDE DIGITOXIGENIN DIGITOXIGENIN-= BISDIGITOXOSIDE DIGITOXIGENIN-= DIGITOXOSIDE DIGITOXIN DIGOXIN DIHYDROOUABAIN HYRCANOSIDE LANATOSIDE-A LANATOSIDE-B LANATOSIDE-C LANATOSIDE-D LANATOSIDE-E LND-796 OUABAIN PST-2107 PST-2238 PST-2744 STROPHANTHIN-H ACETYLMORPHINE-3 ALFENTANIL ALLETORPHINE ALPHAPRODINE ANILERIDINE ASIMADOLINE AZIDOMORPHINE B-777-81 BENZYLMORPHINE BREMAZOCINE BRIFENTANIL BRL-52537 BUPRENORPHINE BUTANOYLMORPHINE-6 BUTORPHANOL BW-373-U-86 CAPPORPHIN CARFENTANIL CHLORBICYCLEN CODEINE CODEINE-EPOXIDE CONORFONE CP-0494 CP-0499 CYCLORPHAN CYPRENORPHINE DESOMORPHINE DEXTRALLORPHAN DEXTROMETHADONE DEXTROMETHORPHAN DEXTRORPHAN DEXTRORPHAN-= GLUCURONIDE DIACETYLMORPHINE DIACETYLNALORPHINE DIALLYLNORMORPHINIUM = BROMIDE DIBUTANOYLMORPHINE DIHYDROCODEINE DIHYDROCODEINE-= GLUCURONIDE-6 DIHYDROETORPHINE DIHYDROMORPHINE DIMEMORFAN DIPRENORPHINE DIVINYL-ETHER DROTEBANOL EMBUTRAMIDE EMD-60400 ESEROLINE ESEROLINE-SALICYLATE ETHYLKETAZOCINE ETHYLMORPHINE ETORPHINE FENARIDINE FENTANYL FUNALTREXAMINE-ALPHA FUNALTREXAMINE-BETA GEMAZOCINE GI-90291 GR-103545 GR-38414 GR-45809 GR-86014 GR-89696 GR-91272 HOMPRENORPHINE HYDROCODONE HYDROMORPHINOL HYDROMORPHONE ICI-197067 ICI-199441 ISOSULFORPHANOL = PERCHLORATE KETAZOCINE KETOBEMIDONE KT-90 LEVACETYLMETHADOL LEVALLORPHAN LEVOMETHADONE LEVOMETHORPHAN LEVOPHENACYLMORPHAN LEVORPHANOL LOFENTANIL LORCINADOL LY-136595 LY-136596 METHADONE METHYLDESORPHINE METHYLDIHYDROMORPHINE METHYLFENTANYL-ALPHA METHYLMEPTAZINOL-N METHYLNALTRINDOLE-N METOMIDATE METOPON MIRFENTANIL MORPHINE MORPHINE-EPOXIDE MORPHINE-HEXANOATE-3 MORPHINE-= MONONICOTINATE-3 MORPHINE-= MONONICOTINATE-6 MORPHINE-PROPIONATE-3 MORPHINE-SULFATE-3 MORPHINE-SULFATE-6 MORPHINONE MR-1268 MR-2033 MR-2096-CL MR-2097-CL MR-2261 MR-2264-CL MYROPHINE NALBUPHINE

MYOSIN-LIGHT-CHAIN-KINASEINHIBITORS NAIL H-7 LEUKONYCHIA ML-7 MELANONYCHIA ML-9 ONYCHOLYSIS MS-444 ONYCHOMADESIS ONYCHOMYCOSIS MYXOVIRUS PACHYONYCHIA DISTEMPER-VIRUS PARONYCHIA INFLUENZA-A-VIRUS NARCOTICS INFLUENZA-B-VIRUS INFLUENZA-VIRUS ACETORPHINE MEASLES-VIRUS ACETYLMETHADOL MUMPS-VIRUS ACETYLMORPHINE

1190 APPENDIX D NALBUPHINE-= ACETYLSALICYLATE-3 NALMEFENE NALMEXONE NALORPHINE NALORPHINE-6-= GLUCURONIDE NALORPHINE-6-SULFATE NALORPHINE-EPOXIDE-7,8 NALOXONAZINE NALOXONE NALOXONE-= BENZOYLHYDRAZONE NALOXONE-METHOBROMIDE NALTREXONE NALTREXONE-= METHOBROMIDE NALTRIBEN NARCEINE NARCOBARBITAL NICODICODINE NICOMORPHINE NORBUTORPHANOL NORCODEINE NORLEVORPHANOL NORMORPHINE NOSCAPINE OPIUM ORIPAVINE OXILORPHAN OXYCODONE OXYMORPHAZONE OXYMORPHONAZINE OXYMORPHONE PAPAVERETUM PD-123475 PD-123497 PENTAZOCINE PERICALLINE PETHIDINE PHENAZOCINE PHENOMORPHAN PHOLCODINE PICENADOL PIMINODINE RACEMETHORPHAN RACEMORPHAN REMIFENTANIL RO-03-4661 RP-60180 RX-77989 SINOMENINE SPIRADOLINE SUFENTANIL THEBACON THEBAINE TONAZOCINE U-50488 U-50488E U-50488H U-53455E U-62066E U-63639 U-63640 U-69593 UM-1250 XORPHANOL NEMATODE AELUROSTRONGYLUS AMIDOSTOMUM ANCYLOSTOMA ANGIOSTRONGYLUS ANISAKIS APROCTELLA ASCARIDIA ASCARIS ASCAROPS ASCOCOTYLE ASPICULURIS ATRACTIS AUGUSTICAECUM BAYLISASCARIS BRUGIA BUNOSTOMUM CAENORHABDITIS CAMALLANUS CAMELOSTRONGYLUS CAPILLARIA CARDIOFILARIA CENTRORHYNCHUS CHABERTIA COOPERIA CRENOSOMA CYATHOSTOMUM CYLICOCYCLUS CYLICODONTOPHORUS CYLICOSTEPHANUS DICTYOCAULUS DIOCTOPHYMA DIPETALONEMA DIROFILARIA DISPHARYNX DRACUNCULUS DRASCHIA ELAEOPHORA ELAPHOSTRONGYLUS ENTEROBIUS FILARIA FILAROIDES GAIGERIA GANGULETERAKIS GLOBOCEPHALUS GNATHOSTOMA GONGLYONEMA GYALOCEPHALUS HABRONEMA HAEMONCHUS HELIGMOSOMOIDES HETERAKIS HETERODERA HIRSCHMANIELLA HYOSTRONGYLUS IMPALAIA LAGOCHILASCARIS LITOMOSOIDES LOA MACRACANTHORHYNCHUS MANSONELLA MARSHALLAGIA MECISTOCIRRUS MEHDIELLA MELOIDOGYNE METASTRONGYLUS MONANEMA MUELLERIUS NECATOR NEMATODIRELLA NEMATODIRUS NEMATOSPIROIDES NEOASCARIS NEOPLECTANA NIPPOSTRONGYLUS OESOPHAGODONTUS OESOPHAGOSTOMUM OLLULANUS ONCHOCERCA OPHIDASCARIS OSTERTAGIA OXYSPIRURA OXYURIS PARABRONEMA PARAFILARIA PARASCARIS PARELAPHOSTRONGYLUS PELODERA PHILOMETRA PHYSALOPTERA PHYSOCEPHALUS PORROCAECUM POTERIOSTOMUM PROTOSTRONGYLUS PTERYGODERMATITES RHABDITIS SETARIA SKRJABINEMA SPIROCERCA SPLENDIDOFILARIA STEPHANOFILARIA STEPHANURUS STRONGYLOIDES STRONGYLUS SUBULURA SYNGAMUS SYPHACIA TACHYGONETRIA TELADORSAGIA TETRAGOMPHIUS THELAZIA TOXASCARIS TOXOCARA TRICHINELLA TRICHODORUS TRICHONEMA TRICHOSOMOIDES TRICHOSTRONGYLUS TRICHURIS TRIODONTOPHORUS UNCINARIA WUCHERERIA XIPHINEMA NEMATODIASIS ELEPHANTIASIS GAPES LOAIASIS ONCHOCERCIASIS OXYURIASIS TRICHINOSIS NEOPLASM ACANTHOMA ADENOACANTHOMA ADENOCARCINOMA ADENOFIBROMA ADENOMA ALDOSTERONOMA AMELOBLASTOMA ANAPLASIA ANGIOMYOLIPOMA ANGIOSARCOMA APUDOMA BARD-PIC-SYNDROME BLASTOMA CARCINOID CARCINOMA CARCINOSARCOMA CHOLANGIOCARCINOMA CHONDROBLASTOMA CHONDROMA CHONDROSARCOMA CHORDOMA CHORIOCARCINOMA COMEDOCARCINOMA CRANIOPHARYNGIOMA CYSTADENOCARCINOMA CYSTADENOMA diffuse-sym.lipoma EATON-LAMBERT-SYNDROME embryonal-nephroma EPENDYMOBLASTOMA EPITHELIOMA ESTHESIONEUROBLASTOMA

Derwent Drug File 1191 Thesaurus ewing-bone-sarcoma ewing-osteosarcoma FIBROADENOMA FIBROHISTIOCYTOMA FIBROMA FIBROMATOSIS FIBROMYXOSARCOMA FIBROSARCOMA GANGLIONEUROBLASTOMA GANGLIONEUROMA GERMINOMA GLUCAGONOMA HAMARTOBLASTOMA HAMARTOMA head-and-neck-sarcoma HEMANGIOMA HEMANGIOPERICYTOMA HEMANGIOSARCOMA HEPATOBLASTOMA HIDRADENOMA HIPPEL-LINDAU-SYNDROME HISTIOCYTOMA HISTOMA HYDATIDIFORM-MOLE HYPERNEPHROMA KASABACH-MERRITT-= SYNDROME LEIOMYOMA LEIOMYOSARCOMA LIPOMA LIPOSARCOMA LUTEOMA LYMPHANGIOLEIO= MYOMATOSIS LYMPHANGIOMA LYMPHANGIOMYOMATOSIS LYMPHANGIOSARCOMA LYMPHOEPITHELIOMA MACROADENOMA madelung-disease MASTOCYTOMA MEDULLOBLASTOMA MEDULLOEPITHELIOMA MEDULLOMYOBLASTOMA MEIGS-SYNDROME MENINGIOMA MESENCHYMOMA MESOTHELIOMA MICROADENOMA MULT.NEUROFIBROMA MYELOLIPOMA MYELOMA MYOMA MYXOFIBROSARCOMA MYXOMA MYXOSARCOMA NELSON-SYNDROME nephroblastoma NEPHROBLASTOMATOSIS NEPHROMA NEUROBLASTOMA NEUROEPITHELIOMA NEUROFIBROMATOSIS NEUROFIBROSARCOMA NEUROMA ONCOCYTOMA OSTEOCLASTOMA OSTEOMA PANCOAST-SYNDROME PAPILLOMA PARAGANGLIOMA PHEOCHROMOCYTOMA PIETRANTONI-SYNDROME PINEALOMA PINEOBLASTOMA PROLACTINOMA RAYMOND-CESTAN-= SYNDROME RETINOBLASTOMA RHABDOMYOMA RHABDOMYOSARCOMA SARCOMA sarcoma, head and neck SCHWANNOMA SIPPLE-SYNDROME SOMATOSTATINOMA SPONGIOBLASTOMA stewart-treves-syndrome SYRINGOCYSTADENOMA TERATOCARCINOMA TERATOMA THYMOLIPOMA TRICHILEMMOMA TUBEROUS-SCLEROSIS VERNER-MORRISON-= SYNDROME VIPOMA WERMER-SYNDROME wilms-tumor ZOLLINGER-ELLISON-= SYNDROME NEPHROPATHY angara-disease ANURIA BARTTER-SYNDROME CRYSTALLURIA CYLINDRURIA CYSTOPYELITIS CYTURIA diabetic-glomerulosclerosis embryonal-nephroma FANCONI-SYNDROME GLOMERULITIS GLOMERULONEPHRITIS GLOMERULOSCLEROSIS GLYCOSURIA GOODPASTURE-SYNDROME HEMOLYTIC-UREMIC-= SYNDROME HEPATORENAL-SYNDROME HORSESHOE-KIDNEY HYDRONEPHROSIS hydropericardium-syndrome HYPERNEPHROMA INCLUSION-BODY-HEPATITIS kidney-calculi kimmelstiel-wilson-syndrome LIGHTWOOD-ALBRIGHT-= SYNDROME NEPHRITIS nephroblastoma NEPHROBLASTOMATOSIS NEPHROCALCINOSIS NEPHROLITHIASIS NEPHROMA NEPHROSCLEROSIS NEPHROSIS NEPHROSONEPHRITIS NEPHROTIC-SYNDROME NONNENBRUCH-SYNDROME NYCTURIA OLIGURIA osteodystrophia-fibrosa PERINEPHRITIS POLYCYSTIC-KIDNEY POLYURIA PYELONEPHRITIS PYONEPHROSIS RENAL-COLIC RENAL-FAILURE RENAL-INSUFFICIENCY renal-osteodystrophy renal-rachitis renal-rickets RENINOMA SPONGE-KIDNEY UREMIA wilms-tumor NERVE AXON DEAFFERENTATION DENDRITE ELECTROPLAX GANGLION HYPOGLOSSAL-NUCLEUS MOTOR-END-PLATE NEURITE NEUROGLIA NEURON NODE-OF-RANVIER PARAGANGLION SCHWANN-CELL SPINOCERVICAL-TRACT SPINOTHALAMIC-TRACT SYNAPSE VAGUS NEURALGIA HERPES-ZOSTER NEURAMINIDASE-INHIBITORS RWJ-270201 NEUROBLASTOMA C1300-CELL CHP126-CELL M1-CELL M5-CELL NG108-15-CELL NIE115-CELL NS20-CELL NEUROGLIA GLIACYTE NEUROLEPTANALGESIA NEUROLEPTANESTHESIA NEUROLEPTICS 106-689 1192-U-90 4684-RP A-23887 A-31472 A-37850 A-69024 ACEPERONE ACEPROMAZINE ACEPROMETAZINE ACETOPHENAZINE AD-5423 AET AGAROSPIROL AHR-1709 AHR-1900 AL-1612 AL-449 ALENTEMOL ALPIROPRIDE AMINOBENZONITRILE-PARA AMIPERONE AMISULPRIDE AMOXAPINE AMPEROZIDE ANISOPERIDONE ANISOPIROL AZ-21666 AZABUPERONE AZAPERONE BALAPERIDONE BATELAPINE BENPERIDOL BENZQUINAMIDE BIRIPERONE

1192 APPENDIX D BMY-14802 BMY-14802-1 BMY-20551 BMY-20661 BRL-34778 BROMOSPIPERONE-PARA BROMPERIDOL BROMPERIDOL-DECANOATE BUSPIRONE BUTACLAMOL BUTAPERAZINE BUTYLSYMPATON CARFENAZINE CARPERONE CENTPYRAQUIN CHLOROSERPIDINE CHLORPROETHAZINE CHLORPROMAZINE CHLORPROMAZINE-= METHIODIDE CHLORPROTHIXENE CI-1007 CI-905 CI-913 CI-936 CI-943 CICLOFENAZINE CINUPERONE CITATEPINE CLEBOPRIDE CLOFLUMIDE CLOFLUPEROL CLOMACRAN CLOPENTHIXOL CLOPENTHIXOL-DECANOATE CLOPIPAZAN CLOPITHEPIN CLOROPERONE CLOROTEPINE CLOTIAPINE CLOXATHIEPIN CLOXYPENDYL CLOZAPINE CORYTUBERINE CP-135807 CP-88059 CX-516 CYAMEMAZINE DEMETHYLNEMONAPRIDE-N DESERPIDINE DEXCLAMOL DICARBINE DICHLORPROMAZINE DIHYDROBENPERIDOL DIHYDROTETRABENAZINE DIHYDROWISANINE DIMELAZINE DIXYRAZINE DO-897 DOKLOXYTHEPIN DROPERIDOL DU-127090 DUP-734 E-0663 E3-54 ELTOPRAZINE ERIZEPINE ETASULINE EX-11-582A FENAPERONE FH-510 FLA-988 FLB-457 FLB-463 FLUANISONE FLUBEPRIDE FLUCIPRAZINE FLUMEZAPINE FLUOTHEPINE FLUPENTIXOL FLUPENTIXOL-DECANOATE FLUPERLAPINE FLUPHENAZINE FLUPHENAZINE-DECANOATE FLUPHENAZINE-ENANTHATE FLUPIMAZINE FLUPRAZINE FLUSPIPERONE FLUSPIRILENE FLUTIZENOL FR-33 FUROMAZINE G-365 GEVOTROLINE GMC-1-169 GP-45795 GP-50302 GR-103691 GRI-1665 GYKI-22441 HALOPERIDOL HALOPERIDOL-DECANOATE HOMOFENAZINE HP-236 HP-370 HPP HUF-2046 HYDROXYBENZONITRILE-= PARA ILOPERIDONE IMICLOPAZINE IODOPROXYFAN IPROZILAMINE IRFI-165 ISOBUTACLAMOL ISOCLOTHIAPINE ISOFLOXYTHEPIN JINKOH-EREMOL JL-13 L-701324 L-741742 LEK-8829 LENPERONE LEVOMEPROMAZINE LEVOMETIOMEPRAZINE LOXAPINE LU-13-117 LU-14-068 LU-17-151 LU-17-152 LUR-2366 LY-262691 LY-379268 M+B-18706 MAFOPRAZINE MANASSANTIN-A MAROXEPIN MDL-100151 MDL-100907 MDL-28133A MDL-72483 MEFECLORAZINE MELPERONE MEPIPRAZOLE MEPROTIXOL MESMAR MESORIDAZINE METHIOMEPRAZINE METHIOTHEPIN METHOPROMAZINE METIAPINE METOFENAZATE METOSERPATE METOXEPIN MEZILAMINE MGS-0008 MILENPERONE MILIPERTINE MINDOPERONE MJ-13980-1 MJ-7378 MOLINDONE MOPERONE MOSAPRAMINE MS-257 MS-377 NAFADOTRIDE NCQ-318 NEFLUMOZIDE NEMONAPRIDE NERISOPAM NGD-94-1 NNC-0112 NNC-22-0031 NNC-90-3094 NO-01-0756 NONAPERONE NORCHLORPROMAZINE NORTHIORIDAZINE NP-207 NPC-16377 NRA-0045 NRA-0160 NRA-0215 NRA-0562 OCAPERIDONE OLANZAPINE OLANZAPINE ONDANSETRON OPC-14597 OPC-4392 OPROMAZINE ORG-5222 OSU-6162 OXAFLUMAZINE OXIPEROMIDE OXYCLOTHEPINE OXYPERTINE OXYPROTHEPINE OXYPROTHEPINE-= DECANOATE OXYRIDAZINE P-9236 PD-118717 PD-119819 PD-143188 PD-152255 PD-158771 PD-172760 PECAZINE PENFLURIDOL PENTIAPINE PERATHIEPINE PERAZINE PERICIAZINE PERIMETAZINE PERPHENAZINE PERPHENAZINE-DECANOATE PERPHENAZINE-ENANTHATE PIFLUTIXOL PIMOZIDE PINOXEPIN PIPAMPERONE PIPERACETAZINE PIPOTIAZINE PIPOTIAZINE-PALMITATE PIQUINDONE PROCHLORPERAZINE PROFENAMINE PROMAZINE PROPIONYLPROMAZINE PROPYPERONE

Derwent Drug File 1193 Thesaurus PROSULPRIDE PROTHIPENDYL PROTHIXENE PSD-958 PYRICAPIRONE QF-0307-B QF-0313-B QF-2003-B QF-2004-B QM-7184 QUETIAPINE R-24763 R-2572 RED.HALOPERIDOL REMOXIPRIDE RESERPINE RGH-1756 RGH-6141 RILAPINE RIMCAZOLE RISPERIDONE RMI-11974 ROLIPRAM ROMERGOLINE ROXOPERONE RWJ-37796 S-16924 S-18327 SARIZOTAN SAVOXEPIN SB-228357 SB-271046 SB-277011 SCH-23390 SCH-39166 SCH-40853 SDZ-208-911 SDZ-208-912 SDZ-212-327 SEROQUEL SERTINDOLE SETOPERONE SKF-83742 SM-13496 SM-9018 SPICLOMAZINE SPIPERONE SPIRAMIDE SPIRILENE SPIROXATRINE ST-1460 SULFAMOTHEPIN SULFORIDAZINE SULMEPRIDE SULTOPRIDE TEFLUDAZINE TEFLUTIXOL TENILAPINE TEPIRINDOLE TETRABENAZINE THIOPROPAZATE THIOPROPERAZINE THIORIDAZINE THIORIDAZINE-= DISULFOXIDE-2,5 THIORIDAZINE-OXIDE-5 TIAPRIDE TIENOCARBINE TIMELOTEM TIMIPERONE TIOPERIDONE TIOSPIRONE TIOTIXENE TJ-24 TPN-12 TPO-33 TRIFLUOMEPRAZINE TRIFLUOPERAZINE TRIFLUPERIDOL TRIFLUPROMAZINE TRIFLUTHEPIN TRIMOPAM TROPAPRIDE U-101387 U-101958 U-25927 U-99363-E UK-177 UMESPIRONE XANTHIOL Y-20024 YG-19256 YM-43611 ZETIDOLINE ZOLOPERONE ZOTEPINE ZUCLOPENTHIXOL ZUCLOPENTHIXOL-ACETATE ZUCLOPENTHIXOL-= DECANOATE NEUROMEDIN-K-ANTAGONISTS SB-222200 NEUROMUSC. BIVENTER-CERVICIS END-PLATE NEUROMUSC.BLOCKERANTAGONISTS AMINOPYRIDINE-3 AMINOPYRIDINE-4 DIAMINOPYRIDINE-2,4 DIAMINOPYRIDINE-3,4 DIMETHYLAMINOPYRIDINE-4 LF-14 NEUROMUSC.BLOCKERS 202 34-W-89 35-W-89 36-W-89 49-W-89 50-W-89 51-W-89 AF-64A AGATOXIN-ALPHA-489 ALCURONIUM CHLORIDE ANQ-9040 ARGIOTOXIN-636 ATRACURIUM BESILATE BENZOQUINONIUM BOTULINUM-C-TOXIN BW-252-C64 BW-403-C65 BW-A444U CANDOCURONIUM-IODIDE CHANDONIUM CHONDROCURINE CISATRACURIUM BESILATE CORYNEINE CURARE CURARINE CURARINE-C-I CURARINE-C-III CURINE DACURONIUM BROMIDE DECAMETHONIUM BROMIDE DIHYDRO-BETA-= ERYTHROIDINE DIMETHYLTUBO= CURARINIUM CHLORIDE DIPLACIN DIPYRONIUM DOXACURIUM CHLORIDE DUADOR ECHITAMINE ERYSODINE ERYTHROIDINE ERYTHROIDINE-ALPHA ERYTHROIDINE-BETA FAZADINIUM BROMIDE G-1-64 GALLAMINE-TRIETHIODIDE GEPHYROTOXIN-223-AB GW-280430-A HC-15 HEMICHOLINIUM-A-4 HEMICHOLINIUM-A-5 HEXCARBACHOLINE BROMIDE HM-197 HS-342 HS-692 LAUDEXIUM-METILSULFATE LEPTODACTYLINE MEPROADIFEN METHYLOXAMETHONIUM = IODIDE MIVACURIUM CHLORIDE MUREXINE NAM-204 NAM-221 NAM-224 ORG-20059 ORG-20297 ORG-6368 ORG-7268 ORG-7402 ORG-7617 ORG-8715 ORG-8730 ORG-8764 ORG-9273 ORG-9453 ORG-9489 ORG-9616 ORG-9943 ORG-9955 ORG-9991 ORG-NC-58 OXAMETHONIUM IODIDE OXYDIPENTONIUM CHLORIDE PAEONIFLORIGENONE PANCURONIUM BROMIDE PIPECURONIUM PIPROCURARIUM IODIDE PRODECONIUM BROMIDE PUMILIOTOXIN-C PYROCURINE QUALIDIL RAPACURONIUM BROMIDE ROCURONIUM BROMIDE STERCURONIUM IODIDE SUCCINYLMONOCHOLINE SUXAMETHONIUM CHLORIDE SUXAMETHONIUM IODIDE SUXETHONIUM CHLORIDE SZ-1676 TAAC-3 TACRINE TERCURONIUM BESILATE TL-351 TL-363 TL-365 TL-371 TL-381 TOOSENDANIN TRUXICURIUM IODIDE TRUXILLONIUM TRUXIPICURIUM IODIDE TUBEROSTEMONINE

1194 APPENDIX D TUBOCURARINE CHLORIDE VECURONIUM BROMIDE VESAMICOL NEUROMUSC.DISEASE EATON-LAMBERT-SYNDROME MYASTHENIA-GRAVIS SPASMOPHILIA TETANY NEUTRAL-ENDOPEPTIDASEINHIBITORS BMS-182657 CANDOXATRIL CANDOXATRILAT CGS-24592 CGS-26303 CGS-28106 CGS-34043 CGS-35066 ECADOTRIL ER-32935 GEMOPATRILAT MDL-100240 MIXANPRIL OMAPATRILAT PHOSPHORAMIDON RB-105 SCH-32615 SCH-39370 SCH-42354 SCH-42495 SCH-54470 SINORPHAN SQ-28603 THIORPHAN Z-13752-A NF-KAPPA-B-INHIBITORS BAY-11-7085 SN-50 NITRIC-OXIDE-ANTAGONISTS BYAKANGELICOL CORONARIN-E MYRICANOL MYRICANONE PACOVATININ-A TP-151 NITRIC-OXIDE-SYNTHASEINHIBITORS 1400-W ADEFOVIR-DIPIVOXIL AMINOETHYLISOTHIOUREA ANDALUSOL AURANOFIN AVICIN-G BENZOQUINONE BN-80933 BROUSSOCHALCONE-A CMT-8 COSTUNOLIDE FORMAMIDINE GABEXATE GLAUCOLIDE-A GW-274150 HIRSUTANONOL IPRIFLAVONE LY-83583 MAGNOLIALIDE MERCAPTOETHYLGUANIDINE METHYLARGININE-N-G MYRICANOL MYRICANONE NCX-1015 NICOTINAMIDE NITROARGININE-N-G-= METHYLESTER NITROINDAZOLE-7 ONO-1714 OREGONIN PACOVATININ-A PSILOSTACHYIN-A PYRUVATE-ETHYL-ESTER SPIRAFOLIDE TISOCARBAMIDE TRICHODION XANTHOMEGNIN NOOTROPICS ABT-089 ABT-418 ACETYLASPARTATE-N ACETYLGLYCINAMIDE-N ACETYLLEVOCARNITINE ADAFENOXATE AF-150-S AG-4 AIT-082 AKF-94 ALTINICLINE AMBOCARB AMIRIDINE ANIRACETAM AP-521 ARGIPRESSIN-4-9 AWD-52-39 BACOSIDE-A BESIPIRDINE BIIE-0246 BMY-21502 BN-80933 BR-16A BU-224 BY-1947 BY-1949 CEBARACETAM CEP-1347 CGP-36742 CGP-71982 CGS-5649B CHF-2819 CI-933 CL-275838 CR-2249 CROCIN CX-516 DEHYDROEVODIAMINE DENBUFYLLINE DEXEFAROXAN DIMIRACETAM DITHIOPIRACETAM DM-232 DM-235 DMP-543 DU-14 DUPRACETAM DX-9386 E-2030 E-4804 EGIS-8332 EK-49 ETIRACETAM FK-960 FPL-14995 FR-121196 FR-64822 FUB-181 GENIPIN GENIPOSIDATE GLUTAPYRONE GLYCEROPHOSPHORYLSERINE GVS-111 HOE-288 IDRA-21 IRFI-117 JTP-4819 KF-15372 KF-17837 KFM-19 KMBZ-009 KW-6055 L-783281 LEVEMOPAMIL LEVETIRACETAM LINOPIRDINE LY-404187 MCI-225 MDL-26479 METHYLAMINOPHOSPHONO= BUTYRATE-N METHYLAMINOPHOSPHONO= PROPIONATE-N NC-1900 NEBRACETAM NEFIRACETAM NICOMORPHOLINE NOOGLUTYL NS-105 NS-2359 OF-6145 OREXIN-A OXIRACETAM OXYBATE LITHIUM OXYBATELITHIUM PD-142505 PIFITHRIN-ALPHA PIRACETAM PRAMIRACETAM RIVASTIGMINE RO-13-6680 ROLZIRACETAM RS-67333 RS-67532 RU-33965 RU-35929 RU-41656 RU-49041 RU-52583 S-11701 S-12024-2 S-17092 S-18986 S-8510 S-9977 S-9977-2 SA-4503 SABELUZOLE SB-271046 SCH-211803 SIB-1508-Y SIB-1553-A SK-946 SK-9709 SKF-64346 SKF-74652 SM-10888 SM-21 SP-600125 SUN-0588 SURONACRINE T-588 TAK-147 TAMITINOL TAMOLARIZINE TDN-345 TENILOXAZINE TENILSETAM TGS-20 TGS-33 TGS-34 TOLSERINE UCB-11056

Derwent Drug File 1195 Thesaurus VELNACRINE WEB-1881-FU WS-1490 XR-543 NUT PEANUT OBESITY PICKWICK-SYNDROME OBSTETRICS ABORTION ABRUPTIO-PLACENTAE AMNIONITIS CHORIOAMNIONITIS DELIVERY DYSTOCIA ECLAMPSIA ECTOPIC-PREGNANCY EGG-YOLK-PERITONITIS EPISIOTOMY LABOR PLACENTA-RETENTION PREECLAMPSIA PRRS PUERPERIUM ODONTOLOGY CAPDEPONT-SYNDROME CARIES dental-caries DYSODONTIASIS ENAMELOMA MALOCCLUSION MICRODONTIA PERICORONITIS PERIODONTITIS PERIODONTOPATHY PERIODONTOSIS PULPITIS OLIGODEOXYNUCLEOTIDE ISIS-1082 ISIS-11061 ISIS-12449 ISIS-12959 ISIS-13650 ISIS-1570 ISIS-1751 ISIS-1753 ISIS-1755 ISIS-2105 ISIS-2302 ISIS-2503 ISIS-2922 ISIS-3082 ISIS-3521 ISIS-4015 ISIS-8005 ISIS-9044 ISIS-9047 OLIGOPHRENIA cerebral-gigantism CRETINISM debre-semelaigne-syndrome DOLLINGER-= BIELSCHOWSKY-= SYNDROME hypothyroid-myopathy KUFS-DISEASE LESCH-NYHAN-SYNDROME LITTLE-DISEASE MARTIN-BELL-SYNDROME MONGOLISM PHENYLKETONURIA RICHNER-HANHART-= SYNDROME trisomy-21 TUBEROUS-SCLEROSIS WEST-SYNDROME WILLIAMS-BEUREN-= SYNDROME ONCOVIRUS AVIAN-SARCOMA-VIRUS C-TYPE-VIRUS ERYTHROLEUKOSIS-VIRUS FRIEND-VIRUS GROSS-VIRUS KIRSTEN-VIRUS LEUKOSIS-VIRUS MAMMARY-TUMOR-VIRUS MASON-PFIZER-MONKEY-= VIRUS MOLONEY-VIRUS MOUSE-SARCOMA-VIRUS MYELOBLASTOSIS-VIRUS PULMONARY-= ADENOMATOSIS-VIRUS RETICULOENDOTHELIOSIS-= VIRUS ROUS-SARCOMA-VIRUS SIMIAN-SARCOMA-VIRUS SQUIRREL-MONKEY-= RETROVIRUS OPHTHALMOLOGICAL COLLYRIUM OPIOID-ANTAGONISTS CORYNANTHEIDINE HS-378 J-113397 NALMEFENE-GLUCURONIDE NIH-10420 NOCICEPTIN-1-13-NH2 NOCICEPTIN-PSI TRK-851 OPIOIDS 443-C 66A-078 A-3080 ACETORPHAN ADRENORPHIN AKUAMMICINE AMIDORPHIN ASIMADOLINE BAM-12P BAM-18 BAM-22P BC-3016 BIPHALIN BRL-52537 BRL-52656 BRL-53001 BRL-53001A BUBU BW-180C BW-831C BW-942C CASOMORPHIN-BETA-3 CASOMORPHIN-BETA-4 CASOMORPHIN-BETA-4-= HUMAN CASOMORPHIN-BETA-5 CASOMORPHIN-BETA-5-= HUMAN CASOMORPHIN-BETA-6 CASOMORPHIN-BETA-7 CASOPEPTONE CDRI-82-205 CYCLOPROPYLMETHYL= NORMORPHINE CYTOCHROPHIN-4 CYTOCHROPIN-5 DBO-11 DELTAKEPHALIN DELTORPHIN DELTORPHIN,2-D-ALA-4-GLU DELTORPHIN-I DELTORPHIN-II DEMETHYLKETOBEMIDONE DERMORPHIN DERMORPHIN,2-D-ARG DERMORPHIN,2-D-ARG-4-SAR DERMORPHIN,4-TRP-7-ASN DERMORPHIN,6-D-PRO DERMORPHIN,6-HYP DERMORPHIN,7-LYS DERMORPHIN-1-5 DEVALMUCEPTIN DPI-3290-W-93 DSTBULET DYNORPHIN DYNORPHIN-1-10 DYNORPHIN-1-10-AMIDE DYNORPHIN-1-11 DYNORPHIN-1-11-D-PRO-10 DYNORPHIN-1-12 DYNORPHIN-1-13 DYNORPHIN-1-17-D-ALA-2 DYNORPHIN-1-6 DYNORPHIN-1-7 DYNORPHIN-1-8 DYNORPHIN-1-9 DYNORPHIN-2-12 DYNORPHIN-2-13 DYNORPHIN-2-17 DYNORPHIN-3-13 DYNORPHIN-3-8 DYNORPHIN-32 DYNORPHIN-6-17 DYNORPHIN-B DYNORPHIN-B29 EK-209 EK-399 ENDOMORPHIN-1 ENDOMORPHIN-2 ENDORPHIN ENDORPHIN-ALPHA ENDORPHIN-ALPHA-DE-TYR-1 ENDORPHIN-BETA ENDORPHIN-BETA-1-9 ENDORPHIN-BETA-6-16 ENDORPHIN-BETA-ACETYL-N ENDORPHIN-BETA-CAMEL ENDORPHIN-BETA-D-ALA-2 ENDORPHIN-BETA-DE-TYR-1 ENDORPHIN-BETA-ELEPHANT ENDORPHIN-BETA-HORSE ENDORPHIN-BETA-HUMAN ENDORPHIN-BETA-HUMAN-= 1-26 ENDORPHIN-BETA-HUMAN-= 1-27 ENDORPHIN-BETA-HUMAN-= 1-28 ENDORPHIN-BETA-HUMAN-= 28-31 ENDORPHIN-BETA-HUMAN-= 6-31 ENDORPHIN-BETA-HUMAN-= LEU-5 ENDORPHIN-BETA-LEU-5 ENDORPHIN-BETA-OSTRICH ENDORPHIN-BETA-PIG ENDORPHIN-BETA-RAT ENDORPHIN-BETA-TURKEY ENDORPHIN-GAMMA ENDORPHIN-GAMMA-6-17 ENDORPHIN-GAMMA-DE-= TYR-1 ENKEPHALIN ENKEPHALIN,2-D-ALA-5-D-= MET

1196 APPENDIX D ENKEPHALIN,2-D-ALA-5-LEU ENKEPHALIN,2-D-ALA-5-= LEU-6-ARG ENKEPHALIN,2-D-ALA-5-= LEU-6-CYS ENKEPHALIN,2-D-ALA-5-= LEU-6-SER ENKEPHALIN,2-D-ALA-5-MET ENKEPHALIN,2-D-ALA-LEU-= 6-D-ARG ENKEPHALIN,2-D-PEN-5-CYS ENKEPHALIN,2-D-PEN-5-D-= PEN ENKEPHALIN,2-D-PEN-5-PEN ENKEPHALIN,2-D-SER-5-= LEU-6-THR ENKEPHALIN,2-D-THR-5-LEU ENKEPHALIN,2-D-THR-5-= LEU-6-THR ENKEPHALIN-LEU ENKEPHALIN-LEU,DE-TYR ENKEPHALIN-MET ENKEPHALIN-MET,6-ARG ENKEPHALIN-MET,6-ARG-7-= GLY-8-LEU ENKEPHALIN-MET,6-ARG-7-= PHE ENKEPHALIN-MET,6-ARG-7-= PHE-AMIDE ENKEPHALIN-MET,DE-TYR ENKEPHALINAMIDE ENKEPHALINAMIDE,2-D-= ALA-5-D-LEU ENKEPHALINAMIDE,2-D-= ALA-5-DE-LEU ENKEPHALINAMIDE,2-D-= ALA-5-LEU ENKEPHALINAMIDE,2-D-= ALA-5-MET ENKEPHALINAMIDE,2-D-= ALA-5-PRO ENKEPHALINAMIDE,2-D-= MET-5-PRO ENKEPHALINAMIDE-LEU ENKEPHALINAMIDE-MET ES-52 FEDOTOZINE FK-33-824 GR-94839 GYKI-14238 HEMORPHIN-4 HISTORPHIN HP-736 HZ-2 ICI-204448 JOM-13 KEPHALIN-DELTA KT-95 KYOTORPHIN KYOTORPHIN-D LACTORPHIN-ALPHA LEUMORPHIN METKEFAMIDE MITRAGYNINE-= PSEUDOINDOXYL MOL-5210 MORPHICEPTIN MORPHICEPTIN,4-D-PRO MRZ-2549 NEO-ENDORPHIN-ALPHA NEO-ENDORPHIN-BETA NEO-KYOTORPHIN NIFALATIDE NIH-10420 NIH-10741 NIRAVOLINE NOCICEPTIN NOCICEPTIN-1-13-NH2 OCILTIDE OHMEFENTANYL PD-129290 PENTAMORPHONE PEPTIDE-E PEPTIDE-F PL-017 R-84760 RB-38A RETRO-ENKEPHALIN-LEU RIMORPHIN RO-64-6198 RX-783006 RX-783030 SA-4503 SAMERIDINE SB-227122 SC-39566 SD-62 SK-9709 SL-3111 SNC-162 SNC-243-A SNC-80 SYNDYPHALIN-25 SYNDYPHALIN-33 SYNDYPHALIN-34 SYNDYPHALIN-41 SYNDYPHALIN-49 SYNDYPHALIN-6 SYNDYPHALIN-62 TAGEFLAR TAN-67 THIORPHAN TREFENTANIL TRIMU-5 TRK-820 U-54494A VALMUCEPTIN WY-42186 WY-42896 ZP-120-C OPT.ROTATION CIRCULAR-DICHROISM COTTON-EFFECT DICHROISM ORD POLARIMETRY RACEMIZATION ORL EPIGLOTTIS EUSTACHIAN-TUBE GLOTTIS HEARING HYPOLARYNX HYPOPHARYNX LABYRINTH LARYNX NASOPHARYNX OROPHARYNX PHARYNX PIRIFORM-SINUS SEMICIRCULAR-CANAL THROAT TONSIL UVULE VOCAL-CORDS ORL-DISEASE ADENOIDITIS ARYTENOIDITIS atrophic-rhinitis atrophic-rhinitis CARDIOAUDITORY-= SYNDROME CHOLESTEATOMA COMMON-COLD CROUP DEAFNESS dejerine-syndrome DIPHTHERIA diphtheritic-polyneuritis EPIGLOTTIDITIS HAY-FEVER HOARSENESS HYPERACUSIS HYPOACUSIS INCLUSION-BODY-RHINITIS LARYNGISMUS LARYNGITIS LARYNGOPHARYNGITIS LARYNGOTONSILLITIS LARYNGOTRACHEITIS LARYNGOTRACHEOBRONCHITIS LERMOYEZ-SYNDROME MASTOIDITIS MENIERE-DISEASE MYRINGITIS NASOPHARYNGITIS OTITIS OTORRHEA OTOSCLEROSIS PANSINUSITIS PERITONSILLITIS PERTUSSIS PHARYNGITIS PHARYNGOLARYNGEAL-= PARALYSIS-SYNDROME PHARYNGOLARYNGITIS PIETRANTONI-SYNDROME PSEUDOCROUP RHINITIS RHINOPHARYNGITIS RHINOPNEUMONITIS RHINORRHEA RHINOSCLEROMA RHINOTRACHEITIS SINUSITIS SNEEZING TEMPOROMANDIBULAR-= JOINT-SYNDROME TINNITUS TONSILLITIS TROTTER-SYNDROME UVULITIS VERTIGO XEROMYCTERIA ORNITHINE-DECARBOXYLASEINHIBITORS AMINOXYPROPYLAMINE AROTENOID BMY-30047 CHLOROQUINE CHS-828 DEGUELIN EFLORNITHINE ISOTRETINOIN K-1115-A MDL-26752 MDL-27695 MDL-72403 MDL-72430 MEFLOQUINE METHYLORNITHINE-ALPHA MONOFLUOROMETHYLDE= HYDROORNITHINE-ALPHA MOTRETINIDE RETINAL SANTALOL-ALPHA TRETINOIN OSMOSIS HYPEROSMOLAR OSMOLALITY OSMOLARITY

Derwent Drug File 1197 Thesaurus OSTEOMYELITIS PHYSITIS OSTEOPATHY ALGODYSTROPHY ankylosing-hyperostosis BAASTRUP-SYNDROME BONE-CARIES BONE-SPAVIN caffey-silverman-syndrome CONRADI-HUNERMAN-= SYNDROME disseminated-fibrous-osteitis DYSCHONDROSTEOSIS DYSOSTOSIS DZIERZYNSKY-SYNDROME ECTROMELIA ENOSTOSIS EPIPHYSIOLYSIS EPIPHYSITIS ERLACHER-BLOUNT-= SYNDROME ewing-bone-sarcoma ewing-osteosarcoma EXOSTOSIS forestier-rotes-querol-= syndrome FRACTURE FRIEDRICH-SYNDROME HAGLUND-SYNDROME HYPEROSTOSIS hypertrophic-pulmonary-= osteoarthropathy idiopathic-hypertrophic-= osteoarthropathy idiopathic-osteopsathyrosis infantile-cortical-hyperostosis KYPHOSCOLIOSIS KYPHOSIS LARSEN-JOHANNSON-= SYNDROME lobstein-syndrome LORDOSIS marie-bamberger-syndrome MELORHEOSTOSIS MORGAGNI-SYNDROME NAVICULAR-DISEASE OSTEALGIA OSTEITIS OSTEITIS-DEFORMANS OSTEOARTHROPATHY OSTEOBLASTOMA OSTEOCHONDRITIS OSTEOCHONDROSIS OSTEOCLASTOMA osteodystrophia-fibrosa OSTEODYSTROPHY OSTEOLATHYRISM OSTEOMALACIA OSTEOMYELITIS OSTEOMYELOSCLEROSIS OSTEONECROSIS OSTEOPENIA OSTEOPETROSIS OSTEOPHYTOSIS OSTEOPOROSIS OSTEOPSATHYROSIS OSTEOSARCOMA OSTEOSIS PANDIAPHYSITIS PERIOSTITIS PHYSITIS POTOMAC-HORSE-FEVER PROGRESSIVE-DIAPHYSEAL-= DYSPLASIA PSEUDARTHROSIS renal-osteodystrophy renal-rachitis renal-rickets RILEY-SHWACHMAN-= SYNDROME SAPHO-SYNDROME SCOLIOSIS SESAMOIDITIS SPINE-DEFORMITY SPONDYLARTHRITIS SPONDYLARTHROSIS SPONDYLITIS SPONDYLOLISTHESIS SPONDYLOLYSIS SPONDYLOPATHY SPONDYLOSIS SUDECK-DISEASE touraine-solente-gole-= syndrome uehlinger-syndrome wobbler-syndrome OSTEOSARCOMA MG63-CELL RPMI0041-CELL SA2-CELL SA9-CELL TE85-CELL OVARY CHO-CELL CORPUS-LUTEUM GRAAFIAN-FOLLICLE GRANULOSA-CELL HILUS-CELL MESOVARIUM ovarian-follicle OVIDUCT OVULATION OVARY-DISEASE carcinoma, ovary CYSTIC-OVARY DYSGERMINOMA HYPERANDROGENISM HYPERESTROGENISM LUTEOMA MEIGS-SYNDROME OOPHORITIS ovary-carcinoma POLYCYSTIC-OVARY OXIDATION DEHYDROGENATION OXYTOCIN-AGONISTS ANTOCIN-II ARGIPRESTOCIN CARBETOCIN CARGUTOCIN DEMOXYTOCIN DICARBAOXYTOCIN GLUMITOCIN ISOTOCIN MESOTOCIN NACARTOCIN OXYPRESSIN OXYTOCIN OXYTOCIN-1-8 TOCINAMIDE TOCINOATE OXYTOCIN-ANTAGONISTS ATOSIBAN CAP-440 F-123 F-327 L-342643 L-365209 L-366509 L-366682 L-366811 L-366948 L-368899 L-371257 SO-121 P-GLYCOPROTEIN-INHIBITORS AMIODARONE ANDRASTIN-A ATORVASTATIN-METHYL-= ESTER CGP-41251 CICLOSPORIN CLOFAZIMINE COLCHICINE DAUNORUBICIN DEHYDROSTIPIAMIDE-6,7 DENDROAMIDE-A DEXVERAPAMIL DIHYDROXYCHLOR= PROMAZINE-7,8 DOXORUBICIN EPIRUBICIN ER-086526 FLUNARIZINE GF-109203X GF-120918 GRAMICIDIN H-7 H-87 HAPALOSIN KN-62 LAMELLARIN-I LY-335979 MITOMYCIN N-5228 OC-144093 PACLITAXEL QUINIDINE QUININE R-101933 RESERPINE S-23906-1 S-9788 SB-RA-31012 SB-T-1213 U-74389 VALINOMYCIN VALSPODAR VANADATE VERAPAMIL VINBLASTINE XR-9051 XR-9576 PACKAGING LABEL PAF-ANTAGONISTS 48740-RP 52770-RP 59227-RP A-137491 A-85783 ABC-99 ABT-299 ACOPAFANT AGLAFOLINE APAFANT BB-823 BEPAFANT BN-50341 BN-50726 BN-50727 BN-50730 BN-50739 BN-52111 BN-52115 BN-52256 BN-54062

1198 APPENDIX D CIS-19 CK-53 CL-184005 CMI-206 CMI-392 CV-3988 CV-6209 DF-1111301 DIHYDROKAOSURENONE E-5880 E-6123 ECHISTATIN EPIYANGAMBIN FARGESIN FR-49175 FR-900452 FUTOENONE GINKGOLIDE-A GINKGOLIDE-B GINKGOLIDE-C GINKGOLIDE-J GLAUCOCALYXIN-A HISPANOLONE KADSURENONE KO-286011 KW-4679 L-002 L-615919 L-651142 L-652731 L-653150 L-659989 L-668750 L-680573 L-680574 LEXIPAFANT MAGNONE-A MAGNONE-B MEQUITAMIUM IODIDE METHYLPIPERBETOL MIZOLASTINE ONO-6240 PCA-4248 PF-10040 PINUSOLIDE PMS-832 PREDICENTRINE RO-19-1400 RO-19-3704 RO-23-0238 RO-24-0238 RO-24-4637 RO-24-4736 RP-52629 RP-52770 RP-58467 RP-59228 RU-45703 RUPATADINE S35B SB-203347 SCH-37370 SCH-44643 SCH-47918 SDZ-62-434 SDZ-62-694 SDZ-62-759 SDZ-62-826 SDZ-63-135 SDZ-64-412 SELLIGUEAIN SKF-45905 SKF-98625 SL-85-0324 SM-10661 SM-12502 SR-27417 SRI-63-072 SRI-63-119 SRI-63-441 SRI-63-675 STY-2108 SWIETEMAHONIN-A SWIETEMAHONIN-E TCV-309 U-46195 U-66982 U-66985 U-68043 UK-74505 UR-10324 UR-11353 UR-12460 UR-12592 UR-12670 VERAGUENSIN WEB-2118 WEB-2347 Y-24180 YANGAMBIN YM-264 YM-461 ZG-1494-ALPHA PANCREAS BETA-CELL PANCREAS-HORMONE GLUCAGON-AGONIST INSULIN-AGONIST PANCREAS-HORMONES AD-5075 ALX-0600 BM-130913 CHIRO-INOSITOL CLX-0901 DIARGINYLINSULIN ENTEROGLUCAGON EXENDIN-4 GLICENTIN GLUCAGON GLUCAGON-1-21 GLUCAGON-37 GLUCAGON-AGONISTS GLUCAGON-LIKE-PEPTIDE-1 GLUCAGON-LIKE-PEPTIDE-= 1,7-36-AMIDE GLUCAGON-LIKE-PEPTIDE-= 1,7-37 GLUCAGON-LIKE-PEPTIDE-2 GLUCAGON-LIKE-PEPTIDE-= 2-HUMAN HOE-71-GT INSULIN INSULIN-A-CHAIN INSULIN-AGONISTS INSULIN-ASPART INSULIN-B-9-23 INSULIN-B-CHAIN INSULIN-CATTLE INSULIN-CATTLE-A-CHAIN INSULIN-CATTLE-B-CHAIN INSULIN-DETEMIR INSULIN-FOWL INSULIN-GLARGINE INSULIN-GUINEA-PIG INSULIN-HORSE INSULIN-HUMAN INSULIN-HUMAN-A-CHAIN INSULIN-HUMAN-B-CHAIN INSULIN-HUMAN-B10-ASP INSULIN-HUMAN-B10-GLU INSULIN-HUMAN-B28LYS,B29-PRO INSULIN-HUMAN-B9-ASP,= B27-GLU INSULIN-PIG INSULIN-RABBIT INSULIN-RAT INSULIN-SAPG INSULIN-SHEEP L-783281 LY-307161 MERCK-L-7 METHYLCYSTEINE-= SULFOXIDE-S NN-2211 NN-304 PANCREATIC-POLYPEPTIDE PANCREATIC-POLYPEPTIDE-= BIRD PANCREATIC-POLYPEPTIDE-= CATTLE PANCREATIC-POLYPEPTIDE-= FOWL PANCREATIC-POLYPEPTIDE-= HUMAN PANCREATIC-POLYPEPTIDE-= PIG PANCREATIC-POLYPEPTIDE-= RAT PROINSULIN PROINSULIN-CATTLE PROINSULIN-HUMAN PROINSULIN-HUMAN-DE-64-= 65 PROINSULIN-MONKEY PROINSULIN-PIG VANADYL DIPICOLINATE PANCREOPATHY BALSER-NECROSIS BARD-PIC-SYNDROME bronze-diabetes DAWN-PHENOMENON DIABETES diabetic-glomerulosclerosis diabetic-retinopathy GASTRINOMA GLUCAGONOMA HYPERGASTRINEMIA HYPERINSULINISM INSULINOMA INSULITIS metabolic-syndrome METABOLIC-SYNDROME-X MUCOVISCIDOSIS NESIDIOBLASTOSIS PANCREATITIS PANCREOHEPATIC-= SYNDROME SCHWACHMAN-SYNDROME troissier-hanot-chauffard-= syndrome VERNER-MORRISON-= SYNDROME VIPOMA WERMER-SYNDROME ZOLLINGER-ELLISON-= SYNDROME PANCREOZYMIN-ANTAGONISTS A-64718 A-65186 A-67396 ASPERLICIN ASPERLICIN-B ASPERLICIN-C ASPERLICIN-D ASPERLICIN-E BENZOTRIPT BUTABINDIDE BZ-140 CAM-1481 CARBOBENZOTRIPT

Derwent Drug File 1199 Thesaurus CR-2017 DEVAZEPIDE DEXLOXIGLUMIDE FK-480 GE-410 GV-150013 GV-150013-X GW-5823 IQM-95333 JB-93182 JMV-179 KSG-504 L-365031 L-365260 L-368935 L-740093 L-740093-S LORGLUMIDE LOXIGLUMIDE LY-219057 LY-262691 LY-288513 PD-134308 PD-135158 PD-135666 PD-136450 PD-140376 PD-140548 PD-142308 PD-142898 PD-145942 PROGLUMIDE RB-211 RP-69758 S-0509 SPIROGLUMIDE SR-27897 T-0632 TETRONOTHIODIN TOMOGLUMIDE TP-680 YM-022 YM-220 Z-360 PAPOVAVIRUS BK-VIRUS PAPILLOMA-VIRUS POLYOMA-VIRUS SV40-VIRUS PARALYSIS AVELLIS-SYNDROME BABINSKI-NAGEOTTE-= SYNDROME BELLS-PALSY brown-sequard-syndrome CEREBRAL-PALSY CESTAN-CHENAIS-= SYNDROME DEJERINE-KLUMPHE-= SYNDROME DIPLEGIA familial-spastic-paraplegia FOVILLE-SYNDROME HEMIPARAPLEGIA HEMIPARESIS HEMIPLEGIA LITTLE-DISEASE MILLARD-GUBLER-= SYNDROME PARAPLEGIA PARESIS QUADRIPLEGIA spinal-hemiparaplegia struempell-lorrain-disease TETRAPLEGIA PARANOIA EROTOMANIA PARAPROTEINEMIA ALPHA-CHAIN-DISEASE CRYOGLOBULINEMIA GAMMOPATHY HEAVY-CHAIN-DISEASE MACROGLOBULINEMIA WALDENSTROEM-DISEASE PARASYMPATHOLYTICS ADIPHENINE AF-14 AF-DX-384 AF-DX-474 AH-9700 AJ-234 ALVERINE AMBUTONIUM AMIXETRINE APROFENE APROLIDINE AQ-RA-391 AQ-RA-741 ARPENAL ATROMEPINE ATROPINE ATROPINE-ETHIODIDE ATROPINE-METHONITRATE ATROPINE-OXIDE AWD-26-39 AZAPROPHEN BENACTYZINE BENAPRIZINE BENTIPIMINE BENZATROPINE BENZETIMIDE BENZILONIUM BROMIDE BENZILYLCHOLINE BENZOMETHAMINE BENZOPYRRONIUM BROMIDE BEPERIDIUM IODIDE BEVONIUM METILSULFATE BIBN-99 BIPERIDEN BL-14 BM-5 BOK-1 BORNAPRINE BR-370 BS-6181 BUTINOLINE BUTROPIUM BROMIDE BUTYLSCOPOLAMINE BUTYLSCOPOLAMINE = BROMIDE BUZEPIDE-METIODIDE CANDOCURONIUM-IODIDE CARAMIPHEN CATECHOLINE CEB-1957 CHANDONIUM CHLORBENZOXAMINE CHLOROSIL CHLORPHENOXAMINE CI-923 CICLONIUM BROMIDE CIMETROPIUM BROMIDE CLIDINIUM BROMIDE CYCLOPENTOLATE CYCLOPYRRONIUM BROMIDE CYCLOSTELLETTAMINE-A CYCLOSTELLETTAMINE-B CYCLOSTELLETTAMINE-C CYCLOSTELLETTAMINE-D CYCLOSTELLETTAMINE-E CYCLOSTELLETTAMINE-F CYCRIMINE DAC-5945 DAMP-4 DARIFENACIN DECITROPINE DEETHYLOXYBUTYNIN DEMETHYLOXYPHENONIUM DEPTROPINE DEPTROPINE-= METHOBROMIDE DEXETIMIDE DF-594 DIBROMOSCEPTRIN DICARFEN DICYCLOVERINE DIETHAZINE DIFEMERINE DIHEXYVERINE DIMEVAMIDE DIPHEMANIL-METILSULFATE DIPHENYLTROPINE DOMAZOLINE DROCLIDINIUM BROMIDE ELANTRINE ELUCAINE EMEPRONIUM BROMIDE ERYSODINE ET-126 ETEROFEN ETPENAL ETYBENZATROPINE EUCATROPINE FC-18-94 FC-20-94 FENCARBAMIDE FENTONIUM BROMIDE FK-584 FLUOROHEXAHYDRO= DIFENIDOL-PARA FLUOROHEXAHYDRO= DIFENIDOL-PARA FLUOROHEXAHYDROSILA= DIFENIDOL-PARA FLUOROHEXBUTINOL-PARA FLUTROPIUM BROMIDE G-3063 GLYCOPYRRONIUM BROMIDE GUANYLPIRENZEPINE HEMICHOLINIUM HEMICHOLINIUM-15 HEMICHOLINIUM-A-4 HEMICHOLINIUM-A-5 HETERONIUM BROMIDE HEXAHYDRODIFENIDOL HEXAHYDROSILADIFENIDOL HEXASONIUM IODIDE HEXBUTINOL METHIODIDE HEXOCYCLIUM = METILSULFATE HEXOPYRRONIUM BROMIDE HOMATROPINE HOMATROPINE = METHYLBROMIDE HYOSCYAMINE IMPERIALINE IPRAGRATINE IPRATROPIUM BROMIDE ISOPROPAMIDE IODIDE KRP-197 LACHESINE LU-25-109-T LY-315535 LY-316108 MDL-201346 MECLOXAMINE MEFURTRAMINE MELETIMIDE

1200 APPENDIX D MEPENZOLATE BROMIDE MEPIPERPHENIDOL METHAMICIL METHANTHELINIUM = BROMIDE METHOCTRAMINE METHOXYSILAHEXO= CYCLIUM-ORTHO METHSCOPOLAMINE METHYLBENACTYZIUM = BROMIDE METIXENE METOCINIUM IODIDE METOQUIZINE MF-10058 NAM-242 NAM-250 NOLINIUM BROMIDE NS-21 NUVENZEPINE OCTATROPINE-= METHYLBROMIDE OROIDIN ORPHENADRINE OTENZEPAD OXAPIUM IODIDE OXITROPIUM BROMIDE OXYBUTYNIN OXYCLIPINE OXYPHENCYCLIMINE OXYPHENONIUM BROMIDE OXYPYRRONIUM BROMIDE OXYSONIUM IODIDE PARAPENZOLATE BROMIDE PD-102807 PD-150714 PENTAPIPERIDE PENTAPIPERIUM-= METILSULFATE PENTHIENATE PHENGLUTARIMIDE PHENSERINE PIPENZOLATE BROMIDE PIPERIDOLATE PIPETHANATE PIRENZEPINE PIROTRAMINE PLATYPHYLLINE PNU-200577 POLDINE-METILSULFATE PRAMPINE PRIDINOL PRIDINOL-MESILATE PRIFINIUM BROMIDE PROCYCLIDINE PROFENAMINE PROMAZINE PROPANTHELINE PROPANTHELINE BROMIDE PROPYLBENZILYLCHOLINE-= MUSTARD PROPYROMAZINE BROMIDE QUINUCLIDINYL-XANTHENE-= CARBOXYLATE-9 RISPENZEPINE RITROPIRRONIUM BROMIDE RO-2-3308 SALFLUVERINE SCH-211803 SCOPOLAMINE SECOVERINE SILAHEXOCYCLIUM SILAHEXOCYCLIUM-= METILSULFATE SILAPROCYCLIDINE SILATRIHEXYPHENIDYL SINTROPIUM BROMIDE SOPITAZINE SPIROTRAMINE SS-62-4 SS-62-6 SU-740 SULTROPONIUM TELENZEPINE TERODILINE THIAZINAMIUM IODIDE THIAZINAMIUM-= METILSULFATE THIAZINAMIUM-SULFOXIDE THIAZINAMIUM-SULFOXIDE = IODIDE THIENGLUTARIMIDE THIHEXINOL-= METHYLBROMIDE TIEMONIUM IODIDE TIFENAMIL TIGLOIDINE TIMEPIDIUM BROMIDE TIOTROPIUM BROMIDE TIQUINAMIDE TL-402 TOFENACIN TOLTERODINE TOQUIZINE TRANTELINIUM BROMIDE TRIAMPYZINE TRICLAZATE TRICYCLAMOL CHLORIDE TRICYCLAMOL-IODIDE TRIDIHEXETHYL IODIDE TRIHEXYPHENIDYL TRIHEXYPHENIDYL-= METHIODIDE TRIMETHYLDIPHENYL= PROPYLAMINE TROPENZILINE BROMIDE TROPICAMIDE TROPIGLINE TROPINE-BENZILATE TROPIRINE TROPODIFENE TROVENTOL UH-AH-37 UNO-3 VALETHAMATE BROMIDE VAMICAMIDE W-84 XENYTROPIUM BROMIDE YM-53707 YM-905 Z-338 ZAMIFENACIN ZEPASTINE PARASYMPATHOMIMETICS 210-086 A-82695 A-84543 A-85380 ABT-089 ABT-418 ABT-594 ACECLIDINE ACETOXYNORTROPANE-6-= BETA ACETYLCAINE ACETYLCHOLINE ACETYLSELENONIUM-= CHOLINE AF-102B AF-150-S AF-267-B AF-30 AG-4 AH-6405 ALLOMUSCARONE ALTINICLINE AMBENONIUM CHLORIDE AMINOSTIGMINE AMYL-= TRIMETHYLAMMONIUM ANATOXIN-A ARECAIDINE-PROPARGYL-= ESTER ARMINE BETHANECHOL BM-123 BM-123A BM-130 BM-130-A BM-5 BR-100 BR-401 BR-401A BRL-20627 BUTYRYLCHOLINE CARBACHOL CARPRONIUM CHLORIDE CDD-0098-J CHOLINE CHOLINE-ALFOSCERATE CYTISINE DBO-83 DEMECARIUM BROMIDE DEMETHYLXANOMELINE DFP DISTIGMINE BROMIDE DMPP EDROPHONIUM CHLORIDE EPIBOXIDINE ESERIDINE ETHYLCHOLINE EXEPANOL F-2268 FPL-14995 FURTRETHONIUM IODIDE GTS-21 HEPTYLPHYSOSTIGMINE HEXYLTRIMETHYL= AMMONIUM BROMIDE HP-184 HSR-803 HUPRINE-Y HYDROXYMINAPRINE-2+ ICOPEZIL ISOARECOLINE ISOARECOLONE-METHIODIDE ISOPILOCARPINE KW-5092 L-658903 L-660863 L-670207 L-687306 L-689660 LINOPIRDINE LU-25-109-T LY-297802 METANICOTINE METHACHOLINE CHLORIDE METHOXYTACRINE-7 METHYLCARBACHOL-N METHYLFURMETHIDE MF-268 MFS-3 MR-16728 MUSCARINE MUSCARONE NEOSTIGMINE NEOSTIGMINE BROMIDE NEOSTIGMINE = METHYLSULFATE

Derwent Drug File 1201 Thesaurus NICOTINE NICOTINE-POLACRILEX NORPHYSOSTIGMINE OB-47042 OXA-22 OXOTREMORINE OXOTREMORINE-1 OXOTREMORINE-2 OXOTREMORINE-3 PARAOXON PD-142505 PHENTHIMENTONIUM PHENYLTRIMETHYL= AMMONIUM IODIDE PHYSOSTIGMINE PHYSOSTIGMINE-SALICYLATE PILOCARPINE PK-154 PLICATATE PROPIONYLCHOLINE PYRIDOSTIGMINE BROMIDE PYROPHOS RIVASTIGMINE RJR-2429 RS-86 RU-35926 RU-35963 S-6 S-9977-2 SDZ-ENS-163 SIB-1508-Y SIB-1553-A SIB-1765-F SK-946 SLAFRAMINE SM-10888 SM-21 SR-46559-A SR-95639A SUBECHOLINE SUBEROGORGIN SULFOTEPP SUVANINE TAK-147 TEPP THB-013 U-80816 UM-1046 WAL-2014 WEB-1881-FU WIN-3286 XANOMELINE XE-991 XR-543 YM-796 PARATHYROID-DISEASE HYPERPARATHYROIDISM HYPOPARATHYROIDISM WERMER-SYNDROME PARP-INHIBITORS AMINONICOTINAMIDE NU-1025 NU-1064 PD-128763 PARVOVIRUS ADENO-ASSOCIATED-VIRUS ALEUTIAN-DISEASE-VIRUS DERZSY-DISEASE-VIRUS PANLEUKOPENIA-VIRUS PDGF-ANTAGONISTS CT-052923 IMATINIB PEDIATRICS INFANT PELLET MICROPELLET PENETRATION-ENHANCERS BUTYL-LAURATE CAPRATE CAPROYLLYSOLECITIHN CHAPSO CHENODEOXYCHOLATE CITRATE CYCLODEXTRIN-ALPHA-= DIMETHYL DECANOYLPHENYLALANINE DECYL-METHYL-SULFOXIDE DEOXYCHOLATE DIMETHYLSULFOXIDE DODECYL-PYROGLUTAMATE DODECYLAMINE E-414 EDTA EICOSENOATE-11 EMI-1 EMI-2 EMI-3 ENOXOLONE-= MONOHEMIPHTHALATE ETHYL-ALCOHOL ETHYLMENTHOL-O ETHYLPYRROLIDONE-2 EUCALYPTOL GLYCOCHOLATE HEXADECYLMALTOSIDE HEXAMETHYLENELAURAMIDE HEXYLPYRROLIDONE-2 HPE-101 ISOPROPYL-ALCOHOL LAURATE LAUROCAPRAM LAUROYLALANINE LAURYL-SULFATE SODIUM LAURYLPYRROLIDONE-2 LIMONENE-OXIDE MEGA-10 MEGA-8 METHOXYSALICYLATE-5 METHYLPYRROLIDONE-2 NONANE OCTYL-ACETATE OCTYLTHIOGLUCOSIDE OLEATE POLIDOCANOL POLYCARBOPHIL POLYISOPRENE POLYOXYETHYLENE-CETYL= ETHER POLYOXYETHYLENE-= CHOLESTEROL-ETHER POLYOXYETHYLENE-OLEYL-= ETHER POLYOXYETHYLENE-= STEARYL-ETHER PROLINE-METHYL-ESTER PROPYL-LAURATE PROPYLENE-GLYCOL PYRROLIDONE-2 STEAROYLLYSOLECITHIN TAUROCHOLATE TRIMETHYLCHITOSAN-N-= CHLORIDE UREA (Drug) PENIS CORPUS-CAVERNOSUM CORPUS-SPONGIOSUM ERECTION FORESKIN PENIS-DISEASE BALANITIS BALANOPOSTHITIS HYPOSPADIAS PARAMPHIMOSIS PARAPHIMOSIS PHIMOSIS PLASTIC-INDURATION POSTHITIS PRIAPISM PEPTIDE-HYDROLASEINHIBITOR CATHEPSIN-INHIBITOR CHYMOTRYPSIN-INHIBITOR COLLAGENASE-INHIBITOR GELATINASE-A-INHIBITOR GELATINASE-B-INHIBITOR HIV-PROTEASE-INHIBITOR LEUKOCYTE-ELASTASE-= INHIBITOR MATRIXMETALLOPROTEINASE-= INHIBITOR NEUTRAL-ENDOPEPTIDASE-= INHIBITOR NEUTROPHIL-ELASTASE-= INHIBITOR PANCREATIC-ELASTASE-= INHIBITOR STROMELYSIN-1-INHIBITOR STROMELYSIN-2-INHIBITOR STROMELYSIN-INHIBITOR PEPTIDE-HYDROLASEINHIBITORS A-74704 A-75912 A-75925 A-76792 A-76889 A-76890 A-76928 A-77003 A-77212 A-98881 ACETYLCYSTEINE ACETYLPEPSTATIN-N ACETYLSTATINE ADALIMUMAB AERUGINOSIN-298-A AG-1402 AG-555 AG-7088 AK-275 AK-295 ALLICIN ALOXISTATIN AMASTATIN AMIDINOPHENYLPYRUVATE-4 AMPRENAVIR ANTILEUKOPROTEASE ANTIPAIN APC-2059 APROTININ APROTININ-ARG-15 APSTATIN BATIMASTAT BAY-12-9566 BB-16 BB-2275 BB-3103 BILN-303-SE BMS-182193 BMS-182657 BMS-262084 BMS-275291 BMY-44621

1202 APPENDIX D BOROLEUCINE BOWMAN-BIRK-INHIBITOR BU-2743-E BW-175 CA-030 CA-074 CALPAIN-INHIBITOR-I CALPAIN-INHIBITOR-II CALPEPTIN CAMOSTAT CARBOXYPEPTIDASE-= INHIBITOR CATHEPSIN-INHIBITORS CATHESTATIN-A CATHESTATIN-B CE-0265 CE-0266 CE-0267 CGP-53820 CGP-73547 CGS-24592 CGS-25462 CGS-26303 CGS-26670 CGS-27023-A CGS-31447 CHYMOSTATIN CHYMOSTATIN-A CHYMOSTATIN-B CHYMOSTATIN-C CHYMOTRYPSIN-INHIBITORS CIPEMASTAT CMT-7 COLLAGENASE-INHIBITORS CP-471-474 CYSTATIN CYSTATIN-C-HUMAN DESMAL DIDANOSINE DMP-450 DOXYCYCLINE E-3123 E-64 E-64C ECADOTRIL EETI-II EGLIN-C EI-546 ELASNIN ELASTATINAL EP-459 EPIBESTATIN EPIGALLOCATECHIN-GALLATE EPOSTATIN EPOXOMICIN ER-32935 EURYSTATIN-A EURYSTATIN-B FK-448 FLUOSTATIN-A FLUOSTATIN-B FOY-251 FR-134043 FUCOSTEROL FUTOENONE GABEXATE GELATINASE-A-INHIBITORS GELATINASE-B-INHIBITORS GELIN GM-6001 GW-433908 H-19 HIRUGEN HIV-PROTEASE-INHIBITORS HYDROXYACECLOFENAC-4 HYDROXYUBENIMEX-PARA ICI-200355 ICI-200880 INDINAVIR JE-2147 JMV-390-1 JTP-2724 K-11002 K-11777 KAEMPFEROL KB-R-7785 KUNITZ-PROTEASE-INHIBITOR KYNOSTATIN-272 L-373890 L-657229 L-658758 L-659286 L-669844 L-670258 L-679723 L-680831 L-680833 L-680861 L-682271 L-682946 L-683537 L-683557 L-683558 L-683841 L-683845 L-684248 L-684249 L-684481 L-689502 L-691886 L-694458 L-696474 L-805645 LAVENDUSTIN-A LEUCINTHIOL LEUHISTIN LEUKOCYTE-ELASTASE-= INHIBITORS LEUPEPTIN LEUPEPTIN-1 LEUPEPTIN-2 LEX-032 LOPINAVIR LUTIDINATE LY-103629 LY-289612 LY-806303 MAPI-ALPHA MARIMASTAT MATRIX-= METALLOPROTEINASE-= INHIBITORS MC-11 MDL-102111 MDL-102823 MDL-201053 MDL-201404 METHYLSELENOL MG-115 MG-132 MG-262 MICROVIRIDIN-B MICROVIRIDIN-C MICROVIRIDIN-D MICROVIRIDIN-E MICROVIRIDIN-F MINOCYCLINE MIXANPRIL MMI-166 MR-889 NAFAMOSTAT NCO-700 NELFINAVIR NERFILIN-I NERFILIN-II NEUTRAL-ENDOPEPTIDASE-= INHIBITORS NEUTROPHIL-ELASTASE=INHIBITORS NK-3201 NSC-158393 NVP-DPP-728 ONO-3307 ONO-3403 ONO-5046 ONO-6818 ORYZACYSTATIN-I OSCILLAMIDE-Y P-32-98 PANCREATIC-ELASTASE-= INHIBITORS PANTRIPIN PD-166793 PD-178390 PD-178392 PEPSTATIN PEPSTATIN-A PEPSTATINYL-ARGININE-= METHYL-ESTER PGE-4410186 PHELORPHAN PHOSPHORAMIDON PIPERASTATIN-A PLASMINOSTREPTIN PLATYCODIN-D PNU-109112 PNU-99533 POLYACRYLATE POLYPORENATE-C POSTSTATIN POT-II PRINOMASTAT PROBESTIN PROCTOLIN PROTEASOME-INHIBITOR-1 PS-519 QUERCETIN RADIOSUMIN RB-105 RD-3-0174 RHEIN RIFAMPICIN RIFAMYCIN RIFAMYCIN-B RITONAVIR RO-28-2653 RO-32-7315 S-17092 S-2441 SA-7090 SAQUINAVIR SB-203238 SC-37698 SC-39026 SC-44463 SC-52151 SCH-54470 SD-146 SDZ-MTH-958 SECRETORY-= LEUKOPROTEASE-= INHIBITOR SEPIMOSTAT SINORPHAN SPI-501 SQ-28603 SQ-29072 STAVUDINE STROMELYSIN-1-INHIBITORS STROMELYSIN-2-INHIBITORS STROMELYSIN-INHIBITORS SUAM-1221 TALOPEPTIN

Derwent Drug File 1203 Thesaurus TEI-5624 TEI-6344 TENIDAP THEAFLAVIN THEAFLAVIN-DIGALLATE THIOLSTATIN TIAPROFENATE TIPRANAVIR TMC-2-A TMC-2-B TMC-2-C TP-151 TPCK TRANSFORMING-GROWTH-= FACTOR-BETA-1 TRYPSIN-INHIBITOR-CATTLE TRYPSIN-INHIBITOR-CORN TRYPSIN-INHIBITOR-HUMAN TRYPSIN-INHIBITOR-LIMA-= BEAN TRYPSIN-INHIBITOR-= OVOMUCOID TRYPSIN-INHIBITOR-SOY-= BEAN TYRPHOSTIN-B-44 U-103017 U-11790 U-11866 U-18598 U-22312 U-22989 U-24278 U-24279 U-24522 U-24631 U-27391 U-75875 U-80631-E U-96988 UBENIMEX UIC-94003 ULINASTATIN VANADATE WIN-63394 WIN-63759 WIN-64733 WS-1358A1 WS-1358B1 WS-75624-A WS-75624-B XK-216 XR-457 XR-835 XV-638 YM-47141 ZALCITABINE ZIDOVUDINE ZINCOV ZK-805412 ZK-805623 ZL-III-43-A PERIPHERAL-NERVE-DISEASE ADIE-SYNDROME ALLODYNIA ANDRADE-SYNDROME ANOSMIA AREFLEXIA AURICULOTEMPORAL-= SYNDROME BARRE-LIEOU-SYNDROME BELLS-PALSY BERNARD-HORNER-= SYNDROME CARPAL-TUNNEL-SYNDROME CAUSALGIA CERVICAL-SYNDROME charcot-marie-tooth-= syndrome charlin-syndrome ciliary-neuralgia DEJERINE-KLUMPHE-= SYNDROME dejerine-sottas-syndrome dejerine-syndrome DERMATOPOLYNEURITIS diphtheritic-polyneuritis duchenne-erb-paralysis DYSERGIA DYSESTHESIA ENURESIS ERYTHROPROSOPALGIA facial-paralysis facial-trophoneurosis FOIX-SYNDROME fothergill-syndrome GANGLIONITIS GARCIN-SYNDROME GLANZMANN-SALAND-= SYNDROME GRADENIGO-SYNDROME guillain-barre-syndrome HERPES-ZOSTER HOWSHIP-ROMBERG-= SYNDROME HYPERALGESIA HYPERESTHESIA HYPERPATHIA hypertrophic-interstitial-= neuritis hypertrophic-neuritis HYPOESTHESIA INCONTINENCE ISCHIALGIA JEFFERSON-SYNDROME JUGULAR-FORAMEN-= SYNDROME KEY-GASKELL-SYNDROME MEIGE-SYNDROME MELKERSSON-ROSENTHAL-= SYNDROME NEURALGIA NEURITIS NEUROCIRCULATORY-= COMPRESSION-= SYNDROME NEUROLIPOMATOSIS neuropathic-musc.atrophy NUMBNESS OPTIC-NEUROMYELOPATHY orthostatic-dysautonomic-= hypotension orthostatic-hypotension PARALYSIS PARESTHESIA PARINAUD-SYNDROME PHARYNGOLARYNGEAL-= PARALYSIS-SYNDROME PIETRANTONI-SYNDROME POLYNEURITIS POLYNEUROPATHY POLYRADICULONEURITIS PROGRESSIVE-TORSION-= SPASM putti-syndrome RADICULITIS RADICULOPATHY RESTLESS-LEGS RETROPAROTID-SPACE-= SYNDROME rheumatic-sciatica RILEY-SHWACHMAN-= SYNDROME romberg-syndrome roussy-cornil-syndrome ROUSSY-LEVI-SYNDROME SCIATICA shingles SHOULDER-HAND-= SYNDROME shy-drager-syndrome sluder-disease sphenopalatine-neuralgia STIFF-MAN-SYNDROME SUBACUTE-MYELOOPTIC-= NEUROPATHY SUDECK-DISEASE SYMPATHETICOTONIA tic-douloureux trigeminal-neuralgia TRISMUS TROPHONEUROSIS TROTTER-SYNDROME VAGOACCESSORY-= HYPOGLOSSAL-= SYNDROME VAGOACCESSORY-= SYNDROME VAGOHYPOGLOSSAL-= SYNDROME VAGOTONIA WALLERIAN-DEGENERATION WARTENBERG-DISEASE WRIGHT-SYNDROME PEROXIDASE MYELOPEROXIDASE PERSONALITY-DISORDER NARCISSISM PH-PK ACIDITY ALKALINITY BUFFER PHAGE PROPHAGE PHARM.PREP. BALM BULLET CAPSULE CHEWING-GUM COLLYRIUM CREAM DEPOT DOUCHE DRAGEE DROPS DURULE ELIXIR GARGLE GELULE GRANULE IMMUNOLIPOSOME INJECTABLE JELLY LINIMENT LIPSTICK LOTION LOZENGE LYOC MICROBEAD MICROCAPSULE MICROGRANULE MICROPELLET NANOCAPSULE NANOPELLET NIOSOME OINTMENT OVULE PASTE PASTILLE PELLET PESSARY POMADE POWDER

1204 APPENDIX D SPRAY STICK SUPPOSITORY SYRUP TABLET TINCTURE TISANE PHARMACEUTICS ANISOTROPY ANTISTATIC AUXILIARY-INGREDIENT BINDER BREAKING-STRENGTH BULK-DENSITY BULK-VOLUME CAPSULATION CAST COACERVATION COATING COMPACTING COMPRESSIBILITY COMPRESSION CONSISTENCY CRUSHING DESICCANT DISINTEGRANT DISINTEGRATION ENCAPSULATION FILLER FORMULATION FRIABILITY GRANULATION GRINDING HARDNESS HOMOGENIZATION HUMECTANT MICROENCAPSULATION MICROPARTICLE MICROPELLETIZATION MICROPELLETIZATION MILLING NANOENCAPSULATION NANOPARTICLE PARTICLE-SIZE PELLETIZATION POROSITY PRECOMPRESSION SOFTNESS SPHERONIZATION SPRAY-EMBEDDING TABLETTING TACKINESS PHARMACOECONOMICS COST COST-EFFECTIVENESS PHARMACOKINETICS distribution-volume HALF-LIFE volume-of-distribution PHEOCHROMOCYTOMA PC12-CELL PHOSPHODIESTERASEINHIBITORS 349U85 661U88 A-802715 AAL-05 ABC-99 ADIBENDAN AH-P-719 ALBANOL-B AMENTOFLAVONE-= HEXAACETATE AMINOPHYLLINE AMRINONE ANTIARRHYTHMIC-PEPTIDE ATZ-1993 AWD-12-281 B-9004-070 BEFURALINE BEMORADAN BMY-43351 CD-349 CDP-840 CH-102 CHALCOMORACIN CHOLINE-THEOPHYLLINATE CI-1018 CI-931 CILOMILAST CILOSTAZOL CIPAMFYLLINE CK-2130 CL-06A CL-42A CL-68A CL-860201 CP-248 CP-461 CP-77059 CYCLOMORUSIN D-22888 D-4030 DA-8159 DC-TA-46 DIHYDROPAPAVERINE DIPYRIDAMOLE DN-9693 DPN-205-734 E-4010 E-4021 EMD-57033 EMD-57439 ENOXIMONE FENOXIMONE GRISEOLATE-A GS-389 GW-3600 GYKI-52843 HCL-31-D HFV-1017-C ICI-118233 ICI-153110 ICI-58301 ICI-61129 ICI-63197 IMAZODAN ISOFRAXIDIN K-259-2 KF-17625 KF-19514 KS-501 KS-502 KS-504A KS-504B KS-504D KS-504E KS-505A KS-619-1 KURARIDIN KURARINONE KUSHENOL-B KUSHENOL-E KUSHENOL-H KUWANON-C KUWANON-E KUWANON-G KUWANON-H KUWANON-J L-0066 L-686398 L-826141 LEVOSIMENDAN LIXAZINONE LP-805 LY-186126 MEP-1 MERIBENDAN MILRINONE MIMAX MORACHALCONE-A MORUSIN MULBERROFURAN-J MY-5445 N-3601 NITRAQUAZONE NOR-KURARINONE NSP-804 NSP-805 OPC-13135 OPC-3911 ORG-20241 ORG-20494 ORG-9935 PAB-110 PAB-12 PAB-13 PAB-23 PAB-30 PAB-40 PDE-I PDE-II PINORESINOL PIROXIMONE PS-990 PV-2 R-80122 RA-642 REN-1053 RO-15-2041 RO-20-1724 RO-20-2926 ROFLUMILAST RP-73401 RS-1893 RS-25344 RX-RA-69 RX-RA-85 RX-RE-92 S-9795 SANGGENON-B SANGGENON-C SANGGENON-D SB-207499 SC-2964 SCA-41 SCA-44 SCH-351591 SCH-365351 SCH-51866 SCH-59498 SEQUOIAFLAVONE SH-869 SIGUAZODAN SILDENAFIL SKF-94120 SKF-96231 SQ-20006 SQ-65442 SR-24870 SURFACTIN T-1032 T-440 TADALAFIL THEOPHYLLINE

Derwent Drug File 1205 Thesaurus THEOPHYLLINE-LYSINE THEOPHYLLINE-SODIUM-= ANISATE THEOPHYLLINE-SODIUM-= GLYCINATE THIOCAFFEINE-6 THIOTHEOPHYLLINE-6 TIBENELAST TOLAFENTRINE TREQUINSIN TZC-5665 UK-14275 UK-1745 UK-343664 VARDENAFIL VK-744 VK-774 WAY-PDA-641 XT-611 Y-590 ZAPRINAST ZARDAVERINE ZSY-27 PHOSPHOLIPASE-INHIBITORS BILOBALIDE BMS-181162 CACOSPONGIONOLIDE CURCUMIN D-609 FPL-67047-XX FUROSEMIDE MANOALIDE MASTICADIENONATE MEPACRINE MORELLOFLAVONE NEOMYCIN PARAOXON PINITOL PMS-832 SB-203347 SB-435495 SURAMIN U-73122 VARIABILIN WA-8242-A1 WA-8242-A2 WA-8242-B PHOSPHOLIPID CARDIOLIPIN PLASMALOGEN PHOTOCHEM. PHOTOAFFINITY-LABELED PHOTOLYSIS PHOTOSYNTH. HILL-REACTION PHYS.CHEM. SURFACE-TENSION PHYSICOTHERAPY BALNEOTHERAPY CHIROPRACTIC GYMNASTICS MASSAGE PHYTONCIDES AKUAMMIDINE ALLICIN ALLIXIN ANTOFINE ARENARIN ARGENTATIN-A ARISTOLOCHATE-I ARISTOLOCHATE-IA ARISTOLOCHATE-II ASEBOGENIN ATHEROSPERMININE ATHEROSPERMININE-N-OXIDE BAKUCHIOL BASIL-OIL BATATASIN-III BIDWILLON-A BISNORDIHYDROTOXIFERINE BOUVARDIN BROUSSOCHALCONE-A BUDDLEDIN-A BUDMUNCHIAMINE-A CARDAMONIN CHONEMORPHINE CLAUSSEQUINONE CRINAMINE CRINITOL CRYPTOTANSHINONE CURINE CYCLOEUDESMOL CYCLOVIROBUXEINE-F CYPERONE-ALPHA DAPHNODORIN-B DEHYDROFALCARINDIOL DENTATIN-A DERMOCEPT DIALLYL-TETRASULFIDE DIALLYL-TRISULFIDE DICRANENONE-A DIHYDROTANSHINONE-I DIMETHOXYBENZO= QUINONE-2,5 DIOSQUINONE DIPLOICIN DRIMENINE DRUMMONDIN-A DRUMMONDIN-B DRUMMONDIN-C DRUMMONDIN-F DYSOXYSULFONE ENMEIN EPIPOLYGODIAL EUCHRESTAFLAVANONE-A EUROPINE FALCARINDIOL FORSYTHIASIDE FRONTALIN FULVOPLUMIERIN GARLIC-EXTRACT GIRINIMBINE GLABRENE GLABRIDIN GLYCYCOUMARIN HALIMEDATRIAL HALLERIDONE HELENIN HINESOL HISPANOLONE HUMULONE HYDROXYACTEOSIDE-BETA HYDROXYDERRICIN-4 HYPERFORIN ISOISOVELLERAL ISOXANTHOHUMOL JULIFLORINE JUNCUSOL KANUKA-OIL KOBOPHENOL-A KOLAVENOL LANIGEROL LASIOCARPINE-N-OXIDE LICOCHALCONE-A LICOCHALCONE-B LICOCOUMARONE LIRIODENINE LONGIKAURIN-A LONGIKAURIN-B LUPULONE MAACKIAIN MACROCARPAL-A MACROCARPAL-B MACROCARPAL-C MACROCARPAL-D MACROCARPAL-E MACROCARPAL-G MACROCARPAL-H MALABARICONE-C MALYNGOLIDE MANGIOSTIN MANUKA-OIL MARCHANTIN-A MELIACIN METHYLACRYLYLPLENOLIN-= 6-O METHYLGALANGIN-3-O METHYLGLABRIDIN-4+-O MICROSTEGIOL MIYABENOL-C MONOGAGAINE MYRTUCOMMULONE-A MYRTUCOMMULONE-B NEOCRYPTOLEPINE NIAOULI-OIL NORDENTATIN OBOVATOL OCHROLIFURANINE-A OLEANOLATE-ACETATE ONOPORDOPICRIN PAEPALANTINE PECTINOLIDE PETALOSTEMUMOL PETALOSTEMUMOL-G PHAEANTHARINE PHENYLHEPTATRIYNE PICLAVINE-A1 PICLAVINE-A2 PIPERADUNCIN-B PISATIN PISIFERATE PLUMERICIN POLYGODIAL POLYPHENON-60 PRENYLNARINGENIN-8 PROTOANEMONIN PROTOLICHESTERATE PSEUDOLARATE-B PSEUDOLARATE-C RAMONTOSIDE RAPANONE RUTAEVIN SALVIN SAMPANGINE SANGUINARINE SANTALOL SCOULERINE SHINJUDILACTONE SIGMOIDIN-A SIGMOIDIN-B SOPHORAFLAVONE-G STRYCHNOPENTAMINE SUGIOL SUSPENSASIDE TABULIN TANACHIN TELEKIN TETRAHYDROSECAMINE TETRANDRINE THIARUBRINE-A THUJAPLICIN-BETA THUNBERGINOL-A THUNBERGINOL-B THUNBERGINOL-F TOMATINE

1206 APPENDIX D TRICHOSETIN TRICOLORIN-A TULIPALIN-A TYLOPHORINIDINE UMBELLIFERONE UMBROSONE UNCINATONE USAMBARENSINE USAMBARINE USNATE UVARETIN VIOLACEIN VIRGAUREASAPONIN-1 VIRGAUREASAPONIN-2 WOODFORDIN-A WOODFORDIN-C WYERONE XANTHATIN XANTHOANGELOL XANTHOCHYMOL XANTHOHUMOL XANTHOXYLIN YOMOGIARTEMIN ZOSTERIN PHYTOTOXINS AMANITIN AMANITIN-ALPHA AMANITIN-BETA CICUTOXIN COTYLEDOSIDE CROTON-OIL CYCASIN DEMETHYLPHALLOIN EUROPINE FRAXINELLONE FUSICOCCIN-A GOSSYPOL GOSSYPOL-ACETATE HOMOLYCORINE HYMENOXON HYPOGLYCIN-A HYPOGLYCIN-B ICI-D-0490 INOPHYLLOLIDE LASIOCARPINE-N-OXIDE LOLITREM-B LYONIOL-A LYONIOL-D MEZEREIN MONOCROTALINE NGAIONE PHALLOIDIN PHALLOIN PHASIN PHYTAGGLUTININ PHYTOHEMAGGLUTININ PICROTOXININ POKEWEED-MITOGEN PTAQUILOSIDE RADICININ RICIN RICIN-A-CHAIN RICIN-A-CHAIN-= DEGLYCOSYLATED RICIN-B-CHAIN RICIN-BLOCKED SAPORIN STEMPHONE TAXINE-II TRICHOKIRIN VISCOTOXIN VISCOTOXIN-A2 VISCOTOXIN-A3 VISCOTOXIN-B PICORNAVIRUS COXSACKIE-VIRUS ECBO-VIRUS ECHO-VIRUS EMC-VIRUS ENCEPHALOMYELITIS-VIRUS ENTEROVIRUS ERC-VIRUS MENGO-VIRUS POLIOMYELITIS-VIRUS RHINO-VIRUS SMEDI-VIRUS TESCHEN-DISEASE-VIRUS PIGMENTATION DYSCHROMIA HYPERCHROMATISM HYPERPIGMENTATION HYPOPIGMENTATION LENTIGINOSIS LEUKODERMA LIPOFUSCINOSIS MELANODERMA MELANONYCHIA MELASMA VITILIGO PITUITARY PARS-INTERMEDIA PITUITARY-DISEASE ACROMEGALY AHUMADA-DEL-CASTILLO-= SYNDROME ARGONZ-DEL-CASTILLO-= SYNDROME CHIARI-FROMMEL-= SYNDROME DIAB.INSIP. DWARFISM dwarfism,pituitary HYPERPROLACTINEMIA hypophyseal-dwarfism hypophyseal-gigantism HYPOPHYSITIS HYPOPITUITARISM HYPOPROLACTINEMIA KALLMANN-SYNDROME launois-syndrome lorain-levi-syndrome NELSON-SYNDROME PANHYPOPITUITARISM pituitary-dwarfism postpartum-= panhypopituitarism RENON-DELILLE-SYNDROME sheehan-syndrome SOMATOTROPINOMA WERMER-SYNDROME PITUITARY-HORMONE ACTH-AGONIST GONADOTROPIN INTERMEDIN-AGONIST OXYTOCIN-AGONIST PROLACTIN-AGONIST SOMATOTROPIN-AGONIST THYROTROPIN-AGONIST VASOPRESSIN-AGONIST PITUITARY-HORMONE-METAB. GONADOTROPIN-METAB. PITUITARY-HORMONES ACTH ACTH-1-10 ACTH-1-13 ACTH-1-13-AMIDE ACTH-1-14 ACTH-1-16 ACTH-1-16-AMIDE ACTH-1-18 ACTH-1-4 ACTH-11-24 ACTH-4-10 ACTH-4-10,7-D-PHE ACTH-4-11 ACTH-4-7 ACTH-5-10 ACTH-5-24 ACTH-6-9 ACTH-7-24 ACTH-7-38 ACTH-AGONISTS ACTH-CATTLE ACTH-HUMAN ACTH-PIG-A ACTH-PIG-BETA ACTH-SHEEP ALSACTIDE ANTOCIN-II ARGIPRESSIN ARGIPRESSIN-1-8 ARGIPRESSIN-VAL-4 ARGIPRESTOCIN BA-44680 BETA-CELL-TROPIN CARBETOCIN CARGUTOCIN CLIP CODACTIDE COHERIN DEMOXYTOCIN DESMOPRESSIN DICARBAOXYTOCIN EBIRATIDE FELYPRESSIN FSH FSH-ALPHA FSH-BETA FSH-CATTLE FSH-HORSE FSH-HUMAN FSH-PIG FSH-RAT FSH-SHEEP GIRACTIDE GLUMIPRESSIN GLUMITOCIN GONADOTROPINS HHG HP-466 HYPOPHYSIN ICSH ICSH-BETA ICSH-CATTLE ICSH-HORSE ICSH-HUMAN ICSH-PIG ICSH-SHEEP INTERMEDIN INTERMEDIN,4-NLE-7-D-PHE INTERMEDIN-AGONISTS INTERMEDIN-ALPHA INTERMEDIN-BETA INTERMEDIN-BETA-CATTLE INTERMEDIN-BETA-HORSE INTERMEDIN-BETA-HUMAN INTERMEDIN-BETA-MONKEY INTERMEDIN-BETA-PIG INTERMEDIN-GAMMA INTERMEDIN-GAMMA-3 ISOTOCIN L-163191 LIPOTROPIN LIPOTROPIN-BETA LIPOTROPIN-BETA-HUMAN

Derwent Drug File 1207 Thesaurus LYPRESSIN MESOTOCIN NACARTOCIN NC-1900 NORLEUSACTIDE ORG-2766 ORG-5667 ORNIPRESSIN OXYPRESSIN OXYTOCIN OXYTOCIN-1-8 OXYTOCIN-AGONISTS PITUITRIN PRESSINAMIDE PRESSINOATE PROLACTIN PROLACTIN-AGONISTS PROLACTIN-CATTLE PROLACTIN-HUMAN PROLACTIN-PIG PROLACTIN-RAT PROLACTIN-SHEEP SEMAX SERACTIDE SOMATOTROPIN SOMATOTROPIN-31-44 SOMATOTROPIN-77-107 SOMATOTROPIN-AGONISTS SOMATOTROPIN-CATTLE SOMATOTROPIN-DE-MET SOMATOTROPIN-FOWL SOMATOTROPIN-HUMAN SOMATOTROPIN-METHIONYL SOMATOTROPIN-PIG SOMATOTROPIN-RAT SOMATOTROPIN-SHEEP SOMATOTROPIN-TROUT SOMATOTROPIN-TURKEY SOMATREM SOMAVUBOVE SOMETRIBOVE SOMETRIPOR SOMIDOBOVE TERLIPRESSIN TETRACOSACTIDE TGS-34 THYROTROPIN THYROTROPIN-AGONISTS THYROTROPIN-CATTLE THYROTROPIN-HUMAN THYROTROPIN-RAT TOCINAMIDE TOCINOATE TOSACTIDE TRICOSACTIDE VASOPRESSIN VASOPRESSIN-AGONISTS PLACENTA CHORION TROPHOBLAST UMBILICAL-CORD PLANT-GROWTH-FACTORS ABSCISATE BENZYLADENINE CYTOKININ GIBBERELLATE GIBBERELLIN INDOLEACETATE INDOLEBUTYRATE KINETIN MEFLUIDIDE PLANT-SUBSTANCE CASCARA GINSENG UROL PLASMA-PROTEIN ALPHA-1-ACID-= GLYCOPROTEIN ALPHA-1-= ANTICHYMOTRYPSIN ALPHA-1-ANTITRYPSIN ALPHA-1-PROTEASE-= INHIBITOR ALPHA-2-ANTIPLASMIN ALPHA-2-GLYCOPROTEIN ALPHA-2-MACROGLOBULIN ANTITRYPSIN APOPROTEIN-A APOPROTEIN-AI (endogenous) APOPROTEIN-AII APOPROTEIN-B APOPROTEIN-B-100 APOPROTEIN-C APOPROTEIN-CII APOPROTEIN-CIII APOPROTEIN-D (endogenous) APOPROTEIN-E BETA-2-MICROGLOBULIN COLECALCIFEROL-BINDING-= GLOBULIN HISTIDINE-RICH-= GLYCOPROTEIN PREALBUMIN PREGNANT-ZONE-PROTEIN PROTEIN-C (Endogenous) PROTEIN-S (Endogenous) RETINOATE-BINDING-PROTEIN RETINOL-BINDING-PROTEIN SEX-HORMONE-BINDING-= GLOBULIN SP-1 THYROXINE-BINDING-= GLOBULIN THYROXINE-BINDING-= PREALBUMIN PLASMACYTOMA MOPC-CELL MOPC173-CELL TEPC15-CELL PLASTICIZER DIETHYL-PHTHALATE OCTICIZER PLATELET THROMBOPOIESIS PNEUMONIA LEGIONNAIRE-DISEASE PNEUMOPATHY allergic-alveolitis ALVEOLITIS ASBESTOSIS aspiration-pneumonitis ASTHMA ATELECTASIS AYERZA-SYNDROME bronchial-pneumonia BRONCHIECTASIS BRONCHITIS BRONCHOMALACIA BRONCHORREA BRONCHOSPASM caplans-syndrome carcinoma, lung CAVITATION ceelen-gellerstedt-syndrome CYSTIC-FIBROSIS diffuse-interstitial-= pulmonary-fibrosis EATON-LAMBERT-SYNDROME EMPHYSEMA EMPYEMA eosinophilic-pneumonitis ess.pulmonary-hemosiderosis farmers-lung GOODPASTURE-SYNDROME hamman-rich-syndrome HYDROPNEUMOTHORAX IBR INFLUENZA KARTAGENER-SYNDROME LARYNGOTRACHEOBRONCHITIS LEGIONNAIRE-DISEASE LEITNER-SYNDROME LEWIS-LUNG-CARCINOMA loeffler-syndrome loehr-kindberg-syndrome lung-carcinoma maedi mendelson-syndrome OCULO-RESPIRATORY-= SYNDROME PANCOAST-SYNDROME PARAINFLUENZA PERTUSSIS pleural-edema PLEURISY PLEUROPERICARDITIS PLEUROPNEUMONIA PNEUMOCONIOSIS PNEUMONIA PNEUMONITIS PRRS PULMONARY-= ADENOMATOSIS pulmonary-edema pulmonary-embolism pulmonary-eosinophilia-= syndrome pulmonary-eosinophilic-= infiltration PULMONARY-FIBROSIS pulmonary-proteinosis PYOPNEUMOTHORAX RESPIRAT.DISTRESS-= SYNDROME rheumatic-pneumoconiosis RHINOPNEUMONITIS rosen-castleman-liebow-= syndrome SHAVER-SYNDROME SHIPPING-FEVER SIDEROSIS SILICOSIS TRACHEITIS TRACHEOBRONCHITIS POLYPOSIS GARDNER-SYNDROME PORPHYRIA COPROPORPHYRIA PORPHYRIA-CUTANEA-TARDA PROTOPORPHYRIA POTASSIUM-ANTAGONISTS NIFEKALANT POTASSIUM-CHANNELRECEPTOR HERG-CHANNEL POTATO SWEET-POTATO POXVIRUS CAMELPOX-VIRUS COWPOX-VIRUS LUMPY-SKIN-DISEASE-VIRUS

1208 APPENDIX D MOLLUSCUM-= CONTAGIOSUM-VIRUS MOUSEPOX-VIRUS MYXOMATOSIS-VIRUS ORF-VIRUS PAPULAR-STOMATITIS-VIRUS PIGEONPOX-VIRUS PIGPOX-VIRUS PSEUDO-COWPOX-VIRUS SMALLPOX-VIRUS VACCINIA-VIRUS PPAR-AGONIST PPAR-GAMMA-AGONIST PPAR-AGONISTS A-320454 AZ-242 DRF-2725 FARGLITAZAR GW-0072 GW-1929 GW-347845-X GW-409544 GW-510516 GW-7647 GW-7845 L-165041 L-805645 PHYTANATE ROSIGLITAZONE PPAR-ANTAGONISTS BISPHENOL-A-DIGLYCIDYL-= ETHER GW-0072 PGJ2-DEOXY-15-DELTA-12,14 PRESERVATION DEEP-FREEZING PROGESTOGEN-ANTAGONISTS DILAPAN HRP-2000 LG-100127 LILOPRISTONE MIFEPRISTONE NORETHISTERONE-OXIME-3 ONAPRISTONE ORG-31376 ORG-31710 RU-42698 RU-42698 ZK-112993 ZK-115716 ZK-136799 PROGESTOGENS ACETOMEPREGENOL ALGESTONE ALGESTONE-ACETONIDE ALGESTONE-ACETOPHENIDE ALLYLESTRENOL ALTRENOGEST AMADINONE AMADINONE-ACETATE ANAGESTONE ANAGESTONE-ACETATE BL-141 CHLORMADINOL-ACETATE CHLORMADINONE CHLORMADINONE-ACETATE CHLORSUPERLUTIN CINGESTOL CISMADINONE CISMADINONE-ACETATE CLOGESTONE CLOGESTONE-ACETATE CLOMEGESTONE CLOMEGESTONE-ACETATE DELMADINONE DELMADINONE-ACETATE DEMEGESTONE DESOGESTREL DEXTRONORGESTREL DIENOGEST DIHYDROPROGESTERONE-= 20-ALPHA DIHYDROPROGESTERONE-= 3-ALPHA DIHYDROPROGESTERONE-= 5-ALPHA DIMETHISTERONE DU-41164 DU-41165 DYDROGESTERONE EDOGESTRONE ELTANOLONE EPIPREGNANOLONE-3 ETHISTERONE ETHYNERONE ETYNODIOL FLUGESTONE-ACETATE FLUMEDROXONE FLUMEDROXONE-ACETATE GESTACLONE GESTADIENOL GESTODENE GESTONORONE-CAPROATE GR2-1159 HALOPROGESTERONE HYDROMADINONE HYDROMADINONE-ACETATE HYDROXYMETHYL= HISTERONE-2 HYDROXYPROGESTERONE HYDROXYPROGESTERONE-= 11-ALPHA HYDROXYPROGESTERONE-= 11-BETA HYDROXYPROGESTERONE-= ACETATE HYDROXYPROGESTERONE-= CAPROATE HYDROXYPROGESTERONE-= HEPTANOATE KETONORGESTIMATE-3 LEVONORGESTREL LEVONORGESTREL-ACETATE LEVONORGESTREL-= BUTYRATE LEVONORGESTREL-= CAPROATE LEVONORGESTREL-= CYCLOBUTANOATE LEVONORGESTREL-= CYCLOHEXANOATE LEVONORGESTREL-= CYCLOPENTANOATE LEVONORGESTREL-= CYCLOPROPANOATE LEVONORGESTREL-= PENTANOATE LEVONORGESTREL-= PROPIONATE LG-100128 LG-120746 LYNESTRENOL MEDROGESTONE MEDROXYPROGESTERONE MEDROXYPROGESTERONE-= ACETATE MEGESTROL MEGESTROL-ACETATE MELENGESTROL MELENGESTROL-ACETATE MEPREGNOL-ACETATE MEPREGNOL-DIACETATE METHYLENEANDROSTENE= DIONE-6 METHYLENE= PROGESTERONE-6 METHYLESTRENOLONE METHYLPROGESTERONE-= 16-ALPHA METYNODIOL-DIACETATE NOMEGESTROL NOMEGESTROL-ACETATE NORELGESTROMIN NORETHISTERONE NORETHISTERONE-ACETATE NORETHISTERONE-= ACETATE-OXIME NORETHISTERONE-BENZOATE NORETHISTERONE-= ENANTHATE NORETHISTERONE-= PHENYLACETATE NORETYNODREL NORGESTERONE NORGESTIMATE NORGESTOMET NORGESTREL NORGESTREL-ACETATE NORGESTREL-OXIME NORGESTRIENONE NORVINISTERONE ORG-2058 ORG-30659 ORG-OH-06 OXODESOGESTREL-3 OXOGESTONE OXOLVEN PENTAGESTRONE PENTAGESTRONE-ACETATE PREGNANEDIOL PREGNANEDIONE PROGESTERONE PROLIGESTONE PROMEGESTONE QUINGESTANOL QUINGESTANOL-ACETATE QUINGESTRONE RENANOLONE RETROPROGESTAGEN RTI-3021-020 RU-25253 RU-3097 SANDOZ-45249 SH-D-510 ST-1435 STS-737 TIGESTOL TRENGESTONE TRIMEGESTONE TX-045 TZP-4238 WY-4355 ZK-30595 PROLACTIN-AGONISTS PROLACTIN PROLACTIN-CATTLE PROLACTIN-HUMAN PROLACTIN-PIG PROLACTIN-RAT PROLACTIN-SHEEP PROLACTIN-ANTAGONISTS 201-403 6605-VUFB BAM-1110 BROMOCRIPTINE CABERGOLINE CGP-19984 DCN-203-922

Derwent Drug File 1209 Thesaurus DEPRENON DISULERGINE DOCARPAMINE DOPAMINE ETISULERGINE FCE-27395 HA-114 HA-117 HA-118 HACHIMIJIOGAN LERGOTRILE MASTODYNON MERGOCRIPTINE MESULERGINE PRAMIPEXOLE PROLACTIN-HUMAN-G129R PROTERGURIDE QUINAGOLIDE TERGURIDE VUFB-10726 PROLACTOLIBERIN-AGONISTS PROLACTOLIBERIN PROPELLANT DICHLORODIFLUOROMETHANE FREON-113 FREON-114 FREON-21 TRICHLOROFLUOROMETHANE PROSTACYCLIN-AGONISTS 15-AU-81 ATAPROST BERAPROST BMY-42393 BUTAPROST BW-245C CARBACYCLIN CG-4303 CICAPROST CIPROSTENE CS-570 CU-23 CU-602 EMD-42501 EMD-46335 EP-035 EP-157 EPTALOPROST FCE-21258 FCE-22509 ILOPROST ISOCARBACYCLIN ISOCARBACYCLIN-METHYL-= ESTER KETOPROSTACYCLIN-7 KETOPROSTACYCLIN-7 = EPHEDRINE KP-10614 METHYLCARBACYCLIN-9-= BETA METHYLENEISOCARBA= CYCLIN-5,5 MM-706 NAXAPROSTENE NILEPROST ONO-AP-227 ONO-AP-324 ONO-AP-437 OP-2507 PGE1-KETO-6 PGI1 PGI1-BETA-6 PGI3 PIMILPROST PROSTACYCLIN PROSTACYCLIN-METHYL-= ESTER RS-93427 RS-953 SC-39902 SM-10906 TAPROSTENE TEI-1324 TEI-3356 TEI-9063 TILSUPROST TRY-200 U-68215 UT-15 ZK-36375 PROSTAGLANDIN PROSTACYCLIN-AGONIST THROMBOXANE-AGONIST PROSTAGLANDIN-ANTAGONIST CYCLOOXYGENASE-1-= INHIBITOR CYCLOOXYGENASE-2-= INHIBITOR CYCLOOXYGENASE-= INHIBITOR THROMBOXANE-= ANTAGONIST PROSTAGLANDINANTAGONISTS ACECLOFENAC AF-2259 AGNUSIDE AJULEMATE ALCLOFENAC AMENTOFLAVONE AMPIROXICAM AMTOLMETIN GUACIL APYRAMIDE ASPIRIN AURANOFIN AZAPROPAZONE AZAPROSTANOATE-13 BDH-7538 BENDAZAC BENDAZAC-LYSINE-SALT BENORILATE BENOXAPROFEN BENZOFENAC BENZOFUROCAINE BF-389 BI-RM-270 BM-500 BM-519 BM-567 BM-573 BMY-30094 BRL-10720 BROMFENAC BROUSSOAURONE-A BROUSSOFLAVONOL-F BUCLOXATE BUDDLEDIN-A BUFEXAMAC BW-540C BW-A868C CANNFLAVIN-A CARPROFEN CBS-1108 CBS-113A CENTAUREIDIN CGP-47969-A CGS-11776 CHF-1194 CI-986 CICLOPROFEN CINNOPENTAZONE CL-28A CLIDANAC CLONIXIN CLOPIRAC CO-1828 CP-14304 CYCLOOXYGENASE-1-= INHIBITORS CYCLOOXYGENASE-2-= INHIBITORS CYCLOOXYGENASE-= INHIBITORS CYPERONE-ALPHA DAISAIKOTO DARBUFELONE DICLOFENAC DICLOFENAC HYDROXY= ETHYLPYRROLIDINE DIFLUMIDONE DIFLUNISAL DIFTALONE DIPHLORETIN-PHOSPHATE DITAZOLE DROXICAM E-5110 E-6080 E-6087 EMORFAZONE ENFENAMATE EPIAFZELECHIN EPIRIZOLE ESCULETIN ETODOLAC ETORICOXIB F-1067 FCE-22176 FELBINAC FENBUFEN FENCLOFENAC FENCLOZATE FENDOSAL FENFLUMIZOLE FENOPROFEN FEPRAZONE FERULOYLTYRAMINE-N FK-3311 FLOSULIDE FLUFENAMATE FLURBIPROFEN FLURBIPROFEN-ETHYL-ESTER FPL-62064 FR-122047 FR-123826 FR-140423 FUREGRELATE FUROBUFEN FUROFENAC GLYCITEIN GP-53633 GX-258 HAI-105 HCT-3012 HR-546 HSR-284 HYDROXYACECLOFENAC-4 IBUFENAC IBUPROFEN IBUPROFEN LYSINE INDOMETACIN INDOMETACIN MEGLUMINE INDOMETACIN-FARNESIL INDOPROFEN IRISOLIDON ISOXEPAC ISOXICAM JTE-522 KB-3022 KETOPROFEN KETOPROFEN LYSINE

1210 APPENDIX D KME-4 L-636499 L-640035 L-651392 L-651896 L-655240 L-657925 L-657926 L-745296 L-745337 L-746483 L-761066 L-768277 LAGASCATRIOL LG-82-4-00 LG-82-4-01 LICOFELONE LIGSTROSIDE LM-1228 LOXOPROFEN LUMIRACOXIB LY-178002 LY-256548 M-5011 MASTICADIENONATE MB-432 MECLOFENAMATE MEFENAMATE MELOXICAM METBUFEN METOXIBUTROPATE MF-TRICYCLIC MK-966 MOFEZOLAC N-0164 NABUMETONE NAFAZATROM NAPROXEN NB-431 NCX-4016 NCX-701 NEPAFENAC NEUTROPHIL-INHIBITORY-= FACTOR NICTINDOLE NIFLUMATE NIMESULIDE NITROACETYLSALICYLATE NORARTOCARPANONE NQ-Y-15 NS-398 ONO-3144 ONO-3708 ONO-8711 ONO-NT-012 OSTHENOL OXAGRELATE OXEPINAC OXYPHENBUTAZONE P-8977 PARADOL-8 PARECOXIB PC-88 PD-138387 PD-164387 PGV-20229 PHENYLBUTAZONE PHENYLBUTAZONE = PIPERAZINE PIMETACIN PINADOLINE PIROXICAM PIROXICAM-CINNAMATE PIRPROFEN POLYPHLORETIN-PHOSPHATE PRAVADOLINE PROCYANIDIN PROCYANIDIN-B2 PRODOLATE PROQUAZONE R-830 RHAPONTIGENIN RIDOGREL RO-22-4679 RO-3-1314 RO-3-1428 ROFECOXIB RU-29693 RU-43526 RUTECARPINE RWJ-63556 S-2474 S-6907 S35B SC-19220 SC-236 SC-299 SC-51089 SC-51234A SC-560 SC-57666 SC-58125 SC-58236 SC-58560 SCYPHOSTATIN SERATRODAST SKF-104493 SKF-105561 SKF-105809 SKF-106978 SKF-86002 SKF-86002-A2 SOPHORAFLAVONE-G SP-600125 SQ-28852 SUDOXICAM SULFINPYRAZONE SULINDAC SULINDAC-SULFIDE SULOTROBAN SUPROFEN T-614 TA-60 TECTORIDIN TENOXICAM TEPOXALIN THIELAVIN-A THIELAVIN-B THROMBOXANE-= ANTAGONISTS TIARAMIDE TILOMISOLE TINORIDINE TIOPINAC TOLMETIN TOLMETIN-GLYCINE-AMIDE TOMOXIPROLE TRICHODION TRIFENAGREL TRIFLUMIDATE TROPESIN TX-11027 TZI-615 U-2021 U-54874 UFENAMATE UK-141161 UK-147535 UR-8880 VALDECOXIB WITHAFASTUOSIN-E WY-47288 WY-48090 WY-49232 XU-745 Y-23023 YM-26734 YM-57158 Z-335 ZIDOMETACIN ZOLIPROFEN PROSTAGLANDIN-RECEPTOR PROSTACYCLIN-RECEPTOR PROSTAGLANDINS 15-AU-81 192C86 AE-1734 AGN-191976 AGN-192093 AH-13205 ALFAPROSTOL ALPROSTADIL ARBAPROSTIL AS-013 ATAPROST AY-16809 AY-20524 AY-21669 AY-21670 AY-22093 AY-23578 AY-23626 BERAPROST BMY-42393 BUTAPROST BW-245C CARBACYCLIN CARBOCYCLIC-= THROMBOXANE-A2 CARBOPROST CARBOPROST-METHYL CG-4303 CICAPROST CIPROSTENE CL-115129 CL-115574 CL-116147 CLOPROSTENOL CS-570 CU-23 CU-602 DEHYDROTHROMBOXANE-= B2-11 DELPROSTENATE DEPROSTIL DICALCIPHOR DIMOXAPROST DINORTHROMBOXANE-B2-2,3 DOXAPROST EMD-42501 EMD-46335 ENISOPROST ENPROSTIL EP-011 EP-031 EP-035 EP-109 EP-157 EP-171 EPTALOPROST ETIPROSTON FCE-20700 FCE-21258 FCE-22177 FCE-22509 FENPROSTALENE FLUNOPROST FLUPROSTENOL FROXIPROST GEMEPROST

Derwent Drug File 1211 Thesaurus GR-63799X I-BOP ICI-74205 ICI-79939 ICI-80205 ICI-86841 ILOPROST IOS-4074 IOS-4732 ISOCARBACYCLIN ISOCARBACYCLIN-METHYL-= ESTER KETOPROSTACYCLIN-7 KETOPROSTACYCLIN-7 = EPHEDRINE KP-10614 L-644122 LATANOPROST LEVUGLANDIN-D2 LEVUGLANDIN-E2 LIMAPROST LUPROSTIOL M+B-28767 METENEPROST METHYLCARBACYCLIN-9-= BETA METHYLENEISOCARBA= CYCLIN-5,5 MEXIPROSTIL MISOPROSTOL MISOPROSTOL-FREE-ACID MM-706 MR-256 MR-356 NAXAPROSTENE NEPP-11 NILEPROST NOCLOPROST OC-2186 OC-5181 OC-5186 ONO-8815-LY ONO-AE-1-259 ONO-AE-1-329 ONO-AE-248 ONO-AP-227 ONO-AP-324 ONO-AP-437 OP-1206 OP-2507 ORNOPROSTIL OXAPROSTYNOATE PENPROSTENE PGA PGA1 PGA1-DELTA-7 PGA1-DELTA-7-METHYL-= ESTER PGA1-DIMETHYL-16,16 PGA2 PGA2-DIMETHYL-16,16 PGA2-ISOPROPYL-ESTER PGB PGB1 PGB1-KETO-15 PGB2 PGBX PGC1 PGC2 PGD1 PGD2 PGD2-METHYL-ESTER PGD3 PGE PGE1-DELTA-17 PGE1-DEOXY-11 PGE1-DIHYDRO-13,14 PGE1-DIMETHYL-16,16 PGE1-DIMETHYL-16,16-= METHYL-ESTER PGE1-KETO-15 PGE1-KETO-15-DIHYDRO-= 13,14 PGE1-KETO-6 PGE1-METHYL-15 PGE1-METHYL-ESTER PGE2 PGE2-DEOXY-11 PGE2-DIMETHYL-16,16 PGE2-DIMETHYL-16,16-= METHYL-ESTER PGE2-KETO-15 PGE2-KETO-15-DIHYDRO-= 13,14 PGE2-METHYL-15-= METHYL-ESTER PGE2-METHYL-ESTER PGE2-TRIMETHYL-11,16,16 PGE3 PGF1 PGF1-ALPHA PGF1-ALPHA-KETO-6 PGF1-BETA PGF2 PGF2-ALPHA PGF2-ALPHA-DIMETHYL-= 16,16 PGF2-ALPHA-EPI-11 PGF2-ALPHA-EPI-8 PGF2-ALPHA-ISOPROPYL-= ESTER PGF2-ALPHA-KETO-15 PGF2-ALPHA-KETO-15-= DIHYDRO-13,14 PGF2-ALPHA-METHYL-ESTER PGF2-BETA PGF2-BETA-METHYL-ESTER PGF3-ALPHA PGG1 PGG2 PGH1 PGH2 PGH2-AZO-9,11 PGH3 PGI1 PGI1-BETA-6 PGI3 PGJ2 PGJ2-DELTA-12 PGJ2-DEOXY-15-DELTA-12,14 PIMILPROST PIRIPROST PROSTACYCLIN PROSTACYCLIN-AGONISTS PROSTACYCLIN-METHYL-= ESTER PROSTALENE PROSTANOATE PROSTIANOL RIOPROSTIL RO-22-1327 RO-22-6923 ROSAPROSTOL RS-86505-007 RS-86505-008 RS-86812-007 RS-86812-008 RS-93427 RS-953 SC-30249 SC-36067 SC-39902 SC-46275 SM-10906 SQ-26655 STA-2 SU-840 SULPROSTONE TAPROSTENE TEI-0303 TEI-1324 TEI-3356 TEI-5178 TEI-9063 TEI-9826 TFC-612 THROMBOXANE-A1 THROMBOXANE-A2 THROMBOXANE-AGONISTS THROMBOXANE-B1 THROMBOXANE-B2 TIAPROST TILSUPROST TIPROSTANIDE TOK-4528 TRIMOPROSTIL TRY-200 U-38833 U-43728 U-44069 U-46619 U-47473 U-56467 U-62840 U-68215 UNOPROSTONE UNOPROSTONE-= ISOPROPYLESTER UT-15 VIPROSTOL WY-17186 WY-18189 WY-19068 WY-19110 WY-40659 ZK-111298 ZK-112151 ZK-115886 ZK-118182 ZK-36375 ZK-71677 PROSTATE DUNNING-R3327H PROSTATE-DISEASE DUNNING-R3327H PROSTATE-HYPERPLASIA PROSTATE-HYPERTROPHY PROSTATITIS PROTEIN GLOBIN GLOBULIN MACROGLOBULIN MICROGLOBULIN NUCLEOPROTEIN PROPERDIN PROTEIN-KINASE-C-INHIBITORS AG-1007 AG-1024 AG-1034 AG-1049 AG-126 AG-1478 AG-17 AG-528 AG-879 AG-879 AMILORIDE BALANOL

1212 APPENDIX D BATZELLADINE-A BATZELLADINE-B CEP-1347 CGP-41251 CGP-42700 CGP-60474 CISPLATIN CKI-7 DIHYDROSPHINGOSINETHREO FUROSEMIDE FUROSEMIDE GOE-6976 GOE-6983 GOE-7874 H-7 H-9 HIRSUTANONOL HYDROXYTAMOXIFEN ISIS-3521 JM-34 KN-93 L-86-8275 LY-333531 MDL-27032 MITOXANTRONE MLR-52 NA-382 NSC-115290 NSC-639366 OLOMOUCINE OREGONIN OXOSTAUROSPORINE-7 P-9782 PKC-412 POLYMYXIN-B PROCYANIDIN-B2-DIGALLATE PROSTRATIN RO-31-8830 RO-32-0432 SPC-100270 SPC-100271 STAUROSPORINE TAMOXIFEN TMB-8 TRICOLORIN-A TX-1123 VERAPAMIL PROTEIN-METAB.DISORDER AMYLOIDOSIS ANDRADE-SYNDROME DYSPROTEINEMIA HYPOPROTEINEMIA MICROALBUMINURIA MYOGLOBINURIA PERIODIC-DISEASE PROTEINOSIS PROTEINURIA pulmonary-proteinosis rosen-castleman-liebow-= syndrome PROTOZOACIDE AMEBICIDE PROTOZOACIDES 102-198 150C47 225-144 261-115 98-202 A-9145C ABRUQUINONE-A ABT-773 ACEDAPSONE ACETARSOL ACONITATE-TRANS ACRANIL ACRONYCINE AKLOMIDE ALLOPURINOL-RIBOSIDE AM-92008 AMARIIN AMBROSIN AMEBICIDES AMICARBALIDE AMINAZOLINE AMINITROZOLE AMINOACRIQUINE AMINOQUINOL AMODIAQUINE AMOPYROQUINE AMPROLIUM AMQUINATE ANDROGRAPHISIDE ANTIMONYLGLUCONATE = SODIUM APICIDIN APICIDIN-A APLASMOMYCIN ARSANILATE ARSANILATE SODIUM ARSTHINOL ARTEETHER ARTEETHER-BETA ARTEFLENE ARTEFLENE ARTEINCULTON ARTELINATE ARTEMETHER ARTEMISININ ARTESUNATE ASCOSFEROL ATALAPHILLIDINE ATALAPHILLININE ATOVAQUONE AZACRIN AZAINOSINE-8 AZANIDAZOLE AZOMYCIN AZURE-A AZURE-B BA-41799 BAMNIDAZOLE BAY-B-1694 BAYG-7183 BECLOTIAMINE BENZNIDAZOLE BENZOXAZOLINONE-2 BG-237 BG-289 BG-325 BG-374 BG-958 BIALAMICOL BIKAVERIN BISDEETHYLCHLOROQUINE BP-12231 BRINDOXIME BRL-50395 BRL-50523 BRL-50551 BRL-50702 BRL-50714 BRL-50715 BRL-50717 BRL-51136 BRL-51334 BRL-6231 BRUCEANTINOL BRUCEIN-A BRUCEIN-B BRUCEIN-C BRUCEIN-D BS-1-81 BTI-2286E BUPARVAQUONE BUQUINOLATE BUTAMIDINE BW-568C BW-58C BW-826C CAERULOMYCIN-A CALOTHRIXIN-A CARBARSONE CARBIDIUM CARNIDAZOLE CARYOPHYLLENE-ALPHA-= OXIDE CASPOFUNGIN CDRI-80-53 CDRI-87-209 CEPHAELINE CG-10248 CG-8935 CG-9442 CGP-33829-A CGP-35753-A CGP-39937-A CGP-40-215 CGP-40-215-A CHAMUVARETIN CHIMANINE-A CHIMANINE-B CHIMANINE-D CHINATIN CHLORBETAMIDE CHLORCYCLOGUANIL CHLOROQUINE CHLORPROGUANIL CHONEMORPHINE CINCHONAMINE CINCHONIDINE CINCHONINE CIPROQUINATE CITPRESSINE-I CITPRESSINE-II CITRACRIDONE-II CITRUSININE-I CL-64855 CLAMOXYQUINE CLAZURIL CLEFAMIDE CLOCIGUANIL CLOPIDOL CLOQUINATE CM-6606 CNI-H-0294 COCSOLINE CONESSINE CORYNANTHEIDINE CP-25415 CRL-81-31 CRL-81-42 CRL-85-221 CURINE CUSPARINE CYCLOGUANIL CYCLOGUANIL EMBONATE CYCLOLEUCINE CYMELARSAN DABEQUINE DB-289 DEAZAINOSINE-7 DEAZAINOSINE-9 DECOQUINATE DEETHYLAMODIAQUINE DEETHYLCHLOROQUINE DEHYDROBRUCEIN-A DEHYDROEMETINE DEHYDROTELOBINE-1,2 DEOXOARTEMISININ

Derwent Drug File 1213 Thesaurus DEOXYURIDINE-3+ DIAVERIDINE DIBROMPROPAMIDINE DICHLORQUINAZINE DIFETARSONE DIFORMYLDAPSONE DIHYDROARTEMISININ DIHYDRONEPLANOCIN-D DIHYDROQUININE DILOXANIDE DILOXANIDE-FUROATE DIMETHIALIUM DIMETRIDAZOLE DIMIDIUM DIMINAZENE DIMINAZENE-ACETURATE DINSED DIONCOPELTINE-A DIONCOPHYLLINE-B DIONCOPHYLLINE-C DIOSPYRIN DIOSPYROL DIPI DIUVARETIN ECHINATIN EFLORNITHINE EMETINE EMIMYCIN ENDOCHIN ENPIROLINE EPI-OLEANOLATE EPINIGERICIN ES-242-6 ES-242-8 ESPINTANOL ETHOPABATE ETOFAMIDE EURYCOMANOL FEBRIFUGINE FERRUGININ-B FEXINIDAZOLE FISTULARIN-3 FLOXACRINE FLUNIDAZOLE FLUORODEOXYINOSINE-3+ FLUOROMISONIDAZOLE FORMINITRAZOLE FORMYCIN-B-= MONOPHOSPHATE FORMYCIN-= MONOPHOSPHATE FORMYCIN-TRIPHOSPHATE FR-160 FTI-2153 FURAZOLIDONE GALLOCYANINE GEDUNIN GENTIOPICROSIDE GILLETINE GLAUCARUBIN GLYCARBYLAMIDE GLYCOBIARSOL GLYCOBISMINE-A GLYCOCITRINE-I GLYFOLINE GM-193663 GM-237354 GRANDISINE-I GRANDISINE-II GRANDISININE HAEMOSPORIDIN HALOFANTRINE HALOFUGINONE HEDERACOLCHISID-A1 HEDERACOLCHISIDE-A HEDERIN-BETA HEPTYLCHAPARRINONE-15-= BETA HEXAMIDINE HOMIDIUM BROMIDE HOMIDIUM CHLORIDE HORMINONE HYDROXYCHLOROQUINE HYDROXYCRYPTOLEPINE-11 HYDROXYMETRONIDAZOLE HYDROXYPIPERAQUINE HYDROXYPRIMAQUINE-5 HYDROXYQUININE-3 HYDROXYSTILBAMIDINE HYDROXYVERNOLIDE ICI-153066 ICI-3327 IMIDOCARB IMIDOCARB-DIPROPIONATE IMINOLANOSTEROL-24,25 IMOL-881 INSULARINE IODOAZOMYCIN-RIBOSIDE IPRONIDAZOLE IRAMINE ISOBRUCEINE-A ISOFEBRIFUGINE ISOLASALOCID-A ISOMETAMIDIUM CHLORIDE ISOMETRONIDAZOLE ISONOTHOLAENATE ISOPENTAQUINE ISOTRIUVARETIN K-11777 K-120 K-137 KISIMICIN KORUPENSAMINE-B KORUPENSAMINE-B KY-62 KYNOSTATIN-227 L-611744 L-634549 L-651582 L-652042 L-652069 L-6678 L-687781 L-688786 L-693989 L-733560 L-8580 L-8711 LAGOSIN LAPACHOL LAPINONE LASALOCID LASALOCID-A LASALOCID-B LASALOCID-C LASALOCID-D LASALOCID-E LICARIN-A LISSOCLINOTOXIN-A LONIDAMINE LUMEFANTRINE LY-303366 M+B-35769 M+B-39434 MAGAININ-1 MAGAININ-2 MAGAININ-A MAGAININ-B MAGAININ-G MAGAININ-H MANSONONE-F MAP-1987 MASTICADIENONATE MDL-19152 MDL-20828 MDL-26547 MDL-26752 MDL-27391 MDL-27693 MDL-27695 MDL-27700 MDL-27701 MDL-27994 MDL-28842 MDL-73811 MEFLOQUINE MEGLUMINE STIBONATE MELARSEN MELARSENOXIDE MELARSOMINE MEN-10706 MENOCTONE MEPACRINE METHYLCHLOROQUINE METHYLDINITROBENZAMIDE METHYLENE-VIOLET METHYLPRIMAQUINE-4 METRONIDAZOLE METRONIDAZOLE-BENZOATE METRONIDAZOLE-= PHOSPHATE METRONIDAZOLE-SUCCINATE MICONIDIN MIKS-10 MIKS-9 MISONIDAZOLE MK-436 MOXIPRAQUINE MOXNIDAZOLE MP-90 MSI-103 MSI-94 MT-81 MYRALACT NARDOSINONE NEOANDROGRAPHOLIDE NEOCRYPTOLEPINE NEQUINATE NEUROLENIN-B NEW-METHYLENE-BLUE NICARBAZIN NIFLURIDIDE NIFURATEL NIFURSEMIZONE NIFURSOL NIFURTIMOX NIMBOLIDE NIMORAZOLE NIRIDAZOLE NITARSONE NITHIAZIDE NITRAZOLE NITROMIDE NITROPHENIDE NITROQUINE NORACRONYCINE NSC-118203 NSC-125358 NSC-128189 NSC-211327 NSC-232965 NSC-235777 NSC-3077 NSC-330465 NSC-35843 NSC-402538 NYASOL OBAMEGINE OBIOPEPTIDE-1 ORNIDAZOLE P-1266 P-1995

1214 APPENDIX D P-536 PAMAQUINE PANIDAZOLE PARVAQUONE PENTAMIDINE PENTAQUINE PENTATROXANE PEROXYACHILIFOLIDE-ALPHA PHANQUINONE PHASEOLINONE PHENAMIDINE PHENARSONE-SULFOXYLATE PIPERAQUINE PIRINIDAZOLE PNEUMOCANDIN-A1 PNEUMOCANDIN-A2 PNEUMOCANDIN-A3 PNEUMOCANDIN-A4 PNEUMOCANDIN-B0 PNEUMOCANDIN-B2 PNEUMOCANDIN-C0 POLYBENZARSOL POLYHEXAMETHYLENE-= BIGUANIDE PREUSSOMERIN-E PREUSSOMERIN-F PREUSSOMERIN-G PREUSSOMERIN-H PREUSSOMERIN-I PRIMAQUINE PRIMIN PROGUANIL PROPIDIUM IODIDE PROQUINOLATE PS-15 PSEUDOBAPTIGENIN PURVALANOL-A PURVALANOL-B PYRIMETHAMINE PYRITIDIUM BROMIDE PYRONARIDINE QUINAPYRAMINE QUINDOLINE QUINFAMIDE QUINIDINONE QUINIFURIL QUININE QUININE-ETHYLCARBONATE QUINOCIDE QUINURONIUM RANALEXIN RAPANONE RC-12 RETUSIN RGW-806 RHODOQUINE RL-712 RO-11-8958 RO-15-0216 RO-19-9638 RO-41-3118 RO-47-0543 RO-47-7737 RO-47-9396 ROBENIDINE RONIDAZOLE ROXARSONE RUFIGALLOL RUGOSAL-A S-75-0400A SATRANIDAZOLE SB-37 SB-59 SECNIDAZOLE SENEGALENE SEPTICINE SERGEOLIDE SETAMYCIN SEVERIFOLINE SHIVA-1 SHIVA-10 SIMALIKALACTONE-D SKF-3301-A SN-10275 SN-12108 SN-6911 SPIROTRYPAN STEVALADIL STIBAMINE-GLUCOSIDE STIBOGLUCONATE SODIUM STIBOPHEN STIBOSAN STILBAMIDINE ISETIONATE STIRIMAZOLE STRYCHNOPENTAMINE SULAZURIL SULFAMOYLDAPSONE SULNIDAZOLE SURAMIN SURAMIN SODIUM SYMETINE TAFENOQUINE TAGITININ-C TAURINE-CHLORAMINE TEBUQUINE TECLOZAN TENONITROZOLE TETRAHYDROECHINO= CANDIN-B THALIFENDINE THALRUGOSINE THIODIHYDROOROTATE-6 THIOFORMYCIN-B TIABENDAZOLE TIAZURIL TINGENONE TINIDAZOLE TN-108 TN-109 TN-112 TN-121 TN-77 TN-78 TN-79 TN-80 TOLTRAZURIL TOSULUR TRICHOMONACID TRYPAN-RED UK-5099 UR-9825 UREA-STIBAMINE USAMBARENSINE USAMBARINE VERNOLIDE VIOLACEIN VISMIONE-A VISMIONE-B WR-106147 WR-122455 WR-15081 WR-158122 WR-159412 WR-165355 WR-172435 WR-175412 WR-177602 WR-178460 WR-181023 WR-182232 WR-182234 WR-182393 WR-183489 WR-184806 WR-188438 WR-190420 WR-194965 WR-199385 WR-199507 WR-199507 WR-199508 WR-212579 WR-216804 WR-224097 WR-225448 WR-226253 WR-242511 WR-243251 WR-250016 WR-250547 WR-250548 WR-30090 WR-3090 WR-33063 WR-40070 WR-49577 WR-5677 WR-5990 WR-6026 WR-6881 WR-93133 WR-9792 WR-99662 WS-5995A WS-5995B WS-5995C YINGZHAOSU-C ZK-28943 ZL-III-43-A PROTOZOON ACANTHAMOEBA AEGYPTIANELLA AMEBA BABESIA BALANTIDIUM BESNOITIA BLASTOCYSTIS CHILODONELLA CILIATA COLPODA COSTIA CRITHIDIA CRYPTOBIA CRYPTOCARYON CRYPTOSPORIDIUM CYCLOSPORA DIENTAMOEBA EIMERIA ENCEPHALITOZOON ENTAMOEBA ENTODINIUM EPIDINIUM GIARDIA GYMNODINIUM HAEMOPROTEUS HAMMONDIA HARTMANELLA HENNEGUYA HEPATOZOON HERPETEMONAS HERPETOMONAS HEXAMITA HISTOMONAS ICHTHYOPHTHIRIUS ISOSPORA ISOTRICHA LANKESTERELLA LEISHMANIA LEUKOCYTOZOON MALPIGHIELLA MASTIGOPHORA

Derwent Drug File 1215 Thesaurus MYXOBOLUS MYXOSOMA MYXOSPORIDIA NAEGLERIA NEOSPORA NOSEMA OODINIUM PARAMECIUM PLASMODIUM PNEUMOCYSTIS POLYPLASTRON SARCOCYSTIS SARCOSPORIDIUM SPORIDIUM SPOROZOA TETRAHYMENA THEILERIA TOXOPLASMA TRICHODINA TRICHOMONAS TRITRICHOMONAS TRYPANOSOMA PSEUDOHERMAPHRODITISM REIFENSTEIN-SYNDROME PSYCHOLOGY PSYCHOANALYSIS PSYCHOSEDATIVE NEUROLEPTIC TRANQUILIZER PSYCHOSEDATIVES 10184-CERM 106-689 1192-U-90 340125 450247 450304 450789 450790 4684-RP 52-522 709-W-92 A-23887 A-31472 A-37850 A-69024 A-80426 ABECARNIL ABT-418 AC-3579 ACAPRAZINE ACEPERONE ACEPROMAZINE ACEPROMETAZINE ACETOPHENAZINE AD-5423 ADATANSERIN ADINAZOLAM AEC AET AHR-14042 AHR-1709 AHR-1900 AL-1612 AL-449 ALENTEMOL ALIMEMAZINE ALOZAFONE ALPERTINE ALPIDEM ALPIROPRIDE ALPRAZOLAM AMBOCARB AMINOBECLAMIDE-PARA AMINOBENZONITRILE-PARA AMIPERONE AMISULPRIDE AMOXAPINE AMPEROZIDE AMPHENIDONE ANISOPERIDONE ANISOPIROL ANTALARMIN AP-159 AP-521 ARFENDAZAM AWD-131-138 AZ-21666 AZABUPERONE AZACYCLONOL AZAPERONE AZAQUINZOLE B-20991 BALAPERIDONE BARAKOL BATELAPINE BENACTYZINE BENPERIDOL BENTAZEPAM BENZINDOPYRINE BENZOCTAMINE BENZQUINAMIDE BIRIPERONE BMS-184111 BMY-14802 BMY-14802-1 BMY-20551 BMY-20661 BRL-20596 BRL-34778 BRL-46470 BRL-46470A BROMAZEPAM BROMOPRIDE BROMOSPIPERONE-PARA BROMPERIDOL BROMPERIDOL-DECANOATE BROTIZOLAM BTG-1501 BUCLIZINE BURAMATE BUSPIRONE BUTACLAMOL BUTAMOXANE BUTAPERAZINE BUTYLSYMPATON CAMAZEPAM CAMPIRONE CARBURAZEPAM CARFENAZINE CARPERONE CENTAZOLONE CENTPYRAQUIN CGP-49823 CGS-17867A CGS-20625 CGS-9896 CHLORDIAZEPOXIDE CHLORFENETHAZINE CHLORMEZANONE CHLOROSERPIDINE CHLORPHENESIN-= CARBAMATE CHLORPROETHAZINE CHLORPROMAZINE CHLORPROMAZINE-= METHIODIDE CHLORPROTHIXENE CI-1007 CI-905 CI-913 CI-936 CI-943 CICLOFENAZINE CICLOTIZOLAM CIDOXEPIN CINITAPRIDE CINOCTRAMIDE CINPERENE CINTRAMIDE CINUPERONE CIPRAZAFONE CIPROXIMIDE CITATEPINE CL-218872 CL-273547 CLAZOLAM CLEBOPRIDE CLOBAZAM CLOFLUMIDE CLOFLUPEROL CLOMACRAN CLOPENTHIXOL CLOPENTHIXOL-DECANOATE CLOPERIDONE CLOPIMOZIDE CLOPIPAZAN CLOPITHEPIN CLORAZEPATE CLOROPERONE CLOROTEPINE CLOTIAPINE CLOTIAZEPAM CLOTIXAMIDE CLOXATHIEPIN CLOXAZOLAM CLOXYPENDYL CLOZAPINE CO-134444 CORYTUBERINE CP-135807 CP-141938 CP-154526 CP-88059 CP-93393 CP-93393-1 CRA-1000 CRA-1001 CX-516 CYAMEMAZINE CYCLARBAMATE CYCLOBENZAPRINE CYCLOPREGNOL CYPRAZEPAM DAA-1097 DAA-1106 DECLENPERONE DELORAZEPAM DEMETHYLCLOBAZAM DEMETHYLDOXEPIN DEMETHYLFLUDIAZEPAM DEMETHYLNEMONAPRIDE-N DEMOXEPAM DESERPIDINE DETOMIDINE DEXCLAMOL DIAMIPHENE DIAZEPAM DICARBINE DICHLORMEZANONE DICHLORPROMAZINE DICLOMETIDE DIFENCLOXAZINE DIFLUANAZINE DIHYDROBENPERIDOL DIHYDROFENAZEPAM DIHYDROHONOKIOL-B DIHYDROMAGNOLOL DIHYDROTETRABENAZINE DIHYDROWISANINE

1216 APPENDIX D DIMELAZINE DIMEPROZAN DIPHOXAZIDE DIXYRAZINE DIZOCILPINE DO-897 DOKLOXYTHEPIN DOXEFAZEPAM DOXEPIN DROPERIDOL DTZ-323 DU-127090 DULOZAFONE DUP-734 E-0663 E3-54 ECTYLUREA ELENOSIDE ELFAZEPAM ELTOPRAZINE EMYLCAMATE ENCIPRAZINE ENCYPRATE ENPIPRAZOLE ERIZEPINE ESTAZOLAM ETAFENOXIN ETASULINE ETAZOLATE ETHOMOXANE ETIFOXINE ETIZOLAM ETODROXIZINE ETOPERIDONE ETYMEMAZINE EX-11-582A FENAPERONE FENAZEPAM FENHARMANE FENIBUT FENIMIDE FENMETRAMIDE FENOBAM FG-8205 FG-9202 FH-510 FLA-988 FLB-457 FLB-463 FLUANISONE FLUBEPRIDE FLUCIPRAZINE FLUDIAZEPAM FLUMEZAPINE FLUNITRAZEPAM FLUORESONE FLUOTHEPINE FLUOTRACEN FLUPENTIXOL FLUPENTIXOL-DECANOATE FLUPERLAPINE FLUPHENAZINE FLUPHENAZINE-DECANOATE FLUPHENAZINE-ENANTHATE FLUPIMAZINE FLUPRAZINE FLUSPIPERONE FLUSPIRILENE FLUTAZOLAM FLUTIZENOL FLUTOPRAZEPAM FLUTROLINE FOSAZEPAM FOSENAZIDE FR-33 FUROMAZINE G-365 GANAXOLONE GEPIRONE GEVOTROLINE GIDAZEPAM GINDARINE GIRISOPAM GLAZIOVINE GMC-1-169 GP-41299 GP-45795 GP-50302 GR-100679 GR-103691 GR-159897 GRAYANOTOXIN-III GRI-1665 GV-150013 GV-150013-X GVS-111 GYKI-22441 HALAZEPAM HALOPEMIDE HALOPERIDOL HALOPERIDOL-DECANOATE HOMOCHLORCYCLIZINE HOMOFENAZINE HP-236 HP-370 HPP HS-2314 HT-90-B HUF-2046 HYDAZEPAM HYDROXYALPRAZOLAM-= ALPHA HYDROXYBENZONITRILE-= PARA HYDROXYCAMAZEPAM HYDROXYFENAZEPAM-3 HYDROXYZINE ICI-190622 ICLAZEPAM ID-4708 ID-495-37 ILOPERIDONE IMICLOPAZINE IMIDOLINE IODOPROXYFAN IPROZILAMINE IPSAPIRONE IRAZEPINE IRFI-165 ISAMOLTAN ISOBUTACLAMOL ISOCLOTHIAPINE ISOFLOXYTHEPIN JL-13 KC-3756 KETAZOLAM KW-6002 L-663581 L-701324 L-741742 LEK-8829 LENPERONE LESOPITRON LEVOMEPROMAZINE LEVOMETIOMEPRAZINE LEVOPROTILINE LEVOSULPIRIDE LITHIUM-NICOTINATE LOFENDAZAM LOFLAZEPATE-ETHYL LOMETRALINE LONETIL LOPIRAZEPAM LOPRAZOLAM LORAZEPAM LORZAFONE LOXAPINE LU-13-117 LU-14-068 LU-17-151 LU-17-152 LU-28-179 LUR-2366 LY-262691 LY-333068 LY-354740 LY-379268 M+B-18706 MAFOPRAZINE MANASSANTIN-A MAROXEPIN MDL-100151 MDL-100907 MDL-105519 MDL-28133A MDL-72483 MDL-73005 MDL-73005EF MDL-73450 MDL-74217 MEBICAR MEBUTAMATE MECLONAZEPAM MECLORALUREA MEDAZEPAM MEDIFOXAMINE MEFECLORAZINE MELPERONE MEPHENOXALONE MEPIPRAZOLE MEPROBAMATE MEPROTIXOL MERAZOLAM MESMAR MESORIDAZINE METACLAZEPAM METAGLYCODOL METAXALONE METHINDIONE METHIOMEPRAZINE METHIOTHEPIN METHOPROMAZINE METIAPINE METOFENAZATE METOPIMAZINE METOSERPATE METOXEPIN MEXAZOLAM MEZEPINE MEZILAMINE MGS-0008 MGS-0028 MIDAFLUR MIDAZOLAM MILENPERONE MILIPERTINE MILTIRONE MINAPRINE MINDOPERONE MJ-13653 MJ-13980-1 MJ-7378 MOLINDONE MONODEMETHYLDOXEPIN MOPERONE MOSAPRAMINE MOTRAZEPAM MS-257 MS-377 NABILONE NAFADOTRIDE NAPRODOXIME

Derwent Drug File 1217 Thesaurus NARANOL NCQ-318 NDO-008 NE-100 NEFLUMOZIDE NELEZAPRINE NEMONAPRIDE NERISOPAM NEUROLEPTICS NGD-94-1 NIMETAZEPAM NISOBAMATE NITRAZEPATE NITRAZEPATE POTASSIUM NKP-608 NNC-0112 NNC-22-0031 NNC-90-3094 NO-01-0756 NONAPERONE NORCHLORPROMAZINE NORDAZEPAM NORTETRAZEPAM NORTHIORIDAZINE NP-207 NPC-16377 NRA-0045 NRA-0160 NRA-0215 NRA-0562 OCAPERIDONE OLANZAPINE OLANZAPINE ONDANSETRON OPC-14597 OPC-4392 OPROMAZINE ORG-2305 ORG-37684 ORG-5222 OSU-6162 OXAFLUMAZINE OXANAMIDE OXAZEPAM OXAZOLAM OXIPEROMIDE OXYCLOTHEPINE OXYFENAMATE OXYPERTINE OXYPROTHEPINE OXYPROTHEPINE-= DECANOATE OXYRIDAZINE P-2565 P-9236 PANADIPLON PANCOPRIDE PAZINACLONE PD-118717 PD-119819 PD-135666 PD-142898 PD-143188 PD-152255 PD-158771 PD-172760 PECAZINE PENFLURIDOL PENTABAMATE PENTAMOXANE PENTIAPINE PERATHIEPINE PERAZINE PERICIAZINE PERIMETAZINE PERPHENAZINE PERPHENAZINE-DECANOATE PERPHENAZINE-ENANTHATE PHENAGLYCODOL PHENPROBAMATE PIFLUTIXOL PIMOZIDE PINAZEPAM PINOXEPIN PIPAMPERONE PIPEQUALINE PIPERACETAZINE PIPETHANATE PIPOTIAZINE PIPOTIAZINE-PALMITATE PIQUINDONE PIVAGABINE PIVOXAZEPAM PK-9084 PRAZEPAM PREMAZEPAM PROCHLORPERAZINE PROFENAMINE PROFLAZEPAM PROMAZINE PROMOXOLANE PROPIONYLPROMAZINE PROPYPERONE PROSULPRIDE PROTHIPENDYL PROTHIXENE PSD-958 PYRICAPIRONE PYRIDARONE PYRIMIDINYLPIPERAZINE QF-0307-B QF-0313-B QF-2003-B QF-2004-B QM-7184 QUETIAPINE R-24763 R-2572 RED.HALOPERIDOL REMOXIPRIDE RESCINNAMINE RESERPINE RGH-1756 RGH-6141 RILAPINE RIMCAZOLE RIPAZEPAM RISPERIDONE RMI-11974 RO-11-7800 RO-17-1812 RO-19-5686 RO-21-6347 RO-21-8384 RO-22-3245 RO-23-0364 RO-4-1284 RO-4-9040 RO-48-6791 RO-48-8684 RO-5-2904 RO-5-2925 RO-5-3590 RO-5-4528 RO-5-4864 RO-60-0175 RO-64-6198 RO-7-5205 ROLIPRAM ROMERGOLINE ROXOPERONE RP-59037 RP-60503 RU-31719 RU-32514 RU-32698 RU-32759 RU-33203 RU-33368 RU-33543 RWJ-37796 RWJ-45788 S-14506 S-16924 S-18327 SARIZOTAN SAS-646 SAVOXEPIN SB-200646-A SB-206553 SB-228357 SB-271046 SB-277011 SC-32855 SCH-23390 SCH-39166 SCH-40853 SDZ-208-911 SDZ-208-912 SDZ-212-327 SEDONIUM SERAZEPINE SEROQUEL SERTINDOLE SETOPERONE SIB-1553-A SKF-10812 SKF-83742 SM-13496 SM-9018 SP-904 SPICLOMAZINE SPIPERONE SPIRAMIDE SPIRILENE SPIROXATRINE SQ-10996 SR-41378 SSR-149415 ST-1460 STACHYDRINE STIRIPENTOL SUANZAORENTANG SULAZEPAM SULFAMOTHEPIN SULFORIDAZINE SULMEPRIDE SULPIRIDE SULTOPRIDE SUN-8399 SUNEPITRON SURICLONE SZJ-3361 SZJ-3388 TACLAMINE TANDOSPIRONE TEFLUDAZINE TEFLUTIXOL TEMAZEPAM TENILAPINE TEPIRINDOLE TETRABENAZINE TETRAZEPAM THIOPROPAZATE THIOPROPERAZINE THIORIDAZINE THIORIDAZINE-DISULFOXIDE-= 2,5 THIORIDAZINE-OXIDE-5 TIAGABINE TIAPRIDE TIENOCARBINE

1218 APPENDIX D TIMELOTEM TIMIPERONE TIOPERIDONE TIOSPIRONE TIOTIXENE TJS-010 TOFISOLINE TOFISOPAM TOLBOXANE TOLPIPRAZOLE TPN-12 TPO-33 TRACAZOLATE TRANQUILIZERS TRAZODONE TRIACETONAMINE TRICLODAZOL TRIFLUBAZAM TRIFLUOMEPRAZINE TRIFLUOPERAZINE TRIFLUPERIDOL TRIFLUPROMAZINE TRIFLUTHEPIN TRIMETOZINE TRIMOPAM TROPAPRIDE TUCLAZEPAM TYBAMATE U-101017 U-101387 U-101958 U-25927 U-43465F U-92016-A U-93385 U-99363-E UK-177 ULDAZEPAM UMESPIRONE VA-21-B7 VALNOCTAMIDE WAY-100289 WAY-100635 WE-1008 WY-48723 XANTHIOL Y-20024 Y-23684 YG-19256 YM-43611 ZALOSPIRONE ZETIDOLINE ZK-91296 ZK-93423 ZK-95962 ZOLAZEPAM ZOLOPERONE ZOLPIDEM ZOPICLONE ZOTEPINE ZUCLOPENTHIXOL ZUCLOPENTHIXOL-ACETATE ZUCLOPENTHIXOL-= DECANOATE PSYCHOSTIMULANT ANTIDEPRESSANT PSYCHOTONIC PSYCHOSTIMULANTS 19148-RP 19749-RP 23669-RP 680-C-91 709-W-92 A-1866 A-80426 AB-15 ACEGLUTAMIDE ACETYLGLUTAMINE-N ADAFENOXATE ADEPREN ADINAZOLAM AGAROSPIROL AGN-2979 ALAPROCLATE ALFETAMINE ALGINOSIDE ALMOXATONE ALTINICLINE AMEDALIN AMFETAMINIL AMFONELATE AMIFLAMINE AMINEPTINE AMINOCYCLOPROPANE= CARBOXYLATE-1 AMITRIPTYLINE AMITRIPTYLINOXIDE AMIXETRINE AMOXAPINE AMPHETAMINE AMPYZINE ANTIDEPRESSANTS ANTIFFEIN APTAZAPINE AS-8 AZ-16596 AZABON AZAPHEN AZEPINDOLE AZIPRAMINE B-193 B-777-81 BAY-1433 BAZINAPRINE BCE-001 BEFLOXATONE BEFURALINE BENMOXIN BENZAPRINOXIDE BENZPHETAMINE BIFEMELANE BINEDALINE BISORCIC BL-KR-140 BMS-181101 BN-50043 BN-50156 BRL-14831 BRL-16644 BROMANTANE BROMOMETHYLPHENIDATE= PARA BUDIPINE BUFENOXATE BUFOTENINE BUPROPION BUTACETIN BUTRIPTYLINE BW-1370U87 BW-1555-U-88 BW-17U BW-287U BW-306U BW-616U76 BW-A-494U BY-1947 BY-1949 C-153 C-307 C-383 C-394 C-395 CAFFEINE CAFFEINE-SODIUM-= BENZOATE CAFFEINE-SODIUM-= SALICYLATE CAPROXAMINE CARBENZIDE CAROXAZONE CARPIPRAMINE CARTAZOLATE CATHINE CATHINONE CENTPROPAZINE CEPHEDRINE CERICLAMINE CGP-12104-A CGP-12104A CGP-22364A CHLORDESIPRAMINE CHLOROAMPHETAMINE CI-933 CIANOPRAMINE CICLAZINDOL CICLINDOLE CICLOPRAMINE CIDOXEPIN CILOBAMINE CIMEMOXIN CIMOXATONE CINFENINE CIPROXIMIDE CITALOPRAM CL-255663 CLEMEPROL CLOCAPRAMINE CLODAZON CLOFENCICLAN CLOFEXAMIDE CLOMIPRAMINE CLORGILINE CLOVOXAMINE COR-3224 COTININE COTRIPTYLINE CP-154526 CP-66713 CP-77059 CP-93393 CRA-1000 CRA-1001 CRL-40827 CYCLAZODONE CYPENAMINE CYPRODENATE CYPROLIDOL DALEDALIN DANITRACEN DAPOXETINE DAZADROL DAZEPINIL DEANOL DEANOL-ACEGLUMATE DEMANYL-PHOSPHATE DEMETHYLDOSULEPIN DEMETHYLDOXEPIN DENBUFYLLINE DEOXYPIPRADOL DESIPRAMINE DEXAMISOLE DEXAMPHETAMINE DEXIMAFEN DEXOXADROL DIBENZEPIN DICLOFENSINE DIMETACRINE DIMETHAMPHETAMINE DIMETHAZAN DIOXADROL

Derwent Drug File 1219 Thesaurus DITRAN DMP-229 DOSULEPIN DOXEPIN DR-250 DU-127090 DULOXETINE E-2011 E-6006 ECLANAMINE EGYT-2760 EGYT-3615 EK-49 ELANZEPINE EMD-68843 ENILOSPIRONE ENPRAZEPINE EPROBEMIDE ESCITALOPRAM ETOPERIDONE ETRYPTAMINE EXP-561 F-13714 FA-37 FANTRIDONE FEMOXETINE FENBUTRAZATE FENCAMFAMIN FENETYLLINE FENGABINE FENMETOZOLE FENOXYPROPAZINE FENOZOLONE FENPENTADIOL FEZOLAMINE FI-4501 FI-4503 FIPEXIDE FLA-289 FLA-299 FLA-314 FLA-334 FLA-336 FLA-365 FLA-384 FLA-405 FLA-417 FLA-450 FLA-463 FLA-558 FLA-668 FLA-717 FLA-727 FLA-788 FLEROBUTEROL FLETAZEPAM FLUACIZINE FLUBANILATE FLUCINDOL FLUOROTRANYLCYPROMINE FLUOTRACEN FLUOXETINE FLUPERLAPINE FLURADOLINE FLUVOXAMINE FR-121196 FS-32 FTORMETAZINE FTORPROPAZINE FURFENOREX GAMFEXINE GC-46 GC-94 GERFONAL GUANOXYFEN HEPZIDINE HEXACYCLONATE HEXACYCLONATE SODIUM HEXAPRADOL HOMOPIPRAMOL HOPANTENATE HP-505 HT-90-B HYDROTHIADENE HYDROXINDASOL HYDROXYAMOXAPINE-7 HYDROXYAMOXAPINE-8 HYDROXYMAPROTILINE HYDROXYTRYPTOPHAN-= ETHYL-ESTER HYDROXYTRYPTOPHAN-= METHYL-ESTER HYPERICIN IEM-487 IEM-508 IEM-611 IF-C-45 IFOXETINE IMAFEN IMIPRAMINE IMIPRAMINE-METHIODIDE IMIPRAMINOXIDE INDALPINE INDATRALINE INDELOXAZINE INDOPAN INDRILINE INN-00835 INTRIPTYLINE IODOCLORGYLINE IPRINDOLE IPROCLOZIDE IPRONIAZID ISOCARBOXAZID IVOQUALINE J-508 J-512 J-516 JB-835 JINKOH-EREMOL JL-3 KETIMIPRAMINE L-783281 LEVOFACETOPERANE LEVOPROTILINE LEVOXADROL LI-160 LILLY-51641 LIS-30 LITHIUM-ASPARTATE LITHIUM-CARBONATE LITHIUM-CHLORIDE LITHIUM-CITRATE LITHIUM-HYDROXYBUTYRATE LITHIUM-NITRATE LITHIUM-SALT (Drug) LITHIUM-SULFATE LITHIUM-TRYPTOPHANATE LITOXETINE LITRACEN LK-63 LOFEPRAMINE LOMEVACTONE LORTALAMINE LOSINDOLE LU-10-134-C LU-11-109 LU-11-161 LU-11-305 LU-17-133 LU-3-009 LU-43706 LY-113821 LY-154045 LY-227942 LY-51641 MAPROTILINE MAZINDOL MCI-225 MCN-4187 MCN-4612-Z MCN-5652-Z MCN-5707 MCN-5908 MD-240098 MD-240233 MD-760548 MDL-19660 MDL-26479 MDL-72394 MDL-72974 MEBANAZINE MECLOFENOXATE MECLOSULFONATE MEDIFOXAMINE MEFEXAMIDE MELITRACEN MEMANTINE MEQUITAZINE MESOCARB METAPRAMINE METHAMPHETAMINE METHASTYRIDONE METHYLAMINOPHOSPHONO= BUTYRATE-N METHYLAMINOPHOSPHONO= PROPIONATE-N METHYLPHENIDATE METRALINDOLE MIANSERIN MILNACIPRAN MIRTAZAPINE MK-0869 MK-306 (psychostimulant) MK-869 MKC-242 MOCLOBEMIDE MODAFINIL MODALINE MONODEMETHYLDOXEPIN MONOMETACRINE NAFENODONE NAPACTADINE NAPAMEZOLE NBF-003 NBF-008 NBF-021 NDO-008 NEBRACETAM NEFAZODONE NEFOPAM NIALAMIDE NICOTINOYLALANINE NISOXETINE NITRAFUDAM NITROXAZEPINE NOMELIDINE NOMIFENSINE NORANTIFFEIN NORCLOMIPRAMINE NORFEMOXETINE NORFLUOXETINE NORTRIPTYLINE NOXIPTILINE NS-105 NSD-2023 NUCLOTIXENE OCTAMOXIN OCTRIPTYLINE OF-6145 OF-743 OI-77

1220 APPENDIX D OMILOXETINE OPC-14117 OPC-14523 OPIPRAMOL ORG-4428 ORG-6582 ORG-6906 OXAFLOZANE OXAPROTILINE OXIFENTOREX OXITRIPTAN PANURAMINE PARAXAZONE PARGYLINE PAROXETINE PEMOLINE PEMOLINE MAGNESIUM PERAFENSINE PERIVINE PF-257 PHENATINE PHENDIMETRAZINE PHENELZINE PHENIPRAZINE PIBERALINE PIM-35 PIPOFEZINE PIPRADROL PIRACETAM PIRANDAMINE PIRLINDOLE PIZOTIFEN PR-881-884A PRAMIRACETAM PRAZEPINE PRAZITONE PRIDEFINE PRINDAMINE PROCYMATE PROLINTANE PROPIZEPINE PROTRIPTYLINE PSILOCIN PSYCHOTONICS PYRIDAZOLE PYRITINOL QUINUPRAMINE RAN-113 REBOXETINE RIBAMINOL RO-4-4318 RO-4-6861 RO-60-0175 ROLICYPRINE ROLZIRACETAM ROSAVIN ROSIN ROSIN-X ROSIRIDIN RS-2232 RTI-113 RU-41656 SABELUZOLE SAFRAZINE SALIDROSIDE SB-224289 SB-271046 SELEGILINE SEPROXETINE SERTRALINE SETIPTILINE SIB-1508-Y SIB-1553-A SIBUTRAMINE SIDNOFEN SKF-25971 SPIROXEPIN SU-11739 SUCCINONITRILE SULTOPRIDE SUNEPITRON SYNHEXYL TABERNAMINE TALOPRAM TALSUPRAM TAMITINOL TAMPRAMINE TANDAMINE TENILSETAM TENOILOXAZINE TETRINDOLE THIONISOXETINE TIANEPTINE TIAZESIM TIENOPRAMINE TIFEMOXONE TIFLUCARBINE TIOMERGINE TISOCROMIDE TJS-010 TOFENACIN TOLOXATONE TOLQUINZOLE TOMOXETINE TOZALINONE TRACAZOLATE TRANYLCYPROMINE TRAZODONE TREBENZOMINE TRELIBET TRIMIPRAMINE TRIZOXIME TROCIMINE TV-3326 TZ-650 U-1424 U-22394A U-23807A U-48753E U-93385 UP-614-04 VALDIPROMIDE VENLAFAXINE VERATRYLHYDRAZINE VILOXAZINE VIQUALINE VUFB-15468 WF-31 WIN-35004 WIN-35065-2 WIN-35065-3 WIN-35140 WIN-35428 WY-25093 WY-27587 WY-45233 YM-08054-1 YM-35992 ZAFULEPTINE ZE-117 ZIMELDINE ZOMETAPINE ZYLOFURAMINE PSYCHOTIC-DISORDER BRIEF-PSYCHOTIC-DISORDER CAPGRAS-SYNDROME catatonic-schizophrenia DELUSIONAL-DISORDER EROTOMANIA PARANOIA paranoid-schizophrenia PARAPHRENIA psychosis SCHIZOAFFECTIVE-DISORDER SCHIZOPHRENIA SCHIZOPHRENIFORM-= DISORDER PSYCHOTOMIMETICS ANANDAMIDE BL-3912 BROLAMFETAMINE CANNABICHROMENE CANNABICYCLOL CANNABIDIOL CANNABIDIOL-= MONOMETHYL-ETHER CANNABIGEROL CANNABINOL CP-47497 CZ-74 DEACETYLLEVONANTRADOL DIMOXAMINE DIPROPYLTRYPTAMINE DOET DOI DOM DRONABINOL HASHISH HYDROXYTETRAHYDROCANNABINOL11 ISOLYSERGATE LSD LY-154045 LYSERGAMIDE LYSERGATE MACROMERINE MESCALINE METHYLENEDIOXYETIL= AMPHETAMINE-3,4 METHYSERGIDE NL-105 NL-106 NORMACROMERINE PIRNABIN PSILOCYBINE SALVINORIN-A SALVINORIN-B SP-111A TENAMFETAMINE TETRAHYDROCANNABINOL-= DELTA-8 TETRAHYDROCANNABINOL-= DELTA-9-11 TETRAHYDROCANNABINOL-= HEMISUCCINATE TETRAHYDROCANNABIVARIN V-111 PSYCHOTONICS ACEGLUTAMIDE ACETYLGLUTAMINE-N AMFETAMINIL AMFONELATE AMINEPTINE AMPHETAMINE AMPYZINE ANTIFFEIN AZABON BENZPHETAMINE BROMOMETHYLPHENIDATE-= PARA BUFOTENINE CAFFEINE CAFFEINE-SODIUM-= BENZOATE CAFFEINE-SODIUM-= SALICYLATE CHLOROAMPHETAMINE CLOFEXAMIDE CYCLAZODONE CYPRODENATE DEANOL

Derwent Drug File 1221 Thesaurus DEANOL-ACEGLUMATE DEMANYL-PHOSPHATE DEOXYPIPRADOL DEXAMPHETAMINE DIMETHAMPHETAMINE DIMETHAZAN ENILOSPIRONE ETRYPTAMINE FENBUTRAZATE FENCAMFAMIN FENETYLLINE FENOZOLONE FIPEXIDE FLUCINDOL FURFENOREX HEXAPRADOL HOPANTENATE HYDROXINDASOL IEM-487 IEM-508 IEM-611 IMIPRAMINE INDOPAN INDRILINE MECLOFENOXATE MECLOSULFONATE MEFEXAMIDE MESOCARB METHAMPHETAMINE METHASTYRIDONE METHYLPHENIDATE MODAFINIL NORANTIFFEIN OPC-14117 OXAFLOZANE OXIFENTOREX PEMOLINE PEMOLINE MAGNESIUM PHENATINE PIPRADROL PRINDAMINE PROCYMATE PROLINTANE PSILOCIN PYRITINOL RIBAMINOL SELEGILINE SYNHEXYL TOFENACIN VALDIPROMIDE ZYLOFURAMINE PURINE-ANTAGONIST ADENOSINE-ANTAGONIST PURINE-ANTAGONISTS A-720287 ADENOSINE-ANTAGONISTS APEC ARC-69931-MX BST-101 BW-A-1433 BW-A-1433U BW-A522U BW-A844U BW-A947U CGS-15943 CGS-15943A CHICAGO-ACID CP-66713 CS-747 CVT-124 DIMETHYLPROPARGYL= XANTHINE FK-352 FK-453 FK-838 FPL-66096 FPL-67085 FR-113452 IRFI-117 IRFI-165 KF-15372 KF-17837 KFM-19 KN-04 KW-3902 KW-6002 L-249313 MDL-102234 MRS-1067 MRS-1097 MRS-1191 MRS-1220 MRS-1754 MRS-2179 MRS-2257 MRS-2286 N-0840 N-0861 NF-023 NF-037 NF-279 PD-115199 PD-116948 PD-81723 PHENYLTHEOPHYLLINE-8 PROCION-BLUE-HB R-99224 SCH-58261 VUF-8501 VUF-8504 VUF-8505 VUF-8507 WRC-0342 WRC-0571 XAMR-0716 XT-044 ZM-241385 PURINE-METAB.DISORDER GOUT HYPERURICEMIA HYPERURICURIA HYPOURICEMIA LESCH-NYHAN-SYNDROME XANTHINURIA PURINERGIC ADENOSINE-AGONIST PURINERGICS ADENOSINE ADENOSINE-AGONISTS ADENYLOSUCCINATE ADP-METHYLENE-= ALPHA,BETA AGR-529 ALLYLADENOSINE ARISTEROMYCIN ATL-193 ATP-METHYLENE-= ALPHA,BETA ATP-METHYLENE-= BETA,GAMMA ATP-METHYLTHIO-2 B-744-96 BENZYLADENOSINE-6 CARBOXAMIDOADENOSINE CGS-21680 CGS-21680A CGS-21680C CGS-22492 CGS-22988 CGS-22989 CHLOROADENOSINE-2 CI-936 CVT-3033 CVT-313 CVT-3146 CVT-510 CYCLOBUTYLADENOSINE CYCLOHEXYLADENOSINE CYCLOPENTYLADENOSINE DADP DIADENOSINE-= PENTAPHOSPHATE DIADENOSINE-= TETRAPHOSPHATE DINECA DWH-146-E FPL-67156 GP-1-515 GR-190178 GR-79236 IBMECA INS-365 LUF-5407 MDL-201112 MDV-1 METHYLADENOSINE-N-6 METHYLCARBOXAMIDE-= ADENOSINE MRE-0470 MRS-1760 NNC-21-0238 NNC-53-0055 NNC-53-0082 NNC-90-1515 OXAZOFURIN PD-117519 PD-125944 PHENYLADENOSINE-6 PHENYLETHYLADENOSINE-= N-6 PHENYLISOPROPYL= ADENOSINE RG-14123 RG-14202 RPR-100579 SCH-59761 SDZ-WAG-994 THIOPHENFURINE UP-20256 WRC-0090 WRC-470 XYLOADENINE YT-146 YT-146 PURPURA HENOCH-SCHOENLEIN PYRIMIDINE-METAB.DISORDER PYRIMIDINEMIA PYRIMIDINURIA QUALITY-CONTROL CONTENT-UNIFORMITY RADIOACTIVITY RADIOENZYME-DET. RADIOENZYME-IMMUNODET. RADIORECEPTOR-DET. RADIOLESION ALVELD CHRYSIASIS HYDROA PHOTODERMATITIS PHOTODERMATOSIS RADIATION-SICKNESS RADIODERMATITIS SUNBURN RADIOPAQUES 2-5410-4A ACETRIZOATE SODIUM

1222 APPENDIX D ADIPIODONE ADIPIODONE MEGLUMINE ADIPIODONE-ETHYL-ESTER AG-52-315 ALBUNEX AMIDOTRIZOATE AMIDOTRIZOATE LYSINE AMIDOTRIZOATE = MEGLUMINE AMIDOTRIZOATE SODIUM ANGIOVIST BARIUM-SULFATE BROMOHIPPURATE BUNAMIODYL CARTRIZOATE-ETHYL DIMETHIODAL SODIUM DIODONE DIPROTRIZOATE DOCETRIZOATE-PROPYL ECHOGEN EDTA-CHROMIUM ETHIODOL ETHYL-IOPANOATE ETIOTRAST FP-736-03 FP-736-04 GADOLINIUM-DOTA GADOLINIUM-OXALATE GADOPENTETATE IOBENGUANE IOBENZAMATE IOBITRIDOL IOBUTOATE IOCARMATE IOCARMATE MEGLUMINE IOCETAMATE IODAMIDE IODAMIDE MEGLUMINE IODAMIDE SODIUM IODECIMOL IODETRYL IODIXANOL IODIZED-OIL IODOHIPPURATE IODOPHENYLPENTA= DECANOATE-ORTHO IODOPHTHALEIN SODIUM IODOXAMATE IODOXAMATE MEGLUMINE IODOXYL IOFENDYLATE IOGLICATE IOGLUCOL IOGLUCOMIDE IOGLUNIDE IOGLYCAMATE IOGLYCAMATE MEGLUMINE IOGULAMIDE IOHEXOL IOLIDONATE IOLIXANATE IOMEGLAMATE IOMEPROL IOMORINATE IOPAMIDOL IOPANOATE IOPANOATE SODIUM IOPANOATE-CHOLESTERYL IOPENTOL IOPHENOATE IOPODATE IOPODATE CALCIUM IOPODATE SODIUM IOPROCEMATE IOPROMIDE IOPRONATE IOPYDOL IOPYDONE IOSARCOL IOSEFAMATE IOSERATE IOSIMIDE IOSULAMIDE IOSUMETATE IOTALAMATE IOTALAMATE MEGLUMINE IOTALAMATE SODIUM IOTASUL IOTETRATE IOTRANATE IOTRIZOATE IOTROLAN IOTROXATE IOVERSOL IOXAGLATE IOXAGLATE MEGLUMINE IOXAGLATE SODIUM IOXILAN IOXITALAMATE IOXITALAMATE MEGLUMINE IOXITALAMATE SODIUM IOXOTRIZOATE IOZOMATE IPODATE-ETHYL LEVOVIST METHIODAL SODIUM METRIZAMIDE METRIZOATE METRIZOATE CALCIUM METRIZOATE MAGNESIUM METRIZOATE MEGLUMINE METRIZOATE SODIUM NP-59 P-308 P-530 P-743 PERFLUBRON PERFLUOROHEXYLBROMIDE PERFLUTREN PHENIODOL SODIUM PHENOBUTIODIL PROPYLIODONE RP-30A SH-771 SQ-32014 TYROPANOATE TYROPANOATE SODIUM YTTERBIUM-DTPA RADIOPROTECTIVES ABSOL ACTINOQUINOL AET AGL-517 AMIFOSTINE AVOBENZONE BATILOL BGP-15 BORNELONE BUMETRIZOLE CHLOROTRYPTAMINE-5 CINOXATE DIOXYBENZONE DROMETRIZOLE ETOCRILENE EUSOLEX-232 EUSOLEX-6300 EUSOLEX-8020 GEROQUINOL GLUTAURINE GLYCERYL-PABA HOMOSALATE I-102 KERATINOCYTE-GROWTH-= FACTOR-2 MERCAPTOBENZ= IMIDAZOLE-2 MERCAPTOETHYLGUANIDINE MEXAMINE MEXENONE NEO-HELIOPAN OCTABENZONE OCTOCRILENE OCTRIZOLE OCTYL-METHOXY= CINNAMATE OXYBENZONE PADIMATE PADIMATE-O PALLIRAD PEUCEDANIN PHOSPHOTYROSINE-O SALOL SESAMOL SULISOBENZONE U-75412E UVINUL-T150 WITISOL WR-1065 WR-151326 WR-3689 WR-638 WR-77913 RADIOSENSITIZERS AK-2123 AMINOLEVULINATE-DELTA-= HEXYL-ESTER AMINOLEVULINATE-DELTA-= METHYL-ESTER ANGELICIN AQ4N AZOMYCIN-RIBOSIDE BACTERIOCHLORIN-A BACTERIOCHLOROPHYLL-A BENZOPORPHYRIN-= DERIVATIVE BERGAPTEN BPD-MA CCI-103F CHLORIN-P6-LYSYL CHLOROALUMINUM-= DISULFOPHTHALOCYANINE CHLOROALUMINUM-= MONOSULFOPHTHALO= CYANINE CHLOROALUMINUM-= PHTHALOCYANINE CHLOROALUMINUM-= SULFOPHTHALOCYANINE CHLOROALUMINUM-= TETRASULFOPHTHALO= CYANINE CHLORODEOXYCYTIDINE-5 CI-1010 CITROPTEN CL-315555 CL-315585 DEUTEROPORPHYRIN-IX-= 2,4-BIS-GLYCOL DEUTEROPORPHYRIN-IX-TIN DIHEMATOPORPHYRIN-ETHER DIIODODEUTERO= PORPHYRIN-TIN DIMEGIN ETANIDAZOLE ETIOPURPURIN-TIN FTI-277 GADOLINIUM TEXAPHYRIN HEMATOPORPHYRIN-= DERIVATIVE HYDROXYMETHYLTRIOXY= SALEN-4+ HYDROXYMETRONIDAZOLE HYPOCRELLIN-A

Derwent Drug File 1223 Thesaurus HYPOCRELLIN-B ICRF-186 ILX-23-7553 KIH-200 KIH-201 KIH-202 KIH-802 KIN-804 KU-2285 L-8580 LIMETTIN LONIDAMINE LUMIDOXYCYCLINE LUTETIUM-TEXAPHYRIN MESOPORPHYRIN-TIN METHOXSALEN METHYLISOPSORALEN-5 METRONIDAZOLE METRONIDAZOLE-= PHOSPHATE METRONIDAZOLE-SUCCINATE MISONIDAZOLE MONOASPARTYLCHLORIN-E6 MV-6401 NDH-3080 NILE-BLUE-A NIRIDAZOLE NITROIMIDAZOLE-4 NSC-676418 NU-1025 NU-1064 NU-7026 NU-7163 PD-128763 PD-144871 PD-146923 PD-183805 PH-1008 PHEOPHORBIDE-A PHOTOSAN PHTHALOCYANINE PIMONIDAZOLE PKC-412 PLATONIN POLYHEMATOPORPHYRIN PORPHYRIN-C PR-350 PSORALEN R-6998 R-7000 RB-6145 RB-7040 RK-28 RO-03-8800 RO-3-6156 RO-31-0368 RO-5-9963 RSR-13 RSU-1069 RSU-1131 RSU-1137 RSU-1150 RSU-1164 RSU-1165 RSU-1170 RSU-1172 SR-2555 SUBEROYLANILIDE-= HYDROXAMATE TBI-361 TEMOPORFIN TERTHIENYL-ALPHA TETRAPHENYLPORPHYCENE TETRASULFOPHENYLPORPHINE THIOPYRONINE TOLYPORPHIN-A TRIMETHYLANGELICIN-4,6,4+ TRIMETHYLAZAPSORALEN-= 4,4+,5+ TRIOXYSALEN UROPORPHYRIN-I VICTORIA-BLUE-BO ZINC-PHTHALOCYANINE-= TETRASULFONATE RADIOTHERAPY RADIOCHEMOTHERAPY RADIOIMMUNOTHERAPY RECEPTOR ACTH-RECEPTOR ADRENERGIC-RECEPTOR ALDOSTERONE-RECEPTOR alpha4beta1 AMPA-RECEPTOR ANDROGEN-RECEPTOR ANF-RECEPTOR ANGIOTENSIN-2-RECEPTOR ANGIOTENSIN-RECEPTOR ANTIESTROGEN-RECEPTOR ATP-RECEPTOR atrial-natriuretic-factor-= receptor AUTORECEPTOR BENZODIAZEPINE-RECEPTOR BOMBESIN-RECEPTOR BRADYKININ-RECEPTOR CALCIFEROL-RECEPTOR CALCITONIN-RECEPTOR CALCIUM-CHANNELRECEPTOR CALMODULIN-RECEPTOR CANNABINOID-RECEPTOR CARDIOGLYCOSIDE-= RECEPTOR cd49d-cd29 CHEMOKINE-RECEPTOR CHEMOTACTIC-FACTOR-= RECEPTOR CHLORIDE-CHANNEL-= RECEPTOR CHOLINERGIC-RECEPTOR COMPLEMENT-RECEPTOR CORTICOLIBERIN-RECEPTOR CORTICOSTEROID-RECEPTOR CXC-RECEPTOR DEATH-RECEPTOR digitalis-receptor DOPAMINE-RECEPTOR EGF-RECEPTOR ENDOTHELIN-RECEPTOR ENZYME-RECEPTOR-DET. ESTROGEN-RECEPTOR FC-RECEPTOR FSH-RECEPTOR GABA-RECEPTOR GASTRIN-RECEPTOR GASTRIN-RELEASING-= PEPTIDE-RECEPTOR GLUCAGON-RECEPTOR glucocorticoid-receptor GLUTAMATE-RECEPTOR GLYCINE-RECEPTOR GLYCINE-RECEPTOR GONADOLIBERIN-RECEPTOR GONADOTROPIN-RECEPTOR GPIIB-IIIA-RECEPTOR HERG-CHANNEL HISTAMINE-RECEPTOR ICSH-RECEPTOR IMIDAZOLINE-RECEPTOR INSULIN-RECEPTOR INTERFERON-RECEPTOR INTERLEUKIN-2-RECEPTOR INTERLEUKIN-RECEPTOR KAINATE-RECEPTOR LEUKOTRIENE-RECEPTOR LIPOPROTEIN-RECEPTOR LIVER-X-RECEPTOR LULIBERIN-RECEPTOR MELANOCORTIN-RECEPTOR MELATONIN-RECEPTOR METHYLASPARTATE-N-= RECEPTOR MOTILIN-RECEPTOR MOTILIN-RECEPTOR NEUROMEDIN-RECEPTOR NEUROPEPTIDE-Y-RECEPTOR NEUROTENSIN-RECEPTOR OPIOID-RECEPTOR OXYTOCIN-RECEPTOR PAF-RECEPTOR PANCREOZYMIN-RECEPTOR PARATHORMONE-RECEPTOR PHENCYCLIDINE-RECEPTOR POTASSIUM-CHANNEL-= RECEPTOR PPAR-ALPHA PPAR-DELTA PPAR-GAMMA PROGESTOGEN-RECEPTOR PROLACTIN-RECEPTOR PROSTACYCLIN-RECEPTOR PROSTAGLANDIN-RECEPTOR PURINE-RECEPTOR QUISQUALATE-RECEPTOR RETINOIC-ACID-RECEPTOR RETINOID-RECEPTOR RETINOID-X-RECEPTOR RYANODINE-RECEPTOR SECRETIN-RECEPTOR SEROTONIN-RECEPTOR SIGMA-RECEPTOR SODIUM-CHANNEL-= RECEPTOR SOMATOMEDIN-C-RECEPTOR SOMATOSTATIN-RECEPTOR SOMATOTROPIN-RECEPTOR SUBSTANCE-K-RECEPTOR SUBSTANCE-P-RECEPTOR TGF-RECEPTOR THROMBIN-RECEPTOR THROMBOXANE-RECEPTOR THYROLIBERIN-RECEPTOR TNF-RECEPTOR TRANSFERRIN-RECEPTOR TRIIODOTHYRONINE-= RECEPTOR TRYPTAMINE-RECEPTOR VANILLOID-RECEPTOR vasoact.intest.peptide-= receptor VASOPRESSIN-RECEPTOR VIP-RECEPTOR vitamin-a-receptor vitamin-d-receptor VLA-4 REDUCTION HYDROGENATION REFLEX BLINKING REGULATION AUTOREGULATION RELAXANTS 340125 450247 450304 450789 450790 58-112 AD-2239

1224 APPENDIX D AFLOQUALONE AGATOXIN-ALPHA-489 AGELASIMINE-A AGELASIMINE-B AHR-2666 AMBENOXAN ANETHOCURARIUM ANQ-9040 AZUMOLENE BA-28882 BACLOFEN BM-519 BN-063 BROFOXINE CARAMIPHEN CARISOPRODOL CHLORPHENESIN-= CARBAMATE CHLORZACETAMOL CHLORZOXAZONE CILTOPRAZINE CINNAMAMIDE CISATRACURIUM BESILATE CLIMAZOLAM CLODANOLENE CLOFEVERINE CNIDILIDE CONDELPHINE CYCLOBENZAPRINE D-174 D-175 DANTROLENE DECADONIUM IODIDE DENPIDAZONE DEXTROFEMINE DIADONIUM DIAZEPAM DICHLORMEZANONE DIPYRANDIUM DORIDOSINE ELATINE EMYLCAMATE ENANTALDEHYDE EPERISONE ETOMIDOLINE FEBARBAMATE FENYRAMIDOL FENYRIPOL FLETAZEPAM FLUCARBRIL FLUMETRAMIDE FLUNITRAZEPAM GABA-LINOLEAMIDE GRAYANOTOXIN-III GUAIFENESIN GUANABENZ GYKI-52466 HB-218 HEXAFLURONIUM BROMIDE HONOKIOL HYDROXYDANTROLENE-5 IDPH-791 IDROCILAMIDE INAPERISONE IPROZILAMINE ISOFLURANE KOJIC-AMINE LANPERISONE LEFETAMINE LIGUSTILIDE LINDOLDHAMINE LORBAMATE MAGNOLOL MDL-105519 MDL-27531 MEBEZONIUM IODIDE MELADRAZINE MELLICTINE MENITRAZEPAM MEPHENESIN MEPHENOXALONE METAXALONE METHOCARBAMOL MEZILAMINE MLV-3076 MLV-5860 MLV-6976 MS-322 NABILONE NAFOMINE NCX-950 NEFOPAM NELEZAPRINE NK-422 NK-433 NORDAZEPAM NS-1608 PARSALMIDE PHENPROBAMATE PIFEXOLE PIPECURONIUM PIRIQUALONE POPISONINE PRAZEPAM PRIDINOL-MESILATE QUILOFLEX R-8110 RACEFEMINE RGH-5002 RJ-64 RO-22-8349 RO-5-4864 RO-5-5115 RO-5-6669 RO-5-6945 RO-5-6993 ROLODINE RS-722 RU-31719 SENKYUNOLIDE SO-121 STIRIPENTOL STYRAMATE TAAC-3 TETRAZEPAM THIOCOLCHICOSIDE TIZANIDINE TK-11 TMB-5 TOLOXATONE TOLPERISONE TYBAMATE XILOBAM ZOXAZOLAMINE RELEASING-FACTOR CORTICOLIBERIN-AGONIST FOLLIBERIN-AGONIST GONADOLIBERIN-AGONIST LULIBERIN-AGONIST MELANOLIBERIN-AGONIST PROLACTOLIBERIN-AGONIST SOMATOLIBERIN-AGONIST THYROLIBERIN-AGONIST RELEASING-FACTOR-INHIBITOR CORTICOLIBERIN-= ANTAGONIST FOLLIBERIN-ANTAGONIST GONADOLIBERIN-= ANTAGONIST LULIBERIN-ANTAGONIST MELANOSTATIN-AGONIST SOMATOSTATIN-AGONIST RELEASING-FACTORINHIBITORS 204-090 ABARELIX ACYLINE AG-045572 AN-238 ANTALARMIN ANTARELIX ANTIDE ANTISAUVAGINE-30 ASTRESSIN AZALINE AZALINE-B BIM-23003 BIM-23003 BIM-23023 BIM-23026 BIM-23027 BIM-23034 BIM-23056 BIM-23127 BIM-23190 BIM-23197 BM-2-28 BM-23014 CDB-2085A CETRORELIX CGP-15425 CGP-23996 CH-288 CORTICOLIBERIN-12-41,D-PHE CORTICOLIBERIN-9-41 CORTICOLIBERIN-= ANTAGONISTS CORTISTATIN CP-154526 CRA-1000 CRA-1001 DC-13-57 DC-23-99 DETIRELIX DETIRELIXACETATE EC-5-20 FOLLIBERIN-ANTAGONISTS GANIRELIX GONADOLIBERIN-= ANTAGONISTS JV-1-36 L-362855 L-779976 LANREOTIDE LULIBERIN-ANTAGONISTS MELANOSTATIN MELANOSTATIN-AGONISTS MELANOSTATIN-I MI-1544 MK-363-301 MK-678 MZ-4-71 MZ-5-156 NAL-ARG-LULIBERIN NAL-GLU-LULIBERIN NC-8-12 OCTREOTIDE ORF-18260 ORF-21243 ORG-30093 ORG-30276 PENTETREOTIDE PROSOMATOSTATIN PROSOMATOSTATIN-1-12 PROSOMATOSTATIN-II-= ANGLERFISH QUADRIGEMINE-C RC-101-I RC-121 RC-160-II

Derwent Drug File 1225 Thesaurus RC-98-I RWJ-47428-021 SANDOZ-201995 SB-29 SB-30 SB-88 SC-241 SD-357 SDZ-207-895 SDZ-212-610 SDZ-215-811 SDZ-217-704 SDZ-CO-611 SEGLITIDE SOMATOSTATIN SOMATOSTATIN-AGONISTS SOMATOSTATIN-D-TRP-8 SOMATOSTATIN-LINEAR SOMATOSTATIN-PHE-4 SP-904 TEVERELIX TT-232 TX-44 TX-51 TX-53 TYROSYL-MELANOSTATIN VAPREOTIDE WY-18185 WY-41747 WY-45760 RELEASING-FACTORS ACTIVIN AN-207 AY-25205 BI-679 BUSERELIN CORTICOLIBERIN CORTICOLIBERIN-AGONISTS CORTICOLIBERIN-CATTLE CORTICOLIBERIN-HUMAN CORTICOLIBERIN-SHEEP CYCLO-HIS-PRO DEAMIDOLULIBERIN DEAMIDOTHYROLIBERIN DESLORELIN DN-1417 FERTIRELIN FOLLIBERIN FOLLIBERIN-AGONISTS G-7039 G-7203 G-7502 GHRELIN-HUMAN GONADOLIBERIN GONADOLIBERIN-AGONISTS GONADOLIBERIN-SALMON GONAVET GOSERELIN HEXARELIN HISTRELIN JG-73 JTP-2942 L-162752 L-163191 L-163540 L-692429 L-692585 L-700653 LEUPRORELIN LULIBERIN LULIBERIN-3-10 LULIBERIN-4-10 LULIBERIN-AGONISTS LULIBERIN-D-ALA-6 LULIBERIN-D-LYS-6 LULIBERIN-D-PHE-6 LULIBERIN-D-SER-6 LULIBERIN-FOWL LULIBERIN-I-FOWL LULIBERIN-II-FOWL LUTRELIN LY-444711 MELANOLIBERIN MELANOLIBERIN-AGONISTS MINILULIBERIN MK-0677 MK-771 MONTIRELIN MONTIRELIN MZ-2-51 MZ-2-75 MZ-2-87 NAFARELIN OROTIRELIN OVURELIN PHYLADOX PRALMORELIN PROLACTOLIBERIN PROLACTOLIBERIN-AGONISTS RO-23-7863 RS-49947 RX-77368 SKF-110679 SM-130686 SOMATOCRININ SOMATOCRININ-CATTLE SOMATOCRININ-HUMAN SOMATOLIBERIN SOMATOLIBERIN-1-29 SOMATOLIBERIN-1-29-AMIDE SOMATOLIBERIN-1-29-= AMIDE,NLE-27 SOMATOLIBERIN-1-40 SOMATOLIBERIN-1-44 SOMATOLIBERIN-2 SOMATOLIBERIN-AGONISTS SOMATOLIBERIN-HUMAN-= PANCREATIC-1-29 SOMATOLIBERIN-HUMAN-= PANCREATIC-1-37 SOMATOLIBERIN-HUMAN-= PANCREATIC-1-40 SOMATOLIBERIN-PIG-1-44 SOMATOLIBERIN-RAT SOMATOLIBERIN-RAT-1-29 SOMATOLIBERIN-RAT-1-43 SOMATOLIBERIN-SHEEP-1-44 SUPERGESTRAN TA-0910 TABIMORELIN THYROLIBERIN THYROLIBERIN-AGONISTS THYROLIBERIN-T TRIPTORELIN UROCORTIN YM-14673 RENIN-INHIBITORS A-65137 A-68064 A-72517 A-74273 BILA-2157-BS CGP-29287 CGP-38560 CGP-38560A CGP-44099A CP-71362 CP-80794 CYCLOTHIAZOMYCIN DITEKIREN ENALKIREN ES-1005 ES-295 ES-300 ES-305 ES-313 ES-316 ES-317 ES-6864 ES-8891 H-113 H-261 JTP-2724 KRI-1177 KRI-1314 PD-132002 PD-134672 RO-42-5892 SC-45075 SC-46507 SC-46944 SCRIP SPP-100 SQ-33800 SR-42128 SR-42128A SR-43845 U-71909E U-73777-E U-77455-E U-77647E REOVIRUS BLUE-TONGUE-VIRUS BLUECOMB-VIRUS EPIZOOTIC-HEM.DISEASE-= VIRUS IBARAKI-VIRUS INFECTIOUS-BURSAL-= DISEASE-VIRUS ROTA-VIRUS REPTILE ALLIGATOR RES HISTIOCYTE KUPFFER-CELL MACROPHAGE MICROGLIA OSTEOCLAST PHAGOCYTE RESISTANCE R-FACTOR RESPIRAT.TRACT HYOID-ARCH TRACHEA RESPIRATION ACCELERATION-INDEX AIRWAY-COMPLIANCE AIRWAY-CONDUCTANCE AIRWAY-RESISTANCE BREATHING CAROTID-BODY-REFLEX dynamic-compliance MINUTE-VOLUME peak-flow-rate TIDAL-VOLUME VITAL-CAPACITY RESPIRATION-DISORDER altitude-anoxia ANOXIA APNEA ASPHYXIA BRADYPNEA CARDIAC-ASTHMA DECOMPRESSION-SICKNESS DYSPNEA HYPERCAPNIA HYPEROXIA

1226 APPENDIX D HYPERPNEA HYPERVENTILATION HYPOCAPNIA HYPOVENTILATION HYPOXIA idiopathic-alveolar-= hypoventilation MOUNIER-KUHN-SYNDROME mountain-sickness ondine-curse ORTHOPNEA RESPIRAT.ARREST RESPIRAT.DEPRESSION SLEEP-APNEA STRIDOR TACHYPNEA RETINOBLASTOMA Y79-CELL RETINOID-RECEPTOR RETINOIC-ACID-RECEPTOR RETINOID-X-RECEPTOR RETROVIRUS LENTIVIRUS REVERSE-TRANSCRIPTASEINHIBITORS 306 739-W-94 ABACAVIR ALIZARIN-COMPLEXONE ALIZARIN-S AMBIGOL-A AMBIGOL-B AMINOTHYMIDINE-3+ ANHYDROZIDOVUDINE-5+,2 ANOLIGNAN-A ATEVIRDINE AZIDODIDEOXY= GUANOSINE-2+,3+ B-041 B-059 B-239 B-442 BCH-189-TRIPHOSPHATE BI-RJ-70 CALANOLIDE-A CARBOVIR CARBOVIR-TRIPHOSPHATE CGP-53437 CORDATOLIDE-A CORDATOLIDE-B COSALANE CS-85 CS-87 CS-87-TRIPHOSPHATE CURDLAN-ARABINOSE-= SULFATE CURDLAN-GALACTOSE-= SULFATE CURDLAN-SULFATE DELAVIRDINE DEOXYCARBOVIR-6 DIDEOXY-GTP DIDEOXY-ITP DIDEOXY-TTP DIDEOXY-UDP DIDEOXY-UMP DIDEOXY-UTP DMP-963 DPC-082 DPC-083 DPC-961 EA-521 EFAVIRENZ EMTRICITABINE-= TRIPHOSPHATE ETHOXIDINE FLUORODIDEOXY-CTP-5 FLUORODIDEOXY-= VIDARABINE-= 2+TRIPHOSPHATE FLUORODIDEOXYCYTIDINE-= 2+ FPMPA FTC HBY-097 HEPT HI-236 HI-253 HI-280 INOPHYLLUM-B INOPHYLLUM-P IVX-E-59 JANIEMYCIN JM-1590 JM-1591 JM-1596 JM-2815 JM-2820 L-693593 L-696040 L-696229 L-697639 L-697661 L-697695 L-702007 L-737126 L-738372 LAMIVUDINE LAMIVUDINE-TRIPHOSPHATE LY-300046 LY-300082 LY-73497 MAP-30 MEN-10690 METHOXYDODECANOATE-12 MICHELLAMINE-A MICHELLAMINE-B MKC-442 MSC-206 MSH-372 NEVIRAPINE NF-201 NF-503 NF-504 NF-506 NIGRANOATE NSC-287474 NSC-615985 NSC-624231 NSC-648400 OENOTHEIN-B OXOCALANOLIDE-A-12 PD-134922 PD-135390 PETROSYNOL PM-19 PMPDAP PNU-142721 POLYVINYLSULFONATE = SODIUM R-82150 R-86183 R-88703 R-89439 RD-42024 RO-24-5098 RS-980 RUBROMYCIN-ALPHA RUBROMYCIN-BETA RUBROMYCIN-GAMMA S-2720 SALASPERMATE SCHIZOPHYLLAN-SULFATED SJ-3366 SQ-34676 STAVUDINE SWERTIFRANCHESIDE TENOFOVIR TENOFOVIR-DIPHOSPHATE THIELAVIN-A THIELAVIN-B TIBO TMC-125 TOXICOL-A TOXICOL-B TOXIUSOL U-104489 U-88204 U-88204E U-95133 UC-040 UC-10 UC-284 UC-42 UC-781 VF-1634 WHI-07 ZIDOVUDINE ZIDOVUDINE-ISOLEUCINE ZIDOVUDINE-TRIPHOSPHATE RHABDOMYOSARCOMA A204-CELL RD-CELL RHABDOVIRUS AMERICAN-EEL-VIRUS BIVENS-ARMS-VIRUS DUVENHAGE-VIRUS EUROPEAN-EEL-VIRUS FLURY-VIRUS HEM.SEPSIS-VIRUS INFECTIOUS-= HEMATOPOIETIC-= NECROSIS-VIRUS MOKOLA-VIRUS PIKE-FRY-DISEASE-VIRUS RABIES-VIRUS SPRING-VIREMIA-VIRUS THREE-DAY-SICKNESS-VIRUS VESICULAR-STOMATITIS-= VIRUS RHEOLOGY COHESION FLOW RHEOPEXY SHEAR-FLOW SHEAR-STRESS SPREADABILITY THIXOTROPY VISCOSITY RHEUMATOID FELTY-SYNDROME RHINITIS INCLUSION-BODY-RHINITIS RIBOZYME MAXIZYME RICKETTSIALES ANAPLASMA CHLAMYDIA chlamydia-psittaci chlamydia-trachomatis COLESIOTA COWDRIA COXIELLA CYTOECETES EHRLICHIA EPERYTHROZOON GRAHAMELLA

Derwent Drug File 1227 Thesaurus HAEMOBARTONELLA NEORICKETTSIA ornithosis-virus RICKETTSIA RICKETTSIELLA ROCHALIMAEA SYMBIOTES trachoma-inclusion-= conjunctivitis-agent tric-agent WOLBACHIA RODENTICIDES BROMADIOLONE BROMETHALIN CRIMIDINE PYRINURON WARFARIN RUBEFACIENTS CANTHARIDIN CAPSAICIN CAPSICUM SALIVA PTYALISM SALIVATION SARCOMA EMT6-CELL M5076-SARCOMA RIF1 RIF1-CELL RR1022-CELL SARCOMA-180 SARCOMA-180-CELL SARCOMA-37 SARCOMA-37-CELL SARCOMA-45 SARCOMA-45-CELL XC-CELL YOSHIDA-SARCOMA YOSHIDA-SARCOMA-CELL SEDATIVES 340125 450247 450304 450789 450790 ACEBROCHOL ACECARBROMAL ACEVALTRATE ALLOBARBITAL ALONIMID ALOZAFONE AMINOGLUTETHIMIDE AMOBARBITAL APIOLE-DILL APOMORPHINE APROBARBITAL APRONALIDE AR-A-008055 AZAPERONE BALDRIANOL BALDRINAL BARBEXACLONE BARBITAL BARBITAL SODIUM BARBITURATE BASON BENZOBARBITAL BENZYLURIDINE-3 BERSALDEGENIN-= ORTHOACETATE BIGLUMIDE BORNYVAL BRALLOBARBITAL BROMAMID BROMISOVAL BROMOBUTANOL BROMOCAMPHOR BROMOFORM BROMOLACTOBIONATE = CALCIUM BUCOLOME BUTALBITAL BUTALLYLONAL BUTHALITAL SODIUM BUTOBARBITAL BUTOCTAMIDE BUTOCTAMIDE-SUCCINATE C-720045 CAMAZEPAM CAPTODIAME CAPURIDE CARBOCLORAL CARBROMAL CARBROMIDE CARBUBARB CARFIMATE CELUCLORAL CENTALUN CESEDON CETOHEXAZINE CG-601 CHLORAL-HYDRATE CHLORALODOL CHLORALOSE CHLOROBUTANOL CHLORPROMAZINE CHLORPROMAZINE-= METHIODIDE CHROMOCARB CIMEPANOL CL-284846 CLAZOLAM CLIDAFIDINE CLIMAZOLAM CLOMETHIAZOLE CLOPERIDONE CLORAZEPATE CLORETATE CLOTIAZEPAM CO-134444 CROTARBITAL CYCLOBARBITAL CYCLOPENTOBARBITAL DAA-1097 DAA-1106 DAIGREMONTIANIN DAMOTEPINE DEALKYLFLURAZEPAM DETOMIDINE DIALLYLPENTOBARBITAL DIAZEPAM DICHLORALPHENAZONE DIDROVALTRATE DIFEBARBAMATE DIHYPRYLONE DIMETHYLPHENOBARBITAL DIPHENHYDRAMINE DORMOVIT DOXYLAMINE E-350 EA-1465 EA-1476 ECTYLUREA ENALLYPROPYMAL EPINOVAL ETAQUALONE ETEROBARB ETHCHLORVYNOL ETHINAMATE ETHYLAL ETHYPICONE ETODROXIZINE ETOMIDATE ETYMEMAZINE FEBARBAMATE FELBAMATE FENADIAZOLE FEPITRIZOL FLUPERLAPINE FLURAZEPAM FOSAZEPAM FUMARILINE GINGEROL-6 GLOMERIN GLUTETHIMIDE GP-41299 HALOXAZOLAM HAPLOPINE HD-233 HEPTABARB HEPTOBARBITAL HEXAPROPYMATE HEXETHAL HEXOBARBITAL HOMOGLOMERIN HYDROXYCAMAZEPAM HYDROXYPHENOBARBITAL-= PARA IB-503 IBROTAMIDE IDOBUTAL IMINOPHENIMIDE INDOPINE ISOVALEROXYHYDROXY= DIDROVALTRATE ISOVALTRATE K-2604 LONETIL LOPRAZOLAM LORMETAZEPAM MAGNOLOL MATHALLATAL MEBUTAMATE MECLOQUALONE MECLOXAMINE MECLOZINE MEDETOMIDINE MENTHOVAL MEPENTAMATE MEQUITAZINE METHALLATAL METHAPYRILENE METHAQUALONE METHARBITAL METHITURAL METHOHEXITAL METHYLCHROMONE METHYLCYCLOBARBITAL-N METHYLPENTYNOL METHYLPHENOBARBITAL METHYPRYLON METOMIDATE MORPHINE MPV-2426 MUREXIDE NARCEINE NARCOBARBITAL NEALBARBITAL NERAMEXANE NF-2 NIAPRAZINE NIMETAZEPAM NISOBAMATE NITRAMARINE NITRAZEPAM NORCHLORPROMAZINE NORHEXOBARBITAL OXOMEMAZINE OXOQUAZEPAM-2

1228 APPENDIX D OXYBATE SODIUM OXYCODONE OXYLIDINE PARALDEHYDE PENTABAMATE PENTENAL PENTHRICHLORAL PENTOBARBITAL PERISOXAL PERLAPINE PETRICHLORAL PHENALLYMAL PHENOBARBITAL PHENOBARBITAL SODIUM PHETHARBITAL PHYTONOXON PIMETHIXENE PROBARBITAL SODIUM PROFEXALONE PROMETHAZINE PROPALLYLONAL PROPIOMAZINE PROPOXATE PROPYLBARBITAL PROXIBARBAL PYRITHYLDIONE QUAZEPAM R-8110 RAPIDORM RECTIDON REPOSAMAL RILMAZAFONE RO-41-3290 RO-41-3696 RO-48-6791 RO-48-8684 RO-5-4864 RO-7-2750 ROLETAMIDE ROMIFIDINE RUPATADINE SANJOININE-G1 SCH-50971 SCOPOLAMINE SECBUTABARBITAL SECOBARBITAL SEDONIUM SHOGAOL-6 SIGMODAL SKF-5390 SR-41378 SULFONALONE SUPIDIMIDE SURICLONE SX-3228 TAK-375 TALBUTAL TAMERIDONE TETRABARBITAL THALIDOMIDE THIALBARBITAL THIOAMOBARBITAL THIOBARBITAL THIOBARBITURATE-2 THIOTETRABARBITAL TIXADIL TOLOXATONE TOLOXYCHLORINOL TOPRILIDINE TRIAZOLAM TRICETAMIDE TRICLOFOS TRIFLUBAZAM TRIONALONE TRK-820 U-90042 URAMIL URETHANE VALDISPERT VALERANONE VALERENATE VALIRACYL VALPERINOL VALTRATE VALTROXAL VINBARBITAL VINYLBITAL WU-385 XYLAZINE ZK-93423 ZOLOPERONE ZOLPIDEM ZOPICLONE SEDIMENTATION CENTRIFUGATION ULTRACENTRIFUGATION SELECTIN-ANTAGONISTS COLCHICINE OC-229-648 P-SELECTIN-GLYCO= PROTEIN-LIGAND-1 TOCOPHEROL SELECTIVE-ESTROGENRECEPTOR-MODULATORS ARZOXIFENE SEROLOGY COMPLEMENT-FIXATION COOMBS-TEST ELISA EMIT ENZYME-IMMUNODET. GONOZYME HEMADSORPTION HEMAGGLUTINATION IMMUNOADSORPTION IMMUNODET. IMMUNODIFFUSION IMMUNOELECTROPHORESIS IMMUNOFLUORESCENCE IMMUNOPRECIPITATION PETINIA PRECIPITIN-REACTION RADIOALLERGOSORBENT RADIOENZYME-IMMUNODET. RADIOIMMUNODET. RADIOIMMUNOSORBENT SEROTONINERGICS 4991-W-93 723-C-86 A-80426 ADATANSERIN ALEPH-2 ALK-3 ALMOTRIPTAN ALNESPIRONE AMINOTRYPTAMINE-5 ANGOLENSATE-METHYL AP-159 AP-521 AS-8 AZ-16596 B-20991 B-695-40 BA-43582A BAY-R-1531 BAY-X-3702 BEA-1654 BEFIPERIDE BENZYLOXYTRYPTAMINE-5 BIMT-17 BIMU-0001 BIMU-1 BIMU-8 BMS-181885 BMS-184111 BP-554 CARBAMOYLTRYPTAMINE-5 CGP-6085-A CGP-6085A CGS-12066A CGS-12066B CGS-18102-A CHLOROPHENYLBIGUANIDE-= META CHLOROPHENYLPIPERAZINE= META CIANOPRAMINE CM-57373 CM-57493 CP-108509 CP-122288 CP-132484 CP-135807 CP-93129 CP-93393 CP-94253 CP-96501 DAU-6236 DIPROPYL-CARBAMOYL= TRYPTAMINE-5 DOI DU-124884 DU-24565 DU-29894 E-3620 ELETRIPTAN ELTOPRAZINE EMD-68843 ERGOVALINE F-13714 FG-5974 GALDANSETRON GR-151004-B GR-46611 GR-49336 HT-90-B HYDROXYDIPROPYLAMINO= TETRALIN-8 HYDROXYTRYPTAMINE-4 HYDROXYTRYPTAMINE-6 IPSAPIRONE KAMPIRONE KAPLAPIRONE KF-66854 L-694247 L-741519 L-741604 L-775606 LEK-8804 LEVOPIRONE LINTOPRIDE LM-5005 LY-228729 LY-274601 LY-301317 LY-315535 LY-334370 LY-344864 LY-41 LY-55 MDL-72832 MDL-73005 MDL-73450 MDL-74217 METHOXYDIMETHYLTRYPTAMINE METHYLAPLYSINOPSIN METHYLQUIPAZINE-N

Derwent Drug File 1229 Thesaurus METHYLSEROTONIN-2 METHYLSEROTONIN-ALPHA METHYLSEROTONIN-N METHYLTRYPTAMINE METHYLTRYPTAMINE-5 METHYLTRYPTOPHAN-ALPHA MJ-13653 MK-462 MKC-242 MKC-733 ML-10302 NDO-008 NS-2359 OLEOYLETHANOLAMINE-N OPC-14523 ORG-37684 PD-158771 PHENYLBIGUANIDE PNU-109291 PRUCALOPRIDE PYRIMIDINYLPIPERAZINE PYRIMIDINYLPIPERAZINE R-76186 RG-12718 RO-60-0175 ROXINDOLE RS-17017 RS-23597 RS-30199-193 RS-42358-197 RS-56532 RS-56812-197 RS-67333 RS-67506 RTI-353 RU-24969 RU-28253 S-14489 S-14506 S-14671 S-15535 S-15931 S-20244 S-20500 S-8849 SANUMGERMAN SARIZOTAN SB-209509 SC-49518 SC-50410 SC-53116 SC-53117 SEROTONIN SEROTONIN-CREATININE-= SULFATE SKF-103829 SKF-99101-H SKK-47029 SN-308 SR-57227A SR-57746A SUMATRIPTAN SUN-8399 SUN-N-4057 SUNEPITRON TEGASEROD TKS-159 TRIFLUOROMETHYLPHENYL= PIPERAZINE-META U-66444B U-92016-A U-93385 WF-31 WY-26157 WY-48723 YM-31636 YM-35992 ZOLMITRIPTAN SERPES-SIMPLEX herpes-keratitis SHOCK GRAY-SYNDROME SICKLE-CELL HEMOGLOBIN-S SKIN DERMIS EPIDERMIS KERATINOCYTE LANGERHAN-CELL MERKEL-CELL STRATUM-CORNEUM STRATUM-SPINOSUM SKIN-TEST MANTOUX-TEST SLEEP DREAMING INSOMNIA NARCOLEPSY NIGHTMARE PARONIRIA REM SLEEP-APNEA SLOW-WAVE SOMNAMBULISM SMELL DYSOSMIA SMOOTH-MUSCLE ANOCOCCYGEUS NICTITATING-MEMBRANE RECTOCOCCYGEUS SOMATOLIBERIN-AGONISTS G-7039 G-7203 G-7502 GHRELIN-HUMAN HEXARELIN JG-73 L-162752 L-163191 L-163540 L-692429 L-692585 L-700653 LY-444711 MK-0677 MZ-2-51 MZ-2-75 MZ-2-87 PRALMORELIN RO-23-7863 SKF-110679 SM-130686 SOMATOCRININ SOMATOCRININ-CATTLE SOMATOCRININ-HUMAN SOMATOLIBERIN SOMATOLIBERIN-1-29 SOMATOLIBERIN-1-29-AMIDE SOMATOLIBERIN-1-29-= AMIDE,NLE-27 SOMATOLIBERIN-1-40 SOMATOLIBERIN-1-44 SOMATOLIBERIN-2 SOMATOLIBERIN-HUMAN-= PANCREATIC-1-29 SOMATOLIBERIN-HUMAN-= PANCREATIC-1-37 SOMATOLIBERIN-HUMAN-= PANCREATIC-1-40 SOMATOLIBERIN-PIG-1-44 SOMATOLIBERIN-RAT SOMATOLIBERIN-RAT-1-29 SOMATOLIBERIN-RAT-1-43 SOMATOLIBERIN-SHEEP-1-44 TABIMORELIN SOMATOSTATIN-AGONISTS 204-090 AN-238 BIM-23003 BIM-23003 BIM-23023 BIM-23026 BIM-23027 BIM-23034 BIM-23056 BIM-23127 BIM-23190 BIM-23197 BM-2-28 BM-23014 CGP-15425 CGP-23996 CH-288 CORTISTATIN DC-13-57 DC-23-99 EC-5-20 JV-1-36 L-362855 L-779976 LANREOTIDE MK-363-301 MK-678 MZ-4-71 MZ-5-156 NC-8-12 OCTREOTIDE PENTETREOTIDE PROSOMATOSTATIN PROSOMATOSTATIN-1-12 PROSOMATOSTATIN-II-= ANGLERFISH RC-101-I RC-121 RC-160-II RC-98-I SANDOZ-201995 SDZ-207-895 SDZ-212-610 SDZ-215-811 SDZ-217-704 SDZ-CO-611 SEGLITIDE SOMATOSTATIN SOMATOSTATIN-D-TRP-8 SOMATOSTATIN-LINEAR SOMATOSTATIN-PHE-4 TT-232 VAPREOTIDE WY-41747 SOMATOTROPIN-AGONISTS L-163191 SOMATOTROPIN SOMATOTROPIN-31-44 SOMATOTROPIN-77-107 SOMATOTROPIN-CATTLE SOMATOTROPIN-DE-MET SOMATOTROPIN-FOWL SOMATOTROPIN-HUMAN SOMATOTROPIN-PIG SOMATOTROPIN-RAT SOMATOTROPIN-SHEEP SOMATOTROPIN-TROUT SOMATOTROPIN-TURKEY

1230 APPENDIX D SOMATREM SOMAVUBOVE SOMETRIBOVE SOMETRIPOR SOMIDOBOVE SOMATOTROPINANTAGONISTS B-2036 CGP-19984 PEGVISOMANT SOMATOTROPIN-HUMAN-= ARG-120 SPASMOLYTICS A-278637 A-29-LUNDBECK AC-119 ACLATONIUM NAPADISILATE ADIPHENINE AF-14 AF-DX-384 AGELASIDINE-A AGELASIDINE-C AGELASIMINE-A AGELASIMINE-B AH-9700 AKLONIN ALBUTOIN ALVERINE AMBUCETAMIDE AMBUTONIUM AMIFLOVERINE AMIKHELLINE AMINOCARBOFLUORENE AMINOPROMAZINE AMIXETRINE AMYL-NITRITE ANDOPAN ANETHOCURARIUM ANGOLENSATE-METHYL APOATROPINE APROFENE APROLIDINE ARPENAL ASPAMINOL ATROMEPINE ATROPINE ATROPINE-ETHIODIDE ATROPINE-METHONITRATE ATROPINE-OXIDE AURAPTEN AURAPTENAL AURICULARATE BAMIFYLLINE BARETTIN BARETTINE BARVERINE BENACTYZINE BENAPRIZINE BENCYCLANE BENDAZOL BENTIPIMINE BENZATROPINE BENZETIMIDE BENZILONIUM BROMIDE BENZILYLCHOLINE BENZOMETHAMINE BENZOPYRRONIUM BROMIDE BENZOYLSCOPOLAMINE BENZYL-ALCOHOL BENZYLMANDELATE BEPERIDIUM IODIDE BEVONIUM METILSULFATE BICYCLOPHENAMINE BIETAMIVERINE BIMAKALIM BIPERIDEN BL-14 BM-5 BOK-1 BORNAPRINE BOTULINUM-A-TOXIN BR-370 BUFLOMEDIL BURODILINE BUTAVERINE BUTETAMATE BUTINOLINE BUTROPIUM BROMIDE BUTYLSCOPOLAMINE BUTYLSCOPOLAMINE = BROMIDE BUZEPIDE-METIODIDE CALCISEPTINE CAMIVERINE CAMYLOFIN CARAMIPHEN CAROVERINE CARZENIDE CAVIDINE CESEDON CHELIDONINE CHLORACYZINE CHLORBENZOXAMINE CHLORBICYCLEN CHLOROSIL CHLORPHENOXAMINE CHLORPROETHAZINE CI-923 CICLACTATE CICLONICATE CICLONIUM BROMIDE CICLOTROPIUM BROMIDE CIMETROPIUM BROMIDE CINNAMAMIDE CINNAMAVERINE CINNAMEDRINE CITRACRIDONE-1 CLIDINIUM BROMIDE CLOFEVERINE CR-1034 CR-1098 CR-1166 CROMAKALIM CYCLANDELATE CYCLARBAMATE CYCLODRINE CYCLOPENTOLATE CYCLOPYRRONIUM BROMIDE CYCRIMINE CYVERINE DAMP-4 DARIFENACIN DECIMEMIDE DECITROPINE DEETHYLOXYBUTYNIN DEHYDROCAVIDINE DEMELVERINE DEMETHYLBUFLOMEDIL-4 DEMETHYLTRIMEBUTINE-N DENAVERINE DEPTROPINE DEPTROPINE-= METHOBROMIDE DEXETIMIDE DEXTROFEMINE DF-594 DIAMIPHENE DICARFEN DICYCLOVERINE DIETHAZINE DIFEMERINE DIHEXYVERINE DIHYDROPAPAVERINE DIISOPROMINE DIMECROTATE DIMENOXADOL DIMEPROZAN DIMETHYLGLYCYLPHENOTHIAZINE DIMETHYLGLYCYLPHENOTHIAZINE DIMETHYLPYRAZINE-2,5 DIMETIPIRIUM BROMIDE DIMEVAMIDE DIMOXYLINE DIOXAPHETYL-BUTYRATE DIPHEMANIL-METILSULFATE DIPHEMIN DIPHENYLTROPINE DIPIPROVERINE DIPONIUM BROMIDE DIPROFENE DISPASMOL DKJ-21 DOMAZOLINE DOTEFONIUM BROMIDE DROCLIDINIUM BROMIDE DROFENINE DROTAVERINE DROTAVERINE-= THEOPHYLLINE-ACETATE ELANTRINE EMEPRONIUM BROMIDE ERITRITYL-TETRANITRATE ET-126 ETAMIPHYLLIN ETEROFEN ETHAVERINE ETOMIDOLINE ETYBENZATROPINE EUCATROPINE EUPAVERIN FC-18-94 FC-20-94 FEBUVERINE FENALAMIDE FENCARBAMIDE FENCLEXONIUM-= METILSULFATE FENOVERINE FENPIPRAMIDE FENPIPRANE FENPIVERINIUM BROMIDE FENTONIUM BROMIDE FISETINIDOL FK-1052 FK-584 FLAMENOL FLAVAMINE FLAVOXATE FLOPROPIONE FLOVERINE FLUOROHEXAHYDRO= SILADIFENIDOL-PARA FLUTROPIUM BROMIDE FUBROGONIUM IODIDE FUROSPONGIN-1 G-3063 GEFARNATE GEPHYROTOXIN GLYCOPYRRONIUM BROMIDE GOE-5438 GUAIACTAMINE GUANYLPIRENZEPINE H-47 H-74 HEMICHOLINIUM HEMICHOLINIUM-15 HEMICHOLINIUM-A-4 HEMICHOLINIUM-A-5 HEPTAVERINE HETERONIUM BROMIDE HEXAHYDRODIFENIDOL

Derwent Drug File 1231 Thesaurus HEXAHYDROSILADIFENIDOL HEXASONIUM IODIDE HEXOCYCLIUM = METILSULFATE HEXOPYRRONIUM BROMIDE HIMBACINE HIMBADINE HOMATROPINE HOMATROPINE = METHYLBROMIDE HYMECROMONE HYOSCYAMINE IBUVERINE IDAVERINE IMIPRAMINE-METHIODIDE IPRAGRATINE IPRATROPIUM BROMIDE ISOMETHEPTENE ISOMYLAMINE ISOPETASIN ISOPROPAMIDE IODIDE JB-318 JB-336 JB-336-4 K-4300 KHELLIN KW-5139 LACHESINE LANPERISONE LEIOPYRROLE LEVCROMAKALIM LEVOMENOL LEVOSULPIRIDE LIPOACONITINE LIPOMESACONITINE LONARID LUFFARIELLOLIDE LY-316108 MANNITOL-HEXANITRATE MARMIN MDL-12330A MDV-2 MEBEVERINE MECINARONE MECLOXAMINE MEFURTRAMINE MELADRAZINE MELETIMIDE MEN-10627 MEPENZOLATE BROMIDE MEPHENOXALONE MEPIPERPHENIDOL METAMIZOLE SODIUM METHAMICIL METHANTHELINIUM = BROMIDE METHOCARBAMOL METHOCTRAMINE METHOXYSILAHEXO= CYCLIUM-ORTHO METHSCOPOLAMINE METHYLBENACTYZIUM = BROMIDE METHYLCHROMONE METINDIZATE METIXENE METOCINIUM IODIDE METOQUIZINE MILVERINE MIMAX MJ-1991 MOBENZOXAMINE MOFLOVERINE MOXAVERINE MYRTECAINE N-1005 N-1024 N-718 NAFIVERINE NAM-204 NAM-224 NAM-242 NAM-250 NARCEINE NICEVERINE NITRAMARINE NITROGLYCEROL NOLINIUM BROMIDE NV-14 NV-15 NV-4 NV-6 OCTAMYLAMINE OCTATROPINE-= METHYLBROMIDE OCTAVERINE OLEUROPEIN ONITIN ORPHENADRINE OTENZEPAD OTILONIUM BROMIDE OXAPIUM IODIDE OXITEFONIUM BROMIDE OXITROPIUM BROMIDE OXYBUTYNIN OXYCLIPINE OXYPHENCYCLIMINE OXYPHENONIUM BROMIDE OXYPYRRONIUM BROMIDE OXYSONIUM IODIDE PAB-12 PAB-13 PAB-13 PAB-23 PAB-23 PAPAVERINE PARAPENZOLATE BROMIDE PARGEVERINE PEDIPHEN PENTAPIPERIDE PENTAPIPERIUM-= METILSULFATE PENTHIENATE PETASIN PETHIDINE PHENGLUTARIMIDE PHENTHIMENTONIUM PHENYTHILONE PHETHARBITAL PHLOROGLUCINOL PICOBENZIDE PIMETREMIDE PINAVERIUM BROMIDE PIPENZOLATE BROMIDE PIPERIDOLATE PIPETHANATE PIPOXOLAN PIRENZEPINE PIROTRAMINE PITOFENONE PK-97 PLATYPHYLLINE POLDINE-METILSULFATE POSKINE PRAMIVERINE PRAMPINE PRENOVERINE PRIDINOL PRIDINOL-MESILATE PRIFINIUM BROMIDE PROCYCLIDINE PROFENAMINE PROMAZINE PROMOXOLANE PROPANTHELINE PROPANTHELINE BROMIDE PROPERIDINE PROPIVANE PROPIVERINE PROPYLBENZILYLCHOLINE-= MUSTARD PROPYROMAZINE BROMIDE PROSPASMIN PROXAZOLE PROXYPHYLLINE PROZAPINE PV-2 PYROPHENDANE QUINOPARINE QURACOL-A QURACOL-B RACEFEMINE RETRACTOR-PENIS-= INHIBITORY-FACTOR RISPENZEPINE RITROPIRRONIUM BROMIDE RO-2-3308 ROCIVERINE S-0121 SALFLUVERINE SALVERINE SAUVAGINE SCOPOLAMINE SECOVERINE SILAHEXOCYCLIUM SILAPROCYCLIDINE SINTROPIUM BROMIDE SOPITAZINE SP-725 SPIROTRAMINE STILONIUM IODIDE STYRAMATE SULPIRIDE SULTROPONIUM SX-284 T-451 TAK-637 TELENZEPINE TERFLAVOXATE TERODILINE THIAZINAMIUM IODIDE THIAZINAMIUM-CHLORIDE THIAZINAMIUM-= METILSULFATE THIAZINAMIUM-SULFOXIDE THIAZINAMIUM-SULFOXIDE = IODIDE THIHEXINOL-= METHYLBROMIDE THYRONAMINE TIEMONIUM IODIDE TIEMONIUM METILSULFATE TIFEMOXONE TIFENAMIL TIGLOIDINE TIMEPIDIUM BROMIDE TIOTROPIUM BROMIDE TIPETROPIUM TIQUINAMIDE TIQUIZIUM BROMIDE TIROPRAMIDE TL-402 TMB-8 TOFENACIN TOLTERODINE TOQUIZINE TRANTELINIUM BROMIDE TREPIBUTONE TREPTILAMINE TRIACANTHINE TRIAMPYZINE TRICLAZATE

1232 APPENDIX D TRICYCLAMOL CHLORIDE TRICYCLAMOL-IODIDE TRIDIHEXETHYL IODIDE TRIETHYLCHOLINE TRIHEXYPHENIDYL TRIMEBUTINE TRIMETHYLDIPHENYL= PROPYLAMINE TRIXOLANE TROPANYL TROPENZILINE BROMIDE TROPICAMIDE TROPIGLINE TROPINE-BENZILATE TROPIRINE TROPODIFENE TROSPIUM CHLORIDE U-247-125 U-247-90 U-247-95 U-247-96 UH-AH-37 UK-84149 UNO-3 UR-8225 UROL VALETHAMATE BROMIDE VAMICAMIDE VETRABUTINE VIQUIDIL W-84 WAY-133537 WAY-151616 WIN-2299 WIN-4981 XENYTROPIUM BROMIDE Y-27632 YENHUSOMINE ZAMIFENACIN ZD-6021 ZD-6169 ZEPASTINE ZICONOTIDE ZOLENZEPINE SPERM POLYSPERMY SPERMATID SPERMATOCYTE SPERMATOGENESIS SPERMATOGONIUM SPERMATOCIDES ALKYLOXYNOL-741 APOGOSSYPOL CDRI-84-35 CELLULOSE-SULFATE CLORINDANOL DIALLYL-TRISULFIDE DL-204-IT GOSSYPOL GOSSYPOL-ACETATE GOSSYPOLONE LONIDAMINE MALVIDIN MENFEGOL NIM-76 NONOXINOL NONOXINOL-10 NONOXINOL-11 NONOXINOL-15 NONOXINOL-20 NONOXINOL-30 NONOXINOL-4 NONOXINOL-40 NONOXINOL-5 NONOXINOL-6 NONOXINOL-9 OCTOXINOL-9 POLIDOCANOL RS-37367 SP-562 SP-563 SP-564 WHI-07 SPINAL-CORD RENSHAW-CELL SPINOCERVICAL-TRACT SPINOTHALAMIC-TRACT WHITE-MATTER ZONA-INTERMEDIA SPINAL-CORD-DISEASE AMYOTROPHIC-LATERAL-= SCLEROSIS AMYOTROPHIC-SYPHILITIC-= MYELITIS ARACHNOIDITIS brown-sequard-syndrome charcot-marie-tooth-= syndrome DANA-SYNDROME ENCEPHALOMYELITIS ENCEPHALOMYELOPATHY familial-spastic-paraplegia FRIEDREICH-ATAXIA HEMIPARAPLEGIA HYPERREFLEXIA LOCOMOTOR-ATAXIA LOUPING-ILL MENINGOENCEPHALOMYELITIS MENINGOMYELOCELE MORVAN-DISEASE MOTOR-NEURON-DISEASE MYELITIS MYELODYSPLASIA MYELOMENINGOCELE neurogenic-bladder neuropathic-musc.atrophy OPTIC-NEUROMYELOPATHY POLIOMYELOMALACIA POLYRADICULONEURITIS RADICULOMYELOENCEPHALITIS RADICULOMYELOPATHY RUST-DISEASE SPINA-BIFIDA spinal-hemiparaplegia struempell-lorrain-disease SUBACUTE-MYELOOPTIC-= NEUROPATHY SYRINGOMYELIA TABES-DORSALIS TESCHEN-DISEASE urinary-retention URINARY-URGENCY WERDNIG-HOFFMANN-= DISEASE SPINAL-FLUID PLEOCYTOSIS SPIROCHAETALES BORRELIA CRISTISPIRA LEPTOSPIRA SERPULINA SPIROCHAETA TREPONEMA SPLEEN MA108-CELL MA200-CELL SPLEEN-DISEASE banti-syndrome chron.congestive-= splenomegaly HEPATOSPLENOMEGALY HYPERSPLENISM SPLENITIS SPLENOMEGALY SPORTS-MED. ATHLETE DOPING SQUALENE-SYNTHASEINHIBITORS BMS-187745 BMS-188494 CP-294838 CP-340868 ER-27856 IBANDRONATE J-104118 RPR-107393 YM-53601 ZARAGOZATE-A ZARAGOZATE-C STABILITY CORROSION DECAY DISCOLORATION SHELF-LIFE STORAGE STEREOCHEM. CIS-ISOMER CONFIG. CONFORMATION D-ISOMER DEXTRO-ISOMER DIASTEREOISOMER L-ISOMER LEVO-ISOMER REGIOSELECTIVE STEREOISOMER STEREOSELECTIVE STEREOSPECIFIC TRANS-ISOMER STEREOISOMER CIS-ISOMER D-ISOMER DEXTRO-ISOMER DIASTEREOISOMER L-ISOMER LEVO-ISOMER TRANS-ISOMER STERILIZATION DISINFECTION PASTEURIZATION STOMACH ABOMASUM ANTRUM CHIEF-CELL FUNDUS GIZZARD OMASUM PARIETAL-CELL PYLORUS RETICULUM STOMATOLOGY APHTHA BAELZ-SYNDROME CHEILITIS CHEILOSIS GINGIVITIS GLOSSITIS GLOSSODYNIA GLOSSOPYROSIS HARELIP LEUKOPLAKIA

Derwent Drug File 1233 Thesaurus malignant-erythema-= multiforme PYOSTOMATITIS RANULA RINDERPEST stevens-johnson-syndrome STOMATITIS STOMATODYNIA URANITIS XEROSTOMIA STROMELYSIN-1-INHIBITORS CGS-27023-A GW-4459 HYDROXYACECLOFENAC-4 PD-166793 STROMELYSIN-INHIBITOR STROMELYSIN-1-INHIBITOR STROMELYSIN-2-INHIBITOR STROMELYSIN-INHIBITORS CGS-27023-A SC-44463 STROMELYSIN-1-INHIBITORS STROMELYSIN-2-INHIBITORS STRUCT.ACT. FREE-WILSON HANSCH SUBCELL.STRUCT. CELL-WALL CHLOROPLAST CHROMATID CHROMATIN CHROMOSOME CYTOPLASM CYTOSOL ENDOPLASMIC-RETICULUM fimbria FLAGELLA GLYOXYSOME GOLGI-APPARATUS HYDROGENOSOME KINETOPLAST LININ LYSOSOME MEMBRANE MICRONUCLEUS MICROSOME MITOCHONDRIA NUCLEOLUS NUCLEOPLASM NUCLEOSOME NUCLEUS PEROXISOME PHAGOLYSOSOME PILUS POLYRIBOSOME SUBSTANCE-P-AGONISTS MDL-103392 NEUROPEPTIDE-GAMMA SENKTIDE SEPTIDE SUBSTANCE-P SUBSTANCE-P-1-4 SUBSTANCE-P-1-6 SUBSTANCE-P-1-7 SUBSTANCE-P-1-8 SUBSTANCE-P-1-9 SUBSTANCE-P-2-11 SUBSTANCE-P-3-11 SUBSTANCE-P-4-11 SUBSTANCE-P-5-11 SUBSTANCE-P-5-9 SUBSTANCE-P-6-11 SUBSTANCE-P-7-11 SUBSTANCE-P-8-11 SUBSTANCE-P-9-11 SUBSTANCE-P-9-PRO SUBSTANCE-P-METHYL-= ESTER SUBSTANCE-P-ANTAGONISTS ANTAGONIST-G APREPITANT CAM-2445 CGP-49823 CJ-12458 CP-100263 CP-141938 CP-96344 CP-96345 CP-99994 CP-II FK-224 FK-888 FR-113680 GR-100679 GR-203040 PROTOPLASM RIBOSOME SPHEROBLAST SUBSTANCE-K-AGONISTS MDL-103392 SUBSTANCE-K-ANTAGONISTS LANEPITANT MEN-10376 MEN-10627 NEPADUTANT SCH-217048 SCH-62373 SR-48968 UK-224671 ZD-6021 GR-205171 HSP-117 L-732138 L-733060 L-741671 L-742694 L-754030 L-758298 LANEPITANT LY-303870 MDL-105212-A MDL-29913 MEN-11149 MK-0869 MK-869 NEPADUTANT NKP-608 PD-154075 RP-67580 RP-68651 RPR-100893 S-18523 S-19752 SCH-62373 SDZ-NKT-343 SPANTIDE SPANTIDE-2 SPANTIDE-2-D-PRO SPANTIDE-5-D-PHE SR-140333 SR-140603 SR-142801 SR-142806 SR-48968 SUBSTANCE-P-2-D-PRO-7,9-= D-TRP SUBSTANCE-P-2-D-PRO-7-= D-PHE-9-D-TRP SUBSTANCE-P-4-11,4-D-= PRO-7,9,10-D-TRP SUBSTANCE-P-7,9,10-D-TRP TAK-637 WIN-51708 WIN-64821 WIN-66306 WS-9326A ZD-6021 SUICIDE-GENE-THERAPY GDEPT SURFACTANTS ABIL-B-8852 ABIL-B8842 ABIL-EM-90 ABIL-WE-09 AMINOXID-WS-35 AMPHOSOL-SP AMPHOTENSIDE ARLATONE-289 ARLATONE-985 ARQUAD-2HT-75 ATLAS-SCS-2054 BKH-14 BL-9 BRIJ-36T C31G CAPMUL-MCM CAPTEX-355 CETIOL-HE CETOMACROGOL CETOSTEARYL-SULFATE CETOSTEARYL-SULFATE = SODIUM CETRIMONIUM CHLORIDE CETYL-BETAINE CHAPSO CHOLYLSARCOSINE CO-610 COCAMIDOPROPYLBETAINE CREMOPHOR-RH40 CREMOPHOR-RH60 CUROSURF DECYL-SULFATE SODIUM DIMETHYLDIOCTADECYL= AMMONIUM BROMIDE DIMODAN-S DISINTEGRON-O DOCUSATE SODIUM DODECLONIUM BROMIDE DODECYLTRIMETHYL= AMMONIUM BROMIDE DODECYLTRIMETHYL= AMMONIUM CHLORIDE EMULGATOR-BTO EMULGIN-B3 EMULPHOR-EL-719 ENTSUFON ETASULFATE SODIUM ETHYLENE-GLYCOL-= MONOSTEARATE FC-72 GENAPOL-PF-10 GLUCAM-E10 HCO-10 HCO-40 HCO-60 HOSTAPHAT-KL340N HOSTAPHAT-KW340N IGEPON-AC-78 L-101 L-121 LAPIRIUM CHLORIDE LAURIMINODIPROPIONATE = SODIUM LAUROYLPROLINE LAUROYLSARCOSINE LAURYL-SULFATE SODIUM

1234 APPENDIX D LAURYL-SULFATE = TRIETHANOLAMINE LUBROL-PX LUNG-SURFACTANT MEGA-10 MEGA-8 MENFEGOL MIRANOL-C2M-CONC.N.P. MIRANOL-MHT MONOOLEIN MONOSTEARIN MUKUROZI-SAPONIN-Y1 MUKUROZI-SAPONIN-Y2 MYRTENAL MYRTENOL MYS-40 MYVACET-9-40 NEONOL-AF9 NIKKOL-AM-101 NIKKOL-SBL-4N NIKKOL-VIFPANT-N NONIDET-P40 NONOXINOL NONOXINOL-10 NONOXINOL-11 NONOXINOL-15 NONOXINOL-20 NONOXINOL-30 NONOXINOL-4 NONOXINOL-40 NONOXINOL-5 NONOXINOL-6 NONOXINOL-9 OCTADECYLTRIMETHYL= AMMONIUMCHLORIDE OCTOXINOL OCTOXINOL-9 OCTYL-GLUCOSIDE OLEYL-SULFATE SODIUM OS-20 P-414 PALMITOYLOLEOYLPHOSPHATI= DYLGLYCEROL PENDECAMAINE PINOCARVEOL POLIDOCANOL POLOXALENE POLOXAMER POLOXAMER-101 POLOXAMER-105 POLOXAMER-108 POLOXAMER-122 POLOXAMER-123 POLOXAMER-124 POLOXAMER-181 POLOXAMER-182 POLOXAMER-184 POLOXAMER-185 POLOXAMER-188 POLOXAMER-215 POLOXAMER-217 POLOXAMER-231 POLOXAMER-234 POLOXAMER-235 POLOXAMER-237 POLOXAMER-238 POLOXAMER-282 POLOXAMER-288 POLOXAMER-331 POLOXAMER-333 POLOXAMER-334 POLOXAMER-335 POLOXAMER-338 POLOXAMER-402 POLOXAMER-403 POLOXAMER-407 POLOXAMER-409 POLOXAMINE-1508 POLOXAMINE-304 POLOXAMINE-904 POLYOXYETHYLENE-= CETOSTEARYL-ETHER POLYOXYETHYLENE-= CETYL-ETHER POLYOXYETHYLENE-= GLYCEROL-MONOLAURATE POLYOXYETHYLENE-= GLYCEROL-MONOOLEATE POLYOXYETHYLENE-= GLYCEROL-= MONORICINOLEATE POLYOXYETHYLENE-= GLYCEROL-= MONOSTEARATE POLYOXYETHYLENE-= GLYCEROL-TRIOLEATE POLYOXYETHYLENE-= GLYCERYL-= MONOISOSTEARATE POLYOXYETHYLENE-= LAURATE POLYOXYETHYLENE-= LAURYL-SULFATE POLYOXYETHYLENE-OLEATE POLYOXYETHYLENE-= OLEYL-ETHER POLYOXYETHYLENE-= STEARATE POLYOXYETHYLENE-= STEARYL-ETHER POLYSORBATE POLYSORBATE-80 PROPYLENEGLYCOL-= MONOLAURATE PROPYLENEGLYCOL-= MONOSTEARATE PROXANOL PROXANOL-168 PROXANOL-268 REWOTERIC-AM-2L ROFETAN-OM ROKOPOL RS-37367 SEBACOYL-CHLORIDE SOLUTOL-HS15 SORBITAN-MONOLAURATE SORBITAN-MONOOLEATE SORBITAN-MONOPALMITATE SORBITAN-MONOSTEARATE SORBITAN-SESQUIOLEATE SORBITAN-TRIOLEATE SORBITAN-TRISTEARATE STANDAPOL-AB45 STEAROYL-LACTYLATE SODIUM SUCROSE-MONOLAURATE SUCROSE-PALMITATE SURFACTANT-KL-4 SURFACTANT-PROTEIN-B SURFACTANT-PROTEIN-B-= HUMAN SURFACTANT-PROTEIN-C SURFACTANT-PROTEIN-C-= CATTLE SURFACTANT-PROTEIN-C-= HUMAN SURFACTIN SURVANTA SYNDET T150R1 TEEPOL TEFOSE TEGIN-M TEGINACID-ML TEGO-BETAIN-L7 TETRABUTYLAMMONIUM TETRADECYLTRIMETHYL= AMMONIUM BROMIDE TEXTAMINE-OXIDE-MP TONZONIUM BROMIDE TRITON-CG-110 TRITON-X-45 TYLOXAPOL VERBENOL VERBENONE WMAP-10 ZLATEMUL-KH50 ZLATEMUL-KHT ZWITTERGENT-3-12 ZWITTERGENT-3-14 ZWITTERGENT-3-16 SURGERY ADENOIDECTOMY AMPUTATION APPENDECTOMY ARTHROPLASTY CAPSULOTOMY CIRCUMCISION COLECTOMY COLPORRHAPHY CONIZATION CRANIOTOMY CRYOSURGERY CRYOTHERAPY CURETTAGE CYSTOLITHECTOMY DEBRIDEMENT DENTISTRY ENUCLEATION EPISIOTOMY ESOPHAGECTOMY EXENTERATION GASTROPLASTY GASTROSTOMY HERNIORRHAPHY HERNIOTOMY HYSTERECTOMY LAPAROTOMY LARYNGECTOMY MASTECTOMY MENISCECTOMY MICROSURGERY NEUROSURGERY OMENECTOMY ORCHIOPEXY PARACENTESIS PNEUMONECTOMY POLYPECTOMY SALPINGO-OVARIECTOMY SIALECTOMY SPHINCTEROTOMY STERNOTOMY SYNOVECTOMY THORACOTOMY THROMBECTOMY TONSILLECTOMY TRABECULECTOMY TRABECULOPLASTY URETHROTOMY VASECTOMY VENECTOMY VENTRICULOTOMY VITRECTOMY SWEAT DIAPHORESIS HYPERHIDROSIS HYPOHIDROSIS PERSPIRATION SWEATING SWEATING HYPERHIDROSIS HYPOHIDROSIS

Derwent Drug File 1235 Thesaurus SYMPATHOLYTICS ACAPRAZINE BOL-148 BUNAZOSIN BUPRANOLOL BUTIDRINE CYVERINE DIBOZANE DIHYDROERGOTAMINE DSP-4 EF-10750 GD-131 GUANETHIDINE H-35-25 IPROXAMINE IPS-339 JCF-9 K-4423 K-4540 KOE-1030 KOE-1313 KOE-1439 KOE-1500 KOE-1560 KOE-1561 KOE-589 KOE-612 KOE-707 L-2 L-741519 L-8040 LY-78335 MA-540 METIROSINE-METHYLESTER PIPEROXAN PIPRATECOL PRANOLIUM CHLORIDE PROSYMPAL RO-3-3528 S-18327 S-464 SANUMGERMAN SKF-7698 SY-14 WR-149024 WR-1729 WR-2823 XYLOCHOLINE YOHIMBATE SYMPATHOLYTICS-ALPHA 1045-U-85 A-119637 A-131701 A-55453 A-75200 A-80426 AAPTAMINE ABANOQUIL ABT-866 ACC-7513 ADIMOLOL AGELASIMINE-A AGELASIMINE-B AH-11110-A AJ-2615 AKUAMMIGINE ALLOYOHIMBINE AMOSULALOL APTAZAPINE AR-C-239 AROTINOLOL ATIPAMEZOLE ATIPROSIN AY-28925 AZAPETINE BAM-1110 BAM-1303 BC-681 BDF-6100 BDF-7572 BDF-8933 BE-1726 BE-2222 BE-2247 BE-2254 BE-2391 BE-2392 BE-2414 BE-6143 BE-7420 BENEXTRAMINE BENOXATHIAN BMY-20064 BREFONALOL BRL-41992 BRL-44408 BRL-44409 BROMERGURIDE BROMOERGOSINE BU-224 BU-E-75 BUTANSERIN BUTIROXAN CGS-10078B CI-927 CL-284027 CP-2907 CP-93393 CRYPTOLEPINE CS-263 CS-265 CYCLAZOSIN D-2343 DA-VIII-MBR DAPIPRAZOLE DC-015 DEMETHYLNAFTOPIDIL DEXEFAROXAN DIHYDROCORYNANTHEINE DIHYDROERGOCORNINE DIHYDROERGOCRISTINE DIHYDROERGOCRYPTINE DIHYDROERGOCRYPTINE-= ALPHA DIHYDROERGOCRYPTINE-= BETA DIHYDROERGOSINE DIHYDROERGOSININE DIHYDROERGOTOXINE DILEVALOL DOXAZOSIN EFAROXAN EPIALLOYOHIMBINE ERGOCORNINE ERGOCRISTINE ERGOCRYPTINE ERGOCRYPTINE-ALPHA ERGOCRYPTINE-BETA ERGOSINE ERGOSININE ERGOTOXINE FCE-22716 FENSPIRIDE FIDUXOSIN FLUPAROXAN FLUPROFYLLINE FR-35447 GW-1818 GYKI-12743 HP-370 HV-723 HYDROXYINDORAMIN-6 HYDROXYTOLAZOLINE-= ALPHA HYDROXYYOHIMBINE-11 HYMENIN IDAZOXAN IK-29 IMILOXAN INDORAMIN IP-66 JTH-601 K-3827 K-4011 K-42999 K-4300 KF-4307 KF-4317 KF-4942 KMD-3213 L-639019 L-654284 L-657743 L-659066 L-762459 L-765314 LABEDIPINEDILOL-A LABETALOL LR-693 LY-062 LY-134046 LY-158A LY-165163 LY-253352 MEDROXALOL METAZOSIN METHYLDOBUTAMINE-O-3 METHYLURAPIDIL-5 MIDAGLIZOLE MK-467 MONATEPIL MOXISYLYTE N-1518 NAFTOPIDIL NAPAMEZOLE NESAPIDIL NIGULDIPINE NNC-22-0031 NORHARMAN OPC-28326 PHENOXYBENZAMINE PHENTOLAMINE PRAZOSIN PROMETHAZINE-= HYDROXYETHYL PROROXAN PROXODOLOL PSEUDOYOHIMBINE PYREXTRAMINE PYRROXANE QF-503 QF-603 QF-607 R-51703 REC-0-0232 REC-15-2615 REC-15-2627 REC-15-2636 REC-15-2739 REC-15-2802 REC-15-2841 REC-15-3039 ROPINIROLE RP-55462 RS-100975 RS-15385-197 RS-17053 RS-79948-197 RU-49041 RU-52583 RX-801074

1236 APPENDIX D RX-801079 RX-811005 RX-811033 RX-811054 RX-811059 RX-821002 RX-821002-A RX-821037A S-10089 S-18327 S-2150 S-9871 SATERINONE SB-216469-S SC-46264 SGB-1534 SGB-483 SHI-437 SKF-101253 SKF-104078 SKF-104856 SKF-550 SKF-625A SKF-85738 SKF-89124 SL-860714 SL-860715 SL-890591 SM-2470 SM-911 SNAP-1069 SNAP-5089 SNAP-5150 SNAP-5399 SNAP-5582 SNAP-6201 ST-89 SUNEPITRON SY-28 SZL-49 TAMSULOSIN TETRAHYDROCOPTISINE TETRAHYDRONORHARMAN TIBALOSIN TIPENTOSIN TOLAZOLINE TOLNAPERSINE TRIMAZOSIN TRIPAMIDE WB-4085 WB-4093 WB-4101 WB-4109 WY-25309 WY-26392 WY-26703 WY-27127 XB-513 YM-11133 YM-12617 YOHIMBINE YOHIMBINE-ALPHA ZK-112566 ZK-33839 SYMPATHOLYTICS-BETA 18-502 20-785 204-155 204-545 21009 AC-623 ACC-9129 ACC-9369 ACEBUTOLOL ADAPROLOL ADIMOLOL AFUROLOL AH-3474 ALPRENOLOL ALPRENOLONE-METHOXIME ALPRENOXIME AMOSULALOL APOYOHIMBINE ARNOLOL AROTINOLOL ATENOLOL AY-28925 B-24-76 BEFUNOLOL BENZYLAMINOCHLORETHYL BETAXOLOL BEVANTOLOL BFE-37 BFE-41 BFE-47 BFE-55 BFE-61 BFE-69 BFE-72 BISOPROLOL BL-343AC BL-443 BM-140830 BOMETOLOL BOPINDOLOL BOPINDOLOL-HYDROLYZED BORNAPROLOL BREFONALOL BROMOACETYLALPRENOLOL= MENTHANE BROMOACETYLPINDOLOL= MENTHANE BUCINDOLOL BUCUMOLOL BUFETOLOL BUFURALOL BUNITROLOL BUNOLOL BUTOCROLOL BUTOFILOLOL BUTOXAMINE BW-A575C BW-B385C CAPSINOLOL CARAZOLOL CARPINDOLOL CARTEOLOL CARVEDILOL CAS-413 CELIPROLOL CETAMOLOL CGP-12177 CGP-12177A CGP-12388 CGP-17582B CGP-20712A CGP-26505 CGS-10078B CICLOPROLOL CK-3579 CLORANOLOL CYANOPINDOLOL DEACETYLMETIPRANOLOL DEMETHYLCARVEDILOL DENITRONIPRADILOL DEXPROPRANOLOL DIACETOLOL DICHLOROISOPRENALINE DIHYDROALPRENOLOL DIHYDROLEVOBUNOLOL DILEVALOL DIOXADILOL DIOXIFEDRINE DOXAMINOL DRAQUINOLOL EPANOLOL ESMOLOL ESPROQUINE EUGENOLOL EXAPROLOL EXP-063 FA-33 FALINTOLOL FLESTOLOL FLUMOLOL FLUSOXOLOL FP-33 GI-104313 H-105-22 H-119-66 H-29-50 H-64-52 H-87-07 HX-CH-44-BS HYDROXYALPRENOLOL-4 HYDROXYBENZYLPINDOLOL HYDROXYBEVANTOLOL-4 HYDROXYCARTEOLOL-8 HYDROXYMETOPROLOL-= ALPHA HYDROXYPROPRANOLOL HYDROXYTERTATOLOL-4 I-06 ICI-118551 ICI-147798 ICI-46037 ICI-89406 IDROPRANOLOL INDENOLOL IODOAMINOFLISOPOLOL IODOPINDOLOL IPROCROLOL ISAMOLTAN KF-4317 KOE-1124 KOE-1350 KOE-1411 KOE-3290 L-643717 L-653328 LABEDIPINEDILOL-A LABETALOL LEVOBUNOLOL LEVOMOPROLOL LK-203-030 LL-21945 LY-377604 MEDROXALOL MEPINDOLOL METALOL METHYLSEROTONIN-ALPHA METIPRANOLOL METOPROLOL MINDODILOL MJ-7434-1 MK-761 MOPROLOL MY-336-A N-1518 NADOLOL NAFETOLOL NAPHTHOXYLACTATE NEBIVOLOL NIFENALOL NIPRADILOL ONO-1101 ONO-SA-132 OXPRENOLOL P-0160 P-11 PAFENOLOL

Derwent Drug File 1237 Thesaurus PAMATOLOL PARGOLOL PENBUTOLOL PENIROLOL PH-QA-33 PHENITRONE PICODRALAZINE PINDOLOL PRACTOLOL PRIMIDOLOL PRIZIDILOL PROCINOLOL PRONETALOL PROPRANOLOL PROPRANOLOL-ACETATE PROXODOLOL R-67138 R-67145 RIDAZOLOL RO-3-7410 RO-3-7894 RO-31-1118 SKF-95018 SOLYPERTINE SOQUINOLOL SOTALOL SPIRENDOLOL SR-59230-A TA-073 TALINOLOL TE-176 TERTATOLOL TIENOXOLOL TILISOLOL TIMOLOL TIMOLOL-BUTYRATE TIPRENOLOL TOLAMOLOL TOLIPROLOL TZC-1370 TZC-5665 UK-1745 USVC-6524 VANINOLOL XIBENOLOL XIPRANOLOL YM-151 YM-16151-1 YM-430 ZAMI-1305 ZAMI-1327 SYMPATHOMIMETICS A-61603 AA-497 ABIADIN ALFETAMINE BAMETHAN BRL-35135A BUTYLETHARINE CC-34 DIMETHYLADRENALINE DIPIVEFRINE ETHYLNORANTIFEINE FLUORODOPAMINE-6 H-75-12 H-77-77 HIGENAMINE HORDENINE HYDROXYDOPAMINE-5 INDOPAN ISOPHENEPHRINE JOD-173 KWD-2312 L-4035 M-6434 M-8 METATEROL METHOXYPHEDRINE METHYLAMINOREX-4 MJ-7999-1 NORPSEUDOEPHEDRINE NS-2359 NS-49 OENETHYL OXIDOPAMINE PIVENFRINE QH-25 S-18149 SKF-88444 SM-220-CL ST-585 TK-174 TL-102 TL-137 TL-140-III TL-224 TL-259 TL-334 TYROSINE-METHYLESTER UK-14819 WIN-513 XYLOPROPAMINE SYMPATHOMIMETICS-ALPHA 44-549 A-53693 A-54741 A-57219 A-61603 A-68930 ABT-866 ADRAFINIL ADRENALINE ADRENALONE AGN-190851 AGN-191103 AGN-193080 AMEZINIUM METILSULFATE AMIDEFRINE MESILATE AMPHETAMINE APRACLONIDINE AZEPEXOLE AZIDOCLONIDINE-PARA BDF-7579 BENAZOLINE BHT-958 BRIMONIDINE CENTAQUINE CENTHAQUIN CH-38083 CIRAZOLINE CLONIDINE CLONIDINE-DISPLACING-= SUBSTANCE CORBADRINE COUMAZOLINE CYCLOPENTAMINE DEOXYADRENALINE DEXAMPHETAMINE DEXMEDETOMIDINE DIMETOFRINE DJ-7141 DOCARPAMINE DOPAMINE DQ-2511 EPHEDRINE EPINEPHRYL-BORATE ETILEFRINE ETILEFRINE-PIVALATE FENOXAZOLINE FLUORONORADRENALINE-6 FLUOROPHENYLEPHRINE-2 FLUOROPHENYLEPHRINE-4 FLUOROPHENYLEPHRINE-6 FLUTONIDINE GEPEFRINE GUANABENZ GUANFACINE HP-184 HYDROXYAMPHETAMINE HYDROXYEPHEDRINE IBOPAMINE ICI-101187 ICI-106270 IDRALFIDINE INDANIDINE IODOCLONIDINE-PARA ISOMETHEPTENE ISOPROPYLMETHOXAMINE K-6341 K-6343 KABI-2023 L-762459 LD-2855 LEVOMEDETOMIDINE LOFEXIDINE M-7 MEDETOMIDINE MEPHENTERMINE METANEPHRINE METARAMINOL METHAMPHETAMINE METHOXAMINE METHYLADRENALINE METHYLDOPA MIDODRINE MIVAZEROL MODAFINIL MOXONIDINE MPV-1440 MPV-207 MPV-2426 MPV-295 MPV-304 MPV-305 MPV-390 NAPHAZOLINE NORADRENALINE NOREPHEDRINE NORFENEFRINE NORMETANEPHRINE OCTODRINE OCTOPAMINE OXYMETAZOLINE P-5369 PHENAMAZOLINE PHENPROMETHAMINE PHENYLEPHRINE PHOLEDRINE PNO-49-B PROPYLHEXEDRINE PSEUDOEPHEDRINE RILMENIDINE ROMIFIDINE RX-801074 S-12813-4 S-8350 SDZ-NVI-085 SKF-102652 SKF-35886 SKF-89748 SKF-89748-A ST-1059 ST-1943 ST-450 ST-464 ST-475 ST-476 ST-587 ST-606 ST-666

1238 APPENDIX D ST-732 ST-91 ST-95 STH-2100 STH-2169 STH-2224 SYNEPHRINE TALIPEXOLE TETRAMINOL TETRYZOLINE TIAMENIDINE TIZANIDINE TL-232 TL-333 TOLONIDINE TRAMAZOLINE TUAMINOHEPTANE TYMAZOLINE TYRAMINE UCB-22073 UK-11957 UK-15121 WHR-1049 WHR-1370A XYLOMETAZOLINE SYMPATHOMIMETICS-BETA ADRENALINE AFORMOTEROL AH-3021 ALIFEDRINE AMPHETAMINE AR-C-68397-AA ARBUTAMINE ASL-7022 BITOLTEROL BMS-210285 BRL-26830-A BRL-26830A BRL-28410 BRL-35113 BRL-35135 BRL-37344 BRL-37344-A BRL-47672 BROXATEROL BUPHENINE BUTYLOCTOPAMINE-N-TERT. CARBUTEROL CC-25 CIMATEROL CL-316243 CLENBUTEROL CLORPRENALINE COLTEROL CRL-40827 D-2343 DENOPAMINE DETERENOL DEXAMPHETAMINE DIOXETHEDRIN DOBUTAMINE DOCARPAMINE DOPAMINE DOPEXAMINE EPHEDRINE EPINEPHRYL-BORATE ETAFEDRINE ETANTEROL ETHYLNORADRENALINE ETILEFRINE ETILEFRINE-PIVALATE FENOTEROL FLUOROMETARAMINOL-6 FLUORONORADRENALINE-2 FLUOROPHENYLEPHRINE-2 FLUOROPHENYLEPHRINE-6 FORMOTEROL GP-2-128 GP-2-128-7 HEXOPRENALINE HSR-81 HYDROXYAMPHETAMINE HYDROXYEPHEDRINE IBUTEROL ICI-198157 ICI-201651 ICI-215001 ICI-D-7114 ISOETARINE ISOPRENALINE JOD-176 KM-13 KUR-1246 KWD-2016 KWD-2023 KWD-2027 KWD-2110 KWD-2131 KWD-2313 KWD-2314 L-640033 L-644969 L-665871 L-755507 L-770644 L-796568 LEVOSALBUTAMOL LY-206243 LY-377604 LY-79771 MABUTEROL ME-506 MELUADRINE MEPHENTERMINE METARAMINOL METHAMPHETAMINE METHOXYPHENAMINE METHYLADRENALINE METHYLEPHEDRINE NAMINTEROL NORBUDRINE NOREPHEDRINE ORCIPRENALINE P-5369 PHOLEDRINE PICUMETEROL PIRBUTEROL PRENALTEROL PROCATEROL PROTOKYLOL PSEUDOEPHEDRINE R-0363 REPROTEROL RIMITEROL RITODRINE RO-16-8714 RO-363 RO-40-2148 RU-42173 SALBUTAMOL SALMEFAMOL SALMETEROL SM-11044 SOM-1122 SOM-1397-CL SOTERENOL SR-58306A SR-58372 SR-58373-A SR-58373A SR-58375A SR-58539B SR-58572A SR-58575A SR-58589 SR-58590 SR-58611A SR-58612A SR-58613A SR-58825A SR-59104-A SR-59119-A SULFONTEROL T-0509 T-1583 T-3660 TA-2005 TERBUTALINE TJ-15 TRETOQUINOL TULOBUTEROL TV-399 TYRAMINE XAMOTEROL ZD-2079 ZD-9989 ZINTEROL SYNERGISTS AG-2037 AHC-52 ALPHA-D-MANNOSIDASE ALRT-1550 ARC-69931-MX AVI-4126 BAL-9611 BENZYLGUANINE-O-6 BETAMIPRON BIBW-22-BS BIRICODAR BL-P-2013 BMS-214662 BNP-7787 BRL-42715 BROBACTAM BROMOPENICILLANATE-6-= BETA BX-471 CARBOXYPEPTIDASE-G2 CD-2247 CERAMIDE-C6 CFT-1201 CGX-571 CHS-828 CILASTATIN CL-329753 CLAVULANATE CMT-1 CP-461 CRONAXIL CS-834 CV-787 DC-101 DEHYDROSTIPIAMIDE-6,7 DEXTRANASE DMP-963 DPC-083 DPC-961 ENIPORIDE FLT-3-LIGAND FLUMECINOL FOSCOLATE GALACTOSE-OXIDASE GAR-936 GD-40 GIMERACIL GP-27 GW-8510 GW-974 H-87 HAPALOSIN

Derwent Drug File 1239 Thesaurus HATOMARUBIGIN-B HATOMARUBIGIN-C HERVELINE-A HERVELINE-B HERVELINE-C HEXENAL-2 HX-600 HX-630 HYB-190 I-152 ILX-23-7553 INTERLEUKIN-18 IROFULVEN JENISSEENSOSIDE-C JENISSEENSOSIDE-D L-778123 LFM-A-13 LILLY-18947 LUF-5484 LY-301621 LY-329146 LY-335979 LY-465803 LY-487355 LY-509207 LYSINE-COPPER MC-02479 MDL-201307 MGK-264 MICAFUNGIN MK-789 MS-209 MYELOPOIETIN N-5228 NAPHTHOFLAVONE-ALPHA NB-1011 NK-250 NK-252 NLCQ-1 NSC-330507 NU-1025 NU-1064 OC-144093 ORI-1202 PD-0183085 PD-184352 PI-88 PIPERAFIZINE-A PIPERONYL-BUTOXIDE PIVSULBACTAM PKI-166 PROADIFEN PROLINE-DITHIOCARBAMATE PROXIFEINE R-101933 RESOBENE RO-15-1903 RS-33295-198 RS-74513-000 RUBIGINONE-A1 RUBIGINONE-A2 RUBIGINONE-B1 RUBIGINONE-B2 RUBIGINONE-C1 RUBIGINONE-C2 RVC-556 S-16317 S-16324 S-9788 SARCOSINE-= DITHIOCARBAMATE SB-214751 SB-218018 SB-RA-31012 SCH-56582 SESAMEX SESAMOLIN SF-2103A SIB-1508-Y SKF-8742-A SQ-28504 SQ-28546 SR-11238 SULBACTAM SULFAMETHOXAZOLE-= HYDROXYLAMINE SULPHIMIDAZOLE SYN-2190 TAZOBACTAM TORILIN TP-72 TST-220 TST-334 UC-781 VALSPODAR VATALANIB VX-710 XR-9051 XR-9576 ZD-6126 SYPHILIS AMYOTROPHIC-SYPHILITIC-= MYELITIS BABINSKI-SYNDROME bayle-disease CHANCRE CLUTTON-SYNDROME LOCOMOTOR-ATAXIA NEUROSYPHILIS paralytic-dementia TABES-DORSALIS TABLET DRAGEE TELOMERASE-INHIBITORS CERAMIDE-C6 CISPLATIN NSC-714187 RO-25-4020 TELOMESTATIN TEMPERATURE COLD COOLING CRYOSCOPY CRYOTHERAPY HEAT HEATING WARM TERATOGENESIS CLEFT-LIP CLEFT-PALATE ECTRODACTYLY TERATOMA TERA-C-CELL TESTIS EPIDIDYMIS LEYDIG-CELL MESORCHIUM MUELLERIAN-DUCT SCROTUM seminal-vesicle SERTOLI-CELL SPERMATIC-CORD VAS-DEFERENS TESTIS-DISEASE CRYPTORCHIDISM EPIDIDYMITIS EPIDIDYMO-ORCHITIS EUNUCHOIDISM FERTILE-EUNUCH-SYNDROME FUNICULITIS HYDROCELE ORCHIALGIA ORCHITIS PERIORCHITIS SEMINOMA TESTICULAR-DYSGENESIS-= SYNDROME VARICOCELE THALAMUS HABENULA THERMODYNAMICS ENTHALPY ENTROPY FREE-ENERGY THIRST ADIPSIA HYPERDIPSIA POLYDIPSIA THROMBIN-INHIBITORS ARGATROBAN BCH-2763 BOTHROJARACIN CRC-220 CVS-995 DUP-714 EFEGATRAN HEPARIN HEPARIN SODIUM HIRUDIN HIRUDIN-LYS-47 HIRULOG-1 INOGATRAN INTIMATAN LB-30057 MELAGATRAN NAPSAGATRAN RWJ-56110 RWJ-58259 S-2238 S-2366 TRIABIN THROMBOLYTICS A-74187 ACYLSTREPTASE AK-124 ALTEPLASE ANISTREPLASE ANNEXIN-II ARC-69931-MX ASTRAGALOSIDE AT-1015 ATROXASE AVELIZINE BISOBRIN BITISTATIN BM-06-021 BM-06-022 BM-573 BRINASE BRL-26920 BRL-33575 BX-807834 CERASTASE-F4 CGP-42934 CGP-42935 CLOTTING-FACTOR-XA CP-2129-AL CS-747 CVS-1123

1240 APPENDIX D CVS-995 D-K2P DEFIBRINOTIDE DIAMIPHENE DPC-423 DUTEPLASE E-6010 ECKOL ECOTIN EFEGATRAN EICOSAPENTAENOATE-= ETHYL-ESTER ELAROFIBAN FIBROLASE FXV-673 G-11021 G-11035 GALACTAN-POLYSULFATE GEA-3175 GT-12 HEMENTIN HFV-1017-C HIRUGEN HYALURONIDASE INICARONE K2P L-722151 LEPIRUDIN LONGOLYTIN LOTRAFIBAN LU-58463 LY-210825 MONTEPLASE MORIKRASE NATTOKINASE ORBOFIBAN ORG-36764 P-SELECTIN-GLYCO= PROTEIN-LIGAND-1 PEROXYNITRITE PLACTIN-D PLASMIN PLASMINOGEN-ACTIVATOR PLASMINOGEN-ACTIVATOR-= BAT PLASMINOGEN-ACTIVATOR-= DELTA-FE1X PLASMINOGEN-ACTIVATOR-= DELTA-FE3X PLASMINOGEN-ACTIVATOR-= GLU-275 PLASMINOGEN-ACTIVATOR-= HUMAN PLASMINOGEN-ACTIVATOR-= MELANOMA PLASMINOGEN-ACTIVATOR-= TNK PLASMINOGEN-LYS PRO-UROKINASE PRO-UROKINASE-HUMAN PROTEASE-C RETEPLASE ROXIFIBAN RPR-110173 RPR-130737 RWJ-56110 S-18204 S-18326 SARUPLASE SB-214857 SC-49992 SDZ-MTH-958 STAPHYLOKINASE STREPTOKINASE STREPTOKINASE-PLASMIN-= ACTIVATOR SUN-9216 TENECTEPLASE TERRILYTINE TRIDEGIN U-46195 UROKINASE WB-3559-A WB-3559-B WB-3559-C WB-3559-D XR-1853 XR-334 XR-5082 XR-5118 XT-199 YM-337 YM-866 THROMBOSIS AIR-EMBOLISM CESTAN-CHENAIS-= SYNDROME FAT-EMBOLISM HUGHES-STOVIN-SYNDROME LERICHE-SYNDROME PHLEBOTHROMBOSIS pulmonary-embolism THALAMIC-SYNDROME THROMBOANGIITIS THROMBOENDOCARDITIS THROMBOPHLEBITIS THROMBUS THROMBOXANE-AGONISTS AGN-191976 AGN-192093 DEHYDROTHROMBOXANE-= B2-11 DINORTHROMBOXANE-B22,3 EP-011 EP-031 EP-109 EP-171 I-BOP ICI-79939 ICI-86841 PGH2-AZO-9,11 SQ-26655 STA-2 THROMBOXANE-A1 THROMBOXANE-A2 THROMBOXANE-B1 THROMBOXANE-B2 U-44069 U-46619 THROMBOXANEANTAGONISTS ACETYLEUGENOL AH-19437 AH-23848 AH-23848B AR-12-456 AR-12463 AZAPROSTANOATE-13 BAY-U-3405 BENZYLIMIDAZOLE-1 BM-500 BM-519 BM-531 BM-567 BM-573 BMS-180291-02 BREVISCAPINE BW-755C C-85 CBS-1108 CGS-12970 CGS-15435-A CGS-15435A CGS-22652 CINNAMOPHILIN CK-53 CL-871502 CV-6504 DALTROBAN DAZMEGREL DAZOXIBEN DT-TX-30 DT-TX-30-SE E-3040 EP-035 EP-045 EP-092 EP-157 F-1322 FCE-22178 FCE-24265 FCE-27262 FR-140423 FUREGRELATE G-25671 G-31442 G-33378 G-619 GR-32191B GR-36246 HN-11500 HOE-944 IBI-P-05006 ICI-159995 ICI-180080 ICI-185282 ICI-192605 ICI-D1542 IFETROBAN IMIDAZOLE (Drug) IMIDAZOLE SALICYLATE ISBOGREL KDI-792 KF-4939 KME-4 KT-2-962 KW-3635 KW-4099 L-636499 L-641953 L-655240 L-657925 L-657926 L-670596 LCB-2853 LIGSTROSIDE LINOTROBAN MASTICADIENONATE MIDAZOGREL MR-948 N-0164 NAFAGREL NAFAZATROM NITROACETYLSALICYLATE NIZOFENONE NQ-Y-15 OKY-1580 OKY-1581 ON-579 ONO-11120 ONO-1301 ONO-3708 ONO-8809 ONO-NT-126 OZAGREL PC-88 PINANE-THROMBOXANE-A2 PIRMAGREL RIDOGREL RO-22-7878

Derwent Drug File 1241 Thesaurus RO-23-0238 RO-23-3423 RO-24-0238 RS-5186 RWJ-63556 S-145 S-1452 S-18204 S-18886 SC-38249 SCH-37224 SERATRODAST SKF-88046 SQ-26536 SQ-27427 SQ-28668 SQ-28852 SQ-29535 SQ-29548 SQ-30741 SQ-33261 SQ-33552 SQ-33961 SULOTROBAN TEI-4120 TER-930180 TERBOGREL TICLOPIDINE TRILOBINE U-51605 UK-101613 UK-102333 UK-141161 UK-147535 UK-49883 UP-116-77 VAPIPROST Y-19018 Y-19432 Y-20811 YM-57158 Z-335 ZK-110841 THYMIDINE-KINASEINHIBITORS L-653180 ZIDOVUDINE THYMIDYLATE-SYNTHASEINHIBITORS 1843U89 AG-331 AG-337 BW-1843U89 CB-300638 CB-300907 CB-30900 FLUORODEOXYCYTIDINE-= PHOSPHATE FLUOROURACIL FOLINATE CALCIUM ICI-198583 LY-231514 MOBILETREX NB-1011 RALTITREXED TYLOPHORINIDINE ZD-9331 THYMOCYTE CD4+-CELL CD8+-CELL HELPER-CELL MT4-CELL SUPPRESSOR-CELL TH1-CELL TH2-CELL THYMOCYTIC EB-LYMPHOMA ESB-LYMPHOMA THYMOMA EL4-CELL THYMUS TLX5 THYMUS-DISEASE NEZELOF-SYNDROME THYMIC-ALYMPHOPLASIA THYMOMA TLX5 THYMUS-HORMONES IRI-426 LEUCOGENENOL PARATHYMOSIN-ALPHA PROTHYMOSIN-ALPHA RGH-0205 RGH-0206 THYMALINE THYMIC-FACTOR THYMIC-FACTOR-GAMMA-2 THYMOGEN THYMOHEXIN THYMOLYMPHOTROPIN THYMOMODULIN THYMOPENTIN THYMOPOIETIN THYMOPOIETIN-II THYMOPTIN THYMOSIN THYMOSIN-ALPHA-1 THYMOSIN-ALPHA-11 THYMOSIN-BETA-10 THYMOSIN-BETA-4 THYMOSIN-BETA-9,MET THYMOSIN-V THYMOTROPIN THYMULIN THYMUS-EXTRACT THYROID-DISEASE CRETINISM debre-semelaigne-syndrome GOITER HYPERTHYROXINEMIA hypothyroid-myopathy HYPOTHYROIDISM PENDRED-SYNDROME THYROIDITIS THYROTOXICOSIS THYROID-HORMONES CALCITONIN CALCITONIN-EEL CALCITONIN-FOWL CALCITONIN-HUMAN CALCITONIN-PIG CALCITONIN-RAT CALCITONIN-SALMON CALCITONIN-SALMON-I DESICCATED-THYROID DEXTROTHYROXINE SODIUM DIIODOTHYRONINE DIIODOTYROSINE DIMIT ELCATONIN LEUCOGENENOL LEVOTHYROXINE SODIUM MONOIODOTHYRONINE RATHYRONINE SKF-L-12276 THYROGLOBULIN THYROIDIN THYRONINE THYROPROPATE THYROXINE TRIIODOTHYRONINE TRIIODOTHYRONINE-REVERSE THYROIDITIS hashimoto-thyroiditis THYROLIBERIN-AGONISTS CYCLO-HIS-PRO DEAMIDOTHYROLIBERIN DN-1417 JTP-2942 MK-771 MONTIRELIN MONTIRELIN OROTIRELIN PHYLADOX RX-77368 TA-0910 THYROLIBERIN THYROLIBERIN-T YM-14673 THYROMIMETICS CGS-26214 IODINATED-CASEIN PROLONIUM IODIDE SKF-L-94901 TIRATRICOL TYROMEDAN THYROTROPIN-AGONISTS THYROTROPIN THYROTROPIN-CATTLE THYROTROPIN-HUMAN THYROTROPIN-RAT TIME PHOTOPERIOD TISSUE-CULTURE 1321N1-CELL 3LL-CELL 3T3-CELL 3T6-CELL 9L-CELL A15-CELL A1847-CELL A204-CELL A253-CELL A31-CELL A427-CELL A549-CELL ABPL2-CELL AD6-CELL AH130-CELL AH66-CELL AKR-CELL AP9-CELL B16-CELL B16A-CELL B35M-CELL B4-CELL B4976-CELL B82-CELL BCL1-CELL BE-CELL BEN-CELL BHK-CELL BHK21-CELL BT20-CELL BT474-CELL BW5147-CELL C1300-CELL C3H2K-CELL C6-GLIAL-CELL CACO2-CELL

1242 APPENDIX D CAOV-CELL CASKI-CELL CBT-CELL CC531-CELL CCD18-CELL CCF-CELL CCL84-CELL CCRF-CEM-CELL CH23-CELL CHO-CELL CHP126-CELL CLOUDMAN-CELL CLOUDMAN-S91-CELL CO115-CELL CT26-CELL CV1-CELL DAUDI-CELL DETROIT-562-CELL DLD1-CELL DON-CELL DT5-CELL DU145-CELL DUNNING-R3327H-CELL EB-CELL EB2-CELL EHB-CELL EHRLICH-ASCITES-CELL EL4-CELL ELCO2-CELL EMT6-CELL ESB-CELL FIBROBLAST FLOW2002-CELL FRIEND-LEUKEMIA-CELL FSD1-F4-CELL G-CELL G8-CELL GLV3-CELL GM258-CELL GROSS-LEUKEMIA-CELL H157-CELL H35-CELL H4-CELL HAB-CELL HAK-CELL HARDING-PASSEY-CELL HBT3-CELL HCCL-CELL HCT-CELL HCT116-CELL HCT8-CELL HEK-CELL HELA-CELL HEP-G2-CELL HEP2-CELL HEPA1-CELL HEY-CELL HL60-CELL HOC1-CELL HOC7-CELL HRIK-CELL HSO578-CELL HT1080-CELL HT29-CELL HTC-CELL HUT102B2-CELL HUT11-CELL HUTU80-CELL huvec HX13-CELL HX18-CELL HX29-CELL IBRS2-CELL IM9-CELL J111-CELL JEG3-CELL JURKAT-CELL K562-CELL KB-CELL KG1-CELL KPI-CELL KU1-CELL L-CELL L1210-CELL L12R4-CELL L132-CELL L1321-CELL L2C-CELL L40-CELL L5222-CELL L929-CELL LAZ007-CELL LEWIS-LUNG-CARCINOMA-= CELL LLC-MK2-CELL LLC-PK1-CELL LLC-RK1-CELL LM-CELL LOVO-CELL M1-CELL M109-CELL M21-CELL M5-CELL MA104-CELL MA108-CELL MA160-CELL MA200-CELL MBL2-CELL MBT2-CELL MC5-5-CELL MC7-CELL MCB6-1-CELL MCF7-CELL MDBK-CELL MDCK-CELL ME180-CELL METH-A-CELL MG34-CELL MG63-CELL MGH41-CELL MGHV1-CELL MH134-CELL MKN1-CELL MKN28-CELL MKN45-CELL ML1-CELL MM253-CELL MOLT3-CELL MOLT4-CELL MOPC-CELL MOPC173-CELL MORRIS-HEPATOMA-CELL MOT-CELL MPC11-CELL MT4-CELL NEMETH-KELLNER-CELL NG108-15-CELL NH1K-3025-CELL NIE115-CELL NOVIKOFF-HEPATOMA-CELL NS1-CELL NS20-CELL OVCAR2-CELL OVCAR3-CELL OVCAR4-CELL OVCAR5-CELL P388-CELL P815-CELL P815Y-CELL PC1-CELL PC10-CELL PC12-CELL PC9-CELL PK15-CELL POC-CELL QG56-CELL QG90-CELL R3230AC-CELL RAG-CELL RAJI-CELL RD-CELL RIF1-CELL RK13-CELL RNF22-CELL RPMI0041-CELL RPMI1346-CELL RPMI1846-CELL RPMI2650-CELL RPMI6410-CELL RPMI8402-CELL RR1022-CELL RT112-CELL RTG2-CELL S49-CELL S91-CELL SA1-CELL SA2-CELL SA5-CELL SA9-CELL SARCOMA-180-CELL SARCOMA-37-CELL SARCOMA-45-CELL SF126-CELL SF375-CELL SF407-CELL SH3-CELL SK-HEP1-CELL SK-MEL28-CELL SK-MEL37E-CELL SK-OV-CELL SKL2-CELL SKL5-CELL ST-BALB-CELL ST-CELL SV80-CELL SW1271-CELL SW403-CELL SW48-CELL SW480-CELL SW620-CELL SW900-CELL T24-CELL TA3-CELL TANG-CELL TE85-CELL TEPC15-CELL TERA-C-CELL TLX5-CELL TUMOR-CELL U937-CELL V79-CELL VERO-CELL VX2-CELL W138-CELL WALKER-256-CELL WIDR-CELL WISH-CELL XC-CELL Y79-CELL YOSHIDA-SARCOMA-CELL TOCOLYTICS FENOTEROL HEXOPRENALINE HSR-81 ISOXSUPRINE KUR-1246 L-366509 L-368899 L-371257 LEVOSALBUTAMOL MELUADRINE

Derwent Drug File 1243 Thesaurus MESUPRINE ONO-8815-LY ORCIPRENALINE RITODRINE SALBUTAMOL TERBUTALINE TV-399 VETRABUTINE TONICS ACETYLLEVOCARNITINE AMITRAZ ARICYL BERBERINE BRUCINE BUCLIZINE CACODYLATE CARNITINE CYPROHEPTADINE ELFAZEPAM GERIFORTE GLYCEROPHOSPHATE = MAGNESIUM GLYCEROPHOSPHATE = SODIUM LEVOCARNITINE LSL-60101 PIZOTIFEN SECURININE STRYCHNINE TOLDIMFOS TOOTH DENTAL-FOLLICLE DENTAL-PULP DENTIN ENAMEL TOPOISOMERASE-I-INHIBITORS BMS-250749 BN-80927 BNP-1350 BNPI-1100 CAMPTOTHECIN COUMAMYCIN CT-17 CZ-48 DB-67 DIFLOMOTECAN ED-749 EICOSADIENOATE-11,14 ETHOXIDINE F-11782 ICRF-505 IRINOTECAN J-109404 LAPACHONE-BETA NB-506 NSC-314622 NU-UB-199 NU-UB-31 ST-1481 TAS-103 TOPOTECAN XR-11576 XR-5944 TOPOISOMERASE-IIINHIBITORS AMSACRINE AZATOXIN BISANTRENE BMS-250749 BN-80927 CC-313 CP-115953 DEXRAZOXANE DOXORUBICIN ELLIPTICINE F-11782 GATIFLOXACIN GEMIFLOXACIN GR-122222-X ICRF-154 ICRF-193 IDARUBICIN KW-2170 MERBARONE MITOXANTRONE MST-16 NOVOBIOCIN NSC-655649 NU-UB-199 NU-UB-31 S-16020-2 SAINTOPIN SALVICINE SITAFLOXACIN T-3811-ME TAS-103 WR-242511 XR-11576 XR-5944 TOPOISOMERASE-INHIBITOR TOPOISOMERASE-1-= INHIBITOR TOPOISOMERASE-2-= INHIBITOR TOPOISOMERASE-INHIBITORS ACLARUBICIN ACTINOMYCIN-D AMAROGENTIN AMSACRINE AZATOXIN BIMOLANE BISANTRENE BMS-250749 BN-80927 BNP-1350 BNPI-1100 CAMPTOTHECIN CC-313 COUMAMYCIN CP-115953 CT-17 CZ-48 DB-67 DIFLOMOTECAN DOXORUBICIN DRF-1042 DX-8951 ED-749 EICOSADIENOATE-11,14 ELLIPTICINE EPIRUBICIN ETHOXIDINE ETOPOSIDE F-11782 GATIFLOXACIN GEMIFLOXACIN GR-122222-X ICRF-154 ICRF-193 ICRF-505 IDARUBICIN IRINOTECAN J-109404 KW-2170 LAPACHONE-BETA MERBARONE MITOXANTRONE MST-16 NAPHTHAZARIN NAPHTHOQUINONE-1,4 NB-506 NK-611 NOVOBIOCIN NSC-606174 NSC-655649 NU-UB-199 NU-UB-31 PIRARUBICIN PIRARUBICIN RO-47-3359 S-16020-2 SAINTOPIN SALVICINE SITAFLOXACIN SN-38 ST-1481 T-3811-ME TAS-103 TOPOISOMERASE-1-= INHIBITORS TOPOISOMERASE-2-= INHIBITORS TOPOTECAN WR-242511 XR-11576 XR-5944 ZD-6126 TOX. LD10 LD100 LD50 LD90 TOXINS ACETYL-T2-TOXIN ACETYLDEOXYNIVALENOL-15 ACETYLDEOXYNIVALENOL-3 AFLATOXICOL AFLATOXIN AFLATOXIN-B AFLATOXIN-B1 AFLATOXIN-B2 AFLATOXIN-G AFLATOXIN-G1 AFLATOXIN-G2 AFLATOXIN-M AFLATOXIN-M1 AFLATOXIN-M2 AFLATOXIN-P1 AFLATOXIN-Q1 ARGIOTOXIN-636 ASTELTOXIN AVELLANIN-A BOTULINUM-A-TOXIN BOTULINUM-C-TOXIN BOTULINUM-TOXIN BRYOPHYLLIN-A CHAETOCHROMIN-A CHOLERA-TOXIN CORD-FACTOR CRM-45 CYCLOPIAZONATE CYTOTOXIN DEEPOXYDEOXYNIVALENOL DEOXYNIVALENOL DIHYDROTELEOCIDIN DIPHTHERIA-TOXIN ENDOTOXIN ENTEROTOXIN ENTEROTOXIN-A-STAPH ENTEROTOXIN-A-STAPH EXFOLIATIN FUMONISIN-B1 FUSAROCHROMANONE GELONIN HELMINTHOSPORAL HEMOLYSIN

1244 APPENDIX D HT2-TOXIN LEUKOCIDIN LYCOMARASMIN LYNGBYATOXIN-A MAITOTOXIN MYROTOXIN-A MYROTOXIN-B NEOSOLANIOL OCHRATOXIN OCHRATOXIN-A OCHRATOXIN-B OCHRATOXIN-C PAXILLINE PENITREM-A PEROXISOMICINE-A1 PEROXISOMYCIN PERTUSSIS-TOXIN PHOMOPSIN-A PROCHOLERAGENOID PS.EXOTOXIN PS.TOXIN RUBRATOXIN RUBRATOXIN-B SATRATOXIN-G SATRATOXIN-H SAXITOXIN SCIRPENTRIOL SPORIDESMIN SPOROL STAPHYLOCOCCUS-= ENTEROTOXIN-B STAPHYLOLYSIN STERIGMATOCYSTIN STREPTOLYSIN T2-TETRAOL-TOXIN T2-TOXIN T2-TRIOL-TOXIN TELEOCIDIN TELEOCIDIN-B TETANUS-TOXIN VERRUCAROL TRANQUILIZERS 10184-CERM 340125 450247 450304 450789 450790 52-522 709-W-92 ABECARNIL ABT-418 AC-3579 ACAPRAZINE ADATANSERIN ADINAZOLAM AEC AHR-14042 ALEPH-2 ALOZAFONE ALPERTINE ALPIDEM ALPRAZOLAM AMBOCARB AMINOBECLAMIDE-PARA AMPHENIDONE ANTALARMIN AP-159 AP-521 ARFENDAZAM AWD-131-138 AZACYCLONOL AZAQUINZOLE B-20991 BARAKOL BENACTYZINE BENTAZEPAM BENZINDOPYRINE BENZOCTAMINE BMS-184111 BRL-46470 BRL-46470A BROMAZEPAM BROMOPRIDE BROTIZOLAM BTG-1501 BUCLIZINE BURAMATE BUTAMOXANE CAMAZEPAM CAMPIRONE CARBURAZEPAM CENTAZOLONE CGP-49823 CGS-17867A CGS-20625 CGS-9896 CHLORDIAZEPOXIDE CHLORFENETHAZINE CHLORMEZANONE CHLORPHENESIN-= CARBAMATE CICLOTIZOLAM CIDOXEPIN CINITAPRIDE CINOCTRAMIDE CINPERENE CINTRAMIDE CIPRAZAFONE CIPROXIMIDE CL-218872 CL-273547 CLAZOLAM CLOBAZAM CLOPERIDONE CLOPIMOZIDE CLOPIPAZAN CLORAZEPATE CLOTIAZEPAM CLOTIXAMIDE CLOXAZOLAM CO-134444 CP-141938 CP-93393 CP-93393-1 CRA-1000 CRA-1001 CYCLARBAMATE CYCLOBENZAPRINE CYCLOPREGNOL CYPRAZEPAM DAA-1097 DAA-1106 DECLENPERONE DELORAZEPAM DEMETHYLCLOBAZAM DEMETHYLDOXEPIN DEMETHYLFLUDIAZEPAM DEMOXEPAM DETOMIDINE DIAMIPHENE DIAZEPAM DICHLORMEZANONE DICLOMETIDE DIFENCLOXAZINE DIFLUANAZINE DIHYDROFENAZEPAM DIHYDROHONOKIOL-B DIHYDROMAGNOLOL DIPHOXAZIDE DIZOCILPINE DOXEFAZEPAM DOXEPIN DTZ-323 DU-127090 DULOZAFONE ECTYLUREA EGIS-7056 ELFAZEPAM EMYLCAMATE ENCIPRAZINE ENPIPRAZOLE ESTAZOLAM ETAFENOXIN ETAZOLATE ETHOMOXANE ETIFOXINE ETIZOLAM ETODROXIZINE ETOPERIDONE ETYMEMAZINE FENAZEPAM FENHARMANE FENIBUT FENIMIDE FENOBAM FG-8205 FG-9202 FLUDIAZEPAM FLUNITRAZEPAM FLUORESONE FLUOTRACEN FLUTAZOLAM FLUTOPRAZEPAM FLUTROLINE FOSAZEPAM FOSENAZIDE GABA-LINOLEAMIDE GANAXOLONE GEPIRONE GIDAZEPAM GINDARINE GIRISOPAM GLAZIOVINE GR-100679 GR-159897 GV-150013 GV-150013-X GVS-111 HALAZEPAM HALOPEMIDE HOMOCHLORCYCLIZINE HT-90-B HYDAZEPAM HYDROXYALPRAZOLAM-= ALPHA HYDROXYCAMAZEPAM HYDROXYFENAZEPAM-3 HYDROXYZINE ICI-190622 ICLAZEPAM IMIDOLINE IODOPROXYFAN IPSAPIRONE IRAZEPINE ISAMOLTAN KC-3756 KETAZOLAM L-663581 LESOPITRON LEVOPROTILINE LITHIUM-NICOTINATE LOFENDAZAM LOFLAZEPATE-ETHYL LOMETRALINE LONETIL LOPIRAZEPAM LOPRAZOLAM LORAZEPAM LORZAFONE LU-28-179

Derwent Drug File 1245 Thesaurus LY-333068 LY-354740 MDL-100907 MDL-105519 MDL-73005 MDL-73005EF MDL-73450 MDL-74217 MEBICAR MEBUTAMATE MECLONAZEPAM MEDAZEPAM MEDIFOXAMINE MEPHENOXALONE MEPROBAMATE METACLAZEPAM METAGLYCODOL METAXALONE METHINDIONE METOSERPATE MEXAZOLAM MIDAFLUR MIDAZOLAM MILTIRONE MINAPRINE MJ-13653 MJ-7378 MOLINDONE MONODEMETHYLDOXEPIN MOTRAZEPAM NABILONE NAPRODOXIME NARANOL NDO-008 NELEZAPRINE NERISOPAM NIMETAZEPAM NISOBAMATE NITRAZEPATE NITRAZEPATE POTASSIUM NKP-608 NORDAZEPAM NORTETRAZEPAM ONDANSETRON ORG-2305 ORG-37684 OXANAMIDE OXAZEPAM OXAZOLAM OXYFENAMATE PANADIPLON PANCOPRIDE PAZINACLONE PD-135666 PD-142898 PD-158771 PENTABAMATE PENTAMOXANE PHENAGLYCODOL PHENPROBAMATE PINAZEPAM PIPEQUALINE PIPETHANATE PIVAGABINE PIVOXAZEPAM PK-9084 PRAZEPAM PREMAZEPAM PROFLAZEPAM PROMOXOLANE PYRICAPIRONE PYRIDARONE PYRIMIDINYLPIPERAZINE RESCINNAMINE RESERPINE RIPAZEPAM RO-11-7800 RO-17-1812 RO-19-5686 RO-21-6347 RO-21-8384 RO-22-3245 RO-23-0364 RO-48-6791 RO-48-8684 RO-5-2904 RO-5-3590 RO-5-4864 RO-60-0175 RO-64-6198 RP-59037 RP-60503 RU-31719 RU-32514 RU-32698 RU-32759 RU-33203 RU-33368 RU-33543 RWJ-45788 S-14506 SAS-646 SB-200646-A SB-206553 SB-228357 SC-32855 SEDONIUM SERAZAPINE SP-904 SR-41378 SSR-149415 STACHYDRINE STIRIPENTOL SUANZAORENTANG SULAZEPAM SUN-8399 SUNEPITRON SURICLONE SZJ-3361 SZJ-3388 TACLAMINE TANDOSPIRONE TEMAZEPAM TETRAZEPAM TIAGABINE TIMELOTEM TJS-010 TOFISOLINE TOFISOPAM TOLBOXANE TOLPIPRAZOLE TRACAZOLATE TRAZODONE TRIACETONAMINE TRICLODAZOL TRIFLUBAZAM TRIMETOZINE TUCLAZEPAM TYBAMATE U-101017 U-43465F U-92016-A U-93385 ULDAZEPAM UMESPIRONE VA-21-B7 VALNOCTAMIDE WAY-100289 WAY-100635 WE-1008 WS-1490 WY-47846 WY-48723 Y-23684 ZALOSPIRONE ZK-91296 ZK-93423 ZK-95962 ZOLAZEPAM ZOLPIDEM ZOPICLONE TRANSPLANTATION ALLOGRAFT AUTOTRANSPLANTATION GRAFT GRAFT-REJECTION GRAFT-VERSUS-HOST-= REACTION HETEROGRAFT HOMOGRAFT TREMATODE ALARIA AMPHISTOMUM BRACHYLAEMUS CALICOPHORON CATATROPIS CEYLONOCOTYLE CLONORCHIS COTYLOPHORON DACTYLOGYRUS DICROCOELIUM DIPLOSTOMUM ECHINOSTOMA EURYTREMA FASCIOLA FASCIOLOIDES FASCIOLOPSIS FILICOLLIS FISCHOEDERIUS GASTROTHYLAX GYRODACTYLUS HETEROBILHARZIA HETEROPHYES METAGONIMUS NANOPHYETUS OPISTHORCHIS ORTHOCOELIUM PARAGONIMUS PARAMONOSTOMUM PARAMPHISTOMUM PARASTRIGEA PHARYNGOSTOMUM POSTHARMOSTOMUM SANGUINICOLA SCHISTOSOMA TREMATODIASIS BLACK-DISEASE OPISTHORCHIASIS SCHISTOSOMIASIS TRIAL-PREP. 10184-CERM 102-198 1031-U-89 104 1045-U-85 106-094 106-689 1067-CERM 116-L 1192-U-90 1229-U-91 129-L 130-B 1396-U-88 1400-W 143 15-AU-81 150-49 150C47 153C51

1246 APPENDIX D 156-S 170U88 1799 18-502 183-C-91 1843U89 191-DG 19148-RP 192C86 1935-L 1944-U-88 19749-RP 2-12362 2-169 2-170 2-5410-4A 20-785 20-AET-1 201-106 201-403 201-678 202 202-791 202-791-(+) 202-791-(-) 204-090 204-155 204-545 205-429 205-430 205-501 207-887 208-199 210-086 21009 212-494 216C 217-AO 2242 225-144 230-A 233 2355-S 235C 23669-RP 248U 253-152 254-S 261-115 261-96 272-131 272C 27753-RP 27753-RP 293-B 306 306159 309 313-40 3178-AQ 34-W-89 340125 348U87 349U85 35-W-89 351-A 36-W-89 4030-W-92 4162-W-94 428-U-89 43-U-87 44-549 44081-RP 443-C 447-C-88 450247 450304 450789 450790 4595-RP 4684-RP 48740-RP 49-W-89 4991-W-93 50-235 50-W-89 502-U-83 502U83 506 506-BD 506-U 51-W-89 516 52-522 523-W-91 524-W-91 52770-RP 53-540 543-U-76 57-118 57-118 58-035 58-112 59227-RP 593-A 606-A 6211 6603 6605-VUFB 661U88 66A-078 670C88 68-157 680-C-91 70026 709-W-92 72-70 723-C-86 7351 739-W-94 764-3 773-U-82 7943 8203-HC 8354 8356 8363-S 86-448 86017 882C 9599 97-139 98-202 A-007 A-025 A-10255 A-1062 A-1110U A-119637 A-127722 A-131701 A-134974 A-134U A-137 A-137491 A-145 A-147627 A-151011 A-1576 A-158112 A-16686 A-16686-A1 A-16686-A2 A-16686-A3 A-16886A A-16886B A-171 A-172 A-173508 A-182086 A-1866 A-19009 A-191 A-192 A-192621 A-195 A-204197 A-204A A-20812 A-20832 A-21459-A A-21459-B A-21978-C1 A-21978-C2 A-21978-C3 A-23887 A-249377 A-2545 A-25822-A A-25822-B A-25822-D A-25822-L A-25822-M A-25822-N A-26771B A-277323 A-278637 A-286982 A-29-LUNDBECK A-292949 A-3-P-166 A-3080 A-31472 A-315675 A-320454 A-32390-A A-35512B A-36683 A-3744 A-37536 A-37850 A-3787 A-4-P-73 A-40557 A-40823 A-40926-PA A-41030A A-41030C A-41030D A-41030E A-41030F A-41030G A-477 A-47934 A-49816 A-5021 A-53693 A-54145A A-54145A1 A-54145B A-54145B1 A-54145C A-54145D A-54145E A-54145F A-54741 A-55453 A-56234 A-57219 A-57274 A-58365A A-58365B

Derwent Drug File 1247 Thesaurus A-61603 A-62176 A-62251 A-62514 A-62671 A-62824 A-64718 A-65186 A-65260 A-65317 A-66005 A-66173 A-66193 A-67396 A-68064 A-68684 A-68828 A-68930 A-69024 A-69334 A-69412 A-71378 A-71623 A-71915 A-71984 A-720287 A-723U A-72517 A-72962 A-73209 A-73342 A-74111 A-74186 A-74187 A-74273 A-74704 A-748 A-74932 A-75179 A-75179 A-75200 A-75912 A-75925 A-75962 A-75962 A-75998 A-76792 A-76889 A-76890 A-76928 A-77003 A-771726 A-77212 A-77636 A-779 A-78773 A-78791 A-79175 A-80198 A-802715 A-80426 A-80915A A-80987 A-81229 A-81988 A-82695 A-83586-C A-84543 A-85226 A-85380 A-85783 A-86281 A-86415 A-86719-0 A-86929 A-87049 A-88861 A-91 A-9145C A-924 A-93178 A-9387 A-98881 AA-1777 AA-193 AA-231-1 AA-2379 AA-31 AA-344 AA-497 AA-501 AA-863 AAL-05 AAL-13 AB-118 AB-15 AB-163 AB-23 AB-47 AB-50 AB-85 ABBOTT-29590 ABBOTT-41988 ABBOTT-56234 ABBOTT-63162 ABBOTT-81282 ABC-99 ABIL-B-8839 ABIL-B-8852 ABIL-EM-90 ABIL-WAX-2434 ABT-080 ABT-089 ABT-229 ABT-299 ABT-418 ABT-431 ABT-510 ABT-526 ABT-594 ABT-606 ABT-702 ABT-761 ABT-773 ABT-866 ABT-987 AC-119 AC-3092 AC-3579 AC-394 AC-623 AC-7700 AC-7739 ACA-147 ACC-7513 ACC-9129 ACC-9358 ACC-9369 ACEA-0593 ACEA-0762 ACEA-1011 ACEA-1021 ACEA-1031 ACEA-1328 ACEA-1416 AD-0261 AD-11 AD-1211 AD-143 AD-194 AD-198 AD-199 AD-20 AD-202 AD-2239 AD-2646 AD-280 AD-284 AD-285 AD-288 AD-294 AD-295 AD-312 AD-32 AD-3264 AD-41 AD-4610 AD-48 AD-5 AD-5075 AD-5423 AD-8112 AD-92 ADA-202-718 ADD-17014 ADD-196022 ADD-213063 ADD-213066 ADD-219048 ADN-138 ADR-847 ADR-851 ADR-925 AE-0047 AE-1734 AE-941 AEOL-10113 AEOL-11201 AF-013 AF-0150 AF-05 AF-102B AF-10847 AF-1312-TS AF-13948 AF-14 AF-150 AF-150-S AF-2259 AF-267-B AF-30 AF-64A AF-ABDMP AF-ABDP AF-ABP AF-CX-1325 AF-DX-384 AF-DX-474 AFD-19 AFD-21 AFK-108 AFP-03 AG-041-R AG-045572 AG-1007 AG-1024 AG-1034 AG-1049 AG-1112 AG-114 AG-115 AG-1254 AG-126 AG-1284 AG-1295 AG-1296 AG-1387 AG-1402 AG-14031 AG-1478 AG-1517 AG-17

1248 APPENDIX D AG-1777 AG-1789 AG-1812 AG-1813 AG-1879 AG-1908 AG-1909 AG-2 AG-2000 AG-2034 AG-2037 AG-246 AG-2H AG-30 AG-307 AG-310 AG-331 AG-3340 AG-337 AG-34 AG-370 AG-377 AG-394 AG-4 AG-4263 AG-490 AG-494 AG-514 AG-52-315 AG-528 AG-537 AG-538 AG-555 AG-555 AG-556 AG-568 AG-6084 AG-6840 AG-7088 AG-775 AG-786 AG-81 AG-825 AG-85 AG-879 AG-879 AG-952 AG-957 AG-99 AG-EE-388-ZW AG-EE-623ZW AG-EE-624-ZW AG-EE-86 AGL-1872 AGL-517 AGM-1470 AGM-1883 AGN-1135 AGN-190073 AGN-190089 AGN-190121 AGN-190186 AGN-190299 AGN-190383 AGN-190727 AGN-190742 AGN-190744 AGN-190851 AGN-191103 AGN-191701 AGN-191976 AGN-192093 AGN-192403 AGN-193080 AGN-193109 AGN-193835 AGN-193836 AGN-194078 AGN-194204 AGN-194301 AGN-194310 AGN-195153 AGN-2979 AGR-529 AGR-614 AH-1058 AH-11110-A AH-13205 AH-19437 AH-22216 AH-23848 AH-23848B AH-2835 AH-3021 AH-3474 AH-6405 AH-7725 AH-7921 AH-9679 AH-9700 AH-P-719 AHA-008 AHC-52 AHN-086 AHR-11748 AHR-11797 AHR-12234C AHR-14042 AHR-16303B AHR-1709 AHR-1900 AHR-1911 AHR-2666 AHR-5333 AHR-5360 AHR-5360C AHR-5955 AHR-602 AHR-9294 AI3-36206 AIS-48 AIT-082 AJ-234 AJ-2615 AJ-3941 AJ-76 AK-124 AK-135 AK-165-3 AK-2123 AK-275 AK-295 AK-40 AK-49 AKF-94 AKI-1 AKS-19 AL-01766 AL-03077 AL-03150 AL-03152 AL-03153 AL-0670 AL-0671 AL-136 AL-1567 AL-1612 AL-294 AL-3152 AL-4114 AL-4414-A AL-449 AL-721 AL-87 ALA-251 ALA-54 ALE-36 ALK-3 ALO-3363 ALRT-1550 ALT-4000 ALT-462 ALT-486 ALT-711 ALT-766 ALX-0600 ALX-40-4-C AM-00 AM-1 AM-132 AM-3 AM-32 AM-36 AM-404 AM-55 AM-55-S AM-555 AM-555-S AM-580 AM-590 AM-630 AM-68 AM-682 AM-80 AM-90 AM-92008 AMA-1294 AMA-3176 AMI-121 AMI-227 AMI-25 AMINOINDAZOLE-6 AMO-1618 AMP-22 AMP-67 AMQ-2 AMQ-4 AMQ-5 AN-12 AN-132 AN-152 AN-162 AN-201I AN-201II AN-207 AN-215 AN-238 AN-9 ANK-102 ANQ-11125 ANQ-9040 AO-1100 AO-124 AO-128 AP-0341 AP-1510 AP-159 AP-1903 AP-20187 AP-237 AP-521 AP-5280 AP-539 AP-811 APC-2059 APC-366 APP-201-533 APREPITANT AQ-0145 AQ-11 AQ-AH-208 AQ-RA-391

Derwent Drug File 1249 Thesaurus AQ-RA-721 AQ-RA-741 AQ4 AQM-171 AR-12-456 AR-12455 AR-12460 AR-12463 AR-12464 AR-12465 AR-A-008055 AR-C-239 AR-C-68397-AA AR-L-100-BS AR-L-113-BS AR-L-57 AR-L-57-CL AR-LH-31 AR-R-15896-AR ARB-95-214 ARC-69931-MX ARK-5210 ARK-5211 ARK-5213 ARK-5310 ARK-5311 ARK-5312 ARL-15849-XX ARL-15895-AR ARTEFLENE AS-013 AS-101 AS-35 AS-4370 AS-48 AS-5370 AS-5820 AS-6 AS-601811 AS-602240 AS-701 AS-8 AS-924 ASI-222 ASI-253 ASI-254 ASL-7022 ASL-8123 ASTA-5607 ASTA-5783 ASTA-7037 ASTA-Z-7654 AT-1015 AT-2433-A1 AT-2433-A2 AT-2433-B1 AT-2433-B2 AT-265 AT-486 AT-760 ATF-H-18 ATI-2001 ATL-193 ATZ-1993 AU-1421 AU-8001 AVI-4126 AVS-1018 AW-464 AWD-12-281 AWD-122-239 AWD-131-138 AWD-140-076 AWD-140-190 AWD-160-275 AWD-19-166 AWD-23-111 AWD-26-06 AWD-26-39 AWD-52-39 AWD-625 AWD-627 AWD-G256 AY-14948 AY-16809 AY-18672 AY-20213 AY-20214 AY-20524 AY-21669 AY-21670 AY-22093 AY-22248 AY-23578 AY-23626 AY-24668 AY-25205 AY-25674 AY-28200 AY-28925 AY-29315 AY-30068 AY-31574 AY-31637 AY-9928 AY-9944 AZ-16596 AZ-21666 AZ-242 AZ-80 AZ-DF-265 AZB-017 AZD-2563 B-041 B-059 B-1086 B-120 B-1324 B-15 B-1600 B-1772 B-1865 B-1912 B-193 B-201 B-2036 B-20991 B-220 B-239 B-24-76 B-283 B-2844 B-3-243 B-3-277 B-327 B-3374 B-3640 B-3722 B-3770 B-3779 B-3785 B-3786 B-3814 B-3816 B-3820 B-3824 B-3832 B-3839 B-3878 B-3926 B-3958 B-3970 B-3995 B-3996 B-4019 B-4021 B-4076 B-4087 B-4100 B-4101 B-4144 B-4146 B-4148 B-4152 B-4154 B-4157 B-428 B-429 B-4308 B-4310 B-432 B-433 B-442 B-4759 B-5-49 B-581 B-621 B-623 (benzothiophene) B-628 B-654 B-669 B-670 B-685 B-695-40 B-744-96 B-744-98 B-744-99 B-746 B-749 B-776 B-777-81 B-797 B-813-19 B-826 B-831-56 B-850040 B-859-35 B-9004-070 B-9066 B-9109-012 B-9209-005 B-9340 B-9430 B-9436 B-956 B-9668 B-975-35-2 B-980 B-9812 B-9816 B-9858 B-9958 BA-28882 BA-30515 BA-31531 BA-32248B BA-32476 BA-32641 BA-33902 BA-34358 BA-35597 BA-35969 BA-36204 BA-36208 BA-36435 BA-36644 BA-37215 BA-40922 BA-41799 BA-41899 BA-42517 BA-43582A

1250 APPENDIX D BA-44680 BA-941 BAC-1829 BAL-9141 BAL-9611 BAM-1110 BAM-12P BAM-1303 BAM-18 BAM-2101 BAM-22P BANA-113 BAS-118 BAU-426 BAX-439 BAY-02752 BAY-10-6734 BAY-1099 BAY-11-7085 BAY-11-7821 BAY-12-9566 BAY-1248 BAY-1433 BAY-1518 BAY-3522 BAY-36-7620 BAY-38-3441 BAY-41-2272 BAY-43-9006 BAY-43-9695 BAY-50-4798 BAY-57-1293 BAY-B-1694 BAY-E-5759 BAY-E-6927 BAY-I-1441 BAY-K-8644 BAY-K-9320 BAY-L-3505 BAY-L-8201 BAY-L-9139 BAY-M-4786 BAY-M-5579 BAY-N-1468 BAY-N-5247 BAY-N-5248 BAY-N-6391 BAY-O-5572 BAY-O-6997 BAY-P-8857 BAY-P-9357 BAY-Q-1313 BAY-Q-3542 BAY-R-1531 BAY-R-3783 BAY-R-3964 BAY-R-4407 BAY-R-5417 BAY-R-9425 BAY-S-9435 BAY-T-5006 BAY-U-3405 BAY-U-3625 BAY-U-9773 BAY-V-3522 BAY-W-5035 BAY-W-5037 BAY-W-5434 BAY-X-1005 BAY-X-3702 BAY-X-7195 BAY-X-9228 BAY-Y-1015 BAY-Y-3118 BAY-Y-5959 BAYA-6781 BAYER-9017 BAYER-A139 BAYG-7183 BB-10010 BB-1101 BB-1502 BB-16 BB-2116 BB-2275 BB-3103 BB-823 BBR-2160 BBR-2196 BBR-2197 BBR-2207 BBR-2209 BBR-2220 BBR-2378 BBR-2577 BBR-2778 BBR-2828 BBR-2867 BBR-2868 BBR-2894 BBR-3005 BBR-3171 BBR-3390 BBR-3464 BC-16 BC-197 BC-264 BC-3016 BC-59 BC-60 BC-63 BC-681 BCE-001 BCH-069 BCH-10618 BCH-10619 BCH-1393 BCH-189 BCH-189-TRIPHOSPHATE BCH-2051 BCH-2763 BCH-325 BCH-4556 BCN-326862 BCR-4 BCX-1827 BCX-1898 BCX-1923 BCX-34 BD-1008 BD-1047 BD-1063 BD-1304 BD-737 BD-738 BDB-106 BDB-108 BDB-27 BDB-37 BDB-91 BDF-6100 BDF-7572 BDF-7579 BDF-8784 BDF-8933 BDF-9145 BDF-9148 BDF-9167 BDF-9196 BDF-9198 BDH-2700 BDH-7538 BE-10988 BE-12406A BE-12406B BE-14348-B BE-1726 BE-18257A BE-18257B BE-18591 BE-2222 BE-2247 BE-2254 BE-23372-M BE-23372M BE-2391 BE-2392 BE-2414 BE-3333 BE-373 BE-40644 BE-4444 BE-6143 BE-7420 BEA-1125 BEA-1128 BEA-1654 BF-389 BF-759 BFE-37 BFE-41 BFE-47 BFE-55 BFE-61 BFE-69 BFE-72 BG-104 BG-237 BG-289 BG-31 BG-32 BG-325 BG-374 BG-60 BG-8865 BG-920 BG-9273 BG-958 BG-996 BGP-15 BHT-958 BI-679 BI-L-226XX BI-L-45XX BI-RJ-70 BI-RM-270 BIA-3-202 BIBF-1000 BIBN-4096-BS BIBN-99 BIBO-3304 BIBP-3226 BIBP-3435 BIBS-222 BIBS-39 BIBU-104 BIBU-104-XX BIBU-52 BIBW-022 BIBW-22-BS BIBX-79 BIIB-513 BIIE-0246 BILA-2157-BS BILA-2185-BS BILD-1263 BILD-1351 BILN-303-SE BILS-45-BS BIM-23003 BIM-23003 BIM-23023

Derwent Drug File 1251 Thesaurus BIM-23026 BIM-23027 BIM-23034 BIM-23056 BIM-23127 BIM-23190 BIM-23197 BIM-26189 BIM-26226 BIM-4004-1 BIM-46174 BIMT-17 BIMU-0001 BIMU-1 BIMU-8 BIRB-796 BK-129 BK-21070 BKH-14 BL-11778 BL-14 BL-141 BL-1743 BL-194 BL-20803 BL-2338 BL-2365 BL-269 BL-343AC BL-3459 BL-3912 BL-443 BL-473 BL-5255 BL-554 BL-562 BL-6341A BL-6783 BL-9 BL-KR-140 BL-P-2013 BL-P-875 BL-S-217 BL-S-339 BM-01014 BM-01044 BM-06-021 BM-06-022 BM-106 BM-11 BM-11189 BM-113 BM-121307 BM-123 BM-123A BM-130 BM-130-A BM-130907 BM-130913 BM-140830 BM-14515 BM-14686 BM-15 BM-15-0639 BM-15766 BM-16-2056 BM-16-2266 BM-16-2287 BM-16-2353 BM-16-2354 BM-16-2374 BM-17 BM-2-28 BM-20 BM-20-1140 BM-208 BM-21-23 BM-23014 BM-24 BM-27 BM-34 BM-42304 BM-5 BM-500 BM-500430 BM-51097 BM-51158 BM-51334 BM-51335 BM-519 BM-531 BM-567 BM-573 BM-8 BM-910183 BM-910228 BM-920700 BML-130 BMS-180291-02 BMS-180448 BMS-180560 BMS-180680 BMS-180742 BMS-180820 BMS-181101 BMS-181162 BMS-181163 BMS-181165 BMS-181167 BMS-181184 BMS-181321 BMS-181681 BMS-181885 BMS-182123 BMS-182178 BMS-182193 BMS-182248-01 BMS-182657 BMS-182874 BMS-183240 BMS-183920 BMS-184111 BMS-184476 BMS-184481 BMS-184698 BMS-185411 BMS-185660 BMS-186318 BMS-187745 BMS-188494 BMS-188667 BMS-188797 BMS-189365 BMS-191095 BMS-191352 BMS-192548 BMS-193884 BMS-204352 BMS-208782 BMS-210285 BMS-214662 BMS-224818 BMS-239091 BMS-247550 BMS-250749 BMS-250904 BMS-262084 BMS-275291 BMS-310705 BMS-753 BMY-14802 BMY-14802-1 BMY-20064 BMY-20551 BMY-20661 BMY-20844 BMY-21502 BMY-21638 BMY-21950 BMY-22089 BMY-25067 BMY-25174 BMY-25271 BMY-25282 BMY-25368 BMY-25405 BMY-25551 BMY-26107 BMY-26517-31 BMY-26605 BMY-28232 BMY-28251 BMY-28271 BMY-28864 BMY-30047 BMY-30094 BMY-30123 BMY-33315 BMY-40062 BMY-40124 BMY-40397 BMY-40662 BMY-41429 BMY-42230 BMY-42393 BMY-43261 BMY-43351 BMY-44621 BMY-45778 BMY-7378 BN-063 BN-1267 BN-1314 BN-50043 BN-50069 BN-50090 BN-50125 BN-50156 BN-50157 BN-50341 BN-50417 BN-50418 BN-50548 BN-50726 BN-50727 BN-50730 BN-50739 BN-52111 BN-52115 BN-52205 BN-52207 BN-52211 BN-52256 BN-54062 BN-80927 BN-80933 BNP-1100 BNP-1350 BNP-7787 BNPI-1100 BO-1165 BO-1166 BO-1236 BO-1341 BO-2727 BO-653 BOF-4269 BOF-4272 BOK-1 BP-12231 BP-179 BP-2-94

1252 APPENDIX D BP-42 BP-554 BPAT-117 BPAT-143 BPDZ-44 BPDZ-62 BPDZ-79 BQ-123 BQ-153 BQ-3020 BQ-485 BQ-610 BQ-788 BQ-928 BR-100 BR-1376 BR-16A BR-227 BR-370 BR-401 BR-401A BRB-I-28 BRC-16-HT BRI-7013 BRIMONIDINE TARTRATE BRL-10720 BRL-10739 BRL-14831 BRL-15572 BRL-16644 BRL-16657 BRL-18725 BRL-19405 BRL-19478 BRL-20459 BRL-20596 BRL-20627 BRL-24649 BRL-25594 BRL-26314 BRL-26830-A BRL-26830A BRL-26920 BRL-27320 BRL-28410 BRL-31532 BRL-31660A BRL-32071 BRL-32077 BRL-32872 BRL-33575 BRL-34778 BRL-35113 BRL-35135 BRL-35135A BRL-36378 BRL-36610 BRL-37344 BRL-37344-A BRL-38226 BRL-39913 BRL-41897A BRL-41897A BRL-41992 BRL-42222 BRL-42245 BRL-42359 BRL-42715 BRL-42715A BRL-43594 BRL-43599 BRL-44154 BRL-44385 BRL-44408 BRL-44409 BRL-46470 BRL-46470A BRL-47672 BRL-47923 BRL-48482 BRL-50395 BRL-50523 BRL-50551 BRL-50702 BRL-50714 BRL-50715 BRL-50717 BRL-51136 BRL-51334 BRL-52537 BRL-52656 BRL-53001 BRL-53001A BRL-54443 BRL-55039 BRL-55730 BRL-55791 BRL-55792 BRL-55834 BRL-57037 BRL-5907 BRL-6231 BRLP-42 BS-1-81 BS-6181 BST-101 BSU-1051 BT-402 BT-563 BT-99-25 BTG-1501 BTI-2286E BTM-1041 BTM-1042 BTM-1086 BTS-53554 BTS-54354 BTS-54505 BTS-63155 BTS-67-582 BTS-72664 BTS-74398 BU-224 BU-239 BU-3129T BU-99006 BU-E-64 BU-E-75 BU-E-76 BW-1003-U-88 BW-1003C87 BW-1024-U-88 BW-1069-C-85 BW-1110U81 BW-1263-W-94 BW-12C BW-1370U87 BW-1552-U-88 BW-1555-U-88 BW-175 BW-17U BW-180C BW-183U88 BW-1843U89 BW-1911-U-90 BW-204-C67 BW-2258-U-89 BW-2258U89 BW-245C BW-252-C64 BW-284-C51 BW-287U BW-306U BW-330-U-88 BW-348U87 BW-373-U-86 BW-380U88 BW-403-C65 BW-494 BW-501 BW-501-C67 BW-534-U-87 BW-540C BW-568C BW-58C BW-61-435 BW-616U76 BW-619-C-89 BW-62-235 BW-62-C47 BW-654 BW-683C BW-737-C BW-755C BW-776-C-85 BW-813U BW-826C BW-831C BW-935-U-83 BW-942C BW-A-1169U BW-A-1261U BW-A-1433 BW-A-1433U BW-A-1454U BW-A-353U BW-A-354U BW-A-424U BW-A-453U BW-A-457U BW-A-466C BW-A-494U BW-A-502U BW-A-503U BW-A-728C BW-A-773U BW-A-822U BW-A-90U BW-A-91U BW-A1117U BW-A137C BW-A256C BW-A444U BW-A4C BW-A522U BW-A575C BW-A589C BW-A616U BW-A78U BW-A797C BW-A7U BW-A844U BW-A868C BW-A947U BW-B218C BW-B385C BW-B429U BW-B70C BWA-270-C BX-471 BX-807834 BXT-51072 BY-101 BY-1947 BY-1949 BY-841 BY-963 BZ-140 BZA-2-B BZA-5-B BZA-7-B C-1005

Derwent Drug File 1253 Thesaurus C-1006 C-1020 C-1027 C-1263 C-1310 C-1311 C-1371 C-153 C-175 C-176 C-18665 C-19393-E5 C-205 C-232 C-257 C-264 C-265 C-27 C-2801-X C-29 C-307 C-308 C-309 C-337 C-338 C-3534 C-3535 C-383 C-394 C-395 C-410 C-4C C-516 C-5720 C-609 C-68-22 C-720045 C-73 C-75 C-780652 C-780698 C-801239 C-829 C-835 C-846 C-849 C-85 C-857 C-863293 C-867 C-873754 C-873786 C-878 C-881 C-883934 C-887 C-894095 C-894144 C-92-4609 C-92-4678 C-921 C-921-78 C3-76 CA-030 CA-074 CAF-603 CAM-1028 CAM-1481 CAM-2291 CAM-2445 CAM-4451 CAN-296 CAP-1 CAP-18-HUMAN CAP-2 CAP-440 CAS-413 CAS-754 CB-10-200 CB-10-252 CB-10-277 CB-10-286 CB-1093 CB-1267 CB-1414 CB-1837 CB-1850 CB-1954 CB-300638 CB-300907 CB-300919 CB-30865 CB-30900 CB-34 CB-3705 CB-3714 CB-3716 CB-3717 CB-3751 CB-3804 CB-3988 CB-7103 CB-7547 CB-7630 CB-7639 CB-7645 CB-7669 CB-7675 CB-7741 CB-874 CB-966 CBM-11 CBS-1108 CBS-1114 CBS-113A CC-1065 CC-25 CC-3052 CC-313 CC-34 CC-4047 CC-5013 CCD-3693 CCI-103F CCI-17810 CCI-22277 CCI-779 CCK-JMV-180 CCRG-82019 CCRL-1002 CCRL-1008 CCRL-1009 CCT-62 CD-2019 CD-2247 CD-2314 CD-2624 CD-2665 CD-270 CD-2809 CD-349 CD-367 CD-388 CD-394 CD-437 CD-564 CD-666 CD-832 CD-86022 CDB-2085A CDC-501 CDD-0098-J CDP-571 CDP-840 CDP-870 CDRI-77-6 CDRI-80-53 CDRI-81-470 CDRI-82-205 CDRI-82-437 CDRI-84-201 CDRI-84-35 CDRI-85-287 CDRI-86-333 CDRI-87-209 CDRI-88-495 CDRI-94-335 CE-0265 CE-0266 CE-0267 CEB-1957 CEDO-8956 CEP-1347 CEP-2563 CEP-5214 CEP-701 CEP-751 CERM-10194 CERM-11888 CERM-11956 CF-1001 CF-1093 CFC-222 CFT-1201 CG-10248 CG-37059 CG-4303 CG-601 CG-662 CG-8840 CG-8935 CG-9442 CGA-19255 CGI-16343 CGI-17658 CGI-18041 CGP-11112 CGP-11130 CGP-11637 CGP-11952 CGP-12104-A CGP-12104A CGP-12177 CGP-12177A CGP-12388 CGP-13231 CGP-15425 CGP-17520 CGP-17582B CGP-18137A CGP-19835 CGP-19835A CGP-19984 CGP-20308 CGP-20309 CGP-20376 CGP-20712A CGP-20909 CGP-21306 CGP-21833 CGP-21835 CGP-22364A CGP-22979A CGP-23518 CGP-23996 CGP-24589 CGP-26505 CGP-26702 CGP-28014 CGP-28237 CGP-28392 CGP-29030-A

1254 APPENDIX D CGP-29287 CGP-29325 CGP-29861 CGP-31362 CGP-31523A CGP-31608 CGP-33101 CGP-33829 CGP-33829-A CGP-34064A CGP-3466 CGP-3466-B CGP-35348 CGP-35753 CGP-35753-A CGP-35949 CGP-36742 CGP-36958 CGP-37849 CGP-38560 CGP-38560A CGP-39551 CGP-39653 CGP-39937-A CGP-40-215 CGP-40-215-A CGP-40116 CGP-41251 CGP-41389 CGP-42112A CGP-42112B CGP-42166 CGP-42700 CGP-42934 CGP-42935 CGP-4303 CGP-43371 CGP-43487 CGP-43902B CGP-44099A CGP-44532 CGP-44533 CGP-44645 CGP-44826 CGP-45715A CGP-46360 CGP-46381 CGP-47072 CGP-47645 CGP-47875 CGP-47969-A CGP-4832 CGP-48506 CGP-48508 CGP-48664 CGP-48664-A CGP-49823 CGP-51176 CGP-520 CGP-52411 CGP-52432 CGP-52608 CGP-53437 CGP-53716 CGP-53820 CGP-54062 CGP-55845 CGP-55845A CGP-56433 CGP-56433A CGP-56999 CGP-56999-A CGP-57698 CGP-57813 CGP-59326 CGP-60261 CGP-6085-A CGP-6085A CGP-61334 CGP-62349 CGP-62706 CGP-645 CGP-6809 CGP-69669-A CGP-69846-A CGP-7040 CGP-71683-A CGP-71982 CGP-73547 CGP-75254-A CGP-8065 CGP-8716 CGS-10078B CGS-11361 CGS-11776 CGS-12066A CGS-12066B CGS-12094 CGS-12970 CGS-13767 CGS-13928C CGS-15435-A CGS-15435A CGS-15529 CGS-15855A CGS-15873A CGS-15943A CGS-17867A CGS-18102-A CGS-18320B CGS-19213 CGS-19281-A CGS-19480A CGS-19755 CGS-20267 CGS-20281 CGS-20625 CGS-21680 CGS-21680A CGS-21680C CGS-22492 CGS-22652 CGS-22745 CGS-22988 CGS-22989 CGS-22996 CGS-23425 CGS-23885 CGS-24128 CGS-24565 CGS-24592 CGS-25015 CGS-25019-C CGS-25019C CGS-25155 CGS-25462 CGS-25659 CGS-26214 CGS-26303 CGS-26393 CGS-26582 CGS-26670 CGS-27023-A CGS-28106 CGS-30440 CGS-31447 CGS-32359 CGS-34043 CGS-35066 CGS-5649B CGS-5677 CGS-7181 CGS-8216 CGS-8515 CGS-9895 CGS-9896 CGX-571 CH-102 CH-127 CH-141 CH-150 CH-20 CH-23 CH-2856 CH-288 CH-30 CH-38083 CH-40 CH-40-S CH-402 CH-55 CH-55-G CH-55-S CH-60 CH-60-G CH-60-S CH-74A CH-80 CH-99A CHF-1035 CHF-1194 CHF-2206 CHF-2819 CHF-3381 CHINOIN-123 CHINOIN-127 CHINOIN-170 CHIRON-2279 CHS-828 CI-1000 CI-1004 CI-1007 CI-1010 CI-1011 CI-1018 CI-201-678 CI-218872 CI-261209 CI-588 CI-624 CI-628M CI-680 CI-750 CI-905 CI-913 CI-922 CI-923 CI-924 CI-925 CI-926 CI-927 CI-930 CI-931 CI-933 CI-934 CI-936 CI-937 CI-943 CI-949 CI-953 CI-958 CI-959 CI-966 CI-972 CI-976 CI-980 CI-986 CI-987 CI-992 CI-996 CIBA-21381-BA CID-85

Derwent Drug File 1255 Thesaurus CIS-19 CJ-12371 CJ-12458 CJM-05 CJM-126 CJS-11 CK-101-A CK-102 CK-103-A CK-113 CK-119 CK-122 CK-123 CK-1649 CK-17 CK-2130 CK-2289 CK-3197 CK-3368 CK-3579 CK-47A CK-53 CK-61A CKD-602 CKI-7 CL-06A CL-115129 CL-115574 CL-116147 CL-13580 CL-1700 CL-184005 CL-218872 CL-228346 CL-232468 CL-242817 CL-246738 CL-255663 CL-259763 CL-273547 CL-274471 CL-275838 CL-277082 CL-283546 CL-283796 CL-283981 CL-284027 CL-284846 CL-284859 CL-286527 CL-28A CL-306293 CL-315555 CL-315585 CL-316243 CL-329167 CL-329753 CL-329998 CL-331002 CL-331928 CL-344677 CL-387626 CL-387785 CL-42A CL-5343 CL-64855 CL-68A CL-77328 CL-860201 CL-868 CL-871502 CL-90100 CLX-0901 CM-101 CM-32191 CM-40142 CM-42641 CM-5637 CM-57373 CM-57493 CM-6 CM-6606 CM-7116 CMI-206 CMI-392 CMI-947 CMN-131 CMT-1 CMT-3 CMT-5 CMT-6 CMT-7 CMT-8 CN-100 CNI-1493 CNI-H-0294 CNI-H-1194 CNS-1102 CNS-1237 CNS-5161 CNS-5161-A CNS-5788 CNV-9203 CO-134444 CO-1408 CO-1828 CO-2-1068 CO-5-2791 CO-610 COBRA-1 COL-3 COMPOUND-102 COMPOUND-1929 COR-3224 CP-0088 CP-0126 CP-0127 CP-02 CP-0347 CP-0364 CP-0494 CP-0499 CP-0597 CP-060 CP-060-S CP-10 CP-10 CP-100263 CP-100356 CP-101606 CP-102 CP-105191 CP-105696 CP-106 CP-107 CP-108509 CP-110 CP-110330 CP-111905 CP-113056 CP-1136S CP-113818 CP-114271 CP-115953 CP-115955 CP-122288 CP-122721 CP-123369 CP-127374 CP-130 CP-132484 CP-135807 CP-141938 CP-14304 CP-146662 CP-148623 CP-154526 CP-162 CP-166572 CP-191166 CP-195494 CP-195543 CP-199331 CP-21 CP-2129-AL CP-22 CP-225917 CP-230821 CP-23445 CP-24 CP-248 CP-25 CP-25415 CP-26 CP-263114 CP-283 CP-2907 CP-293019 CP-294838 CP-30542 CP-316819 CP-331 CP-336156 CP-340868 CP-358774 CP-38 CP-40 CP-41 CP-42096 CP-44 CP-461 CP-465022 CP-46665-1 CP-471-474 CP-47497 CP-502 CP-51 CP-511 CP-52 CP-53261 CP-53607 CP-547632 CP-55244 CP-55940 CP-56667 CP-6162 CP-63956 CP-64131 CP-65207 CP-65526 CP-66713 CP-6679 CP-67015 CP-67804 CP-70429 CP-70490 CP-71362 CP-77059 CP-80794 CP-81054 CP-82009 CP-84657 CP-88059 CP-894S CP-92768 CP-92768 CP-93 CP-93129 CP-93393 CP-93393-1 CP-94 CP-94253

1256 APPENDIX D CP-96 CP-96344 CP-96345 CP-96501 CP-99542 CP-99994 CP-II CPH-82 CPI-0004 CPI-975 CPP-200 CPS-161 CPU-23 CPU-57 CPU-86017 CPW-86363 CQA-206-291 CR-1015 CR-1034 CR-1098 CR-1166 CR-1919 CR-1938 CR-2017 CR-2093 CR-2249 CRA-1000 CRA-1001 CRC-220 CRC-680578 CRE-10086 CRE-1087 CRL-1005 CRL-40467 CRL-40827 CRL-42796 CRL-81-31 CRL-81-42 CRL-8275 CRL-8276 CRL-8277 CRL-8299 CRL-85-221 CRX-103 CS-261 CS-263 CS-265 CS-432 CS-436 CS-437 CS-476 CS-570 CS-61 CS-670 CS-682 CS-747 CS-834 CS-85 CS-87 CS-87-TRIPHOSPHATE CS-905 CS-91 CS-92 CS-940 CT-052923 CT-112 CT-17 CT-1746 CT-2103 CT-2106 CT-2251 CT-2576 CT-2583 CT-2584 CT-3501 CT-3532 CTC-23 CTC-96 CU-23 CU-602 CV-11194 CV-159 CV-1674 CV-1808 CV-3611 CV-3988 CV-5197 CV-5975 CV-6209 CV-6504 CV-787 CVS-1123 CVS-995 CVT-124 CVT-3033 CVT-313 CVT-3146 CVT-510 CVT-P-040 CX-397 CX-397R CX-516 CX-659-S CX-691 CY-1503 CY-208-243 CY-222 CYT-356 CZ-112 CZ-48 CZ-74 D-003 D-0870 D-13223 D-150 D-15413 D-15414 D-15917 D-16120 D-174 D-175 D-17872 D-18024 D-18621 D-18954 D-19575 D-20133 D-20443 D-21266 D-21805 D-22888 D-230 D-2343 D-2439 D-24851 D-2916 D-3187 D-400 D-4026 D-4030 D-435 D-477A D-4975 D-51-4700 D-51-9927 D-528 D-557 D-559 D-573 D-575 D-58 D-595 D-609 D-617 D-620 D-675 D-702 D-784 D-788-1 D-792 D-846 D-890 DA-10 DA-1131 DA-125 DA-1529 DA-1627 DA-1686 DA-3505 DA-3804 DA-3829 DA-3831 DA-3832 DA-3838 DA-3839 DA-3840 DA-3851 DA-3853 DA-3854 DA-3915 DA-4626 DA-4643 DA-5018 DA-8159 DA-9601 DAA-1097 DAA-1106 DAC-5945 DAK-16 DAU-6215 DAU-6236 DAU-6285 DB-174 DB-2073 DB-289 DB-293 DB-67 DBM-819 DBO-11 DBO-83 DC-015 DC-101 DC-13-57 DC-23-99 DC-41-33 DC-81 DC-86-Y DC-92-B DC-92-D DC-TA-46 DCN-203-922 DDE-131 DDS-2700 DEMETHYLIVABRADINE-N DEV-10 DEV-9 DF-100 DF-1111301 DF-129 DF-203 DF-209 DF-229 DF-594 DH-40J DH-6471 DH-990 DHP-218 DIAM-3 DJ-6783 DJ-7041 DJ-7141 DK-118

Derwent Drug File 1257 Thesaurus DK-AH-269 DKA-9 DKJ-21 DL-111-IT DL-204-IT DM-232 DM-235 DM-44 DM-49 DM-75 DM-96 DMP-229 DMP-315 DMP-323 DMP-450 DMP-504 DMP-543 DMP-565 DMP-581 DMP-754 DMP-757 DMP-811 DMP-963 DN-1417 DN-9550 DN-9693 DO-710 DO-897 DOB-41 DOWCO-214 DP-107 DP-432 DPC-082 DPC-083 DPC-423 DPC-961 DPI-3290-W-93 DPN-205-734 DQ-2511 DQ-2556 DR-3438 DR-3862 DRF-1042 DRF-2189 DRF-2725 DS-121 DS-201 DS-210 DS-4152 DS-4524 DS-4574 DS-511 DSB-120 DSP-4 DT-5461 DT-5461-A DT-TX-30 DT-TX-30-SE DTZ-323 DU-1227 DU-124884 DU-125530 DU-127090 DU-14 DU-1777 DU-21117 DU-24565 DU-28663 DU-29894 DU-41164 DU-41165 DU-6668 DU-6681-A DU-6858 DU-717 DU-86 DUP-105 DUP-128 DUP-532 DUP-630 DUP-654 DUP-714 DUP-721 DUP-734 DUP-747 DUP-860 DUP-925 DUP-983 DV-7021 DV-7028 DV-7751 DV-7751-A DW-116 DWA-2114R DWA-2114S DWH-146-E DX-52-1 DX-8739 DX-8951 DX-8951-F DX-9065A DX-9386 DY-9708 DY-9760-E DY-9973 E-0663 E-0702 E-0711 E-0747 E-1020 E-1077 E-1100 E-1101 E-126 E-1309 E-2001 E-2011 E-2030 E-2050 E-3040 E-3123 E-3330 E-350 E-3620 E-3753 E-3846 E-4010 E-4021 E-4031 E-4080 E-414 E-4177 E-4441 E-456 E-4695 E-4701 E-4804 E-4868 E-5050 E-5065 E-5068 E-5090 E-5110 E-5324 E-5510 E-5531 E-5564 E-5880 E-6006 E-6010 E-6080 E-6087 E-6123 E-64 E-64C E-6700 E-7010 E-94 E3-54 EA-1465 EA-1476 EA-521 EB-1053 EB-1213 EB-1231 EB-40 EC-5-20 ED-110 ED-71 ED-749 EF-10750 EG-1088 EGIS-5645 EGIS-7056 EGIS-7229 EGIS-7649 EGIS-8332 EGIS-9377 EGYT-1354 EGYT-1855 EGYT-2474 EGYT-2509 EGYT-2760 EGYT-3615 EI-1511-3 EI-1511-5 EI-1625-2 EI-546 EIPW-111 EK-209 EK-399 EK-49 EKB-569 EL-979 EM-12 EM-138 EM-139 EM-16 EM-170 EM-201 EM-2487 EM-27 EM-311 EM-336 EM-356 EM-405 EM-523 EM-523L EM-536 EM-574 EM-610 EM-65 EM-651 EM-652 EM-776 EM-800 EMD-121974 EMD-122347 EMD-16795 EMD-20262 EMD-21388 EMD-23448 EMD-270179 EMD-28422 EMD-38362 EMD-41000 EMD-41717 EMD-42501 EMD-46335 EMD-46512 EMD-47021 EMD-47499

1258 APPENDIX D EMD-49209 EMD-50689 EMD-50689 EMD-51921 EMD-52-297 EMD-53998 EMD-54622 EMD-54650 EMD-55900 EMD-56133 EMD-57033 EMD-57439 EMD-59730 EMD-60263 EMD-60264 EMD-60400 EMD-66203 EMD-68843 EMD-72000 EMD-85131 EMI-1 EMI-2 EMI-3 EN-105 EN-2260 EN-2265 ENT-51007 ENT-51143 EO-122 EO-15 EO-5A EO-68 EO-72 EO-9 EP-011 EP-031 EP-035 EP-045 EP-092 EP-10045 EP-109 EP-157 EP-171 EP-19-088 EP-459 EPS-2004 EPS-4032 ER-001533 ER-076349 ER-086526 ER-27856 ER-30346 ER-32935 ER-35744 ER-35786 ER-42859 ER-68203-00 ER-69029 ES-1005 ES-242-1 ES-242-2 ES-242-3 ES-242-4 ES-242-5 ES-242-6 ES-242-8 ES-295 ES-300 ES-305 ES-313 ES-316 ES-317 ES-52 ES-6864 ES-8891 ES-921 ES-922 ET-126 ETH-615 EU-4867 EU-5476 EUDRAGIT-P-4135-F EUK-134 EUK-8 EWP-840 EX-10-542A EX-11-582A EX-4877 EX-89 EXBP-68 EXO-226 EXP-063 EXP-132 EXP-3174 EXP-3312 EXP-3892 EXP-561 EXP-597 EXP-6155 EXP-6159 EXP-6803 EXP-7711 EXP-9270 F-0401 F-1044 F-1067 F-10863-C F-10863-D F-11344-A-1 F-11782 F-123 F-12511 F-1322 F-13714 F-1377 F-1394 F-1459 F-1594 F-1603 F-1806 F-1808 F-1839-B F-1839-E F-1893 F-2268 F-2692 F-327 F-36 F-405 F-4168 F-4236 F-4614 F-5 F-6060 F-6103 F-910826 FA-33 FA-37 FA-42 FA-43 FA-45 FA-73 FAD-001 FC-18-94 FC-20-94 FC-3280 FC-726 FC-75 FCC-13 FCC-5 FCE-20635 FCE-20696 FCE-20700 FCE-21258 FCE-21589 FCE-21590 FCE-21904 FCE-22101 FCE-22176 FCE-22177 FCE-22178 FCE-22250 FCE-22509 FCE-22716 FCE-22807 FCE-23762 FCE-24265 FCE-24362 FCE-24561 FCE-24578 FCE-25199 FCE-25217 FCE-25450-A FCE-26176 FCE-26366 FCE-26367 FCE-26541 FCE-26605 FCE-26644 FCE-26743 FCE-26806 FCE-27164 FCE-27262 FCE-27391 FCE-27392 FCE-27395 FCE-27677 FCE-28068 FCE-28164 FCE-28729 FCE-28987 FCE-29006 FCE-29272 FD-008 FD-1 FD-594 FD-891 FG-5803 FG-5865 FG-5893 FG-5974 FG-7098 FG-7106 FG-7142 FG-8205 FG-9041 FG-9065 FG-9067 FG-9202 FGIN-1-27 FH-510 FI-302 FI-4501 FI-4503 FI-6173 FK-037 FK-041 FK-089 FK-1012-H-2 FK-1052 FK-143 FK-156 FK-224 FK-23 FK-33-824 FK-3311 FK-352 FK-409 FK-448 FK-453 FK-480 FK-565

Derwent Drug File 1259 Thesaurus FK-584 FK-613 FK-633 FK-664 FK-706 FK-739 FK-838 FK-888 FK-906 FK-960 FKH-10 FL-120-A FL-120-B FL-120-B+ FL-120-C FL-120-C+ FL-120-D+ FL-120A FL-120B FL-120B+ FL-120C FL-120C+ FL-120D+ FL-155 FL-386 FLA-1085 FLA-1088 FLA-289 FLA-299 FLA-314 FLA-334 FLA-336 FLA-365 FLA-384 FLA-405 FLA-417 FLA-450 FLA-463 FLA-558 FLA-63 FLA-659 FLA-668 FLA-717 FLA-727 FLA-788 FLA-797 FLA-873 FLA-908 FLA-961 FLA-981 FLA-988 FLA-99 FLB-457 FLB-463 FLB-472 FLB-524 FLM-5011 FLU-401 FLU-402 FO-1561 FOY-251 FP-33 FP-736-03 FP-736-04 FPL-12495 FPL-12495-AA FPL-12859 FPL-12860 FPL-13210 FPL-13950 FPL-14995 FPL-15853 FPL-15896-AR FPL-52694 FPL-52757 FPL-55618 FPL-55712 FPL-57231 FPL-62064 FPL-62129 FPL-63012AR FPL-64170-XX FPL-64176 FPL-66096 FPL-66365 FPL-67047-XX FPL-67085 FPL-67156 FPP-028 FR-10024 FR-110302 FR-113452 FR-113680 FR-115092 FR-115427 FR-118487 FR-121196 FR-122047 FR-123826 FR-131535 FR-133605 FR-134043 FR-139317 FR-140423 FR-144420 FR-145237 FR-145715 FR-146801 FR-160 FR-161282 FR-167344 FR-167653 FR-168888 FR-171113 FR-17126 FR-172357 FR-173657 FR-180102 FR-182024 FR-182877 FR-183998 FR-186054 FR-189419 FR-190997 FR-193108 FR-21818 FR-33 FR-35447 FR-46091 FR-46171 FR-46758 FR-47920 FR-48217 FR-49175 FR-64822 FR-66973 FR-66979 FR-66980 FR-71021 FR-76830 FR-860 FR-900109 FR-900359 FR-900405 FR-900411 FR-900452 FR-900482 FR-900483 FR-900490 FR-900523 FR-900840 FR-900848 FR-901228 FR-901451 FR-901463 FR-901464 FR-901465 FR-901469 FR-901483 FR-901537 FR-A-19 FRAN-12 FRG-8813 FS-069 FS-205-397 FS-32 FTI-2148 FTI-2153 FTI-276 FTI-277 FTX-3.3 FTY-720 FUB-181 FUB-360 FUB-373 FUB-407 FUB-451 FUB-86 FX-205-754 FXV-673 G-1-64 G-1026 G-11021 G-11035 G-1460 G-185 G-219 G-229 G-25671 G-264 G-3063 G-3139 G-31442 G-32642 G-33378 G-365 G-4073 G-4120 G-476 G-491 G-512 G-545 G-619 G-6191 G-6249 G-6788 G-7039 G-7203 G-7502 G-871 G-872 G-937 GA-0056 GA-0113 GA-102 GA-3 GA-95 GAP-31 GAR-936 GBC-590 GBR-11513 GBR-12783 GBR-12909 GBR-12921 GBR-12922 GBR-12935 GBR-13069 GBR-13098 GBR-13119 GC-1993 GC-46 GC-94

1260 APPENDIX D GD-131 GD-40 GD-42 GD-7 GE-132 GE-2270-A GE-2270A GE-3 GE-3-B GE-37468-A GE-410 GE-430 GE-68 GE-70 GE-76 GEA-3162 GEA-3175 GEA-3268 GEA-5024 GEA-5145 GEA-857 GEA-968 GEM-132 GEM-231 GEM-91 GERI-BP-001-M GF-109203X GF-120918 GF-120918-A GG-211 GG-745 GGTI-2154 GGTI-286 GGTI-287 GGTI-297 GGTI-298 GH-74 GI-104313 GI-129471 GI-147211 GI-147211-C GI-147211C GI-149893 GI-90291 GK-128 GK-13 GK-206 GL-331 GL-522 GLA-27 GLA-40 GLA-47 GLA-57 GLA-58 GLA-59 GLA-60 GLA-63 GLA-65 GLA-66 GLA-70 GLG-V-13 GLQ-223 GLYCYRRHIZATE-= GLUCURONIDE GM-1077 GM-109 GM-1474 GM-160575 GM-193663 GM-237354 GM-3290 GM-53 GM-6001 GM-611 GMC-5032 GMC-5034 GOE-4902 GOE-5438 GOE-5549 GOE-5584-A GOE-5606 GOE-5806-A GOE-6070 GOE-6976 GOE-6983 GOE-7874 GP-1-343 GP-1-515 GP-1-531 GP-1-668 GP-1447 GP-2-128 GP-2-128-7 GP-27 GP-41299 GP-45699 GP-45795 GP-47779 GP-48989 GP-50302 GP-53633 GP-683 GP-7 GPA-1657 GPA-1658 GPA-1734 GPA-1843 GPA-1847 GPA-1851 GPA-2163 GPI-0100 GPI-1046 GPI-6150 GR-100151 GR-100679 GR-103545 GR-103691 GR-113808 GR-117289 GR-117289-C GR-122222-X GR-125487 GR-125743 GR-127935 GR-138950 GR-138950-C GR-144053 GR-151004-B GR-159897 GR-168320 GR-190178 GR-196429 GR-203040 GR-205171 GR-213907 GR-214060 GR-226206 GR-32191B GR-36246 GR-36264 GR-38414 GR-45809 GR-46611 GR-49336 GR-54374 GR-54374X GR-63799X GR-64349 GR-65630 GR-65630A GR-69153 GR-71251 GR-73632 GR-79236 GR-82334 GR-86014 GR-89696 GR-90291 GR-91272 GR-92132-X GR-92132-X GR-94800 GR-94839 GR-98145 GR-C-507-75 GR2-1159 GRI-1665 GS-13007 GS-1500 GS-1659 GS-389 GS-4071 GS-4104 GS-4116 GS-522 GSC-150 GT-12 GT-165 GT-2227 GT-2331 GT-256729-X GTS-21 GV-104326 GV-118819 GV-129606 GV-150013 GV-150013-X GV-150526-A GV-196771-A GV-213237-A GV-254504 GVS-111 GW-0072 GW-154 GW-158 GW-1818 GW-187 GW-1929 GW-2016 GW-2331 GW-274150 GW-280430-A GW-347845-X GW-3600 GW-409544 GW-420371-X GW-433908 GW-4459 GW-510516 GW-5638 GW-5823 GW-7647 GW-7845 GW-8510 GW-92527 GW-974 GX-258 GY-97 GYKI-11679 GYKI-12735 GYKI-12743 GYKI-13324 GYKI-13380 GYKI-14166 GYKI-14238 GYKI-14451 GYKI-14766 GYKI-21114 GYKI-22441 GYKI-23107 GYKI-24479 GYKI-32084

Derwent Drug File 1261 Thesaurus GYKI-32887 GYKI-35064 GYKI-52466 GYKI-52713 GYKI-52843 GYKI-53405 GYKI-53655 GYKI-53655 GYKI-53784 GYKI-66114 H-100-11 H-104-83 H-105-22 H-105-29 H-1067 H-1075 H-1076 H-113 H-1152 H-117-04 H-117-78 H-119-66 H-119-68 H-119-72 H-1285 H-13-04 H-132-89 H-142 H-151-46 H-151-72 H-151-73 H-152-37 H-152-66 H-155-73 H-160-51 H-168-22 H-168-66 H-170-31 H-173-09 H-186-86 H-19 H-193-10 H-193-12 H-195-60 H-195-80 H-2-G H-200-62 H-200-66 H-200-68 H-215-02 H-22-54 H-224-25 H-256 H-261 H-29-50 H-290-51 H-2954 H-3031 H-335-25 H-35-25 H-4295 H-44-68 H-47 H-5 H-5350 H-59-64 H-635 H-64-52 H-7 H-74 H-75-12 H-76 H-76-8159 H-77 H-77-77 H-774 H-8 H-81-75 H-8208 H-85 H-86 H-87 H-87-07 H-88 H-88-61 H-89 H-9 H-98-52 HA-1004 HA-103 HA-1100 HA-112 HA-113 HA-114 HA-116 HA-117 HA-118 HA-14-1 HA-140 HA-307-319 HA-48 HA-94 HA-966 HA-97 HAI-105 HB-19 HB-218 HB-66 HBY-097 HC-15 HCL-31-D HCO-40 HCT-3012 HD-233 HE-30346 HE-90481 HERCULES-9007 HET-0016 HF-2035 HFV-1017-C HGA-1 HGG-12 HGG-21 HGG-42 HGG-52 HGG-65 HGG-70 HH-38 HI-236 HI-253 HI-280 HI-6 HI-7 HL-004 HL-91 HLOE-7 HM-197 HMN-176 HMR-1098 HMR-1279 HMR-1372 HMR-1402 HMR-1556 HMR-1715 HMR-1794 HMR-3562 HMR-3787 HN-10200 HN-11500 HN-65021 HNS-32 HO-221 HOE-065 HOE-140-DE-ARG-10 HOE-15030 HOE-288 HOE-33342 HOE-36992 HOE-43254 HOE-511 HOE-602 HOE-694 HOE-71-GT HOE-782 HOE-944 HOE-961 HOE-BAY-946 HOE-S616 HOE-S688 HP-184 HP-228 HP-236 HP-370 HP-466 HP-505 HP-573 HP-654 HP-736 HP-7480 HPA-23 HPA-39 HPE-101 HPT-430 HQ-275 HQL-79 HR-2074 HR-2153 HR-2257 HR-546 HR-720 HR-780 HR-916-B HR-979 HRE-664 HRK-055512 HRK-429 HRP-2000 HS-058 HS-12 HS-14 HS-142-1 HS-2314 HS-3 HS-342 HS-37 HS-378 HS-4 HS-6 HS-692 HSP-117 HSR-284 HSR-6071 HSR-609 HSR-803 HSR-81 HSR-903 HT-90-B HU-210 HU-211 HU-213 HUF-2046 HV-723 HW-13 HW-165 HWA-131 HWA-214 HX-0112 HX-1171 HX-600 HX-630 HX-CH-44-BS HYB-101400

1262 APPENDIX D HYB-190 HZ-2 I-06 I-102 I-152 I-537 I-65 IA-3 IA-4 IA-5 IA-6 IB-503 IBI-P-05006 IC-83-1423 ICD-467 ICI-101187 ICI-105552 ICI-106270 ICI-111075 ICI-115432 ICI-118233 ICI-118551 ICI-120518 ICI-130685 ICI-133312 ICI-138061 ICI-139462 ICI-140447 ICI-141389 ICI-142269 ICI-145458 ICI-145663 ICI-145680 ICI-147798 ICI-153066 ICI-153110 ICI-154129 ICI-159995 ICI-162846 ICI-164384 ICI-169369 ICI-170777 ICI-170809 ICI-174864 ICI-180080 ICI-185282 ICI-190622 ICI-192605 ICI-193428 ICI-194008 ICI-195739 ICI-197067 ICI-198157 ICI-198583 ICI-198615 ICI-199441 ICI-200355 ICI-200880 ICI-201651 ICI-204448 ICI-205930 ICI-206970 ICI-207828 ICI-207968 ICI-211965 ICI-213689 ICI-215001 ICI-215918 ICI-216140 ICI-216800 ICI-220800 ICI-230487 ICI-3188 ICI-3327 ICI-42464 ICI-43823 ICI-45337 ICI-46037 ICI-47699 ICI-47776 ICI-49455 ICI-53072 ICI-55548 ICI-58301 ICI-61129 ICI-63197 ICI-65709 ICI-73602 ICI-74205 ICI-77949 ICI-79792 ICI-79939 ICI-80205 ICI-85966 ICI-86841 ICI-89406 ICI-90069 ICI-95527 ICI-A-5165 ICI-D-0490 ICI-D-2138 ICI-D-6888 ICI-D-7114 ICI-D-7288 ICI-D-8731 ICI-D1542 ICIG-1105 ICIG-1163 ICIG-1164 ICN-3952 ICP-1 ICR-170 ICR-191 ICRF-154 ICRF-158 ICRF-186 ICRF-192 ICRF-193 ICRF-197 ICRF-198 ICRF-202 ICRF-226 ICRF-500 ICRF-505 ICRF-510 ICRF-602 ID-1229 ID-17263 ID-17332 ID-4708 ID-495-37 ID-955 IDB-1027 IDB-1031 IDEC-131 IDEC-152 IDN-1965 IDN-5109 IDN-5390 IDPH-791 IDRA-21 IEM-1460 IEM-1592 IEM-1754 IEM-1857 IEM-474 IEM-476 IEM-487 IEM-508 IEM-611 IEM-759 IF-C-45 IG-10 IGN-2098 IH-636 IH-901 IHC-72 IIK-7 IK-29 IK-82029 IKD-8344 IL-40 ILX-23-7553 IM-862 IMET-28-67 IMET-2951 IMET-3164 IMET-3293 IMET-3379 IMOL-881 INN-00835 INO-2628 INO-2628-CZ INS-365 INX-3280 IO-21 IOS-1-1212 IOS-4074 IOS-4732 IP-66 IPD-1151T IPS-1251 IPS-339 IPS-621 IPS-622 IPS-626 IPS-629 IQ-23 IQ-3-B IQB-782 IQB-9302 IQM-95333 IRC-11 IRFI-005 IRFI-016 IRFI-042 IRFI-048 IRFI-117 IRFI-165 IRI-426 IRL-1038 IRL-1620 IRL-1736 IRL-2500 ISA-13-1 ISA-70 ISF-2405 ISIS-1082 ISIS-11061 ISIS-12449 ISIS-12959 ISIS-13650 ISIS-1570 ISIS-1751 ISIS-1753 ISIS-1755 ISIS-2105 ISIS-2302 ISIS-2503 ISIS-2922 ISIS-3082 ISIS-3521 ISIS-4015 ISIS-5320 ISIS-8005 ISIS-9044 ISIS-9047 ISO-DC-81 ISP-I-55 IST-622 IT-066 IT-62-B

Derwent Drug File 1263 Thesaurus ITF-1124 ITF-1300 ITF-1577 ITF-282 ITF-296 ITF-300 ITF-611 ITF-614 ITV-8912 IVX-E-59 IWF-122-14 IWF-122-60 IY-81149 J-104118 J-104132 J-104870 J-109404 J-111225 J-113397 J-114870 J-303 J-508 J-512 J-516 J-628 J-8 J-811 J-824 J-861 J-96 J-995 JB-318 JB-336 JB-336-4 JB-835 JB-93182 JB-9322 JCA-304 JCA-314 JCF-9 JE-2147 JG-365 JG-73 JGC-174 JK-1624-2 JK-1624-3 JL-13 JL-3 JM-1 JM-10 JM-11 JM-118 JM-120 JM-122 JM-125 JM-132 JM-149 JM-1590 JM-1591 JM-1596 JM-1657 JM-185 JM-2 JM-20 JM-216 JM-221 JM-222 JM-223 JM-225 JM-229 JM-231 JM-236 JM-244 JM-251 JM-256 JM-260 JM-262 JM-2644 JM-269 JM-271 JM-273 JM-274 JM-2762 JM-2763 JM-2768 JM-2815 JM-2820 JM-291 JM-2936 JM-3 JM-3100 JM-334 JM-335 JM-34 JM-383 JM-40 JM-407 JM-473 JM-480 JM-5 JM-6 JM-64 JM-68 JM-82 JM-93 JMB-249 JMV-170 JMV-179 JMV-180 JMV-236 JMV-310 JMV-320 JMV-328 JMV-332 JMV-390-1 JMV-449 JO-1605 JO-1717 JO-1783 JOD-173 JOD-176 JOM-13 JPC-266 JPC-6036 JTE-522 JTE-607 JTH-601 JTP-2724 JTP-2942 JTP-4819 JTT-705 JTV-506 JTV-519 JTV-605 JV-1-36 JVA-901 JWH-015 JWH-018 JWH-030 JWH-051 JWH-073 JWH-133 K-107 K-11002 K-11017 K-1115-A K-11777 K-12 K-120 K-122 K-13 K-130 K-137 K-138 K-150 K-185 K-1905 K-191 K-2-9 K-2002 K-2234 K-252B K-252C K-252D K-259-2 K-2604 K-277 K-37 K-38 K-3827 K-4010 K-4011 K-42 K-42999 K-4300 K-4423 K-4540 K-4619 K-50478 K-582-A K-6341 K-6342 K-6343 K-7259 K-76 K-953 K-96 KA-398 KAA-276 KABI-2023 KABI-2161 KAD-1229 KAR-2 KB-1043 KB-2683 KB-2714 KB-2796 KB-3022 KB-5246 KB-5492 KB-5666 KB-6933 KB-R-7785 KB-R-7943 KB-R-8498 KBR-9032 KBT-3022 KC-11404 KC-11458 KC-116 KC-12291 KC-1318 KC-144 KC-146 KC-3755 KC-3756 KC-399 KC-404 KC-515 KC-6141 KC-764 KC-8851 KC-9048 KCA-098 KCB-328 KCD-232 KDI-792 KE-298 KE-748 KE-758 KF-14363 KF-1492

1264 APPENDIX D KF-15372 KF-15570 KF-17625 KF-17837 KF-18259 KF-19514 KF-20170 KF-20405 KF-24345 KF-25706 KF-4307 KF-4317 KF-4939 KF-4942 KF-58333 KF-66854 KFM-19 KGR-1380 KGR-1421 KH-1059 KH-1060 KH-1139 KH-1230 KHL-8425 KHL-8430 KHPC-002 KI-1769 KI-3005 KI-3315 KI-4032 KI-6783 KI-8110 KIH-200 KIH-201 KIH-202 KIH-802 KIN-804 KL-11 KLI-2 KLI-3 KLI-5 KLN-93 KM-13 KM-966 KMBZ-009 KMD-3213 KME-4 KN-04 KN-62 KN-827 KN-93 KNI-102 KNI-144 KNI-174 KNORR-1887 KO-132 KO-134 KO-143 KO-286011 KOE-1030 KOE-1124 KOE-1313 KOE-1350 KOE-1411 KOE-1439 KOE-1500 KOE-1560 KOE-1561 KOE-3290 KOE-589 KOE-612 KOE-707 KP-1019 KP-103 KP-10614 KP-15 KP-21 KP-23 KP-403 KP-418 KP-735 KP-736 KP-840 KR-30450 KR-30818 KR-31372 KR-31378 KRH-594 KRI-1177 KRI-1230 KRI-1314 KRM-1648 KRM-1657 KRM-1668 KRM-1671 KRN-2391 KRN-4884 KRN-5500 KRN-7000 KRN-8602 KRP-197 KS-501 KS-502 KS-504A KS-504B KS-504D KS-504E KS-505A KS-619-1 KS-79 KSG-504 KSU-1415 KT-1-109 KT-1-293 KT-2-962 KT-3-671 KT-3-671 KT-362 KT-3767 KT-3937 KT-4697 KT-4788 KT-5720 KT-5822 KT-5823 KT-5926 KT-6006 KT-6124 KT-6149 KT-6528 KT-7692 KT-90 KT-95 KU-1257 KU-14-R KU-2285 KUM-32 KUR-1246 KV-1360 KW-2170 KW-2189 KW-3033 KW-3196 KW-3407 KW-3433 KW-3600 KW-3635 KW-3902 KW-4099 KW-4679 KW-4994 KW-5092 KW-5139 KW-5805 KW-6002 KW-6055 KW-6629 KWD-2016 KWD-2023 KWD-2027 KWD-2110 KWD-2131 KWD-2312 KWD-2313 KWD-2314 KY-106 KY-556 KY-62 KYN-54 KZ-1026 KZ-111 L-002 L-0066 L-10492 L-10503 L-121 L-154819 L-155175 L-155212 L-156602 L-157012 L-158338 L-158809 L-159689 L-159913 L-16052 L-161177 L-162223 L-162313 L-162389 L-162441 L-162752 L-163017 L-163191 L-163491 L-163540 L-164710 L-165041 L-165461 L-2 L-246736 L-249313 L-30 L-342643 L-362855 L-365031 L-365209 L-365260 L-366012 L-366509 L-366682 L-366811 L-366948 L-367073 L-368899 L-368935 L-370518 L-371257 L-372460 L-373890 L-374087 L-39 L-3937 L-4035 L-44-0 L-48 L-589420 L-593511 L-593754 L-611744 L-615919 L-62208

Derwent Drug File 1265 Thesaurus L-62211 L-628914 L-630571 L-631529 L-632481 L-634549 L-636028 L-636499 L-637146 L-639019 L-640033 L-640035 L-640876 L-641953 L-643411 L-643441 L-643717 L-643799 L-644122 L-644257 L-644711 L-644763 L-6449 L-644969 L-645151 L-645164 L-646462 L-647318 L-648051 L-648865 L-649923 L-651142 L-651392 L-651525 L-651580 L-651582 L-651896 L-652042 L-652069 L-652343 L-652731 L-653150 L-653180 L-653328 L-654284 L-654639 L-654969 L-655238 L-655240 L-655708 L-656224 L-656575 L-657098 L-657229 L-657743 L-657925 L-657926 L-658758 L-658903 L-659066 L-659286 L-659699 L-659837 L-659874 L-659877 L-659989 L-660281 L-660282 L-660343 L-660347 L-660631 L-660711 L-660863 L-662583 L-663581 L-665210 L-665871 L-6678 L-668169 L-668750 L-669572 L-669844 L-670207 L-670258 L-670592 L-670596 L-670602 L-670630 L-671152 L-671776 L-674573 L-674636 L-679336 L-679723 L-680573 L-680574 L-680831 L-680833 L-680861 L-681176 L-682271 L-682946 L-682993 L-683537 L-683557 L-683558 L-683590 L-683841 L-683845 L-683877 L-684248 L-684249 L-684481 L-685818 L-686398 L-686708 L-687306 L-687384 L-687414 L-687781 L-689037 L-689065 L-689502 L-689560 L-689660 L-690330 L-690488 L-691121 L-691816 L-691886 L-692199 L-692429 L-692585 L-693593 L-693612 L-693989 L-694247 L-694458 L-694746 L-695256 L-695902 L-696040 L-696229 L-696474 L-696475 L-697318 L-697639 L-697661 L-697695 L-698544 L-699333 L-699392 L-700417 L-700653 L-701252 L-701273 L-701324 L-701677 L-702007 L-702539 L-702958 L-703014 L-703606 L-703717 L-705022 L-705589 L-706000 L-708541 L-708906 L-709049 L-709780 L-722151 L-731373 L-731723 L-731734 L-731735 L-731988 L-732138 L-733060 L-733061 L-733560 L-733692 L-734217 L-735821 L-736622 L-737126 L-738167 L-738372 L-739010 L-739594 L-739749 L-740093 L-740093-S L-741519 L-741604 L-741626 L-741671 L-741742 L-742694 L-742728 L-743872 L-744832 L-745296 L-745310 L-745337 L-745870 L-746483 L-746530 L-749329 L-749335 L-749345 L-750667 L-751788 L-754030 L-754142 L-754394 L-755507 L-755805 L-758298 L-758354 L-761066 L-762459 L-762745 L-765314 L-767679 L-767685 L-768242 L-768277 L-768673 L-770644 L-775606 L-778123

1266 APPENDIX D L-779976 L-7810 L-783281 L-786392 L-793422 L-796449 L-796568 L-8040 L-805645 L-8109 L-8142 L-826141 L-8412 L-8580 L-86-8275 L-8711 L-9146 LA-15-PH LA-18-PP LAF-389 LAS-30538 LAS-333 LASSBIO-294 LB-10827 LB-145 LB-30057 LB-32841 LB-42908 LB-71148 LB-71350 LBT-44 LC-6 LCB-2183 LCB-2853 LD-2855 LE-300 LE-540 LEA-103 LEF-553 LEK-8804 LEK-8829 LEX-032 LEXIPAFANT LF-1351 LF-14 LF-1695 LF-20254 LFA-703 LFM-A-13 LG-100127 LG-100128 LG-100182 LG-100268 LG-101305 LG-113 LG-114 LG-115 LG-120746 LG-6-101 LG-6-102 LG-63 LG-82-4-00 LG-82-4-01 LG-83-6-05 LGD-1069 LI-132 LI-1370 LI-160 LILLY-18947 LILLY-51641 LILLY-88571 LIV-100 LJP-249 LJP-394 LK-11 LK-203-030 LK-404 LK-409 LK-410 LK-63 LK-903 LL-115 LL-14-I-352-ALPHA LL-14-I-352-BETA LL-1418 LL-21945 LL-AM-374 LL-AM374 LL-C10037-ALPHA LL-D-49194-ALPHA-1 LL-D49194-ALPHA-1 LL-E-19020-ALPHA LL-E-19020-BETA LL-F28249-BETA LL-F28249-GAMMA LL-F28249-LAMBDA LL-S-491-BETA LL-Z-1271-ALPHA LL-Z-1271-GAMMA LL-Z-1272-EPSILON LM-1228 LM-1453 LM-1468 LM-207 LM-246 LM-5005 LM-609 LM-975 LM-985 LMB-7 LN-1643 LN-2833 LN-2839 LN-5330 LND-369 LND-623 LND-796 LNF-209 LOE-908 LON-954 LOS-1-84 LOS-5-79 LP-805 LR-3280 LR-693 LR-99853 LR-B-057 LR-B-081 LS-20 LS-2715 LS-2724 LS-3347 LS-3348 LS-3360 LS-74 LS-93 LSL-60101 LU-10-134-C LU-103793 LU-11-109 LU-11-161 LU-11-305 LU-127043 LU-13-117 LU-135252 LU-14-068 LU-16-073 LU-17-123 LU-17-133 LU-17-151 LU-17-152 LU-18-006 LU-20884 LU-21-099 LU-224332 LU-24-040 LU-2443 LU-25-109-T LU-28-092 LU-28-179 LU-29024 LU-3-009 LU-302146 LU-302872 LU-420627 LU-43706 LU-48895 LU-49667 LU-49888 LU-49938 LU-49940 LU-51903 LU-53439 LU-55446 LU-58463 LU-79553 LUF-5407 LUF-5484 LUR-2366 LW-10078 LW-10079 LW-10086 LW-10121 LW-50020 LY-062 LY-103629 LY-106737 LY-108742 LY-113821 LY-117018 LY-117413 LY-119123 LY-119932 LY-121887 LY-127210 LY-134046 LY-135114 LY-136595 LY-136596 LY-137150 LY-137157 LY-137617 LY-139478 LY-141865 LY-149179 LY-150310 LY-151364 LY-154005 LY-154045 LY-156007 LY-156525 LY-156735 LY-158A LY-163252 LY-163395 LY-163443 LY-164846 LY-165163 LY-171884 LY-173013 LY-175877 LY-177507 LY-178002 LY-178207 LY-180299 LY-181512 LY-181984 LY-181985 LY-183001 LY-186126 LY-186232 LY-186391

Derwent Drug File 1267 Thesaurus LY-186826 LY-189585 LY-189709 LY-190147 LY-191145 LY-191704 LY-193239 LY-193525 LY-195114 LY-195448 LY-195449 LY-195779 LY-197055 LY-197096 LY-197221 LY-197541 LY-201409 LY-201979 LY-202475 LY-202991 LY-202992 LY-203647 LY-203725 LY-206130 LY-206243 LY-207702 LY-210825 LY-211000 LY-211888 LY-212556 LY-213829 LY-214138 LY-214624 LY-215490 LY-215840 LY-217896 LY-219057 LY-219703 LY-221068 LY-221501 LY-222675 LY-223980 LY-223982 LY-225297 LY-227409 LY-227420 LY-227938 LY-227942 LY-228729 LY-231514 LY-231617 LY-233053 LY-233536 LY-235723 LY-235959 LY-243246 LY-249933 LY-253352 LY-253963 LY-254155 LY-254239 LY-254490 LY-255262 LY-255283 LY-255582 LY-256548 LY-256787 LY-257883 LY-258458 LY-262691 LY-264656 LY-264826 LY-266070 LY-266111 LY-267108 LY-269415 LY-274601 LY-274614 LY-275585 LY-278584 LY-278989 LY-280810 LY-281389 LY-281980 LY-288513 LY-289612 LY-290181 LY-290293 LY-290411 LY-293111 LY-293558 LY-293559 LY-294002 LY-294619 LY-295427 LY-295501 LY-297802 LY-298207 LY-300046 LY-300082 LY-300164 LY-300502 LY-300503 LY-301317 LY-301621 LY-301875 LY-302679 LY-303366 LY-303870 LY-306669 LY-307161 LY-307452 LY-307599 LY-307853 LY-309887 LY-314593 LY-315535 LY-315902 LY-316108 LY-316373 LY-317236 LY-317584 LY-317615 LY-320135 LY-326315 LY-326325 LY-329146 LY-333068 LY-333531 LY-334370 LY-335563 LY-335979 LY-338522 LY-339434 LY-341495 LY-343928 LY-344864 LY-34580 LY-353352 LY-353433 LY-354740 LY-357489 LY-367385 LY-377604 LY-379268 LY-389795 LY-393053 LY-404187 LY-41 LY-444711 LY-448212 LY-448731 LY-465803 LY-487355 LY-509207 LY-51641 LY-53857 LY-55 LY-56110 LY-582563 LY-73497 LY-78335 LY-79771 LY-806303 LY-81067 LY-83583 LY-86057 LY-87130 LY-88329 LY-93716 LY-97119 LY-97241 LY-99335 LZ-8 M+B-18706 M+B-28767 M+B-30227 M+B-31426 M+B-35769 M+B-39434 M+B-39890A M+B-4596 M+B-7714 M-12285 M-12325 M-14659 M-15 M-154129 M-16049 M-16209 M-16287 M-1704 M-17055 M-254 M-30 M-32 M-320 M-35 M-40401 M-40403 M-4365-G2 M-5011 M-6007 M-6434 M-66 M-7 M-711 M-79175 M-79193 M-8 M-840 M-9260 MA-540 MA-56 MAP-1987 MAP-4 MAR-99 MAZ-525 MB-3 MB-432 MBI-27 MBI-28 MC-02479 MC-1046 MC-1080 MC-11 MC-1145 MC-1288 MC-1301 MC-62 MC-77 MC-838

1268 APPENDIX D MCC-134 MCC-555 MCI-154 MCI-176 MCI-196 MCI-225 MCI-727 MCI-826 MCN-2165 MCN-2891 MCN-4130 MCN-4187 MCN-4612-Z MCN-5195 MCN-5195-11 MCN-5652 MCN-5652-Z MCN-5655-Z MCN-5691 MCN-5707 MCN-5908 MCN-6186 MCN-A-1293 MCN-A-343 MCN-R-1832-11-98 MD-220661 MD-240098 MD-240233 MD-240928 MD-240931 MD-760548 MD-770222 MDL-100151 MDL-100173 MDL-100240 MDL-100453 MDL-100907 MDL-101002 MDL-101028 MDL-101146 MDL-101731 MDL-102111 MDL-102234 MDL-102382 MDL-102823 MDL-102832 MDL-103323 MDL-103392 MDL-104342 MDL-104653 MDL-104653 MDL-105185 MDL-105212-A MDL-105519 MDL-12330A MDL-14514 MDL-16455-A MDL-17523 MDL-17637 MDL-18341 MDL-18962 MDL-19152 MDL-19438 MDL-19592 MDL-19660 MDL-201012A MDL-201040 MDL-201053 MDL-201112 MDL-201307 MDL-201346 MDL-201404 MDL-201449 MDL-201451 MDL-201484 MDL-20610 MDL-20646 MDL-20828 MDL-25637 MDL-26024-GO MDL-26479 MDL-26508 MDL-26547 MDL-26752 MDL-27032 MDL-27048 MDL-27088 MDL-27192 MDL-27210 MDL-27391 MDL-27531 MDL-27693 MDL-27695 MDL-27700 MDL-27701 MDL-27777 MDL-27994 MDL-28050 MDL-28133A MDL-28170 MDL-28560 MDL-28564 MDL-28574 MDL-28653 MDL-28815 MDL-28842 MDL-29204 MDL-29270 MDL-29311 MDL-29435 MDL-29913 MDL-427 MDL-43305 MDL-43925 MDL-44370 MDL-62208 MDL-62211 MDL-62873 MDL-63246 MDL-71801 MDL-72145 MDL-72175 MDL-72222EF MDL-72274 MDL-72392 MDL-72394 MDL-72403 MDL-72430 MDL-72483 MDL-72521 MDL-72527 MDL-72567 MDL-72638 MDL-72699 MDL-72832 MDL-72912 MDL-72974 MDL-73005 MDL-73005EF MDL-73147 MDL-73404 MDL-73405 MDL-73450 MDL-73492 MDL-73745 MDL-73811 MDL-73945 MDL-74156 MDL-74156EF MDL-74180-DA MDL-74217 MDL-74270 MDL-74366 MDL-74405 MDL-860 MDV-1 MDV-2 MDX-33 MDX-H-210 ME-1207 ME-1228 ME-1401 ME-2303 ME-3221 ME-3229 ME-3277 ME-3407 ME-506 ME-93 MEN-10207 MEN-10208 MEN-10282 MEN-10376 MEN-10397 MEN-10400 MEN-10414 MEN-10567 MEN-10627 MEN-10690 MEN-10700 MEN-10706 MEN-10710 MEN-10755 MEN-11149 MEN-11270 MEP-1 MERCK-L-7 METHOXYDEOXYVASICINONE MF-10058 MF-13 MF-268 MF-5137 MF-922 MF-961 MFS-3 MG-1 MG-115 MG-132 MG-262 MG-341 MG-98 MGK-264 MGN-3 MGS-0008 MGS-0028 MHS-2 MI-1544 MJ-13653 MJ-13980-1 MJ-14030 MJ-1991 MJ-451 MJ-7378 MJ-7434-1 MJ-7999-1 MJ-8592-1 MJ-9444 MJ-9465-2 MK-0591 MK-0677 MK-0852 MK-0869 MK-0963 MK-1-203 MK-1-907 MK-142 MK-212 MK-251 MK-286 MK-306 (psychostimulant) MK-316 MK-351A

Derwent Drug File 1269 Thesaurus MK-363-301 MK-386 MK-410 MK-434 MK-436 MK-447 MK-462 MK-467 MK-473 MK-597 MK-678 MK-711 MK-715 MK-761 MK-771 MK-789 MK-825 MK-830 MK-869 MK-875 MK-886 MK-910 MK-927 MK-954 MK-966 MK-996 MKC-231 MKC-242 MKC-442 MKC-733 MKS-492 MKT-077 ML-10302 ML-1035 ML-10375 ML-23 ML-236A ML-4 ML-7 ML-9 MLM-160 MLR-52 MLV-3076 MLV-5860 MLV-6976 MM-17880 MM-218 MM-22381 MM-22382 MM-44785 MM-44787 MM-4550 MM-46115 MM-706 MMB-4 MMI-166 MNA-279 MNA-715 MNX-160 MOL-5210 MOP-35 MOP-79 MP-2001 MP-3022 MP-90 MPB-07 MPC-2101 MPV-1440 MPV-207 MPV-2213-AD MPV-2426 MPV-295 MPV-304 MPV-305 MPV-390 MR-1-12 MR-1268 MR-1353 MR-1452 MR-1453 MR-16728 MR-2033 MR-2034 MR-2035 MR-20492 MR-2096-CL MR-2097-CL MR-2261 MR-2264-CL MR-2266 MR-2266-BS MR-2267 MR-2549 MR-256 MR-356 MR-566-A MR-566-B MR-714 MR-889 MR-948 MRE-0470 MRL-37 MRS-1067 MRS-1097 MRS-1191 MRS-1220 MRS-1754 MRS-1760 MRS-2179 MRS-2257 MRS-2286 MRX-115 MRX-408 MRZ-2-570 MRZ-2-571 MRZ-2-576 MRZ-2549 MRZ-3-124 MRZ-3124 MS-073 MS-153 MS-209 MS-247 MS-257 MS-27-275 MS-322 MS-325 MS-377 MS-424 MS-430 MS-444 MS-551 MS-681-A MS-681-B MS-681-C MS-681-D MS-818 MS-8209 MS-857 MSC-204 MSC-206 MSD-235-S2 MSD-53 MSD-642317 MSD-819 MSH-372 MSI-103 MSI-1436 MSI-238 MSI-30 MSI-78 MSI-78-A MSI-94 MSI-98 MSL-109 MST-16 MT-0703 MT-81 MTP-1307 MUP-98156 MV-6401 MVE-4 MVT-101 MX MX-1 MX-2 MX-2-120 MX-3350-1 MX-68 MY-103 MY-12-62-C MY-1250 MY-336-A MY-40-20 MY-5 MY-5445 MZ-108 MZ-2-117 MZ-2-123 MZ-2-135 MZ-2-51 MZ-2-57 MZ-2-75 MZ-2-87 MZ-4-243 MZ-4-71 MZ-5-156 N-0164 N-0425 N-0434 N-0435 N-0436 N-0437 N-0438 N-0498 N-0499 N-0724 N-0840 N-0861 N-0918 N-0923 N-0953 N-1005 N-1024 N-1199 N-1518 N-30 N-3256 N-3389 N-3601 N-4472 N-4909 N-5+ N-5228 N-7006 N-718 N-751 N-762-A N-762-B N-789 N-796-A N-796-B NA-0344 NA-0345 NA-0346 NA-0359 NA-0362 NA-22598-A-1 NA-332 NA-379 NA-381 NA-382

1270 APPENDIX D NAB-277 NAM-204 NAM-221 NAM-224 NAM-242 NAM-250 NAN-190 NAP-5 NAP-C-2 NARI-10146 NAT-02-677 NAT-06-097 NB-1011 NB-355 NB-431 NB-506 NB-598 NBF-003 NBF-008 NBF-021 NBF-027 NBO-6 NBQ-38 NBQ-48 NBQ-59 NC-100100 NC-1100 NC-1140 NC-1300 NC-1300-B NC-1300-SULFIDE NC-17 NC-190 NC-1900 NC-8-12 NCC-05-0711 NCO-650 NCO-700 NCQ-115 NCQ-134 NCQ-258 NCQ-298 NCQ-318 NCQ-344 NCQ-436 NCQ-616 NCS-382 NCS-686760 NCX-1000 NCX-1015 NCX-1020 NCX-4016 NCX-4215 NCX-701 NCX-950 ND-186 ND-502 NDH-3080 NDO-008 NE-0080 NE-100 NE-10133 NE-10244 NE-21610 NE-28345 NE-58051 NE-58095 NE-97220 NF-007 NF-018 NF-023 NF-031 NF-032 NF-037 NF-103 NF-110 NF-143 NF-2 NF-201 NF-279 NF-326 NF-449 NF-503 NF-504 NF-506 NG-011 NG-012 NGD-94-1 NGP-1-01 NH-40 NIH-10236 NIH-10420 NIH-10741 NIK-228 NIM-76 NIP-121 NIP-200 NK-104 NK-121 NK-121 NK-122 NK-250 NK-252 NK-3201 NK-422 NK-424 NK-433 NK-611 NKH-477 NKK-100 NKP-608 NL-105 NL-106 NM-324 NM-394 NM-404 NMI-377 NN-2211 NN-304 NNC-01-0687 NNC-0112 NNC-09-0026 NNC-13-8119 NNC-13-8199 NNC-13-8241 NNC-14-0185 NNC-21-0238 NNC-22-0010 NNC-22-0031 NNC-22-0215 NNC-25-2504 NNC-53-0055 NNC-53-0082 NNC-70-0270 NNC-711 NNC-90-1515 NNC-90-3094 NO-01-0756 NO-1886 NO-329 NO-434 NO-437 NO-794 NOC-5 NOC-7 NP-207 NP-252 NP-59 NPB-1 NPC-12626 NPC-14692 NPC-15199 NPC-15437 NPC-15669 NPC-16377 NPC-16570 NPC-16731 NPC-17731 NPC-17742 NPC-17761 NPC-17923 NPC-18521 NPC-18688 NPC-18730 NPC-205 NPC-414 NPC-567 NPC-573 NPF-86-IA NPF-86-IB NPF-86-IIA NPF-86-IIB NPF-86IA NPF-86IB NPF-86IIA NPF-86IIB NPK-1867 NPK-1868 NPK-1882 NPK-1886 NPS-2143 NPS-846 NPS-R-568 NQ-Y-15 NR-583143 NRA-0045 NRA-0160 NRA-0161 NRA-0215 NRA-0562 NRDC-156 NS-004 NS-1 NS-102 NS-105 NS-11 NS-1608 NS-1619 NS-1652 NS-1C NS-1D NS-21 NS-2346 NS-2359 NS-257 NS-398 NS-49 NS-7 NSC-100880 NSC-101327 NSC-107392 NSC-110333 NSC-113423 NSC-114460 NSC-115290 NSC-117614 NSC-118203 NSC-125358 NSC-126771 NSC-127755 NSC-128189 NSC-140117 NSC-140701 NSC-143414 NSC-145813 NSC-146067 NSC-146068 NSC-158197 NSC-158393 NSC-170895 NSC-170898 NSC-170899

Derwent Drug File 1271 Thesaurus NSC-176319 NSC-181928 NSC-191295 NSC-194814 NSC-20625 NSC-211327 NSC-215914 NSC-224070 NSC-224964 NSC-232965 NSC-235777 NSC-23909 NSC-239717 NSC-239851 NSC-246112 NSC-250427 NSC-251635 NSC-255110 NSC-259946 NSC-262666 NSC-267213 NSC-269130 NSC-269416 NSC-271674 NSC-278214 NSC-278467 NSC-278999 NSC-281246 NSC-287474 NSC-289517 NSC-290205 NSC-296964 NSC-303861 NSC-30705 NSC-3077 NSC-311469 NSC-314622 NSC-321567 NSC-321584 NSC-324368 NSC-328002 NSC-330465 NSC-330507 NSC-330770 NSC-335154 NSC-337238 NSC-338600 NSC-338698 NSC-339675 NSC-340307 NSC-341082 NSC-341936 NSC-341964 NSC-343513 NSC-343529 NSC-344270 NSC-344280 NSC-347515 NSC-350102 NSC-350386 NSC-350602 NSC-352683 NSC-352692 NSC-352875 NSC-352876 NSC-353649 NSC-354646 NSC-355277 NSC-357704 NSC-35843 NSC-361456 NSC-364720 NSC-365171 NSC-366140 NSC-370147 NSC-370277 NSC-371168 NSC-373232 NSC-375574 NSC-381577 NSC-38280 NSC-402538 NSC-402666 NSC-4493 NSC-46015 NSC-46015-C NSC-47547 NSC-49272 NSC-521164 NSC-56336 NSC-57153 NSC-57155 NSC-60339 NSC-606174 NSC-606698 NSC-607732 NSC-609974 NSC-612567 NSC-613060 NSC-613862 NSC-613863 NSC-615830 NSC-615831 NSC-615985 NSC-619444 NSC-619446 NSC-619531 NSC-624151 NSC-624152 NSC-624231 NSC-625487 NSC-627505 NSC-628679 NSC-629243 NSC-629971 NSC-630176 NSC-630176D NSC-639366 NSC-639829 NSC-640488 NSC-645306 NSC-647884 NSC-648400 NSC-649488 NSC-651016 NSC-654021 NSC-654261 NSC-655649 NSC-662304 NSC-662306 NSC-663284 NSC-665517 NSC-666724 NSC-667005 NSC-66761 NSC-668380 NSC-676418 NSC-678515 NSC-680434 NSC-680718 NSC-684681 NSC-686288 NSC-693567 NSC-71261 NSC-714187 NSC-76509 NSC-82196 NSC-83265 NSC-84954 NSC-84963 NSC-86047 NSC-87974 NSC-87982 NSC-88104 NSC-95397 NSC-95580 NSC-D-614989 NSC-D-682300-O NSC-D-683663-U NSC-D-699127 NSD-1015 NSD-1024 NSD-1034 NSD-2023 NSD-3004 NSFQ-104 NSFQ-105 NSH-134 NSL-9403 NSP-804 NSP-805 NTE-122 NU-1025 NU-1064 NU-2058 NU-6027 NU-7026 NU-7163 NU-UB-199 NU-UB-31 NV-14 NV-15 NV-4 NV-6 NVP-DPP-728 NVP-VID-400 NXY-059 NY-008 NY-3170 NY-3460 NY-4137 NY-4138 NZ-107 NZ-314 O-129 O-401 O-823 OA-6129A OA-6129B1 OA-6129B2 OA-6129C OA-7653 OB-47042 OC-144093 OC-2186 OC-229-648 OC-5181 OC-5186 OCT-43 ODN-1760 OF-4949-I OF-4949-II OF-4949-III OF-4949-IV OF-6145 OF-743 OF-900 OF-900 OG-21 OG-30 OG-57 OG-90 OGT-719 OH-10172 OH-3984-K-1 OH-3984-K-2 OH-87 OHM-11526 OHM-3295 OHM-3463 OI-77 OK-1035

1272 APPENDIX D OK-431 OKY-1580 OKY-1581 OL-17 OL-2 OL-21 OM-01 OM-163 OM-38 OM-8980 OMS-15 ON-579 ONO-1101 ONO-11120 ONO-1301 ONO-1714 ONO-3122 ONO-3144 ONO-3307 ONO-3403 ONO-3708 ONO-4007 ONO-5046 ONO-6240 ONO-6818 ONO-8711 ONO-8809 ONO-8815-LY ONO-9902 ONO-AE-1-259 ONO-AE-1-329 ONO-AE-248 ONO-AP-227 ONO-AP-324 ONO-AP-437 ONO-EI-601 ONO-LB-457 ONO-NT-012 ONO-NT-126 ONO-RS-347 ONO-SA-132 ONYX-015 OP-1206 OP-2123 OP-2507 OP-386 OP-6 OP-622 OPB-9195 OPC-13015 OPC-13135 OPC-13211 OPC-13213 OPC-13215 OPC-13217 OPC-13326 OPC-13366 OPC-13371 OPC-14117 OPC-14523 OPC-14597 OPC-15161 OPC-18692 OPC-18790 OPC-21268 OPC-28326 OPC-31260 OPC-33509 OPC-3911 OPC-4392 OPC-6535 OPC-7251 OPC-8490 OPC-88117 OR-10141 OR-1246 OR-1364 OR-1855 OR-1896 OR-486 ORF-13811 ORF-13904 ORF-17578 ORF-17910 ORF-18260 ORF-21243 ORF-5330 ORF-5331 ORG-10172 ORG-10325 ORG-20059 ORG-20241 ORG-20297 ORG-20380 ORG-20494 ORG-20549 ORG-2058 ORG-20599 ORG-21465 ORG-2305 ORG-2766 ORG-30029 ORG-30093 ORG-30273 ORG-30276 ORG-30659 ORG-31376 ORG-31540 ORG-31550 ORG-31710 ORG-34006 ORG-36764 ORG-37684 ORG-4094 ORG-4428 ORG-5222 ORG-5667 ORG-6141 ORG-6363 ORG-6368 ORG-6370 ORG-6582 ORG-6906 ORG-6997 ORG-7268 ORG-7402 ORG-7617 ORG-7797 ORG-8715 ORG-8730 ORG-8764 ORG-9273 ORG-9453 ORG-9489 ORG-9616 ORG-9731 ORG-9935 ORG-9943 ORG-9955 ORG-9991 ORG-GC-94 ORG-NC-58 ORG-OH-06 ORH-3088 ORI-1202 ORI-1313 ORI-1327 OSI-774 OSU-6162 OSW-1 OT-24 OT-7100 OX-353 OXA-22 OXI-4503 P-0160 P-0654 P-1005 P-1015 P-10358 P-1060 P-1075 P-11 P-1188 P-1266 P-1368 P-1507 P-1995 P-23 P-2565 P-275 P-280 P-286 P-30 P-308 P-32-98 P-34081 P-371-A-1 P-3924 P-4018 P-414 P-530 P-532 P-536 P-5369 P-5780 P-65 P-743 P-760 P-792 P-86-7480 P-87-7692 P-8714 P-8720 P-8977 P-903 P-9236 P-9782 P-9941 P-BC-264 PAB-110 PAB-12 PAB-13 PAB-13 PAB-23 PAB-23 PAB-30 PAB-40 PAK-104 PAK-104-P PAT-6 PC-1031 PC-766B PC-796 PC-88 PCA-4230 PCA-4248 PCA-50938 PCA-50941 PCF-39 PCR-0665 PCR-2362 PCR-3787 PCR-4499 PCR-5325 PD-0183085 PD-022551 PD-024886 PD-083176 PD-089828 PD-098059 PD-102807

Derwent Drug File 1273 Thesaurus PD-109488 PD-110095 PD-110334 PD-110911 PD-111103 PD-111391 PD-111707 PD-112940 PD-113270 PD-113271 PD-113297 PD-113377 PD-113413 PD-113876 PD-114027 PD-114057 PD-114245 PD-114254 PD-114255 PD-114541 PD-114595 PD-114631 PD-115311 PD-115934 PD-116124 PD-116152 PD-116169 PD-116198 PD-116250 PD-116427 PD-116740 PD-116948 PD-117302 PD-117519 PD-117558 PD-117596 PD-117802 PD-118309 PD-118484 PD-118717 PD-119229 PD-119421 PD-119556 PD-119819 PD-122642 PD-122860 PD-123177 PD-123319 PD-123475 PD-123497 PD-123982 PD-124816 PD-125354 PD-125639 PD-125944 PD-126280 PD-126889 PD-128763 PD-128907 PD-129290 PD-129635 PD-130694 PD-130883 PD-131112 PD-131501-0 PD-131575 PD-131628 PD-131628-2B PD-132002 PD-132301-2 PD-132486 PD-134308 PD-134672 PD-134922 PD-134965 PD-135022 PD-135042 PD-135158 PD-135390 PD-135666 PD-135739 PD-136095 PD-136450 PD-137156 PD-138136 PD-138142 PD-138142-15 PD-138312 PD-138387 PD-138926 PD-139586 PD-140248 PD-140376 PD-140548 PD-141955 PD-141955-2 PD-142308 PD-142505 PD-142893 PD-142898 PD-143188 PD-143289 PD-144550 PD-144795 PD-144871 PD-145065 PD-145942 PD-146176 PD-146415 PD-146923 PD-150606 PD-150714 PD-151242 PD-152247 PD-152255 PD-153035 PD-153717 PD-154075 PD-155080 PD-156202 PD-156252 PD-156707 PD-157570 PD-157655 PD-157672 PD-158473 PD-158771 PD-158780 PD-158804 PD-159020 PD-159206 PD-159433 PD-160793 PD-160874 PD-161176 PD-161182 PD-161314 PD-161374 PD-161570 PD-161956 PD-163070 PD-163637 PD-163639 PD-164387 PD-164488 PD-165557 PD-166285 PD-166793 PD-166866 PD-167462 PD-168368 PD-168393 PD-169451 PD-169540 PD-171026 PD-172760 PD-173074 PD-178390 PD-178392 PD-180970 PD-183805 PD-184352 PD-69405 PD-72953 PD-81723 PD-83176 PD-85639 PD-98059 PE-1001 PEFA-1023 PEFA-1286 PEP-1261 PF-10040 PF-10042 PF-1022A PF-1092-A PF-1092-B PF-1092-C PF-1163-A PF-257 PF-5901 PF-904 PGE-4175997 PGE-4410186 PGE-9262932 PGE-9509924 PGV-20229 PGV-40350 PH-1008 PH-163 PH-776-141 PH-881-7 PH-QA-33 PI-091 PI-201 PI-88 PIM-35 PIMILPROST PIR-87-6-0 PIXY-321 PJ-34 PJ-91 PK-11195 PK-11211 PK-14067 PK-14068 PK-14105 PK-154 PK-9084 PK-97 PKC-412 PKI-166 PKSI-527 PL-017 PL-058 PL-10 PL-385 PLD-118 PM-1 PM-10 PM-1000 PM-102 PM-104 PM-170 PM-19 PM-2 PM-29 PM-3 PM-30 PM-40 PM-43 PM-44

1274 APPENDIX D PM-47 PM-48 PM-504 PM-523 PM-62 PM-63 PM-64 PM-65 PM-66 PM-67 PM-69 PM-72 PM-73 PM-77 PM-8 PM-82 PM-83 PMS-1 PMS-812 PMS-832 PN-203-831 PN-2034 PN-204-144 PN-204-145 PN-204-775 PN-205033 PN-309 PNO-49-B PNU-101383 PNU-106817 PNU-109112 PNU-109291 PNU-140975 PNU-142721 PNU-145156-E PNU-153429 PNU-156804 PNU-157760 PNU-157820 PNU-157924 PNU-159682 PNU-166945 PNU-171933 PNU-172576 PNU-200577 PNU-99533 PO-285 POT-II PR-000001 PR-000608 PR-1501 PR-19 PR-22 PR-23 PR-25 PR-350 PR-39 PR-546 PR-881-884A PR-967-234 PR-967-248 PR-969-566 PR-D-92-EA PRE-084 PRINOMASTAT PRL-2915 PRO-2000 PS-028 PS-15 PS-179 PS-5 PS-519 PS-6 PS-7 PS-990 PSD-958 PST-2107 PST-2238 PST-2744 PT-141 PT-441 PT-523 PT-619 PT-633 PTR-17402 PTT-119 PTU-23 PV-2 PX-12 PXD-101 PY-11 PY-490 PZ-25 PZII-029 Q-12 Q-85 QA-208-199 QF-0307-B QF-0313-B QF-2003-B QF-2004-B QF-303 QF-307 QF-311 QF-313 QF-503 QF-603 QF-607 QH-25 QM-7184 QR-2 QR-4 QR-5 QW-3600 QW-7437 QX-222 QX-314 QX-572 QYL-1064 QYL-685 QYL-769 QYL-941 QYL-972 R-0363 R-101933 R-10233-DA R-102444 R-10556-DA R-1128-A R-1128-B R-1128-C R-1128-D R-11513-DA R-11567-DA R-11877-DA R-14805 R-151885 R-19352 R-24763 R-2572 R-28935 R-2956 R-29814 R-30490 R-37672 R-39519 R-396 R-40519 R-41232 R-43448 R-4407 R-44271 R-45656 R-48455 R-486 R-49285 R-49399 R-5135 R-5144 R-51703 R-51975 R-52163 R-52164 R-52165 R-52166 R-53531 R-5417 R-56413 R-56566 R-56865 R-57720 R-57974 R-59-022 R-59494 R-59949 R-60164 R-6033 R-61837 R-62025 R-62827 R-63373 R-6597 R-665 R-66703 R-66933 R-67041 R-67138 R-67145 R-68151 R-6998 R-7000 R-70380 R-70608 R-715 R-71811 R-72440 R-73335 R-7371 R-73796 R-74774 R-74893 R-76186 R-76713 R-78206 R-80122 R-8110 R-82150 R-82913 R-830 R-83572 R-836 R-83839 R-83842 R-842 R-84760 R-85355 R-86183 R-88703 R-89439 R-91154 R-95288 R-95867 R-99224 RA-159 RA-433 RA-642 RA-7 RA-700 RA-X RAC-109 RAD-150 RAD-154

Derwent Drug File 1275 Thesaurus RAD-179 RAD-240 RAD-241 RAD-242 RAD-243 RAD-244 RAD-393 RAG-505 RAN-113 RB-1000 RB-101 RB-105 RB-120 RB-211 RB-38A RB-6145 RB-7040 RB-90740 RB-91724 RB-92816 RB-93918 RB-94571 RB-95629 RC-101-I RC-12 RC-121 RC-160-II RC-3095 RC-3105 RC-3125 RC-3420 RC-39-2 RC-3940-II RC-3950-II RC-39II RC-98-I RCC-36 RD-11885 RD-12869 RD-211 RD-219 RD-3-0028 RD-3-0174 RD-42024 RD-42217 RD-6-2198 RD-6-5071 RDP-58 RDS-127 RE-1492 RE-2047 RE-244 RE-61 RE-80 REC-0-0232 REC-15-0209 REC-15-2615 REC-15-2627 REC-15-2636 REC-15-2739 REC-15-2802 REC-15-2841 REC-15-3039 REN-1053 RES-1149-1 RES-1149-2 RES-701 RES-701-1 RES-701-2 REV-3579 REV-5901 REV-5901-A REV-6207 RG-12152 RG-12525 RG-12553 RG-12718 RG-12915 RG-12915A RG-12986 RG-13022 RG-13291 RG-14123 RG-14202 RG-14620 RG-14893 RG-16 RG-25 RG-2958 RG-50810 RG-50858 RG-50864 RG-50875 RG-6866 RG-7152 RG-83852 RGH-0205 RGH-0206 RGH-1756 RGH-4615 RGH-5002 RGH-5981 RGH-6141 RGW-2938 RGW-806 RH-5849 RHC-2851 RHC-3024 RHC-3164 RHC-3414 RHC-3454 RHC-80267 RI-331 RI-61 RIG-200 RJ-64 RJR-2429 RK-153 RK-28 RK-286C RK-30 RK-397 RK-682 RL-712 RLH-033 RM-175 RM-O6 RMI-10026 RMI-10393 RMI-10874-DA RMI-11002-DA RMI-11567-DA RMI-11877-DA RMI-11894 RMI-11974 RMI-12366A RMI-12936 RMI-14133A RMI-15307 RMI-15731 RMI-71626 RMI-71645 RMI-71963 RMI-7822 RMI-82249 RMI-9563-DA RMI-9567-DA RMP-7 RNH-6270 RO-03-4661 RO-03-8800 RO-07-1902 RO-07-3149 RO-09-0410 RO-09-0535 RO-09-0680 RO-09-0696 RO-09-0881 RO-09-1168 RO-09-1428 RO-09-3431 RO-09-4889 RO-1-8307 RO-10-1770 RO-11-0503 RO-11-1272 RO-11-1721 RO-11-2616 RO-11-2933 RO-11-3128 RO-11-3624 RO-11-3651 RO-11-4768 RO-11-4791 RO-11-5073-000 RO-11-6893 RO-11-6896 RO-11-7800 RO-11-8284 RO-11-8958 RO-12-0955 RO-12-0995 RO-12-1989 RO-12-4713 RO-12-4825 RO-12-5637 RO-12-7310 RO-12-7554 RO-12-8095 RO-12-9933 RO-13-2389 RO-13-3892 RO-13-4306 RO-13-6307 RO-13-6680 RO-13-7410 RO-13-8320 RO-13-9259 RO-13-9272 RO-14-3168 RO-14-3899 RO-14-5975 RO-14-7437 RO-14-8935-000 RO-14-9012 RO-14-9572 RO-15-0216 RO-15-1549 RO-15-1903 RO-15-2041 RO-15-3505 RO-15-3890 RO-15-4513 RO-15-5458 RO-15-8081 RO-16-3177 RO-16-6491 RO-16-6532 RO-16-8714 RO-17-6661 RO-18-1675 RO-18-3981 RO-18-5362 RO-18-5364 RO-18-6622 RO-18-8093 RO-19-0528 RO-19-0645 RO-19-0645 RO-19-1400 RO-19-3704 RO-19-4603

1276 APPENDIX D RO-19-4787 RO-19-4788 RO-19-5686 RO-19-7224 RO-19-7731 RO-19-8022 RO-19-9638 RO-2-0683 RO-2-3308 RO-2-7239 RO-2-7509 RO-20-1724 RO-20-2926 RO-21-5104 RO-21-6347 RO-21-6583 RO-21-6667 RO-21-7254 RO-21-7634 RO-21-8303 RO-21-8384 RO-22-0654 RO-22-1327 RO-22-3245 RO-22-4679 RO-22-5851 RO-22-6070 RO-22-6162 RO-22-6595 RO-22-6600 RO-22-6923 RO-22-7878 RO-22-8349 RO-22-9194 RO-23-0238 RO-23-0364 RO-23-0983-001 RO-23-1117-000 RO-23-2895 RO-23-3423 RO-23-3571 RO-23-3880-000 RO-23-4293 RO-23-4319 RO-23-6152 RO-23-6457 RO-23-6829 RO-23-7498 RO-23-7553 RO-23-7637 RO-23-7863 RO-23-8525 RO-23-9424 RO-24-0238 RO-24-2090 RO-24-2287 RO-24-2637 RO-24-4383 RO-24-4637 RO-24-4736 RO-24-5098 RO-24-5531 RO-24-5913 RO-24-6173 RO-24-6392 RO-24-7429 RO-24-8138 RO-24-9981 RO-25-1392 RO-25-1553 RO-25-2032 RO-25-3036 RO-25-3562 RO-25-4020 RO-25-5318 RO-25-6603 RO-25-6760 RO-25-6833 RO-25-6981 RO-25-7553 RO-25-9022 RO-25-9887 RO-28-2653 RO-3-1314 RO-3-1428 RO-3-3528 RO-3-6156 RO-3-7410 RO-3-7894 RO-31-0313 RO-31-0368 RO-31-0521 RO-31-1118 RO-31-1215 RO-31-1740 RO-31-1741 RO-31-1749 RO-31-1966 RO-31-2035 RO-31-3294 RO-31-3689 RO-31-4493 RO-31-4724 RO-31-5460 RO-31-6045 RO-31-6930 RO-31-7208 RO-31-7453 RO-31-7467 RO-31-7549 RO-31-8161 RO-31-8220 RO-31-8425 RO-31-8472 RO-31-8830 RO-31-9790 RO-32-0432 RO-32-1520 RO-32-2313 RO-32-3555 RO-32-4397 RO-32-7315 RO-363 RO-4-1284 RO-4-4318 RO-4-5127 RO-4-6824 RO-4-6861 RO-4-8068 RO-4-8932 RO-4-9040 RO-40-0655 RO-40-1021 RO-40-2148 RO-40-3387 RO-40-5966 RO-40-6890 RO-40-6976 RO-40-7591 RO-40-7592 RO-4020 RO-41-0960 RO-41-1049 RO-41-3118 RO-41-3290 RO-41-3399 RO-41-3696 RO-41-4439 RO-41-5253 RO-41-7812 RO-41-9067 RO-42-5892 RO-42-8773 RO-43-0463 RO-43-5054 RO-43-8857 RO-44-3888 RO-44-9375 RO-44-9883 RO-45-2081 RO-46-2005 RO-46-7864 RO-46-8443 RO-47-0543 RO-47-3359 RO-47-5944 RO-47-7737 RO-47-8634 RO-47-9396 RO-48-2249 RO-48-3656 RO-48-5033 RO-48-5695 RO-48-6791 RO-48-8071 RO-48-8684 RO-5-2181 RO-5-2537 RO-5-2752 RO-5-2904 RO-5-2925 RO-5-3335 RO-5-3367 RO-5-3448 RO-5-3464 RO-5-3590 RO-5-3636 RO-5-3663 RO-5-4528 RO-5-4608 RO-5-4864 RO-5-4933 RO-5-5115 RO-5-5119 RO-5-5120 RO-5-5122 RO-5-5340 RO-5-5807 RO-5-5888 RO-5-6524 RO-5-6528 RO-5-6531 RO-5-6669 RO-5-6900 RO-5-6902 RO-5-6945 RO-5-6993 RO-5-9963 RO-60-0175 RO-64-1056 RO-64-6198 RO-66-0376 RO-66-6976 RO-7-2750 RO-7-2956 RO-7-3351 RO-7-5205 RO-7-5220 RO-7-9277 RO-8-4969 RO-8-7699 RO-8-8717 RO-8-9372 RO-8-9750 ROD-185 ROM-126 ROM-131 RP-20132 RP-29753 RP-30 RP-30A RP-32273

Derwent Drug File 1277 Thesaurus RP-35489 RP-36642 RP-444 RP-46166 RP-49356 RP-52629 RP-52770 RP-54275 RP-54745 RP-55462 RP-56142 RP-58467 RP-58802B RP-58866 RP-59037 RP-59228 RP-59500 RP-60180 RP-60475 RP-60503 RP-61419 RP-61499 RP-61605 RP-61969 RP-62203 RP-62373 RP-63165 RP-63600 RP-64477 RP-64966 RP-66471 RP-67580 RP-68651 RP-69698 RP-69758 RP-70676 RP-73163 RP-73401 RPH-2823 RPH-3048 RPR-100579 RPR-100893 RPR-101821 RPR-103611 RPR-104632 RPR-106541 RPR-107393 RPR-108518-A RPR-109039 RPR-109891 RPR-110173 RPR-111423 RPR-111844 RPR-113829 RPR-114334 RPR-121056 RPR-128515 RPR-130737 RPR-208707 RPR-73401 RR-150 RS-0481 RS-100235 RS-10025 RS-100975 RS-102221 RS-10495 RS-10823 RS-130830 RS-15385 RS-15385-197 RS-1541 RS-1653 RS-16566 RS-17017 RS-17053 RS-1893 RS-2039 RS-2131 RS-2135 RS-22-A RS-22-B RS-22-C RS-2232 RS-23597 RS-23597-190 RS-25259-197 RS-25344 RS-25560-197 RS-30026 RS-30199-193 RS-31819 RS-33295-198 RS-33800 RS-37367 RS-37619 RS-39604 RS-4045 RS-42358-197 RS-42358-198 RS-45041-190 RS-49947 RS-504393 RS-51324 RS-5186 RS-56532 RS-56812-197 RS-57639 RS-5773 RS-66331 RS-67333 RS-67506 RS-67532 RS-722 RS-74513-000 RS-79948-197 RS-83277 RS-83287 RS-8359 RS-86 RS-86505-007 RS-86505-008 RS-86812-007 RS-86812-008 RS-87337 RS-91309 RS-93427 RS-93522 RS-953 RS-980 RSD-1000 RSD-1019 RSD-1070 RSD-1235 RSR-13 RSU-1069 RSU-1131 RSU-1137 RSU-1150 RSU-1164 RSU-1165 RSU-1170 RSU-1172 RTI-112 RTI-113 RTI-121 RTI-3021-020 RTI-31 RTI-32 RTI-353 RTI-51 RTI-55 RU-004 RU-13 RU-16117 RU-23345 RU-24213 RU-24926 RU-24969 RU-25055 RU-25159 RU-25253 RU-25328 RU-25519 RU-25593 RU-26752 RU-26988 RU-28111 RU-28253 RU-28362 RU-29065 RU-29693 RU-29702 RU-29717 RU-3097 RU-31719 RU-32007 RU-32514 RU-32698 RU-32759 RU-33094 RU-33203 RU-33356 RU-33368 RU-33543 RU-33697 RU-33965 RU-34000 RU-34113 RU-34347 RU-35926 RU-35929 RU-35963 RU-38796 RU-38882 RU-39001 RU-39411 RU-39419 RU-399 RU-40410 RU-40555 RU-41656 RU-41821 RU-42173 RU-42382 RU-42633 RU-42698 RU-42698 RU-42848 RU-43028 RU-43526 RU-44790 RU-44981 RU-45144 RU-45179 RU-45703 RU-469 RU-49041 RU-5135 RU-52583 RU-56187 RU-58668 RU-58841 RU-64004 RU-66647 RU-69874 RV-538 RVC-556 RVC-588 RWJ-20142 RWJ-22108 RWJ-26629

1278 APPENDIX D RWJ-270201 RWJ-28810 RWJ-29009 RWJ-306490 RWJ-314313 RWJ-37796 RWJ-37868 RWJ-3981 RWJ-45788 RWJ-46458 RWJ-47428-021 RWJ-49815 RWJ-50271 RWJ-56110 RWJ-58259 RWJ-63556 RX-336M RX-67668 RX-72601 RX-77368 RX-77989 RX-783006 RX-783030 RX-8008M RX-801023 RX-801074 RX-801077 RX-801079 RX-811005 RX-811033 RX-811054 RX-811059 RX-821002 RX-821002-A RX-821029 RX-821037A RX-871024 RX-RA-69 RX-RA-85 RX-RE-92 RY-024 S-0121 S-0139 S-0509 S-0773 S-0838 S-10036 S-1006 S-10089 S-1033 S-1090 S-11568 S-11701 S-118 S-1197 S-11978 S-12024-2 S-12362 S-12813-4 S-12967 S-12968 S-13 S-1321 S-1322 S-135 S-137 S-14063 S-14080 S-14280 S-14297 S-14489 S-145 S-14506 S-1452 S-14671 S-14905 S-15176 S-15261 S-15535 S-15931 S-16020-2 S-16118 S-16257 S-16257-2 S-16260-2 S-16317 S-16324 S-16474 S-16924 S-17092 S-17625 S-18149 S-182 S-18204 S-18326 S-18327 S-18523 S-18886 S-18986 S-1924 S-19752 S-20098 S-20242 S-20244 S-20304 S-20478 S-20500 S-20682 S-20749 S-20928 S-21007 S-21357 S-2150 S-21634 S-218 S-22068 S-2238 S-2251 S-2302 S-23515 S-2366 S-23757 S-23906-1 S-2441 S-24623 S-247 S-2474 S-2581 S-25930 S-25932 S-26191 S-26704 S-2720 S-27609 S-28463 S-2864 S-28828 S-3075 S-312 S-312-(+) S-312-(-) S-32502-1 S-33113 S-3473 S-3483 S-3608 S-3744 S-4048 S-4216 S-422 S-4404 S-464 S-4661 S-55 S-5556 S-584 S-6 S-6907 S-7 S-728011 S-75-0400A S-785026 S-7981 S-808314 S-810592 S-811705 S-830544 S-8307 S-8308 S-8350 S-847445 S-8510 S-8666 S-8849 S-9581 S-9788 S-9795 S-9871 S-9977 S-9977-2 S35B SA-1042 SA-130 SA-167 SA-2572 SA-291 SA-3212 SA-333 SA-3443 SA-36 SA-4503 SA-61 SA-62 SA-63 SA-67 SA-672 SA-679 SA-687 SA-7090 SA-738 SA-981 SAD-128 SAE9 SAH-41-178 SANDOZ-201995 SANDOZ-27403 SANDOZ-45249 SANORG-32701 SARI-59801 SAS-597 SAS-599 SAS-645 SAS-646 SAZ-VII-22 SAZ-VII-23 SB-200646 SB-200646-A SB-201823-A SB-202190 SB-202235 SB-202474 SB-203186 SB-203220 SB-203238 SB-203347 SB-203386 SB-203580 SB-204070 SB-204070-A SB-204269 SB-204741 SB-204990

Derwent Drug File 1279 Thesaurus SB-205384 SB-205891 SB-205952 SB-206343 SB-206553 SB-206718 SB-207266 SB-207266-A SB-207499 SB-207710 SB-209509 SB-209670 SB-210396 SB-210661 SB-213068 SB-214751 SB-214857 SB-216469-S SB-216641 SB-216763 SB-217242 SB-218018 SB-219085 SB-219383 SB-220025 SB-220272 SB-222200 SB-223412 SB-224289 SB-22484-1 SB-22484-2 SB-22484-3 SB-22484-4 SB-225002 SB-227122 SB-228357 SB-234551 SB-238039 SB-239063 SB-242084 SB-242784 SB-247083 SB-249417 SB-258585 SB-258719 SB-265123 SB-271046 SB-273005 SB-277011 SB-29 SB-30 SB-328437 SB-334867 SB-357134 SB-37 SB-415286 SB-435495 SB-59 SB-88 SB-RA-31012 SB-T-1213 SB-T-12843 SC-11927 SC-12222 SC-12742 SC-12757 SC-12790 SC-13173 SC-16100 SC-16102 SC-17146 SC-17599 SC-19220 SC-19886 SC-236 SC-241 SC-24813 SC-25111 SC-25152 SC-2644 SC-26519 SC-26962 SC-27169 SC-28538 SC-2964 SC-299 SC-30249 SC-30552 SC-30695 SC-32855 SC-33428 SC-36067 SC-37111 SC-37698 SC-37872 SC-38249 SC-39026 SC-39566 SC-39902 SC-40476 SC-41661A SC-41930 SC-42619 SC-435 SC-44463 SC-4453 SC-45075 SC-45662 SC-46264 SC-46275 SC-46499 SC-46507 SC-46749 SC-46944 SC-47643 SC-49518 SC-49992 SC-50410 SC-50605 SC-51089 SC-51146 SC-51234A SC-51316 SC-52012 SC-52151 SC-52246 SC-5233 SC-52458 SC-52608 SC-53116 SC-53117 SC-53228 SC-53606 SC-54628 SC-54629 SC-54701 SC-54701-A SC-55389A SC-55494 SC-560 SC-56631 SC-57101 SC-57101-A SC-57461 SC-57666 SC-58125 SC-58236 SC-58272 SC-58560 SC-59735 SC-59840 SC-61213 SC-64939 SC-67655 SC-68420 SC-68693 SC-69050 SC-69054 SC-72-14 SC-8076 SC-8092 SC-8109 SC-9022 SCA-40 SCA-41 SCA-44 SCE-20 SCH-00013 SCH-10015 SCH-12679 SCH-15198 SCH-15199 SCH-16423 SCH-18099 SCH-207758 SCH-211803 SCH-21561 SCH-217048 SCH-221 SCH-226374 SCH-23324 SCH-23388 SCH-23389 SCH-23390 SCH-23391 SCH-24518 SCH-24543 SCH-24893 SCH-24937 SCH-25393 SCH-25873 SCH-28080 SCH-28191 SCH-29482 SCH-32260 SCH-32615 SCH-32651 SCH-33256 SCH-34164 SCH-34343 SCH-34826 SCH-350634 SCH-351125 SCH-351591 SCH-365351 SCH-36606 SCH-37137 SCH-37224 SCH-37370 SCH-37398 SCH-38057 SCH-38518 SCH-38519 SCH-38548 SCH-38840 SCH-38840 SCH-39165 SCH-39166 SCH-39304 SCH-39370 SCH-40120 SCH-40853 SCH-40873 SCH-42354 SCH-42426 SCH-42427 SCH-42495 SCH-44342 SCH-44643 SCH-47802 SCH-47918 SCH-48461

1280 APPENDIX D SCH-49648 SCH-50002 SCH-50673 SCH-50911 SCH-50971 SCH-51048 SCH-51866 SCH-53174 SCH-54445 SCH-54470 SCH-56582 SCH-58053 SCH-58235 SCH-58261 SCH-59228 SCH-59498 SCH-59761 SCH-60663 SCH-60677 SCH-61129 SCH-62373 SCH-66336 SCH-66712 SCH-9122 SCHA-123 SCHA-395 SCHA-764 SCHA-87 SD-14045 SD-146 SD-170 SD-217595 SD-3212 SD-357 SD-62 SD-702 SD-894 SDK-103 SDK-110 SDK-12B-13 SDK-12B-5 SDZ-202-791 SDZ-205-557 SDZ-206-792 SDZ-206-830 SDZ-207-895 SDZ-208-911 SDZ-208-912 SDZ-210-096 SDZ-210-204 SDZ-210921 SDZ-212-122 SDZ-212-327 SDZ-214-103 SDZ-215-811 SDZ-216-525 SDZ-216-744 SDZ-216-744 SDZ-217-704 SDZ-217-744 SDZ-217-766 SDZ-220-004 SDZ-220-040 SDZ-220-581 SDZ-224-015 SDZ-266336 SDZ-266337 SDZ-267-489 SDZ-280-446 SDZ-280-636 SDZ-281-240 SDZ-282-870 SDZ-283-053 SDZ-35-682 SDZ-51-641 SDZ-62-434 SDZ-62-694 SDZ-62-759 SDZ-62-826 SDZ-63-135 SDZ-64-412 SDZ-87-469 SDZ-880-431 SDZ-89485 SDZ-90-215 SDZ-ASM-981 SDZ-CO-611 SDZ-CPI-975 SDZ-EAB-515 SDZ-ENS-163 SDZ-FOX-988 SDZ-ICM-567 SDZ-ICT-322 SDZ-LAP-977 SDZ-MRL-953 SDZ-MTH-958 SDZ-NIM-811 SDZ-NKT-343 SDZ-NVI-085 SDZ-PCO-400 SDZ-PGU-693 SDZ-SBA-586 SDZ-SCV-106 SDZ-SER-082 SDZ-WAG-994 SE-1475 SE-16 SE-422 SEF-19 SEK-1005 SEL-2711 SF-2103A SF-2140 SF-2315-A SF-2315B SF-2324 SF-2361 SF-2370 SF-2446-A1 SF-2446-A2 SF-2446-A3 SF-2446-B1 SF-2446-B2 SF-2446-B3 SF-2487 SF-2575 SF-43 SF-44 SF-482 SF-6847 SF-85-190 SF-86-621 SFTX-3.3 SG-103 SG-209 SG-212 SG-86 SG-89 SGB-1534 SGB-483 SGN-10 SH-254 SH-3-24 SH-306 SH-713 SH-771 SH-869 SH-D-510 SHI-437 SHIVA-1 SHL-434A SHL-643-A SHU-454 SHU-508 SHU-508A SHU-555-A SHU-563-A SHU-9119 SIB-1076 SIB-1508-Y SIB-1553-A SIB-1765-F SIB-1893 SIM-2055 SIM-6080 SIN-1A SIN-1C SIPI-549 SJ-3366 SJ-749 SJC-13 SJG-136 SK-31662 SK-31694 SK-549 SK-946 SK-9709 SKF-100273 SKF-100330A SKF-100336 SKF-100398 SKF-10047 SKF-100501 SKF-100561 SKF-100591A SKF-100844A SKF-100885 SKF-101055 SKF-101071 SKF-101132 SKF-101253 SKF-101368 SKF-101485 SKF-101496 SKF-101497 SKF-101498 SKF-101510 SKF-101542 SKF-101772 SKF-101926 SKF-102010 SKF-102048 SKF-102081 SKF-102102 SKF-102229 SKF-102652 SKF-102698 SKF-102912 SKF-102922 SKF-103108A SKF-103561 SKF-103658 SKF-103829 SKF-104069 SKF-104078 SKF-104093 SKF-104146 SKF-104146-D SKF-104214 SKF-104222 SKF-104223 SKF-104241 SKF-104244 SKF-104351 SKF-104353 SKF-104353-Z2 SKF-104373 SKF-104420 SKF-104421 SKF-104428 SKF-104493 SKF-104524

Derwent Drug File 1281 Thesaurus SKF-104662 SKF-104856 SKF-105285 SKF-105494 SKF-105561 SKF-105571 SKF-105657 SKF-105685 SKF-105768 SKF-105809 SKF-105992 SKF-106203 SKF-106615 SKF-106760 SKF-106978 SKF-107260 SKF-107310 SKF-107457 SKF-107461 SKF-107647 SKF-10812 SKF-108738 SKF-108922 SKF-110679 SKF-12185 SKF-12185-D SKF-16467-A SKF-17467 SKF-19086-A SKF-21681 SKF-21687 SKF-22340 SKF-2314 SKF-24260 SKF-25971 SKF-26070 SKF-28393 SKF-29661 SKF-30097 SKF-3301-A SKF-34288 SKF-35886 SKF-36914 SKF-38393 SKF-38393-A SKF-40117 SKF-40117 SKF-40177 SKF-40491 SKF-40539 SKF-45905 SKF-485-A SKF-490 SKF-5390 SKF-550 SKF-56301 SKF-60817 SKF-625A SKF-64139 SKF-64346 SKF-71432-A2 SKF-71481-A2 SKF-7172A SKF-74652 SKF-75670 SKF-7698 SKF-77174 SKF-7732-A3 SKF-77434 SKF-77581 SKF-78729-A SKF-7997-A3 SKF-80019 SKF-80544 SKF-80723 SKF-81297 SKF-82957 SKF-82958 SKF-83189 SKF-83565 SKF-83566 SKF-83692 SKF-83742 SKF-83959 SKF-84210 SKF-85174 SKF-85257 SKF-85626 SKF-85626 SKF-85738 SKF-86002 SKF-86002-A2 SKF-8742-A SKF-87782 SKF-88046 SKF-88070 SKF-88444 SKF-88827 SKF-88864 SKF-89124 SKF-89145 SKF-89615 SKF-89626 SKF-89641 SKF-89748 SKF-89748-A SKF-89976 SKF-89976A SKF-91486 SKF-91487 SKF-91606 SKF-92373 SKF-92408 SKF-92540 SKF-92629 SKF-93241 SKF-93319 SKF-93479 SKF-94120 SKF-94461 SKF-94674 SKF-95018 SKF-95083 SKF-95299 SKF-95456 SKF-95495 SKF-95565 SKF-95601 SKF-95654 SKF-96067 SKF-962-A SKF-96231 SKF-96365 SKF-96365 SKF-97426A SKF-97541 SKF-97574 SKF-98625 SKF-99085 SKF-99101-H SKF-D-83940 SKF-L-12276 SKF-L-39728-A SKF-L-94901 SKF-R-105058 SKF-R-106114 SKF-R-87516 SKF-S-106203 SKF-S-106470 SKI-2053-R SKK-47029 SL-3111 SL-65-0472 SL-78-0622 SL-79-182 SL-80-0522 SL-81-0013 SL-81-0048 SL-81-0196 SL-81-0433 SL-83-0725 SL-83-0912 SL-840418 SL-85-0324 SL-860714 SL-860715 SL-890591 SM-10661 SM-108 SM-10888 SM-10906 SM-11044 SM-11355 SM-12502 SM-130686 SM-13496 SM-15178 SM-18400 SM-20220 SM-20550 SM-21 SM-220-CL SM-2470 SM-266 SM-3163 SM-31900 SM-345 SM-4300 SM-6586 SM-8668 SM-8849 SM-9018 SM-9064 SM-911 SM-9164 SMA-41 SMA-52 SMAP-28 SMAP-29 SMP-300 SMR-2 SMR-6 SMT-487 SN-10275 SN-12108 SN-13553 SN-14771 SN-16507 SN-16713 SN-16814 SN-18071 SN-20779 SN-22 SN-22-NA SN-22981 SN-23862 SN-24771 SN-25084 SN-25261 SN-25341 SN-25507 SN-292 SN-307 SN-308 SN-38 SN-4094 SN-50 SN-602 SN-6053 SN-606078 SN-6113 SN-6131

1282 APPENDIX D SN-6132 SN-6324 SN-6570 SN-6911 SN-6999 SNA-8073-B SNAP-1069 SNAP-5089 SNAP-5150 SNAP-5399 SNAP-5582 SNAP-6201 SNC-121 SNC-162 SNC-243-A SNC-80 SND-919 SNF-8702 SNF-9007 SNK-860 SNX-111 SNX-239 SO-121 SO-324 SO-730 SO-75R1 SOM-1122 SOM-1397-CL SP-100030 SP-111A SP-303 SP-4 SP-4012 SP-500263 SP-562 SP-563 SP-564 SP-600125 SP-725 SP-904 SP-W-5186 SPA-S-565 SPA-S-717 SPA-S-753 SPA-S-843 SPC-100270 SPC-100271 SPC-103600 SPC-3 SPC-5002 SPI-447 SPI-501 SPM-3672 SPM-4744 SPM-5185 SPP-100 SPR-210 SPR-901 SQ-10591 SQ-10996 SQ-11276 SQ-13297 SQ-13863 SQ-14102 SQ-14359 SQ-14534 SQ-14551 SQ-15361 SQ-18506 SQ-19265 SQ-19297 SQ-19300 SQ-19301 SQ-20006 SQ-20204 SQ-20294 SQ-20475 SQ-20661 SQ-20718 SQ-20858 SQ-20859 SQ-20861 SQ-22536 SQ-26180 SQ-26324 SQ-26536 SQ-26559 SQ-26630 SQ-26655 SQ-26668 SQ-26771 SQ-26917 SQ-26992 SQ-27050 SQ-27327 SQ-27427 SQ-27629 SQ-27786 SQ-27860 SQ-28300 SQ-28370 SQ-28504 SQ-28546 SQ-28603 SQ-28668 SQ-28852 SQ-29072 SQ-29535 SQ-29548 SQ-30741 SQ-31360 SQ-31765 SQ-31853 SQ-31854 SQ-31855 SQ-31906 SQ-31945 SQ-32014 SQ-32097 SQ-32547 SQ-32829 SQ-33261 SQ-33351 SQ-33552 SQ-33600 SQ-33800 SQ-33961 SQ-34676 SQ-46542 SQ-65442 SQ-67590 SQ-80338 SQ-81377 SQ-81387 SQ-81402 SQ-81427 SR-11203 SR-11217 SR-11220 SR-11234 SR-11235 SR-11236 SR-11237 SR-11238 SR-11246 SR-11254 SR-11262 SR-11276 SR-11278 SR-11302 SR-11345 SR-11364 SR-120107-A SR-120819-A SR-121463 SR-121463-B SR-121566 SR-121566-A SR-121787 SR-12813 SR-140333 SR-140603 SR-141716-A SR-142801 SR-142806 SR-142948-A SR-144385 SR-144528 SR-146131 SR-16234 SR-24870 SR-2555 SR-25776 SR-25990C SR-26334 SR-2640 SR-27417 SR-27897 SR-27897-B SR-31742A SR-31747 SR-31747-A SR-33510 SR-33671 SR-33805 SR-3722 SR-3745 SR-3745A SR-3772 SR-3773 SR-3775 SR-41378 SR-42128 SR-42128A SR-42641 SR-4317 SR-4330 SR-43845 SR-4452 SR-4482 SR-44866 SR-4554 SR-45813 SR-46349B SR-46559-A SR-47063 SR-4718 SR-48527 SR-48692 SR-4895 SR-48965 SR-48968 SR-49059 SR-49711 SR-57227A SR-57746A SR-58002-C SR-58306A SR-58372 SR-58373-A SR-58373A SR-58375A SR-58539B SR-58572A SR-58575A SR-58589 SR-58590 SR-58611A SR-58612A SR-58613A SR-58825A SR-59104-A

Derwent Drug File 1283 Thesaurus SR-59119-A SR-59230-A SR-80258-A SR-90107 SR-9223-I SR-9223I SR-95195 SR-95639A SRI-2712-24 SRI-4657-47 SRI-5193-34 SRI-5193-43 SRI-5387-31 SRI-5447-28 SRI-5631-96 SRI-5898-21 SRI-5898-71 SRI-6153-40 SRI-62-834 SRI-63-072 SRI-63-119 SRI-63-441 SRI-63-675 SRI-6409-94 SRI-6751-84 SRI-7167-67 SRI-7323-78 SS-202 SS-20846-A SS-228-R SS-228-Y SS-320A SS-56C SS-62-4 SS-62-6 SS-717 SS-750 SSF-109 SSP-11 SSR-149415 SSR-180575 ST-1059 ST-1326 ST-1435 ST-1460 ST-1481 ST-1646 ST-1913 ST-1943 ST-232 ST-271 ST-280 ST-341 ST-363 ST-4250 ST-450 ST-458 ST-464 ST-465 ST-475 ST-476 ST-494 ST-585 ST-587 ST-606 ST-608 ST-630 ST-638 ST-642 ST-666 ST-732 ST-789 ST-80 ST-88 ST-89 ST-91 ST-93 ST-95 STH-2100 STH-2148 STH-2169 STH-2224 STS-153 STS-456 STS-593 STS-64 STS-737 STY-2108 SU-10603 SU-11739 SU-13320 SU-15049 SU-4984 SU-5402 SU-5416 SU-6668 SU-740 SU-8000 SU-840 SU-9055 SU-9516 SUAM-1221 SUMS-1 SUMS-2 SUMS-2P SUMS-3 SUN-0588 SUN-4599 SUN-5555 SUN-8399 SUN-9216 SUN-9221 SUN-C-5174 SUN-N-4057 SUN-N-8075 SUT-8701 SV-4814 SX-284 SX-3228 SY-14 SY-28 SY-6001 SY-640 SY-801 SY-9215 SYM-2081 SYN-2190 SYN-2836 SYN-2869 SYN-2903 SYN-2921 SZ-1676 SZ-48 SZ-51 SZJ-3361 SZJ-3388 SZL-49 T-0115 T-0128 T-0201 T-0509 T-0632 T-0757 T-1032 T-1095 T-121-B T-1218 T-1221 T-1224 T-13 T-138067 T-157602 T-1583 T-162559 T-174 T-1982A T-1982B T-23 T-250 T-2525A T-2588A T-2588F T-283 T-30177 T-30677 T-30695 T-3262A T-3262B T-330 T-3660 T-3811-ME T-44 T-440 T-451 T-477 T-5575 T-588 T-593 T-614 T-686 T-70182 T-72258 T-900607 T-98 T150R1 T22 TA-073 TA-077 TA-078 TA-0910 TA-174 TA-1801 TA-2005 TA-3037A TA-404 TA-5707 TA-5707F TA-60 TA-606 TA-7552 TA-993 TAAC-3 TAD-235 TAI-908 TAK-029 TAK-044 TAK-147 TAK-218 TAK-225 TAK-375 TAK-456 TAK-536 TAK-603 TAK-636 TAK-637 TAK-778 TAK-779 TAN-1030-A TAN-1057-A TAN-1057-B TAN-1057-C TAN-1057-D TAN-1251-A TAN-1518-A TAN-67 TAN-931 TAN-950-A TAS-103 TAS-301 TAT-59 TBC-11192 TBC-11241

1284 APPENDIX D TBC-11251 TBC-1269 TBI-361 TC-13 TCV-116 TCV-295 TCV-309 TDN-345 TE-176 TEI-0303 TEI-1324 TEI-1338 TEI-2306 TEI-3096 TEI-3356 TEI-4120 TEI-5178 TEI-5624 TEI-6344 TEI-6472 TEI-6720 TEI-7322 TEI-8364 TEI-9063 TEI-9647 TEI-9826 TEI-9874 TEL-1338 TER-199 TER-286 TER-930180 TFC-612 TGP-580 TGS-20 TGS-33 TGS-34 TH-1011 TH-1090 TH-1091 TH-1206 TH-1231 TH-1257 TH-1274 TH-142177 TH-1506 TH-91-21 TH-92-20 TH-92-4 THB-013 TI-23 TI-233 TJ-114 TJ-13025 TJ-135 TJ-14 TJ-15 TJ-23 TJ-24 TJ-41 TJ-43 TJ-8007 TJ-8014 TJ-96 TJ-960 TJC-160 TJN-220 TJN-505 TJS-010 TK-11 TK-174 TK-5477 TK-620-9 TKS-159 TL-102 TL-137 TL-140-III TL-224 TL-232 TL-259 TL-302 TL-304 TL-308 TL-312 TL-333 TL-334 TL-350 TL-351 TL-363 TL-365 TL-371 TL-381 TL-402 TL-68 TL-99 TLK-16998 TMB-5 TMB-6 TMB-8 TMC-016 TMC-125 TMC-151-A TMC-151-B TMC-151-C TMC-151-D TMC-151-F TMC-2-A TMC-2-B TMC-2-C TMC-69 TMK-688 TMK-777 TMP-153 TN-108 TN-109 TN-112 TN-121 TN-16 TN-77 TN-78 TN-79 TN-80 TN-871 TNO-1 TNO-38 TNP-351 TOC-39 TOC-50 TOK-4528 TOK-8801 TOP-53 TP-151 TP-40 TP-680 TP-69 TP-72 TP-9201 TPN-12 TPO-33 TR-1722 TR-35 TRI-11 TRI-25 TRI-50-B TRI-59 TRK-219 TRK-710 TRK-820 TRK-851 TRM-115 TRY-200 TS-943 TST-220 TST-334 TT-232 TTA-386 TU-1718B TU-199 TUK-9261 TUK-9262 TV-3326 TV-399 TVP-1022 TW-13 TW-19 TW-22 TW-25 TW-26 TW-32 TW-39 TW-50 TX-045 TX-11027 TX-1123 TX-1856 TX-380 TX-44 TX-51 TX-522 TX-527 TX-53 TY-11345 TY-12533 TYB-2285 TZ-146 TZ-50-2 TZ-650 TZ-93 TZC-1370 TZC-5665 TZI-41127 TZI-615 TZP-4238 TZT-1027 U-0126 U-0521 U-0949 U-10029A U-1003 U-100313 U-101017 U-101033-E U-101387 U-10157 U-101958 U-102466 U-10293 U-103017 U-103264 U-103265 U-104067-F U-104489 U-106305 U-106311-E U-108333-E U-109818 U-11634 U-11790 U-11866 U-11921 U-11973 U-13851 U-1424 U-14624 U-15646 U-16178F U-18 U-18177-A U-18598 U-18666A U-19425 U-20057 U-2021

Derwent Drug File 1285 Thesaurus U-20685 U-2113 U-22105 U-22312 U-22394A U-22989 U-23223 U-23469 U-23807A U-24 U-24278 U-24279 U-24522 U-24568 U-24631 U-247-125 U-247-90 U-247-95 U-247-96 U-25030 U-25166 U-25927 U-26384 U-26727A U-27391 U-30684A U-30870 U-3243 U-34445 U-35122 U-35401 U-37883A U-38658-A U-38833 U-40481 U-42129 U-42352 U-43465F U-43728 U-43795 U-44069 U-46195 U-46619 U-47473 U-48753E U-50488 U-50488E U-50488H U-51605 U-51862 U-53455E U-54494A U-54874 U-56407 U-56467 U-57908 U-62066E U-62168-E U-62168E U-62736 U-62840 U-63360 U-63639 U-63640 U-66226 U-66444B U-66664 U-66694 U-66858 U-66866 U-66982 U-66985 U-67154 U-67786 U-68043 U-68215 U-68415 U-68552B U-68819 U-69593 U-70585 U-71184 U-71185 U-71909E U-72407-E U-72407E U-72408-E U-72408E U-72409-E U-72409E U-72799 U-73122 U-73343 U-73777-E U-74389 U-74389F U-74389G U-74500-A U-75013 U-75014-E U-75302 U-75305 U-75360 U-75412E U-75485 U-75559 U-75875 U-76073 U-76074 U-76088 U-76190 U-76579 U-76915 U-77436 U-77451-E U-77451E U-77455-E U-77646-E U-77646E U-77647E U-77692 U-78057 U-78489 U-78517F U-78518-E U-78518F U-78608 U-79098 U-79206 U-80215-E U-80215E U-80493E U-80631-E U-80816 U-81581 U-81749 U-82208E U-82209E U-82217 U-82579 U-83836 U-83836E U-83892 U-83894 U-84042 U-84645E U-84849 U-85548E U-85549E U-85575 U-86170 U-86170-F U-86983 U-87407 U-87663-E U-87999 U-88204 U-88204E U-88509 U-88566 U-88703 U-88943E U-89232 U-89255 U-89360 U-89678 U-89843 U-89843-A U-89843-D U-89843-E U-90042 U-90167 U-90168 U-91356 U-91356-A U-91502 U-91976 U-92016-A U-92032 U-92593 U-92813 U-93385 U-93631 U-93840 U-93965 U-94430-E U-95133 U-96183 U-96364 U-96988 U-97018 U-97775 U-9888 U-99194-A U-99363-E U-99499 U-99963 UBP-1110 UBP-1111 UBP-1112 UC-040 UC-10 UC-284 UC-42 UC-781 UC-82 UCB-11056 UCB-22073 UCB-28557 UCB-JO28 UCB-L061 UCE-1022 UCE-6 UCF-1-C UCH-9 UCL-1092 UCL-1199 UCL-1285 UCL-1344 UCL-1390 UCL-1495 UCL-1530 UCL-1684 UCN-01 UCN-02 UCT-4B UD-CG-212 UDJO-1311 UH-148 UH-232 UH-242 UH-301

1286 APPENDIX D UH-AH-37 UIC-94003 UK-1 (Cytostatic) UK-101613 UK-102333 UK-103320 UK-11957 UK-141161 UK-14275 UK-147535 UK-14819 UK-15121 UK-1745 UK-177 UK-2-A UK-21 UK-224671 UK-22486 UK-25 UK-279276 UK-3-A UK-343664 UK-34787 UK-36327 UK-3883 UK-47265 UK-49883 UK-5099 UK-52831 UK-55076 UK-57400 UK-61260 UK-63052 UK-65662 UK-66914 UK-69578 UK-69753 UK-74505 UK-84149 UL-AH-99 UL-DF-9 ULFS-49 UM-1037 UM-1046 UM-1250 UM-424 UM-747 UMF-078 UMF-289 UMJD-828 UNO-3 UP-116-77 UP-20232 UP-20256 UP-269-6 UP-614-04 UPF-523 UPF-583 UPF-596 UR-10324 UR-11353 UR-12460 UR-12592 UR-12670 UR-12947 UR-7280 UR-8225 UR-8880 UR-9825 USVC-6524 UT-15 V-10367 V-111 V-33 VA-045 VA-21-B7 VB-11328 VC-1052 VC-15-B VF-122 VF-147 VF-1634 VF-165 VF-233 VG-18563 VICO-81 VJ-45 VJ-52 VJ-53 VJ-58 VJ-60 VK-744 VK-774 VM-44857 VM-44864 VM-44865 VM-44866 VN-85-1 VN-87-1 VNP-20009 VP-343 VP-616-L VP-710-Z VP-712-Z VUF-4567 VUF-4568 VUF-4585 VUF-4591 VUF-4613 VUF-5297 VUF-8294 VUF-8296 VUF-8297 VUF-8298 VUF-8299 VUF-8303 VUF-8401 VUF-8403 VUF-8404 VUF-8405 VUF-8406 VUF-8407 VUF-8411 VUF-8413 VUF-8501 VUF-8504 VUF-8505 VUF-8507 VUF-8514 VUF-8532 VUF-8842 VUF-9019 VUF-9020 VUF-9045 VUF-K-8788 VUFB-10726 VUFB-14170 VUFB-15269 VUFB-15468 VULM-411 VX-497 VX-710 VZ-20 VZ-65 W-12 W-13 W-2531 W-328 W-36017 W-36149 W-36196 W-3795 W-398 W-4010 W-49091 W-49167 W-5 W-66 W-6603 W-68 W-7 W-77 W-8011 W-82139 W-84 WA-8242-A1 WA-8242-A2 WA-8242-B WAL-2014 WAY-100135 WAY-100289 WAY-100579 WAY-100635 WAY-120491 WAY-120739 WAY-121006 WAY-121509 WAY-121520 WAY-123398 WAY-124466 WAY-126227 WAY-133537 WAY-135706 WAY-140424 WAY-151616 WAY-PDA-641 WAY-VPA-985 WB-3559-A WB-3559-B WB-3559-C WB-3559-D WB-4085 WB-4093 WB-4101 WB-4109 WB-4291 WB-4371 WB-608 WE-1008 WE-1061 WE-1064 WE-1073 WE-956 WE-964 WEB-1881-FU WEB-2118 WEB-2347 WF-10129 WF-11605 WF-23 WF-31 WF-3161 WF-3681 WHI-07 WHI-P-111 WHI-P-131 WHI-P-154 WHI-P-180 WHI-P-353 WHI-P-97 WHK-BF-1 WHR-1049 WHR-1049A WHR-1370A WHR-2568 WILD-20 WIN-136455 WIN-17317-3 WIN-18446 WIN-2299 WIN-28929 WIN-3286

Derwent Drug File 1287 Thesaurus WIN-32950 WIN-33123 WIN-33156 WIN-33377 WIN-35004 WIN-35065-2 WIN-35065-3 WIN-35140 WIN-35428 WIN-35439 WIN-35981 WIN-39996 WIN-41258-3 WIN-42610 WIN-44441-2 WIN-4981 WIN-513 WIN-51708 WIN-52035 WIN-52084 WIN-52664 WIN-53024 WIN-53338 WIN-53782 WIN-54954 WIN-55212 WIN-55212-2 WIN-55212-3 WIN-56098 WIN-57007 WIN-57273 WIN-57294 WIN-58161 WIN-63320 WIN-63394 WIN-63395 WIN-63480 WIN-63759 WIN-63843 WIN-64338 WIN-64338 WIN-64593 WIN-64733 WIN-64821 WIN-66306 WIN-67694 WIN-8626 WK-1492 WL-19 WL-22864 WMAP-10 WMC-26 WP-401 WP-546 WP-549 WP-608 WP-631 WP-652 WR-106147 WR-1065 WR-122455 WR-129577 WR-149024 WR-15081 WR-151326 WR-151327 WR-158122 WR-159412 WR-165355 WR-172435 WR-1729 WR-175412 WR-177602 WR-178460 WR-181023 WR-182232 WR-182234 WR-182393 WR-183489 WR-184806 WR-188438 WR-190420 WR-194965 WR-199385 WR-199504 WR-199507 WR-199508 WR-212579 WR-214198 WR-216804 WR-224097 WR-225448 WR-226253 WR-242511 WR-243251 WR-250016 WR-250547 WR-250548 WR-251993 WR-2823 WR-30090 WR-3090 WR-33063 WR-33278 WR-3689 WR-40070 WR-49577 WR-5677 WR-5990 WR-6026 WR-638 WR-6865 WR-6881 WR-6890 WR-77913 WR-93133 WR-9792 WR-99662 WRC-0090 WRC-0342 WRC-0571 WRC-470 WS-009A WS-009B WS-1279 WS-1358A1 WS-1358B1 WS-1442 WS-1490 WS-5995A WS-5995B WS-5995C WS-7338-A WS-7338-C WS-7338-D WS-7528 WS-75624-A WS-75624-B WS-79089-B WS-9326A WS-9659A WS-9659B WS-9761-A WS-9761-B WSP-1 WSP-2 WSP-3 WU-345 WU-385 WV-15 WX-360 WX-UK-1 WY-12556 WY-13876 WY-17186 WY-18185 WY-18189 WY-19068 WY-19110 WY-25093 WY-25110 WY-25309 WY-26157 WY-26392 WY-26703 WY-26769 WY-27127 WY-27587 WY-3457 WY-40659 WY-41195 WY-41747 WY-41770 WY-42186 WY-42896 WY-4355 WY-44221 WY-44329 WY-45086 WY-45233 WY-45494 WY-45662 WY-45727 WY-45760 WY-45881 WY-45911 WY-46689 WY-46965 WY-47288 WY-47766 WY-47877 WY-47894 WY-47961 WY-48090 WY-48723 WY-48986 WY-48989 WY-49051 WY-49232 WY-50295 WY-50295-C WY-50295-T WY-5090 WY-5256 WY-7953 X-14667A X-14868A X-14868B X-14868C X-14868D X-14873A X-14881-D X-14881-E X-14885A X-14889A X-14889C X-14889D X-206 X-50 XAMR-0716 XAMR-0721 XB-277 XB-513 XB-596 XC-164 XC-386 XD-793 XE-991 XJ-735 XJ-754 XJ-757 XK-216

1288 APPENDIX D XK-234 XK-469 XN-482 XR-11576 XR-1853 XR-334 XR-457 XR-5082 XR-510 XR-5118 XR-543 XR-5944 XR-5967 XR-7009 XR-835 XR-9051 XR-9576 XS-361 XT-044 XT-199 XT-403 XT-611 XU-063 XU-745 XV-454 XV-459 XV-638 Y-12141 Y-18598 Y-19018 Y-19432 Y-19638 Y-20024 Y-20487 Y-20811 Y-23023 Y-23684 Y-24180 Y-25130 Y-25510 Y-26611 Y-26763 Y-27152 Y-27632 Y-29794 Y-3310 Y-39041 Y-39241 Y-5554 Y-590 Y-688 Y-8845 Y-9223 Y-9738 YC-1 YC-170 YG-19256 YH-438 YH-439 YJA-20379-1 YJA-20379-8 YL-01869-P YLL-224 YM-022 YM-08054-1 YM-0850 YM-087 YM-099 YM-103 YM-108 YM-11133 YM-114 YM-12617 YM-13115 YM-13650 YM-14471 YM-14673 YM-151 YM-16151-1 YM-16638 YM-175 YM-17690 YM-17E YM-21095 YM-220 YM-264 YM-26567-1 YM-26734 YM-30059 YM-31553 YM-31636 YM-337 YM-358 YM-35992 YM-39558 YM-430 YM-435 YM-43611 YM-461 YM-47141 YM-47522 YM-511 YM-534 YM-53601 YM-53707 YM-57029 YM-57158 YM-60828 YM-62899 YM-75466 YM-75518 YM-796 YM-866 YM-872 YM-900 YM-905 YM-934 YM-95831 YNKO-1 YP-279 YPE-01 YS-035 YS-822A YS-980 YT-1 YT-146 YT-146 YT-615 Z-100 Z-1046 Z-10997-A Z-12000 Z-12001 Z-12007 Z-13752-A Z-300 Z-335 Z-338 Z-360 ZAMI-1305 ZAMI-1327 ZCR-2060 ZD-0947 ZD-1611 ZD-1839 ZD-2079 ZD-2767 ZD-2767-D ZD-2767-P ZD-4190 ZD-5522 ZD-6021 ZD-6126 ZD-6169 ZD-7155 ZD-9331 ZD-9379 ZD-9989 ZE-117 ZG-1494-ALPHA ZG-63 ZH-103 ZIMET-111-74 ZIMET-18-84 ZIMET-19-84 ZIMET-20-84 ZIMET-22-84 ZIMET-25-85 ZIMET-53-84 ZIMET-58-85 ZIMET-61-85 ZIMET-72-85 ZIMET-98-69 ZK-110841 ZK-111298 ZK-112151 ZK-112566 ZK-112993 ZK-114043 ZK-115716 ZK-115886 ZK-118182 ZK-119010 ZK-119095 ZK-132553 ZK-135695 ZK-136799 ZK-138723 ZK-139129 ZK-156718 ZK-158252 ZK-159222 ZK-191703 ZK-28943 ZK-30595 ZK-33839 ZK-36375 ZK-48491 ZK-71677 ZK-805412 ZK-805623 ZK-90798 ZK-90886 ZK-91296 ZK-91587 ZK-93423 ZK-93426 ZK-95962 ZK-97894 ZL-III-43-A ZM-172405 ZM-218463 ZM-226600 ZM-241385 ZM-244085 ZM-249148 ZM-250462 ZM-252868 ZM-258754 ZM-260384 ZM-97480 ZNS-114-666 ZP-120-C ZSY-27 ZTTA-1 ZY-15039 ZY-15850A ZY-17617B TRIPLE-HELIX ANTIGENE-THERAPY

Derwent Drug File 1289 Thesaurus TUBERCULIN PPD TUBERCULOSIS LEITNER-SYNDROME LUPUS-VULGARIS PONCET-DISEASE TUBERCULOSTATICS 27753-RP 27753-RP ACETYLISONIAZID ACONIAZIDE ALLOCUPREIDE SODIUM AMICLENOMYCIN AMINOSALICYLATE SODIUM AMQ-2 AMQ-4 AMQ-5 AW-464 AXISONITRILE-3 AZAROLE AZICEMICIN-A AZICEMICIN-B B-1772 B-1865 B-1912 B-283 B-3722 B-3785 B-4100 B-4101 B-4154 B-4157 B-432 B-433 B-621 B-628 B-654 B-670 B-685 B-746 B-749 B-776 B-797 B-826 B-980 BENFLURON BENZAMIDOSALICYLATE = CALCIUM BOSTRYCOIDIN CAPREOMYCIN CAPREOMYCIN-IA CAPREOMYCIN-IB CAPREOMYCIN-IIA CAPREOMYCIN-IIB CGP-29861 CGP-7040 CITENAZONE CLOFAZIMINE CROTONIAZIDE CYACETACIDE CYCLOSERINE DV-7751 ECTEINASCIDIN-770 ENVIOMYCIN EPI-OLEANOLATE ETHAMBUTOL ETHIONAMIDE ETOCARLIDE FCE-22250 FCE-22807 FENAMISAL FTIVAZIDE GALAPHENYLSULFONE GANGAMICIN GATIFLOXACIN GEMIFLOXACIN GLYCONIAZIDE GRANULYSIN IPRONIAZID ISONIAZID ISONIAZID-MESILATE KAPOSTAT KRM-1648 KRM-1671 LABILOMYCIN LARUSAN MACROCYCLON ME-93 METAZIDE METHANIAZIDE METHYL-SULFOMETURON METHYLGLABRIDIN-4+-O MORINAMIDE NEMOTIN NICOTHIAZONE OLEANONATE OPINIAZIDE PARADOL-6 PAS PAS SODIUM PASINIAZID PD-119421 PD-122642 PD-123982 PD-125354 PD-126889 PD-131575 PD-139586 PD-143289 PD-161314 PELLITORINE PREUSSOMERIN-E PREUSSOMERIN-F PREUSSOMERIN-G PREUSSOMERIN-H PREUSSOMERIN-I PROTIONAMIDE PYRAZINAMIDE RESORCINOMYCIN-A RIFAMPICIN SALINAZID SHINJUDILACTONE SITAFLOXACIN STREPTOMYCIN STREPTONIAZID SUBATHIZONE SULFONIAZIDE T-283 T-3811-ME TELITHROMYCIN TERIZIDONE TETRANDRINE THIOACETAZONE THIOCARBANIDIN THUJAPLICIN-BETA TIOCARLIDE TN-121 TUBERIN VERAZIDE VIOMYCIN VUF-8501 VUF-8514 VUF-8842 TUMOR-CELL 1321N1-CELL 3LL-CELL 9L-CELL A15-CELL A1847-CELL A204-CELL A253-CELL A2780-CELL A427-CELL A549-CELL ABPL2-CELL AH130-CELL AH66-CELL AKR-CELL B16-CELL B16A-CELL B35M-CELL B4-CELL B4976-CELL BCL1-CELL BE-CELL BEN-CELL BT20-CELL BT474-CELL BW5147-CELL C1300-CELL C6-GLIAL-CELL CACO2-CELL CAOV-CELL CASKI-CELL CBT-CELL CC531-CELL CCRF-CEM-CELL CHP126-CELL CLOUDMAN-CELL CLOUDMAN-S91-CELL CO115-CELL CT26-CELL DAUDI-CELL DETROIT-562-CELL DLD1-CELL DT5-CELL DU145-CELL DUNNING-R3327H-CELL EB-CELL EB2-CELL EHRLICH-ASCITES-CELL EL4-CELL ELCO2-CELL EMT6-CELL ESB-CELL FRIEND-LEUKEMIA-CELL FSD1-F4-CELL G-CELL GROSS-LEUKEMIA-CELL H157-CELL H35-CELL H4-CELL HAB-CELL HARDING-PASSEY-CELL HBT3-CELL HCCL-CELL HCT-CELL HCT116-CELL HCT8-CELL HELA-CELL HEP-G2-CELL HEP2-CELL HEPA1-CELL HEY-CELL HL60-CELL HOC1-CELL HOC7-CELL HRIK-CELL HSO578-CELL HT1080-CELL HT29-CELL HTC-CELL HUT102B2-CELL HUT11-CELL HUTU80-CELL HX13-CELL HX18-CELL HX29-CELL J111-CELL

1290 APPENDIX D JEG3-CELL JURKAT-CELL K562-CELL KB-CELL KG1-CELL KPI-CELL KU1-CELL L1210-CELL L12R4-CELL L2C-CELL L40-CELL L5222-CELL LAZ007-CELL LEWIS-LUNG-CARCINOMA-= CELL LOVO-CELL M1-CELL M109-CELL M21-CELL M5-CELL MA160-CELL MBL2-CELL MBT2-CELL MC7-CELL MCB6-1-CELL MCF7-CELL ME180-CELL METH-A-CELL MG34-CELL MG63-CELL MGH41-CELL MGHV1-CELL MH134-CELL MKN1-CELL MKN28-CELL MKN45-CELL ML1-CELL MM253-CELL MOLT3-CELL MOLT4-CELL MOPC-CELL MOPC173-CELL MORRIS-HEPATOMA-CELL MOT-CELL MPC11-CELL NEMETH-KELLNER-CELL NG108-15-CELL NH1K-3025-CELL NIE115-CELL NOVIKOFF-HEPATOMA-CELL NS1-CELL NS20-CELL OVCAR2-CELL OVCAR3-CELL OVCAR4-CELL OVCAR5-CELL P388-CELL P815-CELL P815Y-CELL PC1-CELL PC10-CELL PC12-CELL PC9-CELL POC-CELL QG56-CELL QG90-CELL R3230AC-CELL RAG-CELL RAJI-CELL RAW264-CELL RD-CELL RIF1-CELL RPMI0041-CELL RPMI1346-CELL RPMI1846-CELL RPMI2650-CELL RPMI6410-CELL RPMI8402-CELL RR1022-CELL RT112-CELL S49-CELL S91-CELL SA1-CELL SA2-CELL SA5-CELL SA9-CELL SARCOMA-180-CELL SARCOMA-37-CELL SARCOMA-45-CELL SF126-CELL SF375-CELL SF407-CELL SH3-CELL SK-HEP1-CELL SK-MEL28-CELL SK-MEL37E-CELL SK-OV-CELL SKL2-CELL SKL5-CELL SW1271-CELL SW403-CELL SW48-CELL SW480-CELL SW620-CELL SW900-CELL T24-CELL T47D-CELL TA3-CELL TANG-CELL TE85-CELL TEPC15-CELL TERA-C-CELL TLX5-CELL U937-CELL VX2-CELL WALKER-256-CELL WIDR-CELL XC-CELL Y79-CELL YOSHIDA-SARCOMA-CELL TYROSINE-KINASE-INHIBITORS ADAPHOSTIN AG-1295 AG-1296 AG-1517 AG-17 AG-1879 AG-825 AG-879 AG-957 AGL-1872 CEP-5214 CEP-701 CEP-751 CGP-41251 CGP-53716 CGP-59326 CL-387785 COUMAROYLTYRAMINE-N CP-358774 CP-547632 CT-052923 D-58 DAMNACANTHAL DC-101 DEMETHOXYVIRIDIN EKB-569 EMODIN EPIGALLOCATECHIN-GALLATE GELDANAMYCIN GENISTEIN GW-2016 GW-974 HERBIMYCIN-A IMATINIB K-252B LFM-A-13 LY-294002 NSC-330507 OSI-774 PD-0183085 PD-089828 PD-153035 PD-153717 PD-158780 PD-161176 PD-168393 PD-169540 PD-173074 PD-180970 PD-183805 PKI-166 QUERCETIN RG-13022 RK-682 RPR-108518-A SEMAXANIB SMA-41 ST-638 SU-4984 SU-5402 SU-6668 TX-1123 TYRPHOSTIN-A-47 U-73343 VATALANIB WHI-P-131 WHI-P-97 WORTMANNIN ZD-4190 ZM-252868 ULCER BARRETT-SYNDROME ULTRASONICS SONICATION ULTRASONOGRAPHY URICOSURICS AA-193 BAY-N-1468 BENZBROMARONE BENZIODARONE CIAPILOME CINCHOPHEN COLCHICEINE DITOLAMIDE DR-3438 IRTEMAZOLE ITANOXONE NICOXAMAT OSMADIZONE PROBENECID PYRAZINOATE S-8666 SECLAZONE SODIUM-POTASSIUM-= CITRATE SULFINPYRAZONE TEI-6720 TRAXANOX TRICLACETAMOL URATE-OXIDASE URINARY-TRACT-DISEASE DYSURIA URETERAL-COLIC URETHRAL-SYNDROME URETHRITIS UROLITHIASIS UTEROTONICS

Derwent Drug File 1291 Thesaurus ACETERGAMINE ARDISIACRISPIN-A ARDISIACRISPIN-B CLOQUINOZINE DIHYDROERGOCORNINE DIHYDROERGOCRISTINE DIHYDROERGOCRYPTINE DIHYDROERGOCRYPTINE-= ALPHA DIHYDROERGOCRYPTINE-= BETA DIHYDROERGOSINE DIHYDROERGOTOXINE EPI-OLEANOLATE ERGOMETRINE ERGOSININE ERGOTAMINE ERGOTOXINE HYDROXYMETHYLFURFURAL ISOVERIN METERGOLINE METHYLERGOMETRINE OLEANONATE QUIPAZINE SPARTEINE UTERUS CERVIX DECIDUA ENDOCERVIX ENDOMETRIUM FALLOPIAN-TUBE MYOMETRIUM PARAMETRIUM PERIMETRIUM UTERUS-DISEASE ADENOMYOSIS carcinoma, cervix cervix-carcinoma CHIARI-FROMMEL-= SYNDROME ENDOMETRITIS ENDOMYOMETRITIS HYDROMETRA HYDROSALPINX METRITIS PARAMETRITIS PROLAPSE PYOMETRA TROPHOBLASTIC-DISEASE TUBAL-SPASM VACCINE TOXOID VACCINES AIDS-VACCINE ALLERGOVIT ALLPYRAL ALUTARD AMEBIASIS-VACCINE ANAPLAZ ANJUVAC ANTHRAX-VACCINE ARTERITIS-VACCINE ATROPHIC-RHINITIS-VACCINE BCG BLACK-DISEASE-VACCINE BLACK-QUARTER-VACCINE BLUE-TONGUE-VACCINE BORDER-DISEASE-VACCINE BOTULISM-VACCINE BOVISALORAL BRAXY-VACCINE BRONCASMA BRUCELLOSIS-VACCINE BUCCALIN CAMPYLOBACTERIOSIS-= VACCINE CANDIDIASIS-VACCINE CARCINOMA-VACCINE CARIES-VACCINE CASEOUS-LYMPHADENITIS-= VACCINE CHLAMYDIA-VACCINE CHOLERA-VACCINE COCCIVAC COLOMBOVAC CONJUVAC CONTAGIOUS-AGALACTIA-= VACCINE CORYZA-VACCINE COVEXIN-8 D-53 DENGUE-VACCINE DERMATOPHILOSIS-VACCINE DERZSY-DISEASE-VACCINE DIAVAX-VACCINE DICTOL DIPHTHERIA-VACCINE DISTEMPER-VACCINE DYSENTERY-VACCINE EAST-COAST-FEVER-VACCINE EMC-VACCINE ENCEPHALITIS-VACCINE ENCEPHALOMYELITIS-= VACCINE ENTEROTOXEMIA-VACCINE ENTEROTOXIN-HEAT-= STABLE-E.COLI ENZOOTIC-ABORTION-= VACCINE ERYSIPELAS-VACCINE FURUNCULOSIS-VACCINE GASTRIMMUNE GLAESSER-DISEASE-VACCINE GONORRHEA-VACCINE HEART-WATER-VACCINE HEM.ENTERITIS-VACCINE HEM.SEPSIS-VACCINE HEPATITIS-A-VACCINE HEPATITIS-A-VACCINE HEPATITIS-B-VACCINE HEPATITIS-E-VACCINE HEPATITIS-VACCINE HERPES-SIMPLEX-VACCINE IBR-IPV-VACCINE IBR-VACCINE INFECTIOUS-ANEMIA-= VACCINE INFECTIOUS-BRONCHITIS-= VACCINE INFECTIOUS-BURSAL-= DISEASE-VACCINE INFECTIOUS-PERITONITIS-= VACCINE INFLUENZA-VACCINE IPV-VACCINE IRS-19-VACCINE JAPANESE-B-ENCEPHALITIS-= VACCINE KLEBS.PNEUMONIAE-= VACCINE LARYNGOTRACHEITIS-= VACCINE LASSA-FEVER-VACCINE LEGIONNAIRE-DISEASE-= VACCINE LEISHMANIA-VACCINE LEPROSY-VACCINE LEUKEMIA-VACCINE LEUKOSIS-VACCINE LOUPING-ILL-VACCINE LYME-ARTHRITIS-VACCINE M-PROTEIN-VACCINE MALARIA-VACCINE MALIGNANT-EDEMA-= VACCINE MARBLE-SPLEEN-DISEASE-= VACCINE MASTITIS-VACCINE MEASLES-VACCINE MELANOMA-VACCINE MENINGOENCEPHALITIS-= VACCINE MIGEN MOUSEPOX-VACCINE MUCOSAL-DISEASE-VACCINE MUMPS-VACCINE MURIVAC MYXOMATOSIS-VACCINE ORF-VACCINE P-30 P40 PANLEUKOPENIA-VACCINE PAPILLOMA-VACCINE PARAINFLUENZA-VACCINE PARATUBERCULOSIS-VACCINE PARATYPHOID-VACCINE PASTEURELLOSIS-VACCINE PERTUSSIS-VACCINE PESTE-DES-PETITS-= RUMINANTS-VACCINE PHARMALGEN PIGEONPOX-VACCINE PLAGUE-VACCINE PLEUROPNEUMONIA-= VACCINE POLIOMYELITIS-VACCINE POLITYPHOVAC POTOMAC-HORSE-FEVER-= VACCINE PSEUDORABIES-VACCINE Q-FEVER-VACCINE RABIES-VACCINE REDWATER-VACCINE RESPISURE RESPIVAX RHINOPNEUMONITIS-VACCINE RHINOTRACHEITIS-VACCINE RIFT-VALLEY-FEVER-VACCINE RINDERPEST-VACCINE ROCKY-MOUNTAIN-= SPOTTED-FEVER-VACCINE RUBELLA-VACCINE SCHISTOSOMIASIS-VACCINE SMALLPOX-VACCINE SOLCOUROVAC SPECTRALGEN STRANGLES-VACCINE SUISALORAL TENOSYNOVITIS-VACCINE TESCHEN-DISEASE-VACCINE TETANUS-VACCINE TGE-VACCINE THREE-DAY-SICKNESS-= VACCINE TOXOPLASMOSIS-VACCINE TRACHEOBRONCHITIS-= VACCINE TUBERCULOSIS-VACCINE TULAREMIA-VACCINE TUMOR-CELL-VACCINE TYPHOID-VACCINE TYPHUS-VACCINE UROVAC VARICELLA-VACCINE VEE-VACCINE VESICULAR-STOMATITIS-= VACCINE VIBRIOVAKS WEE-VACCINE YELLOW-FEVER-VACCINE ZOOSAL-ORAL

1292 APPENDIX D VAGINA CLITORIS VULVA VAGINA-DISEASE BARTHOLINITIS IPV VAGINITIS VULVOVAGINITIS VARICES VARICOCELE VASCULAR-DISEASE ACROCYANOSIS ALLERGIC-GRANULOMATOSIS ANEURYSM ANGIODERMATITIS ANGIOSCLEROSIS AORTIC-ARCH-SYNDROME AORTITIS ARTERIOSCLEROSIS ARTERITIS ATHEROSCLEROSIS CAPILLAROSCLEROSIS CAROTID-SINUS-SYNDROME CASSIRER-SYNDROME CLAUDICATION cranial-arteritis-extracranial DETERMANN-SYNDROME diabetic-microangiopathy DICLIDOSTOSIS ENDANGITIS ENDARTERITIS ERYTHROMELALGIA ERYTHROPROSOPALGIA esophageal-varices FAHR-DISEASE GANGRENE GRAY-SYNDROME GSELL-ERDHEIM-SYNDROME HEM.TELANGIECTASIA HEMORRHOID hereditary-hem.telangiectasia horton-disease-extracranial HUGHES-STOVIN-SYNDROME HYPERTENSION hypertensive-ulcus-cruris HYPOTENSION IMMERSION-FOOT intermittent-venous-= claudication ISCHEMIA JEFFERSON-SYNDROME KAWASAKI-DISEASE kussmaul-disease LIPODERMATOSCLEROSIS LYMPHANGIOPHLEBITIS MAFFUCI-SYNDROME martorell-syndrome metabolic-syndrome METABOLIC-SYNDROME-X MICROANGIOPATHY NEUROCIRCULATORY-= COMPRESSION-= SYNDROME orthostatic-dysautonomic-= hypotension orthostatic-hypotension osler-syndrome paget-schroetter-syndrome PERIARTERITIS periarteritis-nodosa PHLEBECTASIA PHLEBITIS PSEUDOANEURYSM PULSELESS-DISEASE RAYNAUD-DISEASE REST-PAIN RESTENOSIS SHOCK shy-drager-syndrome TELANGIECTASIA TELANGIECTASIS temporal-arteritis-= extracranial THROMBOANGIITIS THROMBOPHLEBITIS TROPHIC-ULCER ULCUS-CRURIS VARICES VARICOCELE VARICOSIS VASCULITIS VENA-CAVA-SYNDROME VENO-OCCLUSIVE-DISEASE WEGENER-= GRANULOMATOSIS WRIGHT-SYNDROME VASOCONSTRICTORS 202-791 202-791-(+) A-57219 A-61603 ADRENALINE ADRENALONE ALMOTRIPTAN AMEZINIUM METILSULFATE AMIDEFRINE MESILATE BAY-K-8644 BAY-W-5035 BENAZOLINE BQ-485 CIRAZOLINE CLONAZOLINE CORBADRINE COUMAZOLINE CP-122288 CYCLOPENTAMINE DEOXYADRENALINE DIGOXIGENIN-RHAMNOSIDE DMPP DOMAZOLINE ENDOTHELIN ENDOTHELIN-1 ENDOTHELIN-BIG-HUMAN EPHEDRINE ERGOCORNINE ERGOCRISTINE ERGOCRYPTINE ERGOCRYPTINE-ALPHA ERGOCRYPTINE-BETA ERGOMETRINE ERGOSINE ETIRON FENOXAZOLINE GEPEFRINE GR-49336 HOE-511 INDANAZOLINE IPROHEPTINE ISOMETHEPTENE ISOPROPYLMETHOXAMINE KB-R-8498 L-741519 L-741604 M-6434 MEPHENTERMINE METARAMINOL METHOXAMINE METHYLADRENALINE METRAFAZOLINE MK-462 NAPHAZOLINE NITROARGININE-N-G-= METHYLESTER NORADRENALINE NOREPHEDRINE NORFENEFRINE NORMETANEPHRINE OCTODRINE OXYMETAZOLINE PHENAMAZOLINE PHENPROMETHAMINE PHENYLEPHRINE PHOLEDRINE PNO-49-B PROPYLHEXEDRINE PSEUDOEPHEDRINE RS-30026 S-20749 SB-209509 SKF-102652 SKF-88444 SKF-89748-A SODIUM-ORTHOVANADATE SUMATRIPTAN SYNEPHRINE TEFAZOLINE TETRAMINOL TETRYZOLINE THALICMIDINE TINAZOLINE TISOCARBAMIDE TRAMAZOLINE TUAMINOHEPTANE TYMAZOLINE TYRAMINE U-99963 XYLOMETAZOLINE YC-170 ZOLMITRIPTAN VASODILATORS 1045-U-85 202-791 202-791-(-) 349U85 50-235 661U88 8363-S 97-139 ACOXATRINE ADIBENDAN ADRENOMEDULLIN ADRENOMEDULLIN-HUMAN ADRENOMEDULLIN-RAT AHR-16303B AJ-3941 AL-0671 ALIFEDRINE ALIGERON AMAUROMINE AMINOETHYLISOTHIOUREA AMINOPHYLLINE AMIQUINSIN APOVINCAMINATE APOVINCAMINE APRIKALIM AR-L-100-BS ARAGUSPONGINE-D ARANIDIPINE AZAPETINE B-24-76 BAMETHAN BAY-41-2272 BAY-I-1441 BAY-K-9320 BAY-L-3505 BAY-N-6391 BAY-O-5572 BBR-2160 BELARIZINE

Derwent Drug File 1293 Thesaurus BELFOSDIL BEMARINONE BENCIANOL BENFURODIL-HEMISUCCINATE BENZENESULFOHYDROXAMATE BENZYLAMINOCHLORETHYL BENZYLNICOTINATE BIBP-3226 BIBP-3435 BIMAKALIM BM-531 BMS-180560 BN-50417 BN-50418 BOSENTAN BPDZ-79 BQ-123 BQ-153 BQ-485 BQ-610 BQ-928 BRAZERGOLINE BREFONALOL BRL-55834 BRLP-42 BTS-53554 BUFENIODE BUFLOMEDIL BUPHENINE BUTALAMINE BUTERIZINE BW-654 C-92-4609 C-92-4678 CARBAMOYLTRYPTAMINE-5 CARDIODILATIN-126 CARDIODILATIN-88 CARPRONIUM CHLORIDE CARVEDILOL CAS-754 CD-349 CEDO-8956 CENTAUREIDIN CEREBROCRAST CETIEDIL CGP-18137A CGP-22979A CGS-22492 CGS-34043 CH-102 CH-141 CHF-1035 CHOLINE-THEOPHYLLINATE CI-930 CICLONICATE CICLOSIDOMINE CILOSTAZOL CINEPAZIDE CINNARIZINE CL-860201 CLADIELLOLIDE COHN-FRACTION CP-060-S CPU-23 CROMAKALIM CURCARABRANOL-B CVT-3033 CVT-3146 CYCLANDELATE D-230 DARODIPINE DARUSENTAN DEHYDASAL DEMETHYLBUFLOMEDIL-4 DEMETHYLNAFTOPIDIL DENBUFYLLINE DENITRONIPRADILOL DF-100 DIADENOSINE-= PENTAPHOSPHATE DIADENOSINE-= TETRAPHOSPHATE DIHYDROERGOSINE DIHYDROXYPHENYLLACTATE DIISOCYANOADOCIANE DIISOPROPYLAMINE = DICHLOROACETATE DILEVALOL DINIPROFYLLINE DIPFLUZINE DIPROFENE DIPROPHYLLINE DOTARIZINE DPN-205-734 DROTAVERINE E-4010 E-4021 E-4701 EG-1088 ELEDOISIN ELZIVERINE EMAKALIM ENDOTHELIUM-DERIVED-= RELAXANT-FACTOR ENOXIMONE EPERISONE ER-001533 ERGOSININE ESPROQUINE ETHAVERINE EVOCARPINE EXP-3892 F-0401 F-5 FENOLDOPAM FENOXEDIL FK-409 FLORDIPINE FLOSEQUINAN FLUNARIZINE FPL-63012AR FR-139317 FR-144420 FR-146801 FR-173657 FRAXINELLONE GAPICOMINE GEA-3175 GEA-3268 GEA-5145 GINKGO-BILOBA-EXTRACT GINSENOSIDE-RG5 GLUNICATE GOE-5438 GOUTENIN-4 GOUTENIN-5 GR-117289-C GS-389 GYKI-12743 H-5350 H-7 HA-1004 HA-1100 HEPRONICATE HEPTAMINOL-ACEFYLLINATE HEXAMETHYLENE-= AMILORIDE-5 HF-2035 HFV-1017-C HIRSUTINE HN-10200 HNS-32 HYDROXYINDAPAMIDE-5 HYDROXYPYRIDINE-= TARTRATE ICI-153110 IFENPRODIL IGANIDIPINE INOSITOL-NICOTINATE IODOAMILORIDE-6 IPROXAMINE IRL-1620 IRL-2500 ISOBUTYL-NITRITE ISOCORYNOXEINE ISOCURCUMENOL ISOMANNIDE-MONONITRATE ISOMAZOLE ISOPERISONE ISOPRENALINE ISOXSUPRINE ISRADIPINE J-104132 KB-2796 KHL-8430 KI-1769 KI-3005 KI-3315 KI-4032 KMD-3213 KP-403 KR-30988 KRN-2391 KRN-4884 KW-3196 L-6449 LABETALOL LEMIDOSUL LEVCROMAKALIM LI-1370 LIGUSTRAZINE LIPOXIN-B4 LITHOSPERMATE-B LOMIFYLLINE LP-805 LR-693 LR-B-081 LU-127043 LY-127210 LY-137150 LY-163252 LY-222675 MAXADILAN MCC-134 MDL-27032 MECINARONE MEDULLIPIN-I MEFENIDIL MERIBENDAN MESUDIPINE MESUPRINE METACHROMIN-A METACHROMIN-C METAZOSIN METHYLBULBOCAPNINE-O METHYLCHROMONE METHYLRIPARIOCHROMENE METIAPRIL MIBEFRADIL MIMAX MINDODILOL MJ-1991 MJ-451 MOPIDRALAZINE MOTAPIZONE MPC-2101 MRE-0470 N-1518 NAFTIDROFURYL NAFTOPIDIL NAZLININ NC-1100 NF-023

1294 APPENDIX D NICAMETATE NICARDIPINE NICERGOLINE NICHLOTEST NICOFURANOSE NICOFURATE NICOTAFURYL NICOTINATE NICOTINATE-BENZYL NICOTINATE-BUTYL-ESTER NICOTINATE-ETHYL NICOTINATE-HEXYL NICOTINATE-METHYL NICOTINYL-ALCOHOL NIFEDIPINE-META NIMODIPINE NIP-121 NIPRADILOL NITROIBUPROFEN NITROINDAZOLE-6 NITROSOCAPTOPRIL-S NITROSOCYSTEINE-S NITROSOGLUTATHIONE-S NOC-7 NORUSHINSUNINE NS-004 NSC-110333 NY-008 OF-900 OF-900 OFORNINE OLEUROPEOSIDE ONO-AP-227 OPC-28326 ORG-10325 ORG-20494 ORG-30029 ORG-9935 OXODIPINE P-1060 P-1075 P-1188 PAPAVERINE PAPAVEROLINE PARODILOL PD-145065 PD-166793 PENTIFYLLINE PENTOXIFYLLINE PEROXYNITRITE PGV-40350 PHENOXYBENZAMINE PHYSALEMIN PICODRALAZINE PILDRALAZINE PIMEFYLLINE PINACIDIL PINACIDIL-N-OXIDE PIPRATECOL PIPROFUROL PIRIBEDIL PIROXIMONE PIRSIDOMINE PITENODIL PITUITARY-ADENYLATE-= CYCLASE-ACT.PEPTIDE PRENOVERINE PRIMAPERONE PRIZIDILOL PST-2744 QF-303 QF-307 QF-311 QF-313 QUAZINONE REN-1053 RETRACTOR-PENIS-= INHIBITORY-FACTOR RIG-200 RILMAKALIM RO-20-2926 RO-31-6930 RO-44-9375 RO-46-2005 RP-49356 RP-61419 RPR-100579 RS-91309 RS-93522 RU-42173 RWJ-26629 RWJ-29009 S-0139 S-11568 S-12967 S-12968 S-312 S-312-(+) S-312-(-) SALICYLATE-ETHYL SALSOLIDINE SATERINONE SCH-37398 SCH-54470 SDZ-PCO-400 SIGUAZODAN SILDENAFIL SIM-2055 SIM-6080 SKF-100273 SKF-100885 SKF-101485 SKF-101926 SKF-24260 SKF-85174 SKF-94120 SKF-95018 SKF-R-105058 SKF-R-106114 SKF-R-87516 SL-65-0472 SM-3163 SPM-3672 SPM-4744 SPM-5185 SQ-33961 SR-120819-A SR-44866 SR-47063 SR-49059 SR-59104-A SR-59119-A SULOCTIDIL SUN-C-5174 T-0115 T-0201 T-1032 TA-993 TADALAFIL TAK-044 TCV-295 TENSICOR TETRAMETHYLPYRAZINE TETRANITROMETHANE TEZOSENTAN THEOPHYLLINE THEOPHYLLINE-LYSINE THEOPHYLLINE-SODIUM-= ANISATE THEOPHYLLINE-SODIUM-= GLYCINATE THURFYL-NICOTINATE TIFEMOXONE TINOFEDRINE TIPROPIDIL TIZOPROLATE TJ-8007 TJN-220 TN-871 TOLAZOLINE TOLPERISONE TOPRILIDINE TORBAFYLLINE TR-1722 TREQUINSIN TRIACSIN-C TRIACSIN-D TRIMETAPHAN = NITROPRUSSIDE TROPOXIN U-92032 UK-61260 UK-69578 UNTENOSPONGIN-B UR-8225 UT-15 VA-045 VARDENAFIL VASCULAR-ENDOTHELIAL-= GROWTH-FACTOR VASCULAR-ENDOTHELIAL-= GROWTH-FACTOR-HUM VASONATRIN-PEPTIDE VINCAMINE VINCAMINE ADENYLATE VINCAMINE-TEPROSILATE VINCAMONE VINCANOL VINPOCETINE VINPOLINE VINTOPEROL VIQUIDIL W-66 W-7 WS-009A WS-009B XANTINOL-NICOTINATE XB-513 XESTOSPONGIN-A XESTOSPONGIN-B XESTOSPONGIN-C XESTOSPONGIN-D Y-19638 Y-27632 YAKUCHINONE-A YM-435 YOHIMBINE-BETA YT-146 YT-146 Z-1046 Z-10997-A ZD-6021 ZK-112566 ZK-33839 ZM-172405 ZM-226600 ZOLERTINE ZSY-27 VASOPRESSIN-AGONISTS ARGIPRESSIN ARGIPRESSIN-1-8 ARGIPRESSIN-VAL-4 ARGIPRESTOCIN DESMOPRESSIN FELYPRESSIN GLUMIPRESSIN LYPRESSIN NC-1900 ORG-5667 ORNIPRESSIN OXYPRESSIN

Derwent Drug File 1295 Thesaurus PITUITRIN PRESSINAMIDE PRESSINOATE TERLIPRESSIN TGS-34 VASOPRESSIN VASOPRESSIN-ANTAGONISTS CGP-29325 CONIVAPTAN FR-161282 H-5350 JTV-605 LOE-908 NIRAVOLINE ONO-3122 OPC-21268 OPC-31260 SKF-100273 SKF-100398 SKF-100501 SKF-100885 SKF-101071 SKF-101485 SKF-101496 SKF-101497 SKF-101498 SKF-101926 SKF-103561 SKF-104069 SKF-104146 SKF-104146-D SKF-104222 SKF-104223 SKF-104241 SKF-104244 SKF-105494 SKF-105571 SKF-105768 SKF-88864 SR-121463 SR-121463-B SR-49059 SSR-149415 VP-343 WAY-VPA-985 YM-087 VASOTROPICS ACTOVEGIN ALT-766 BENZARONE BIBN-4096-BS CNS-5788 CYLEXIN DEVARICIN EGIS-8332 EPC-K1 ETHANOLAMINE-OLEATE ETHIBLOC FOLESCUTOL MOBECARB MONOETHANOLAMINE = OLEATE MORRHUATE SODIUM MOXICOUMONE PERSILATE PIBECARB PJ-34 RWJ-56110 SODIUM-IODATE T-0201 TETRADECYLSULFATE = SODIUM TIRILAZAD MESILATE TRIBENOSIDE TY-12533 U-87999 UK-279276 UK-343664 WHI-P-97 XT-199 VCAM-ANTAGONISTS ACETYLCYSTEINE VECTOR VIRAL-VECTOR VEGETABLE BRUSSELS-SPROUT CABBAGE CARROT CUCUMBER LETTUCE ONION PEA POTATO SOY-BEAN SPINACH SUGAR-BEET SWEET-POTATO TOMATO TURNIP VENEREAL-DISEASE AMYOTROPHIC-SYPHILITIC-= MYELITIS BABINSKI-SYNDROME bayle-disease CHANCRE CHANCROID CLUTTON-SYNDROME fitz-hugh-syndrome gonococcal-perihepatitis GONORRHEA LOCOMOTOR-ATAXIA LYMPHOGRANULOMA-= VENEREUM NEUROSYPHILIS paralytic-dementia REITER-SYNDROME SYPHILIS TABES-DORSALIS VESSEL ANGIOGENESIS AORTA ARTERIOLE ARTERY CAPILLARY CORONARY DUCTUS-ARTERIOSUS DUCTUS-VENOSUS MICROVESSEL TRUNCUS-ARTERIOSUS VEIN VENA-CAVA VENULE VIROTHERAPY ONCOLYTIC-VIRUS VIRUCIDES 170U88 2242 306 348U87 44081-RP 523-W-91 524-W-91 6-MFA 739-W-94 882C A-1110U A-134U A-315675 A-36683 A-37536 A-5021 A-723U A-73209 A-74704 A-75912 A-75925 A-76792 A-76889 A-76890 A-76928 A-77003 A-77212 A-78791 A-80987 A-98881 ABACAVIR ABIKOVIROMYCIN ABT-606 ABT-987 ACEMANNAN ACETYLARANOTIN ACICLOVIR ACICLOVIR-PHOSPHATE ACICLOVIR-TRIPHOSPHATE ACID-BLUE-129 ACID-BLUE-40 ACRONYCINE ACTINOHIVIN ADA-202-718 ADAPROMIN ADEFOVIR ADEFOVIR-DIPIVOXIL ADENALLENE AG-1254 AG-1284 AG-1296 AG-1387 AG-1402 AG-6084 AG-6840 AG-7088 AGELIFERIN AHA-008 AL-721 ALIZARIN-BLUE-BLACK ALIZARIN-COMPLEXONE ALIZARIN-S ALOVUDINE ALX-40-4-C AMANTADINE AMANTADINE-GLUCURONIDE AMARIIN AMBIGOL-A AMBIGOL-B AMIDAPSONE AMIDINOMYCIN AMIDOMYCIN AMINOCARBOVIR-6 AMINOTHYMIDINE-3+ AMIPRILOSE AMIXINE AMPRENAVIR ANCITABINE-= MONOPHOSPHATE ANGUIDIN ANHYDROSCHUMANNIFICINE ANHYDROZIDOVUDINE-5+,2 ANOLIGNAN-A APIGETRIN APURINIC-ACID ARABINOSYLHYPOXANTHINE ARABINOSYLSANGIVAMYCIN ARABINOSYLTHYMINE ARABINOSYLTHYMINE-= TRIPHOSPHATE

1296 APPENDIX D ARABINOSYLURACIL ARANOTIN ARB-95-214 ARBIDOL ARBORTRISTOSIDE-A ARBORTRISTOSIDE-B ARBORTRISTOSIDE-C ARILDONE ARJUNOLATE ASPARTATE-= HYDROXAMATE-BETA ASTERRIQUINONE ATALAPHILLIDINE ATALAPHILLININE ATEVIRDINE AVRIDINE AWD-625 AWD-627 AZIDODIDEOXY= GUANOSINE-2+,3+ AZIDOTHYMIDINE-4+ AZODICARBOXAMIDE B-041 B-059 B-220 B-239 B-442 BANA-113 BATZELLADINE-A BATZELLADINE-B BAUERINE-B BAY-43-9695 BAY-57-1293 BC-16 BC-59 BC-60 BC-63 BCH-10618 BCH-10619 BCH-189 BCH-189-TRIPHOSPHATE BCH-4556 BCX-1827 BCX-1898 BCX-1923 BDCRB BENZHYDRAZONE BETA-L-THYMIDINE BI-RJ-70 BILA-2185-BS BILD-1263 BILD-1351 BILS-45-BS BL-1743 BMS-181165 BMS-181167 BMS-182193 BMS-186318 BONAPHTON BRI-7013 BRIVUDINE BRL-42359 BRL-43599 BRL-44385 BRL-47923 BRL-55039 BRL-55791 BRL-55792 BRL-57037 BROMOAGELIFERIN BROMOTOPSENTIN BROMOVINYLARAURIDINE-= TRIPHOSPHATE BROMOVINYLDEOXYCYTIDINE BROMOVINYLDEOXY= URIDINE-DIPHOSPHATE BROMOVINYLDEOXY= URIDINE-= MONOPHOSPHATE BROMOVINYLDEOXY= URIDINE-TRIPHOSPHATE BROMOVINYLURIDINE-5 BROPIRIMINE BROXURIDINE BROXURIDINE-= MONOPHOSPHATE BROXURIDINE-TRIPHOSPHATE BUCICLOVIR BUCICLOVIR-TRIPHOSPHATE BUSATIN BUTYLDEOXYNOJIRIMYCIN-N BW-1110U81 BW-1263-W-94 BW-348U87 BW-683C BW-935-U-83 BW-A1117U BW-B429U CAERIN-1.1 CALANOLIDE-A CALANOLIDE-B CALCIUM-SPIRULAN CALLIPELTIN-A CAPROCHLORONE CARBOVIR CARBOVIR-TRIPHOSPHATE CARBOXYMETHYL= ACRIDANONE-10 CASTANOSPERMINE CC-3052 CD4-PS.EXOTOXIN-A CF-1001 CF-1093 CG-662 CGP-53437 CGP-53820 CGP-57813 CHELIDAMATE CHLORODIDEOXY= GUANOSINE-6 CHLOROETHYLDEOXYURIDINE CHLOROPEPTIN-I CHLOROPURINE-ARABINOSIDE CHLOROTUBERCIDIN-5 CHLOROUS-ACID CHLOROVINYLARAURIDINE-5 CIBACRON-BLUE-3-GA CIDOFOVIR CIPAMFYLLINE CITENAZONE CITPRESSINE-I CITPRESSINE-II CITRACRIDONE-II CITRUSININE-I CL-306293 CL-387626 CLEVUDINE CNI-H-0294 CNI-H-1194 COMPOUND-102 CONIDENDRIN-ALPHA CONOCURVONE CORDATOLIDE-A CORDATOLIDE-B CORNUSIIN-A COSALANE COSTATOLIDE CRAMBESCIDIN-800 CRAMBESCIDIN-816 CS-432 CS-436 CS-437 CS-85 CS-87 CS-87-TRIPHOSPHATE CS-91 CS-92 CT-2576 CTC-23 CTC-96 CURDLAN-ARABINOSE-= SULFATE CURDLAN-GALACTOSE-= SULFATE CURDLAN-SULFATE CYANOVIRIN-N CYCLAM CYCLARADINE CYCLARADINE-METHOXY= ACETATE-5+ CYCLIC-GMP-NOR-2+ CYCLOBUT-A CYCLOBUT-G CYCLODEXTRIN-ALPHA-= SULFATE CYCLODEXTRIN-BETA-= SULFATE CYCLOVIRACIN-B1 CYCLOVIRACIN-B2 CYSTATIN CYSTATIN-C-HUMAN CYTALLENE CYTARABINE CYTARABINE-DIPHOSPHATE CYTARABINE-= MONOPHOSPHATE D-435 D-609 DAMMADIENOL DAMMARENEDIOL-II DAPHNODORIN-A DAPHNODORIN-B DAPHNODORIN-C DEAZAARISTEROMYCIN-3 DEAZAGUANOSINE-3 DEAZAGUANOSINE-7 DEAZANEPLANOCIN-3 DEITIFORIN DELAVIRDINE DEMETHYLCHROMO= MYCIN-A2 DEMETHYLCHROMO= MYCIN-A3 DEMETHYLOLIVOMYCIN-A DEOXYCARBOVIR-6 DEOXYPANCRATISTATIN-7 DEOXYSANGIVAMYCIN-2+ DEOXYTOPSENTIN DEOXYTOYOCAMYCIN-2+ DERCITIN DESCICLOVIR DESTRUXIN-B DEUTIPHORINE DEXTRAN-CM-= BENZYLAMIDE-SULFONATE DEXTRIN-2-SULFATE DIAMINOPHENAZINE-2,3 DIAMINOPURINE-= DIDEOXYRIBOSIDE DIBROMOAGELIFERIN DIBROMOSCEPTRIN DICHLOROFLAVAN DIDANOSINE DIDEMNIN-A DIDEMNIN-B DIDEMNIN-C DIDEOXY-ATP DIDEOXY-ITP DIDEOXY-UDP DIDEOXY-UMP DIDEOXY-UTP DIDEOXYADENOSINE-2+,3+ DIDEOXYCYTIDINENE-2+,3+

Derwent Drug File 1297 Thesaurus DIDEOXYGUANOSINE-2+,3+ DIDEOXYGUANOSINENE-= 2+,3+ DIDEOXYTHYMIDINE-2+,3+ DIHYDROCOSALANE DIHYDROCOSTATOLIDE-7,8 DIHYDROEUPARIN DIHYDRONARCICLASINE-= TRANS DIHYDROXYPROPYL= ADENINE-9 DIMETHYLAMINOPURINE-6ARABINOSIDE DIMETHYLQUERCETIN-3,7 DIOXOLANE-C DIOXOLANE-T DISOXARIL DMP-323 DMP-450 DMP-963 DP-107 DPC-082 DPC-083 DPC-961 DRAGMACIDIN-D DUP-925 EA-521 ECHINOCYSTATE EDOXUDINE EFAVIRENZ EICAR ELENOLATE CALCIUM EM-2487 EMODINBIANTHRONE EMTRICITABINETRIPHOSPHATE ENFUVIRTIDE ENOPEPTIN-A ENVIRADENE ENVIROXIME EOSINOPHIL-DERIVED-= NEUROTOXIN-HUMAN EPERVUDINE EPICASTANOSPERMINE-1 EPMG ERGOSTEROL-PEROXIDE ERMANIN EUDISTOMIN-C EUDISTOMIN-E EUDISTOMIN-F EUDISTOMIN-K EUDISTOMIN-L EUGLOBAL-G5 EXODUS F-36 FAMCICLOVIR FAMOTINE FATTIVIRACIN-FV-8 FEAC FEAU FIAC-TRIPHOSPHATE FIACITABINE FIALURIDINE FIALURIDINE-TRIPHOSPHATE FLAVOFUNGIN FLAVOPENTIN FLOXURIDINE FLUOROARISTEROMYCIN-= 6+BETA FLUORODEOXYADENOSINE-= 3+ FLUORODEOXY= GUANOSINE-2+ FLUORODIDEOXY-CTP-5 FLUORODIDEOXY-= VIDARABINE2+TRIPHOSPHATE FLUORODIDEOXY= ADENOSINE-2+ FLUORODIDEOXY= ARABINOSYLINOSINE-2+ FLUORODIDEOXYCYTIDINE-= 2+ FLUORODIDEOXY= GUANOSINE-3+ FLUORODIDEOXYINOSINE-2+ FLUORODIDEOXY= VIDARABINE-2+ FLUOROTHYMIDINE-= MONOPHOSPHATE FLUOROTHYMIDINE-= TRIPHOSPHATE FLUOROZALCITABINE-5 FLUTIMIDE FLUVIRUCIN-A1 FLUVIRUCIN-A2 FLUVIRUCIN-B1 FLUVIRUCIN-B2 FLUVIRUCIN-B3 FLUVIRUCIN-B4 FMAC-TRIPHOSPHATE FMAU FMAU-TRIPHOSPHATE FOSARILATE FOSCARNET FOSFONET SODIUM FPMPA FPMPDAP FPMPG FRENTIZOLE FTC FUNICULOSIN FURAVIR GANCICLOVIR GANCICLOVIR-DIPROPIONATE GANCICLOVIR-PHOSPHATE GANCICLOVIR-TRIPHOSPHATE GAP-31 GARDENIN-A GEM-132 GEM-91 GLA-27 GLA-40 GLA-57 GLA-58 GLA-59 GLA-60 GLA-63 GLA-66 GLA-70 GLQ-223 GLYCOCITRINE-I GLYCOVIR GLYFOLINE GPI-0100 GRANDISINE-I GRANDISINE-II GRANDISININE GS-1659 GS-4071 GS-4104 GS-4116 GW-433908 H-2-G H-3031 HAEMATOXYLIN HB-19 HBY-097 HELIOXANTHIN HEMINORDIHYDRO= GUAIARETATE HENNOXAZOLE-A HEPT HERACLENOL HERBIMYCIN-A HERBIMYCIN-B HI-236 HI-253 HI-280 HMHBG-2 HOE-602 HOE-961 HOE-BAY-946 HPA-23 HPA-39 HPMPA HPMPDAP HPMPG HS-058 HYB-101400 HYDROXYGLUTAMATE-4 HYDROXYMETHYL= ELLIPTICINE HYDROXYMETHYL= ZALCITABINE-3+ HYDROXYMYRISTATE-2 HYDROXYNORVALINE-BETA HYDROXYPALMITATE-2 HYDROXYPHTHALOYL-= LACTOGLOBULIN-BETA I-152 IBISTEROL-SULFATE ICAM-1 ICI-130685 ICI-65709 ICI-73602 ICN-3952 IDOXURIDINE IDOXURIDINE-= MONOPHOSPHATE IMIQUIMOD IMPACARZINE INDINAVIR INGENOL INGENOL-TRIACETATE INOPHYLLUM-B INOPHYLLUM-P INTERFERON INTERFERON-ALPHA INTERFERON-ALPHA,BETA INTERFERON-ALPHA,BETA-= MOUSE INTERFERON-ALPHA,BETA-= RAT INTERFERON-ALPHA-1 INTERFERON-ALPHA-1-= ALPHA-8-HUMAN INTERFERON-ALPHA-1-= CATTLE INTERFERON-ALPHA-1-= HUMAN INTERFERON-ALPHA-1-= MOUSE INTERFERON-ALPHA-2 INTERFERON-ALPHA-2-1-= HUMAN INTERFERON-ALPHA-2-ARG INTERFERON-ALPHA-2-= HUMAN INTERFERON-ALPHA-2-= MOUSE INTERFERON-ALPHA-2A INTERFERON-ALPHA-2A-= HUMAN INTERFERON-ALPHA-2B INTERFERON-ALPHA-2B-= HUMAN INTERFERON-ALPHA-2C INTERFERON-ALPHA-2C-= HUMAN INTERFERON-ALPHA-4-= HUMAN INTERFERON-ALPHA-4-= MOUSE INTERFERON-ALPHA-4A INTERFERON-ALPHA-54

1298 APPENDIX D INTERFERON-ALPHA-6 INTERFERON-ALPHA-7-= HUMAN INTERFERON-ALPHA-8 INTERFERON-ALPHA-A-D INTERFERON-ALPHA-A-= D(BGL-II) INTERFERON-ALPHA-B INTERFERON-ALPHA-B-D INTERFERON-ALPHA-B-D-= HUMAN INTERFERON-ALPHA-B-= HUMAN INTERFERON-ALPHA-BDBB INTERFERON-ALPHA-C INTERFERON-ALPHA-C-= CATTLE INTERFERON-ALPHA-C-= HUMAN INTERFERON-ALPHA-CATTLE INTERFERON-ALPHA-CON-1 INTERFERON-ALPHA-CON1-= HUMAN INTERFERON-ALPHA-F-D INTERFERON-ALPHA-F-= HUMAN INTERFERON-ALPHA-GAMMA INTERFERON-ALPHA-HUMAN INTERFERON-ALPHA-I INTERFERON-ALPHA-I-= HUMAN INTERFERON-ALPHA-I1 INTERFERON-ALPHA-I1-= CATTLE INTERFERON-ALPHA-II-1 INTERFERON-ALPHA-J INTERFERON-ALPHA-J-C INTERFERON-ALPHA-J1-= SER116 INTERFERON-ALPHA-K INTERFERON-ALPHA-MOUSE INTERFERON-ALPHA-N INTERFERON-ALPHA-N1 INTERFERON-ALPHA-N1-= HUMAN INTERFERON-ALPHA-N3-= HUMAN INTERFERON-ALPHA-PIG INTERFERON-BETA INTERFERON-BETA-1 INTERFERON-BETA-1-HORSE INTERFERON-BETA-1-HUMAN INTERFERON-BETA-1A INTERFERON-BETA-1A-= HUMAN INTERFERON-BETA-1B INTERFERON-BETA-2 INTERFERON-BETA-2-HUMAN INTERFERON-BETA-CAT INTERFERON-BETA-CATTLE INTERFERON-BETA-HUMAN INTERFERON-BETA-MOUSE INTERFERON-BETA-PIG INTERFERON-BETA-SER INTERFERON-BETA-SER-= HUMAN INTERFERON-CAT INTERFERON-CATTLE INTERFERON-CONCENSUS INTERFERON-DELTA-4-= ALPHA-2-ALPHA-1 INTERFERON-GAMMA INTERFERON-GAMMA-1B INTERFERON-GAMMA-4A INTERFERON-GAMMA-= CATTLE INTERFERON-GAMMA-= HUMAN INTERFERON-GAMMA-= MOUSE INTERFERON-GAMMA-PIG INTERFERON-GAMMA-RABBIT INTERFERON-GAMMA-RAT INTERFERON-HUMAN INTERFERON-MOUSE INTERFERON-PI INTERFERON-RAT INTERFERON-TAU INTERFERON-TAU-HUMAN INTERFERON-TAU-SHEEP INTERLEUKIN-13-HUMAN IODODEOXYCYTIDINE IODOVINYLDEOXYURIDINE ISIS-1082 ISIS-1751 ISIS-1753 ISIS-1755 ISIS-2105 ISIS-2922 ISIS-4015 ISIS-5320 ISOCHROMOPHILONE-I ISOCHROMOPHILONE-II ISOELEUTHERIN ISOKAEMPFERIDE ISOMANGIFERIN ISONARCICLASINE IVX-E-59 IZATHIZON JACALIN JARANOL JCA-304 JCA-314 JE-2147 JM-1590 JM-1591 JM-1596 JM-1657 JM-2762 JM-2763 JM-2768 JM-2815 JM-2820 JM-2936 JM-3100 K-12 K-37 K-38 K-42 KAIKASAPONIN-I KARALICIN KETOXAL KISIMICIN KISTAMICIN-A KISTAMICIN-B KNI-102 KNI-144 KNI-174 KP-15 KP-21 KUTAPRESSIN KYNOSTATIN-227 KYNOSTATIN-272 L-653180 L-689502 L-693593 L-694746 L-696040 L-696229 L-696474 L-697639 L-697661 L-697695 L-700417 L-702007 L-708906 L-731723 L-731988 L-737126 L-738372 L-739594 L-754394 L-FMAU LAFARINE LAMIVUDINE LAMIVUDINE-TRIPHOSPHATE LARYPHANE LB-71148 LB-71350 LIGHT-GREEN-SF-YELLOWISH LITHOSPERMATE-B LJ-45 LOBOHEDLEOLIDE LOBUCAVIR LOPINAVIR LY-180299 LY-214624 LY-217896 LY-253963 LY-289612 LY-300046 LY-300082 LY-343928 LY-353352 LY-582563 LY-73497 M+B-7714 M-12325 MACROLACTIN-A MANGIFERIN MAP-30 MAPI-ALPHA MARIBAVIR MDL-101028 MDL-20610 MDL-20646 MDL-28574 MDL-28653 MDL-29204 MDL-29270 MDL-29435 MDL-43305 MDL-44370 MDL-860 MEGALOMICIN-C MELIACIN MEMOTINE MEN-10690 METHANOCARBA= THYMIDINE-N METHISOPRINOL METHOXYDODECANOATE-12 METHOXYPURINE-6-= ARABINOSIDE METHYLANHYDRO= SCHUMANNIFICINE-N METHYLCALOPOCARPIN-O-3 METHYLFORMYCIN-4 METHYLLAUROTETANINE-N METHYLQUERCETIN-3 METHYLSCHUMANNIFICINE-N METISAZONE MGN-3 MICHELLAMINE-A MICHELLAMINE-B MICHELLAMINE-C MKC-442 ML-4 MM-46115 MOLLUGIN MONOLINOLEIN-ALPHA MOPYRIDONE MORONATE

Derwent Drug File 1299 Thesaurus MOROXYDINE MSC-204 MSC-206 MSH-372 MSI-30 MSI-98 MSL-109 MYCALAMIDE-A MYCALISINE-A MYCAPEROXIDE-A MYCAPEROXIDE-B MYCOPHENOLATE NARCICLASINE NARIRUTIN NB-1011 NELFINAVIR NEPLANOCIN-C NEPLANOCIN-D NEURAMIDE NEUTROPHIL-PEPTIDE-= HUMAN-1 NEUTROPHIL-PEPTIDE-= HUMAN-2 NEUTROPHIL-PEPTIDE-= HUMAN-3 NEVIRAPINE NF-201 NF-503 NF-504 NF-506 NIGLIZIN NIGRANOATE NIRURISIDE NITROSOBENZAMIDE-3 NOBOTANIN-B NOBOTANIN-K NONYL-DEOXYNOJIRI= MYCIN-N NORACRONYCINE NORBERGENIN NSC-117614 NSC-158393 NSC-20625 NSC-287474 NSC-4493 NSC-615985 NSC-619531 NSC-624151 NSC-624152 NSC-624231 NSC-625487 NSC-648400 NSC-651016 NSC-654021 NSC-666724 NSC-D-614989 OENOTHEIN-B OL-56 OLOMOUCINE ONCHITRIOL-I ONCHITRIOL-II ONNAMIDE-A ORYZACYSTATIN-I OSELTAMIVIR OXAZINOMYCIN OXETANOCIN-A OXETANOCIN-G OXETANOCIN-GTRIPHOSPHATE OXOCALANOLIDE-A-12 OXOFORMYCIN OXOFORMYCIN-B OXOLIN OXOSTEPHANINE P-4018 P-536 P-9941 PACHYPODOL PACHYSTAUDINE PALIVIZUMAB PD-022551 PD-024886 PD-134922 PD-135390 PD-156202 PD-159206 PD-161374 PD-178390 PD-178392 PENCICLOVIR PENCICLOVIR-TRIPHOSPHATE PENTALENOLACTONE PENTALENOLACTONE-O PENTOSTATIN PEPTIDE-T PEPTIDE-T-4-8 PEPTIDE-T-D-ALA-1 PHENALAMIDE-A1 PHENOXAN PHOSPHONOACETATE PICLAVINE-A1 PICLAVINE-A2 PICLAVINE-A3 PICLAVINE-A4 PIRODAVIR PLAKINIDINE-A PLECONARIL PM-1 PM-102 PM-104 PM-19 PM-2 PM-29 PM-3 PM-30 PM-40 PM-43 PM-44 PM-47 PM-48 PM-504 PM-523 PM-62 PM-63 PM-64 PM-65 PM-66 PM-67 PM-69 PM-72 PM-73 PM-77 PM-82 PM-83 PMEC PMEDAP PMEG PMPDAP PMPG PNU-109112 PNU-142721 PNU-145156-E PODORHIZOL POLY-GA-C POLY-GI-C POLYVINYLSULFONATE = SODIUM PRADIMICIN-A PRADIMICIN-S PRADIMICIN-T1 PRADIMICIN-T2 PRO-2000 PROPHYL PROPYLDEOXYURIDINE-5 PTILOMYCALIN-A PTU-23 PY-11 PYRAZOMYCIN PYRROLIDINEDITHIO= CARBAMATE QUARTROMICIN-A1 QUARTROMICIN-A2 QUARTROMICIN-A3 QUARTROMICIN-D1 QUINIZARIN QUINOBENE QYL-1064 QYL-685 QYL-769 QYL-941 QYL-972 R-60164 R-61837 R-62025 R-62827 R-66703 R-66933 R-67041 R-72440 R-78206 R-82150 R-82913 R-86183 R-88703 R-89439 R-95288 RANTES RD-3-0028 RD-3-0174 RD-42024 RD-42217 RD-6-2198 RD-6-5071 REACTIVE-BLUE-4 REC-15-0209 REISWIGIN-A REISWIGIN-B RESIQUIMOD RESOBENE RIBAMIDINE RIBAVIRIN RIBAVIRIN-DIPHOSPHATE RIBAVIRIN-TRIACETATE RIBAVIRIN-TRIPHOSPHATE RIBONUCLEASE RIDASTINE RIDOSTIN RIFASTINE RIMANTADINE RIODOXOL RITONAVIR RMI-15731 RNA-DOUBLE-STRANDED RO-09-0410 RO-09-0535 RO-09-0696 RO-09-0881 RO-24-5098 RO-24-7429 RO-25-3036 RO-32-1520 RO-32-2313 RO-32-4397 RO-5-3335 ROBUSTAFLAVONE ROSCOVITINE RPR-103611 RPR-111423 RS-980 RUBROMYCIN-ALPHA RUBROMYCIN-BETA RUBROMYCIN-GAMMA

1300 APPENDIX D RWJ-270201 S-26704 S-2720 S-27609 S-28463 S-7 SA-1042 SALASPERMATE SALIREPOSIDE SAMARANGENIN-B SANDWICENSIN SAQUINAVIR SB-203238 SB-203386 SB-205891 SB-206343 SC-52151 SC-55389A SCEPTRIN SCH-350634 SCH-351125 SCH-38057 SCH-47802 SCHIZOPHYLLAN-SULFATED SCOPADULCATE-B SD-146 SD-894 SDZ-282-870 SDZ-283-053 SDZ-35-682 SDZ-NIM-811 SECRETORY-LEUKOCYTE-= PROTEASE-INHIBIT-HU SEVERIFOLINE SF-2140 SF-2324 SF-2361 SF-2487 SIAMYCIN-I SIAMYCIN-II SJ-3366 SKF-107457 SKF-107461 SKF-108738 SKF-108922 SKF-21681 SKF-21687 SKF-30097 SKF-40491 SO-324 SO-730 SORIVUDINE SOULATTROLIDE SP-303 SPC-3 SPIROAMANTADINE SQ-32829 SQ-34676 SR-3722 SR-3745 SR-3745A SR-3772 SR-3773 SR-3775 STACHYFLIN STAVUDINE STROBILURIN-E STROMAL-CELL-DERIVED-= FACTOR-1 STROMAL-CELL-DERIVED-= FACTOR-1-ALPHA SV-4814 SWERTIFRANCHESIDE SY-801 SYNADENOL SYNCYTOL SYNGUANOL SYNTHYMOL SYZYGIOL T-140-POLYPHEMUSIN T-157602 T-30177 T-30677 T-30695 T-70182 T22 TAK-779 TCRB TEBROFEN TENOFOVIR TENOFOVIR-DIPHOSPHATE TENUAZONATE TERNATIN TERPESTACIN TETRAMIN THIANGAZOLE THIOPHENOYLUREA THYMALLENE THYRSIFEROL THYRSIFERYL-ACETATE-23 TIBO TILORONE TIPRANAVIR TJ-13025 TMC-125 TOLYTOXIN TOMEGLOVIR TOPSENTIN TOXICOL-A TOXICOL-B TOXIUSOL TRAPANIN-B TRIBROMOPHLOROGLUCINOL TRICHLOROPHLOROGLUCINOL TRICHLORORESORCINOL TRICHOCARPIN TRIFLUOROMETHYL= DEOXYCYTIDINE TRIFLURIDINE TRIPTERIFORDIN TROMANTADINE TROPHOBLAST-PROTEIN-= SHEEP TUBERCIDIN-= MONOPHOSPHATE TUBERCULATIN U-100313 U-103017 U-104489 U-3243 U-75875 U-76088 U-80493E U-81749 U-84645E U-85548E U-85549E U-88204 U-88204E U-88566 U-89360 U-93840 U-93965 U-95133 U-96988 U-99499 UC-040 UC-10 UC-284 UC-42 UC-781 UC-82 UDJO-1311 UIC-94003 UMJD-828 VALACICLOVIR VALGANCICLOVIR VARIABILIN VARIOLIN-B VB-11328 VENUSTATRIOL VF-1634 VIDARABINE VIDARABINE-ACETATE VIDARABINE-DIACETATE-= 2+,3+ VIDARABINE-OCTANOATE VIDARABINE-PHOSPHATE VIDARABINE-TRIPHOSPHATE VIDARABINE-VALERATE VINYLARABINOSYLURACIL-5 VIOLAMYCIN VIRANTMYCIN VX-497 WHI-07 WIN-52035 WIN-52084 WIN-53338 WIN-54954 WIN-57007 WIN-63843 XENAZOATE XENYGLOXAL XK-216 XK-234 XN-482 XR-457 XR-835 XYLOTUBERCIDIN XYLURE YUCCA-LEAF-PROTEIN ZALCITABINE ZANAMIVIR ZIDOVUDINE ZIDOVUDINE-ISOLEUCINE ZIDOVUDINE-TRIPHOSPHATE ZIMET-111-74 ZIMET-98-69 ZINVIROXIME VIRUS ADENO-ASSOCIATED-VIRUS ADENOVIRUS AKABANE-DISEASE-VIRUS ALEUTIAN-DISEASE-VIRUS AMERICAN-EEL-VIRUS ARBOVIRUS ARENAVIRUS ARTERITIS-VIRUS AVIAN-SARCOMA-VIRUS BACULOVIRUS BIV-VIRUS BIVENS-ARMS-VIRUS BK-VIRUS BLUE-TONGUE-VIRUS BLUECOMB-VIRUS BORDER-DISEASE-VIRUS BORNA-DISEASE-VIRUS BREDA-VIRUS BUNYAMWERA-VIRUS BUSSUQUARA-VIRUS C-TYPE-VIRUS CAE-VIRUS CALICIVIRUS CALIFORNIA-VIRUS CALOVO-VIRUS CAMELPOX-VIRUS CAT-ENTERIC-CORONAVIRUS CAT-SYNCYTIAL-VIRUS CELO-VIRUS CHANNEL-CATFISH-VIRUS CHIKUNGUNYA-VIRUS

Derwent Drug File 1301 Thesaurus COITAL-EXANTHEMA-VIRUS CONGO-VIRUS CORONAVIRUS COWPOX-VIRUS COXSACKIE-VIRUS CYTOMEGALO-VIRUS CYTOPLASMIC-= POLYHEDROSIS-VIRUS DENGUE-VIRUS DERZSY-DISEASE-VIRUS DISTEMPER-VIRUS DUVENHAGE-VIRUS EBHS-VIRUS EBOLA-VIRUS ECBO-VIRUS ECHO-VIRUS EE-VIRUS EMC-VIRUS ENCEPHALITIS-VIRUS ENCEPHALOMYELITIS-VIRUS ENTEROVIRUS EPIZOOTIC-HEM.DISEASE-= VIRUS EPSTEIN-BARR-VIRUS ERC-VIRUS ERYTHROLEUKOSIS-VIRUS EUROPEAN-EEL-VIRUS EVD-VIRUS FIV-VIRUS FLURY-VIRUS FRIEND-VIRUS FROG-VIRUS-3 GETAH-VIRUS GROSS-VIRUS HEM.ANEMIA-SYNDROME-= VIRUS HEM.ENTERITIS-VIRUS HEM.SEPSIS-VIRUS HEMAGGLUTINATING-= ENCEPHALOMYELITIS-= VIRUS HEPATITIS-A-VIRUS HEPATITIS-B-VIRUS HEPATITIS-C-VIRUS HEPATITIS-VIRUS HERPES-SIMPLEX-VIRUS HERPES-SIMPLEX-VIRUS-1 HERPES-SIMPLEX-VIRUS-2 HERPESVIRUS HIV-1-VIRUS HIV-2-VIRUS HIV-VIRUS HTLV-I-VIRUS HTLV-II-VIRUS IBARAKI-VIRUS IBR-IPV-VIRUS ICH-VIRUS INCLUSION-BODY-= HEPATITIS-VIRUS INCLUSION-BODY-RHINITIS-= VIRUS INFECTIOUS-ANEMIA-VIRUS INFECTIOUS-BRONCHITIS-= VIRUS INFECTIOUS-BURSAL-= DISEASE-VIRUS INFECTIOUS-= HEMATOPOIETIC-= NECROSIS-VIRUS INFECTIOUS-= LARYNGOTRACHEITIS-= VIRUS INFECTIOUS-PANCREATIC-= NECROSIS-VIRUS INFECTIOUS-PERITONITIS-= VIRUS INFLUENZA-A-VIRUS INFLUENZA-B-VIRUS INFLUENZA-VIRUS IRIDOVIRUS JAPANESE-ENCEPHALITIS-= VIRUS JUNIN-VIRUS KIRSTEN-VIRUS LANGAT-VIRUS LASSA-FEVER-VIRUS LENTIVIRUS LEUKOSIS-VIRUS LEUKOVIRUS LOUPING-ILL-VIRUS LUMPY-SKIN-DISEASE-VIRUS LYMPHOCYTIC-= CHORIOMENINGITIS-VIRUS MACHUPO-VIRUS MALIGNANT-CATARRHAL-= FEVER-VIRUS MAMILLITIS-VIRUS MAMMARY-TUMOR-VIRUS MAMMILITIS-VIRUS MARBLE-SPLEEN-DISEASE-= VIRUS MASON-PFIZER-MONKEY-= VIRUS MEASLES-VIRUS MENGO-VIRUS MOKOLA-VIRUS MOLLUSCUM-= CONTAGIOSUM-VIRUS MOLONEY-VIRUS MOUSE-HEPATITIS-VIRUS MOUSE-SARCOMA-VIRUS MOUSE-THYMIC-VIRUS MOUSEPOX-VIRUS MUCOSAL-DISEASE-VIRUS MUMPS-VIRUS MYELOBLASTOSIS-VIRUS MYXOMATOSIS-VIRUS MYXOVIRUS NAIROBI-SHEEP-DISEASE-= VIRUS ONCORHYNCHUS-MASOU-= VIRUS ONCOVIRUS ORF-VIRUS PACHECO-DISEASE-VIRUS PANLEUKOPENIA-VIRUS PAPILLOMA-VIRUS PAPOVAVIRUS PAPULAR-STOMATITIS-VIRUS PARAINFLUENZA-VIRUS PARAMYXO-VIRUS PARVOVIRUS PEROMYSCUS-VIRUS PHAGE PICHINDE-VIRUS PICORNAVIRUS PIGEON-HERPESVIRUS PIGEON-PARAMYXO-VIRUS PIGEONPOX-VIRUS PIGPOX-VIRUS PIKE-FRY-DISEASE-VIRUS POLIOMYELITIS-VIRUS POLYOMA-VIRUS POWASSAN-VIRUS POXVIRUS PROGRESSIVE-PNEUMONIA-= VIRUS PROPHAGE PRRS-VIRUS PSEUDO-COWPOX-VIRUS PSEUDORABIES-VIRUS PULMONARY-= ADENOMATOSIS-VIRUS PUNTA-TORO-VIRUS RABIES-VIRUS RAUSCHER-VIRUS REOVIRUS RETICULOENDOTHELIOSIS-= VIRUS RETROVIRUS RHABDOVIRUS RHINO-VIRUS RHINOPNEUMONITIS-VIRUS RHINOTRACHEITIS-VIRUS RIFT-VALLEY-FEVER-VIRUS RILEY-VIRUS RINDERPEST-VIRUS ROTA-VIRUS ROUS-SARCOMA-VIRUS RS-VIRUS RUBELLA-VIRUS SANDFLY-FEVER-VIRUS SEMLIKI-FOREST-VIRUS SENDAI-VIRUS SIALODACRYOADENITIS-= VIRUS SIMIAN-SARCOMA-VIRUS SIMIAN-VARICELLA-VIRUS SINDBIS-VIRUS SIV-VIRUS SMALLPOX-VIRUS SMEDI-VIRUS SNOWSHOE-HARE-VIRUS SPONDWENI-VIRUS SPRING-VIREMIA-VIRUS SQUIRREL-MONKEY-= RETROVIRUS ST.LOUIS-ENCEPHALITIS-= VIRUS STLV-III-VIRUS SV40-VIRUS SV5-VIRUS TACARIBE-VIRUS TAHYNA-VIRUS TESCHEN-DISEASE-VIRUS TGE-VIRUS THREE-DAY-SICKNESS-VIRUS TOBACCO-MOSAIC-VIRUS TRANSMISSIBLE-ENTERITIS-= VIRUS TREMBLING-DISEASE-VIRUS VACCINIA-VIRUS VARICELLA-ZOSTER-VIRUS VE-VIRUS VESICULAR-STOMATITIS-= VIRUS VIRION VISNA-VIRUS WESSELSBRON-DISEASE-= VIRUS WEST-NILE-VIRUS WOODCHUCK-HEPATITIS-= VIRUS YELLOW-FEVER-VIRUS VIRUS-HEPATITIS chron.aggressive-hepatitis SERUM-HEPATITIS VITAMINS ACACETIN AMENTOFLAVONE AMENTOFLAVONE-= HEXAACETATE BILOBETIN BIOFLAVONOIDS CIANIDANOL DIFRAREL DIHYDROFISETIN DIHYDROQUERCETIN DIOSMIN ENDOTELON ESCULIN ETHOXAZORUTOSIDE FLAVODATE

1302 APPENDIX D GINKGETIN GOSSYPETIN GOSSYPIN GUAIJAVERIN HESPERIDIN HESPERIDIN-= METHYLCHALCONE ISOQUERCITRIN ISORHAMNETIN LEUCOCIANIDOL METHYLQUERCETIN-3 MONOXERUTIN MYRICETIN MYRICITRIN NARCISSIN PRUNETIN QUERCETAGITRIN QUERCETIN ROBINETIN RUTOSIDE SCIADOPITYSIN SINENSETIN TANGERETIN TAXIFOLIN TECTORIGENIN TECTORIGENIN-PSI TROXERUTIN VENORUTON-P4 VITAMIN-U Z-12000 Z-12001 Z-12007 VITAMINS-A ACITRETIN ACYCLORETINOATE AGN-190073 AGN-190089 AGN-190121 AGN-190186 AGN-190299 AGN-190727 AGN-191701 AGN-193835 AGN-193836 AGN-194078 AGN-194204 AGN-195153 ALRT-1550 AM-555 AM-590 AROTENOID AROTINOID-ETHYLSULFIDE AROTINOID-ETHYLSULFONE AROTINOID-SULFONATE AZ-80 BMS-181163 BMS-185411 BMY-30047 BUTYLRETINAMIDE-N CAROTENE-BETA CD-2247 CD-2809 CD-394 CD-564 CH-40 DEHYDRORETINAL DEHYDRORETINOATE DEHYDRORETINOL DIDEHYDRORETINOATE-3,4 DIHYDRORETINOATE-9,10 EPOXYRETINOATE-5,6 ETAROTENE ETHYLRETINAMIDE-N ETRETINATE FENRETINIDE HYDROXENIN HYDROXYISOTRETINOIN-4 HYDROXYRETINAL-4 HYDROXYRETINOATE-4 IODOPSIN ISOACITRETIN ISOTRETINOIN ISOTRETINOIN-METHYL-= ESTER ISOTRETINOIN-OXO-4 JUVENILE-HORMONE-III KITOL LG-100182 LG-100268 LG-101305 LGD-1069 LUTEIN METHYL-TRETINOIN METHYLFENRETINIDE-O MOFAROTENE MOTRETINIDE POLYPRENOATE RE-80 RETINAL RETINAL-13-CIS RETINAL-9-CIS RETINAMIDE RETINOATE-9-CIS RETINOL RETINOL-ACETATE RETINOL-GLUCURONIDE RETINOL-HEPTADECANOATE RETINOL-LAURATE RETINOL-LINOLEATE RETINOL-LINOLENATE RETINOL-MYRISTATE RETINOL-OLEATE RETINOL-PALMITATE RETINOL-PALMITOLEATE RETINOL-PHOSPHATE RETINOL-PROPIONATE RETINOL-STEARATE RETINOYL-BETA-GLUCOSE RETINOYL-BETA-= GLUCURONIDE RETINOYL-FLUORIDE RETINOYL-GLYCINE RETINOYL-LEUCINE RETINOYL-PHENYLALANINE RETINYL-METHYL-ESTER RETINYLIDENE-DIMEDONE RETINYLIDENE-= METHYLNITRONE RO-10-1770 RO-11-0503 RO-11-1272 RO-11-4768 RO-11-8284 RO-12-0955 RO-12-0995 RO-12-4825 RO-12-7310 RO-12-7554 RO-12-9933 RO-13-2389 RO-13-4306 RO-13-6307 RO-13-7410 RO-13-8320 RO-13-9272 RO-14-3899 RO-14-9572 RO-15-1549 RO-18-6622 RO-18-8093 RO-19-0645 RO-19-0645 RO-19-4787 RO-19-4788 RO-19-7224 RO-21-6667 RO-22-6595 RO-23-2895 RO-23-3571 RO-23-4293 RO-25-6603 RO-31-3689 RO-4-8068 RO-40-3387 RO-40-6976 RO-47-5944 RO-48-2249 RO-8-4969 RO-8-8717 RO-8-9372 RO-8-9750 SMR-2 SMR-6 SR-11203 SR-11217 SR-11220 SR-11234 SR-11235 SR-11236 SR-11237 SR-11238 SR-11246 SR-11254 SR-11262 SR-11276 SR-11278 SR-11302 SR-11345 SR-11364 SRI-2712-24 SRI-4657-47 SRI-5193-34 SRI-5193-43 SRI-5387-31 SRI-5447-28 SRI-5631-96 SRI-5898-21 SRI-5898-71 SRI-6153-40 SRI-6409-94 SRI-7167-67 SRI-7323-78 ST-80 ST-88 SUMAROTENE TAZAROTENE TEMAROTENE TETRAZOLYLRETINAMIDE-N TRETINOIN TRETINOIN-METHYL-ESTER TRETINOIN-OXO-4 VITAMINS-B B-COMPLEX BIOTIN BIOTIN-METHYL-ESTER CARNITINE CHOLINE DEXPANTHENOL FOLATE FOLINATE FOLINATE CALCIUM GLYCERYL-PABA INOSITOL ISOVALERYLCARNITINE LEVOCARNITINE NICOTINAMIDE NICOTINAMIDE-ASCORBATE NICOTINAMIDE-N-OXIDE NICOTINATE NICOTINATE-BUTYL-ESTER

Derwent Drug File 1303 Thesaurus NICOTINATE-ETHYL NICOTINATE-HEXYL NICOTINATE-METHYL PABA PANTETHEINE-PHOSPHATE-= 4+ PANTETHEINE-SULFONATE PANTETHINE PANTHENOL PANTOTHENATE PANTOTHENATE CALCIUM PHOSPHOPANTOTHENATE-4+ PINITOL VITAMINS-B1 ACETIAMINE BENFOTIAMINE BISBENTIAMINE CETOTIAMINE COCARBOXYLASE CYCOTIAMINE FURSULTIAMINE HYDROXYTHIAMINE MONOPHOSPHOTHIAMINE OCTOTIAMINE THIAMINE THIAMINE-DISULFIDE THIAMINE-MONONITRATE THIAMINE-TRIPHOSPHATE VITAMINS-B12 AQUOCOBALAMIN COBAMAMIDE CYANOCOBALAMIN HYDROXOCOBALAMIN MECOBALAMIN NITROSOCOBALAMIN VITAMINS-B2 BENZAFLAVIN FAD FMN RIBOFLAVIN RIBOFLAVIN-BENZOATE RIBOFLAVIN-BUTYRATE VITAMINS-B6 FLUOROPYRIDOXAL-6 PYRIDOXAL PYRIDOXAL-PHOSPHATE PYRIDOXAMINE PYRIDOXAMINE-PHOSPHATE PYRIDOXATE PYRIDOXINE PYRIDOXINE-PHOSPHATE VITAMINS-C ASCORBATE ASCORBATE-GLUCOSIDE ASCORBATE-PHOSPHATE-2 ASCORBATE-SULFATE-2 ASCORBYL-PALMITATE ASCORBYL-POLYPHOSPHATE ASCORBYL-STEARATE DEHYDROASCORBATE NICOTINAMIDE-ASCORBATE VITAMINS-D ALFACALCIDOL CALCIFEDIOL CALCIFEROL CALCIPOTRIOL CALCITRIOL CB-1093 CB-1267 CB-966 COD-LIVER-OIL COLECALCIFEROL COLECALCIFEROL-ACETATE COLECALCIFEROL-= PROPIONATE DIHYDROERGOCALCIFEROL-= 22,23 DIHYDROTACHYSTEROL DIHYDROXYCOLE= CALCIFEROL-1-A,25,3-EPI DIHYDROXYCOLE= CALCIFEROL-1-ALPHA,24 DIHYDROXYCOLE= CALCIFEROL-1-BETA,25 DIHYDROXYCOLE= CALCIFEROL-1-BETA,25,3-= EPI DIHYDROXYCOLE= CALCIFEROL-23,25 DIHYDROXYCOLE= CALCIFEROL-24,25 DIHYDROXYCOLE= CALCIFEROL-25,26 DIHYDROXYERGO= CALCIFEROL-1-A-25,24-EPI DIHYDROXYERGO= CALCIFEROL-1-ALPHA,24 DIHYDROXYERGO= CALCIFEROL-1-ALPHA,25 DIHYDROXYERGO= CALCIFEROL-24,25 DIHYDROXYERGO= CALCIFEROL-25,26 EB-1213 EB-1231 ED-71 ERGOCALCIFEROL GS-1500 HYDROXYERGO= CALCIFEROL-1-ALPHA HYDROXYERGO= CALCIFEROL-24 HYDROXYERGO= CALCIFEROL-25 HYDROXYVITAMIN-D5,1-= ALPHA ILX-23-7553 JK-1624-2 JK-1624-3 KH-1059 KH-1060 KH-1139 KH-1230 MC-1046 MC-1080 MC-1288 MC-1301 OXACALCITRIOL-22 PARICALCITOL PRECOLECALCIFEROL RO-23-7498 RO-23-8525 RO-24-2090 RO-24-2287 RO-24-2637 RO-24-5531 RO-25-2032 RO-25-4020 RO-25-5318 RO-25-6760 RO-25-7553 RO-25-9022 RO-25-9887 RO-4020 SEOCALCITOL ST-630 TACALCITOL TRIHYDROXYCOLE= CALCIFEROL-1-ALPHA,= 23,25 TRIHYDROXYCOLE= CALCIFEROL-1-ALPHA,= 24,25 TRIHYDROXYCOLE= CALCIFEROL-1-ALPHA,= 25,26 TRIHYDROXYERGO= CALCIFEROL-1,24,25 TRIHYDROXYERGO= CALCIFEROL-1,25-28 TX-522 TX-527 ZK-156718 VITAMINS-D3 RO-23-4319 RO-23-7553 VITAMINS-E MDL-73404 MDL-74270 MDL-74366 TOCOFERSOLAN TOCOPHEROL VITAMINS-K4 MENADIOL MENADIOL-DIACETATE MENADIOL-DIBUTYRATE TOCOPHEROL-ALPHA TOCOPHEROL-ALPHA-= ACETATE TOCOPHEROL-ALPHA-= FUSARATE TOCOPHEROL-ALPHA-= LINOLENATE TOCOPHEROL-ALPHA-= NICOTINATE TOCOPHEROL-ALPHA-= PALMITATE TOCOPHEROL-ALPHA-= PHOSPHATE TOCOPHEROL-ALPHA-= STEARATE TOCOPHEROL-ALPHA-= SUCCINATE TOCOPHEROL-BETA TOCOPHEROL-DELTA TOCOPHEROL-EPSILON TOCOPHEROL-ETA TOCOPHEROL-GAMMA TOCOPHEROL-ZETA-2 TOCOPHERYLHYDROQUINONE TOCOPHERYL-QUINONE TOCOTRIENOL TOCOTRIENOL-ALPHA TOCOTRIENOL-ALPHA TOCOTRIENOL-BETA TOCOTRIENOL-DELTA TOCOTRIENOL-GAMMA VITAMINS-K VITAMIN-K5 VITAMINS-K1 PHYTOMENADIONE PHYTOMENADIONE-OXIDE VITAMINS-K2 MENAQUINONE MENAQUINONE-10 MENAQUINONE-5 MENAQUINONE-6 MENAQUINONE-7 MENAQUINONE-8 MENAQUINONE-9 MENATETRENONE VITAMINS-K3 MENADIONE MENADIONE-BISULFITE = SODIUM MENADOXIME

1304 APPENDIX D MENADIOL-DIPHOSPHATE = SODIUM MENADIOL-SULFATE SODIUM VITRONECTIN-ANTAGONISTS EMD-66203 LOTRAFIBAN SB-265123 SB-273005 VULNERARIES ACEXAMATE ARNEBIN-1 ASIATATE ASIATICOSIDE BISMUTH-SUBGALLATE BRIER-ROSE-OIL CK-103-A CLOSTRIDIOPEPTIDASE-A COLLAGENASE DERMAZELLON DEXTRANOMER DIACETYLAMINOAZOTOLUENE GELIPERM GLUTAURINE KERATINOCYTE-GROWTH-= FACTOR-2 KRILL-PROTEASES KUNITZ-PROTEASE-INHIBITOR LEVOSIN LYSOPHOSPHATIDATE MADECASSATE MADECASSOSIDE MORIKRASE MYTILAN NAKSOL PLATELET-DERIVED-= GROWTH-FACTOR-B-B PLATELET-DERIVED-= WOUND-HEALING-FACTOR POLYVINOX PROTEASE-C QUINAZOPYRINE SEK-1005 SERICATE SERICOSIDE SILVER-NITRATE SILVER-SULFACETAMIDE SILVER-SULFADIAZINE SILVER-SULFATHIAZOLE SILVER-SULFISOMIDINE SUDAN-IV SUTILAINS TETRACHLORODECAOXIDE THIOGLYCEROL TOCORETINATE TRANSFORMING-GROWTH-= FACTOR-BETA-3 TRAP-508 URTIPHYLLIN WILD-ANIMAL DOLPHIN ELK GAZELLE GIRAFFE IMPALA JAGUAR KANGAROO LEMUR MOOSE MOUFLON MUSK-OX PANDA PANTHER RACCOON REINDEER RHINOCEROS SEA-LION SQUIRREL WOOL FLEECE XANTHINE-OXIDASEINHIBITORS ALLOPURINOL AMFLUTIZOLE BOF-4272 BW-776-C-85 DEFEROXAMINE FOLATE OXIPURINOL YEAST HANSENULA NADSONIA NEMATOSPORA PICHIA RHODOTORULA SACCH. SCHWANNIOMYCES ZOOLOGY ACANTHASTER ASTERINA BUFO BUGULA CLAVULARIA CORAL CROTALUS ELECTROPHORUS EUDISTOMA GARVEIA HAEMENTERIA HALICHONDRIA HEMICENTROTUS HIRUDO HYMENIACIDON IGERNELLA LATRUNCULIA LYTECHINUS MACROBDELLA MYOCASTOR NAJA OCTOPUS PHYLLOMEDUSA PRIANUS PSAMMAPLYSILLA PSEUDOPTEROGORGIA RANA SEA-URCHIN SMENOSPONGIA SPODOPTERA STRONGYLOCENTROTUS TEALIA TELESTO TURTLE VIPERA XENOPUS ZOOTOXINS APAMIN BATRACHOTOXIN BEE-VENOM BREVETOXIN-B BUNGAROTOXIN BUNGAROTOXIN-ALPHA CALCISEPTINE CARDIOTOXIN CHARYBDOTOXIN CIGUATOXIN COBRA-VENOM COBRATOXIN CONOTOXIN-GI CROTOXIN DYSIHERBAINE ELEGANTIN ERABUTOXIN-B HOLOTHURIN-A IBERIOTOXIN JORO-TOXIN-3 KRAIT-VENOM LATRUNCULIN-A LOPHOTOXIN MASTOPARAN MCD-PEPTIDE MELITTIN NEOSURUGATOXIN OKADAATE PAHUTOXIN PALYTOXIN PEDERINE PERHYDROHISTRIONICOTOXIN PHILANTHOTOXIN-343 PHILANTHOTOXIN-433 SCORPION-VENOM SEA-ANEMONE-TOXIN-II SNAKE-VENOM SURUGATOXIN TETRODOTOXIN WASP-VENOM ZOOXANTHELLATOXIN-A

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